3A7F - chain A | Serine/threonine kinase 24
Structure information
PDB:3A7F
PubMed:20124694
Release date:2010-02-02
Resolution:1.55 Å
 
Kinase:STK24 (MST3)
Family:STE20
Group:STE
Species:HUMAN
 
Quality Score:8
Missing Residues:0
Missing Atoms:0
DFG conformation:in
αC-helix conformation:in
Salt bridge KIII.17 and EαC.24:Yes (3.1Å)
 
 
ASP rotation (xDFG.81) :21°
PHE rotation (xDFG.82) :16°
Activation loop position:-3.2Å
αC-helix position:18.3Å
 
G-rich loop angle:55.6°
G-rich loop distance:15.7Å
G-rich loop rotation:93.4°
2D & 3D views

The orthosteric binding pocket
Binding pocket waters
The following waters were found in the defined clusters:
I2
H-bond protein
I4
H-bond protein
I5
H-bond protein
I6
No H-bonds
I7
No H-bonds
Binding pocket sequence
UniprotEKIGKGSFGEVFKVAIKIIDIQQEITVLSQCDPYVTKYYGSWIIMEYLGGGSALDLLEPYLHSEKKIHRDIKAANVLLLADFGVA
Structure:EKIGKGSFGEVFKVAIKIIDIQQEITVLSQCDPYVTKYYGSWIIMEYLGGGSALDLLEPYLHSEKKIHRDIKAANVLLLADFGVA


Modified residues
Residue 178 (not in pocket)
Phosphorylated threonine