1GZK - chain A | V-akt murine thymoma viral oncogene homolog 2
Structure information
PDB:1GZK
PubMed:12086620
Release date:2003-05-22
Resolution:2.3 Å
 
Kinase:AKT2
Family:Akt
Group:AGC
Species:HUMAN
 
Quality Score:5.6
Missing Residues:3
Missing Atoms:30
DFG conformation:out
αC-helix conformation:in
Salt bridge KIII.17 and EαC.24:No
 
 
ASP rotation (xDFG.81) :179°
PHE rotation (xDFG.82) :232°
Activation loop position:0.9Å
αC-helix position:19.3Å
 
G-rich loop angle:60.7°
G-rich loop distance:18.2Å
G-rich loop rotation:47.2°
2D & 3D views

The orthosteric binding pocket
Binding pocket waters
The following waters were found in the defined clusters:
I3
H-bond protein
I5
H-bond protein
I6
H-bond protein
I7
H-bond protein
Binding pocket sequence
UniprotKLLGKGTFGKVILYAMKILHTVTESRVLQNTRPFLTALKYACFVMEYANGGELFFHLSRYLHSRDVVYRDIKLENLMLITDFGLC
Structure:KLLGKGTFGKVILYAMKIL__VTESRVLQNTRPFLTALKYACFVMEYANGGELFFHLSRYLHSRDVVYRDIKLENLMLITDFGL_


Modified residues
No modified residues identified.