6BDL - chain B (model A) | Protein kinase, cGMP-dependent, type I
Structure information
PDB:6BDL
PubMed:-
Release date:2018-10-24
Resolution:1.96 Å
 
Kinase:PRKG1 (PKG1)
Family:PKG
Group:AGC
Species:HUMAN
 
Quality Score:9
Missing Residues:0
Missing Atoms:10
DFG conformation:in
αC-helix conformation:in
Salt bridge KIII.17 and EαC.24:Yes (2.9Å)
 
 
ASP rotation (xDFG.81) :347°
PHE rotation (xDFG.82) :18°
Activation loop position:-4Å
αC-helix position:17.3Å
 
G-rich loop angle:61.1°
G-rich loop distance:18.7Å
G-rich loop rotation:50.5°
Other models from this PDB:
2D & 3D views

The orthosteric binding pocket
Binding pocket waters
The following waters were found in the defined clusters:
I11
H-bond protein
Binding pocket sequence
UniprotDTLGVGGFGRVELFAMKILHIRSEKQIMQGAHDFIVRLYRTYMLMEACLGGELWTILRDYLHSKGIIYRDLKPENLILLVDFGFA
Structure:DTLGVGGFGRVELFAMKILHIRSEKQIMQGAHDFIVRLYRTYMLMEACLGGELWTILRDYLHSKGIIYRDLKPENLILLVDFGFA


Modified residues
Residue 517 (not in pocket)
Phosphorylated threonine