5OWQ - chain B (model B) | Serine/threonine kinase 10
Structure information
PDB:5OWQ
PubMed:-
Release date:2017-09-13
Resolution:2.7 Å
 
Kinase:STK10 (LOK)
Family:STE20
Group:STE
Species:HUMAN
 
Quality Score:6
Missing Residues:4
Missing Atoms:23
DFG conformation:na
αC-helix conformation:out
Salt bridge KIII.17 and EαC.24:No (5.3Å)
 
 
ASP rotation (xDFG.81) :°
PHE rotation (xDFG.82) :180°
Activation loop position:0Å
αC-helix position:19.7Å
 
G-rich loop angle:55.1°
G-rich loop distance:16.4Å
G-rich loop rotation:49.9°
Other models from this PDB:
2D & 3D views

The orthosteric binding pocket
Binding pocket waters
No waters were found in the defined clusters
Binding pocket sequence
UniprotGELGDGAFGKVYKAAAKVIDYIVEIEILATCDPYIVKLLGAWIMIEFCPGGAVDAIMLEFLHSKRIIHRDLKAGNVLMLADFGVS
Structure:GELGDGAFGKVYKAAAKVIDYIVEIEILATCDPYIVKLLGAWIMIEFCPGGAVDAIMLEFLHSKRIIHRDLKAGNVLMLAD____


Modified residues
No modified residues identified.
Orthosteric ligand
2D structure of the orthosteric ligand
Ligand HET-code: 38O
Ligand Name: 4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1H-benzimidazol-2-yl]quinolin-2(1H)-one

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  • LABELS
  • KLIFS residue #
  • Amino Acid
  • None
  • COLORS
  • Interaction types
  • KLIFS (all res.)
  • KLIFS (interacting res.)
  • None
  • OTHER
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This ligand targets the following (sub)pockets:
Main pockets
Front

Gate

Back

Subpockets
FP-I

FP-II

BP-I-A

BP-I-B

BP-II-in

BP-II-A-in

BP-II-B-in

BP-II-out

BP-II-B

BP-III

BP-IV

BP-V

Kinase-ligand interactions
Hydrophobic Aromatic face-to-face Aromatic face-to-edge H-bond donor H-bond acceptor Ionic positive Ionic negative
I g.l II III αC
1 G
40
2 E
41
3 L
42
4 G
43
5 D
44
6 G
45
7 A
46
8 F
47
9 G
48
10 K
49
11 V
50
12 Y
51
13 K
52
14 A
62
15 A
63
16 A
64
17 K
65
18 V
66
19 I
67
20 D
77
αC b.l IV
21 Y
78
22 I
79
23 V
80
24 E
81
25 I
82
26 E
83
27 I
84
28 L
85
29 A
86
30 T
87
31 C
88
32 D
89
33 P
91
34 Y
92
35 I
93
36 V
94
37 K
95
38 L
96
39 L
97
40 G
98
IV V GK hinge linker αD αE
41 A
99
42 W
107
43 I
108
44 M
109
45 I
110
46 E
111
47 F
112
48 C
113
49 P
114
50 G
115
51 G
116
52 A
117
53 V
118
54 D
119
55 A
120
56 I
121
57 M
122
58 L
123
59 E
124
60 F
147
αE VI c.l VII VIII x
61 L
148
62 H
149
63 S
150
64 K
151
65 R
152
66 I
153
67 I
154
68 H
155
69 R
156
70 D
157
71 L
158
72 K
159
73 A
160
74 G
161
75 N
162
76 V
163
77 L
164
78 M
165
79 L
173
80 A
174
DFG a.l
81 D
175
82 _
_
83 _
_
84 _
_
85 _
_

Interaction pattern search
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Binding affinities
ChEMBL ID:CHEMBL522892
Bioaffinities: 548 records for 206 kinase(s)

