5U7Q - chain D | Rho associated coiled-coil containing protein kinase 2
Structure information
PDB:5U7Q
PubMed:28284870
Release date:2017-03-29
Resolution:3.15 Å
 
Kinase:ROCK2
Family:DMPK
Group:AGC
Species:HUMAN
 
Quality Score:8
Missing Residues:0
Missing Atoms:0
DFG conformation:in
αC-helix conformation:in
Salt bridge KIII.17 and EαC.24:Yes (2.8Å)
 
 
ASP rotation (xDFG.81) :
PHE rotation (xDFG.82) :
Activation loop position:-4.6Å
αC-helix position:16.3Å
 
G-rich loop angle:58.2°
G-rich loop distance:17.8Å
G-rich loop rotation:77.9°
Other models from this PDB:
2D & 3D views

The orthosteric binding pocket
Binding pocket waters
No waters were found in the defined clusters
Binding pocket sequence
UniprotKVIGRGAFGEVQLYAMKLLFFWEERDIMAFANPWVVQLFYAYMVMEYMPGGDLVNLMSNAIHSMGLIHRDVKPDNMLLLADFGTC
Structure:KVIGRGAFGEVQLYAMKLLFFWEERDIMAFANPWVVQLFYAYMVMEYMPGGDLVNLMSNAIHSMGLIHRDVKPDNMLLLADFGTC


Modified residues
No modified residues identified.