5NG3 - chain A | Receptor interacting serine/threonine kinase 2
Structure information
PDB:5NG3
PubMed:28545134
Release date:2017-06-28
Resolution:2.6 Å
 
Kinase:RIPK2
Family:RIPK
Group:TKL
Species:HUMAN
 
Quality Score:8
Missing Residues:0
Missing Atoms:0
DFG conformation:in
αC-helix conformation:out
Salt bridge KIII.17 and EαC.24:No (11Å)
 
 
ASP rotation (xDFG.81) :289°
PHE rotation (xDFG.82) :313°
Activation loop position:-5.1Å
αC-helix position:21.4Å
 
G-rich loop angle:48.5°
G-rich loop distance:14.6Å
G-rich loop rotation:45.4°
Other models from this PDB:
2D & 3D views

The orthosteric binding pocket
Binding pocket waters
The following waters were found in the defined clusters:
I4
H-bond protein
I11
H-bond protein
Binding pocket sequence
UniprotRYLSRGASGTVSSVAVKHLDVLREAEILHKARSYILPILGIGIVTEYMPNGSLNELLHRHNMTPPLLHHDLKTQNILLIADFGLS
Structure:RYLSRGASGTVSSVAVRHLDVLREAEILHKARSYILPILGIGIVTEYMPNGSLNELLHRHNMTPPLLHHDLKTQNILLIADFGLS


Modified residues
Residue 111 (not in pocket)
Phosphorylated threonine