Species Kinase (ChEMBL naming) Median Min Max Type Records
Homo sapiens3-phosphoinositide dependent protein kinase-1666pKi1
Homo sapiensActivin receptor type-15.95.95.9pKi1
Homo sapiensAdaptor-associated kinase6.86.76.8pKd3
Homo sapiensALK tyrosine kinase receptor5.55.55.5pKd2
Homo sapiensALK tyrosine kinase receptor6.26.26.2pKi1
Homo sapiensAMP-activated protein kinase, alpha-1 subunit6.35.96.3pKd3
Homo sapiensAMP-activated protein kinase, alpha-1 subunit7.17.17.1pKi1
Homo sapiensAMP-activated protein kinase, alpha-2 subunit6.16.16.1pKd2
Homo sapiensAMP-activated protein kinase, gamma-1 subunit666pKd1
Homo sapiensAMP-activated protein kinase, gamma-2 subunit666pKd1
Homo sapiensAnkyrin repeat and protein kinase domain-containing protein 17.17.17.1pKd2
Homo sapiensBMP-2-inducible protein kinase7.37.27.3pKd3
Homo sapiensBone morphogenetic protein receptor type-25.55.55.5pKd2
Homo sapiensBreakpoint cluster region protein4.84.84.8pKd2
Homo sapiensBR serine/threonine-protein kinase 16.46.46.4pKi1
Plasmodium falciparumCalcium-dependent protein kinase 16.26.26.2pKd1
Homo sapiensCaM kinase I gamma999pKd1
Homo sapiensCaM kinase II delta6.56.56.5pKi1
Homo sapiensCaM kinase II gamma6.16.16.1pKi1
Homo sapiensCaM-kinase kinase alpha5.55.55.5pKd2
Homo sapiensCaM-kinase kinase beta6.86.86.8pKi1
Homo sapiensCasein kinase I delta5.85.85.8pKi1
Homo sapiensCasein kinase II alpha5.65.65.9pKd2
Homo sapiensCasein kinase II alpha (prime)5.95.86.7pKd3
Homo sapiensCitron Rho-interacting kinase5.15.15.1pKd2
Homo sapiensc-Jun N-terminal kinase 15.55.55.5pKi1
Homo sapiensc-Jun N-terminal kinase 36.26.26.2pKi1
Homo sapiensCyclin-dependent kinase 35.85.85.8pKd1
Homo sapiensCyclin-dependent kinase 45.55.55.9pKd2
Homo sapiensCyclin-dependent kinase 65.65.65.6pKd1
Homo sapiensCyclin-dependent kinase 75.65.65.6pKd2
Homo sapiensCyclin-dependent kinase 76.66.66.6pKi1
Homo sapiensCyclin-dependent kinase-like 26.86.86.8pKd1
Homo sapiensDeath-associated protein kinase 35.75.75.7pKd1
Homo sapiensDiscoidin domain-containing receptor 25.15.15.1pKd1
Homo sapiensDual specificity mitogen-activated protein kinase kinase 16.35.66.3pKd3
Homo sapiensDual specificity mitogen-activated protein kinase kinase 16.96.96.9pKi1
Homo sapiensDual specificity mitogen-activated protein kinase kinase 26.55.66.5pKd3
Homo sapiensDual specificity mitogen-activated protein kinase kinase 26.86.86.8pKi1
Homo sapiensDual specificity mitogen-activated protein kinase kinase 55.85.87.5pKd2
Homo sapiensDual specificity protein kinase CLK25.85.85.8pKd2
Homo sapiensDual specificity protein kinase CLK26.16.16.1pKi1
Homo sapiensDual specificity protein kinase CLK45.25.25.2pKd2
Homo sapiensDual specificity protein kinase CLK4777pKi1
Homo sapiensDual-specificity tyrosine-phosphorylation regulated kinase 25.25.25.2pKd1
Homo sapiensDual specificty protein kinase CLK15.25.25.2pKd2
Homo sapiensEphrin type-B receptor 66.76.76.7pKd1
Homo sapiensEpidermal growth factor receptor erbB15.95.96pKd2
Homo sapiensEpithelial discoidin domain-containing receptor 15.65.65.6pKd2
Homo sapiensEukaryotic translation initiation factor 2-alpha kinase 46.66.66.6pKd2
Homo sapiensFibroblast growth factor receptor 16.86.86.8pEC501
Homo sapiensFibroblast growth factor receptor 1888.1pIC502
Homo sapiensFibroblast growth factor receptor 16.86.66.8pKd3
Homo sapiensFibroblast growth factor receptor 17.67.67.6pKi1
Homo sapiensFibroblast growth factor receptor 26.46.46.4pKd2
Homo sapiensFibroblast growth factor receptor 38.18.18.5pIC503
Homo sapiensFibroblast growth factor receptor 36.46.46.6pKd4
Homo sapiensFibroblast growth factor receptor 37.47.47.4pKi1
Homo sapiensFibroblast growth factor receptor 45.45.45.4pKd2
Homo sapiensGlycogen synthase kinase-3 beta6.56.56.5pKd2
Homo sapiensG protein-coupled receptor kinase 4777pKd1
Homo sapiensG protein-coupled receptor kinase 75.95.95.9pKd1
Homo sapiensHomeodomain-interacting protein kinase 15.45.45.4pKd1
Homo sapiensHomeodomain-interacting protein kinase 26.36.36.3pKd1
