3TNP - chain F | Protein kinase, cAMP dependent, catalytic, alpha
Structure information
PDB:3TNP
PubMed:22323819
Release date:2012-02-01
Resolution:2.3 Å
 
Kinase:Prkaca (PKACa)
Family:PKA
Group:AGC
Species:MOUSE
 
Quality Score:8
Missing Residues:0
Missing Atoms:0
DFG conformation:in
αC-helix conformation:in
Salt bridge KIII.17 and EαC.24:Yes (2.9Å)
 
 
ASP rotation (xDFG.81) :351°
PHE rotation (xDFG.82) :11°
Activation loop position:-4.1Å
αC-helix position:17.9Å
 
G-rich loop angle:49.5°
G-rich loop distance:15.5Å
G-rich loop rotation:54.9°
Other models from this PDB:
2D & 3D views

The orthosteric binding pocket
Binding pocket waters
The following waters were found in the defined clusters:
I1
H-bond protein
I8
H-bond protein
Binding pocket sequence
UniprotKTLGTGSFGRVMLYAMKILHTLNEKRILQAVNPFLVKLEFSYMVMEYVAGGEMFSHLRRYLHSLDLIYRDLKPENLLIVTDFGFA
Structure:KTLGTGSFGRVMLYAMKILHTLNEKRILQAVNPFLVKLEFSYMVMEYVAGGEMFSHLRRYLHSLDLIYRDLKPENLLIVTDFGFA


Modified residues
Residue 139 (not in pocket)
Phosphorylated serine
Residue 197 (not in pocket)
Phosphorylated threonine
Residue 338 (not in pocket)
Phosphorylated serine