2YHV - chain A | Anaplastic lymphoma receptor tyrosine kinase
Structure information
PDB:2YHV
PubMed:24432909
Release date:2011-05-18
Resolution:1.9 Å
 
Kinase:ALK
Family:ALK
Group:TK
Species:HUMAN
 
Quality Score:6.8
Missing Residues:3
Missing Atoms:0
DFG conformation:in
αC-helix conformation:in
Salt bridge KIII.17 and EαC.24:No (5Å)
 
 
ASP rotation (xDFG.81) :
PHE rotation (xDFG.82) :18°
Activation loop position:-4.3Å
αC-helix position:17.4Å
 
G-rich loop angle:-
G-rich loop distance:-
G-rich loop rotation:-
2D & 3D views

The orthosteric binding pocket
Binding pocket waters
The following waters were found in the defined clusters:
I1
H-bond protein
I4
H-bond protein
I6
H-bond protein
Binding pocket sequence
UniprotRGLGHGAFGEVYEVAVKTLDFLMEALIISKFNQNIVRCIGVFILLELMAGGDLKSFLREYLEENHFIHRDIAARNCLLIGDFGMA
Structure:RGL___AFGEVYEVAVKTLDFLMEALIISKFNQNIVRCIGVFILMELMAGGDLKSFLREYLEENHFIHRDIAARNCLLIGDFGMA


Modified residues
No modified residues identified.