Homo sapiensHomeodomain-interacting protein kinase 35.35.35.3pKd1
Homo sapiensHormonally up-regulated neu tumor-associated kinase6.46.46.4pKd1
Homo sapiensInhibitor of nuclear factor kappa B kinase alpha subunit5.85.85.8pKd1
Homo sapiensInhibitor of nuclear factor kappa B kinase epsilon subunit6.35.86.3pKd3
Homo sapiensInhibitor of nuclear factor kappa B kinase epsilon subunit6.16.16.1pKi1
Homo sapiensInsulin receptor5.85.85.8pKi1
Homo sapiensInterferon-induced, double-stranded RNA-activated protein kinase5.65.65.6pKd2
Homo sapiensInterleukin-1 receptor-associated kinase 16.86.86.8pKd1
Homo sapiensInterleukin-1 receptor-associated kinase 15.95.95.9pKi1
Homo sapiensInterleukin-1 receptor-associated kinase 45.75.76.9pKd2
Homo sapiensLeucine-rich repeat serine/threonine-protein kinase 25.85.86.1pKd2
Homo sapiensLeucine-rich repeat serine/threonine-protein kinase 26.56.56.5pKi1
Homo sapiensLIM domain kinase 15.75.75.7pKi1
Homo sapiensMacrophage colony stimulating factor receptor8.58.59pIC502
Homo sapiensMacrophage colony stimulating factor receptor7.27.27.2pKd2
Homo sapiensMacrophage colony stimulating factor receptor7.47.47.4pKi1
Homo sapiensMacrophage-stimulating protein receptor7.67.67.6pKi1
Homo sapiensMAP/microtubule affinity-regulating kinase 25.85.15.8pKd3
Homo sapiensMAP/microtubule affinity-regulating kinase 26.96.96.9pKi1
Homo sapiensMAP/microtubule affinity-regulating kinase 45.85.86pKd3
Homo sapiensMAP/microtubule affinity-regulating kinase 4777pKi1
Homo sapiensMaternal embryonic leucine zipper kinase5.85.55.8pKd3
Homo sapiensMaternal embryonic leucine zipper kinase7.57.57.5pKi1
Homo sapiensMicrotubule-associated serine/threonine-protein kinase 17.47.47.4pKd1
Homo sapiensMisshapen-like kinase 1778pKd2
Homo sapiensMisshapen-like kinase 1888pKi1
Homo sapiensMitogen-activated protein kinase kinase kinase 105.85.85.8pKi1
Homo sapiensMitogen-activated protein kinase kinase kinase 115.75.75.9pKd3
Homo sapiensMitogen-activated protein kinase kinase kinase 125.75.75.7pKd1
Homo sapiensMitogen-activated protein kinase kinase kinase 136.86.86.8pKd1
Homo sapiensMitogen-activated protein kinase kinase kinase 27.27.27.2pKd1
Homo sapiensMitogen-activated protein kinase kinase kinase 45.35.35.3pKd2
Homo sapiensMitogen-activated protein kinase kinase kinase 76.26.26.2pKd1
Homo sapiensMitogen-activated protein kinase kinase kinase 9555pKd2
Homo sapiensMitogen-activated protein kinase kinase kinase kinase 17.477.4pKd3
Homo sapiensMitogen-activated protein kinase kinase kinase kinase 25.55.55.7pKd2
Homo sapiensMitogen-activated protein kinase kinase kinase kinase 26.26.26.2pKi1
Homo sapiensMitogen-activated protein kinase kinase kinase kinase 36.36.16.3pKd3
Homo sapiensMitogen-activated protein kinase kinase kinase kinase 46.86.86.8pKd3
Homo sapiensMitogen-activated protein kinase kinase kinase kinase 47.67.67.6pKi1
Homo sapiensMitogen-activated protein kinase kinase kinase kinase 56.266.2pKd3
Homo sapiensMitogen-activated protein kinase kinase kinase kinase 57.57.57.5pKi1
Homo sapiensMixed lineage kinase 75.15.15.1pKi1
Homo sapiensMuscle, skeletal receptor tyrosine protein kinase6.16.16.1pKd2
Homo sapiensMyosin light chain kinase8.78.78.7pKd1
Homo sapiensmyosin light chain kinase 2777pKd2
Homo sapiensMyosin light chain kinase family member 47.17.17.1pKd2
Gallus gallusMyosin light chain kinase, smooth muscle8.78.78.7pKd1
Homo sapiensMyosin light chain kinase, smooth muscle5.55.55.5pKd2
Homo sapiensNerve growth factor receptor Trk-A75.77pKd3
Homo sapiensNerve growth factor receptor Trk-A6.66.66.6pKi1
Homo sapiensNeurotrophic tyrosine kinase receptor type 26.16.16.1pKd2
Homo sapiensNeurotrophic tyrosine kinase receptor type 2777pKi1
Homo sapiensNT-3 growth factor receptor6.76.76.7pKd2
Homo sapiensNT-3 growth factor receptor6.76.76.7pKi1
Homo sapiensNUAK family SNF1-like kinase 16.66.66.6pKd2
Homo sapiensNUAK family SNF1-like kinase 26.95.46.9pKd3
Homo sapiensPhosphatidylinositol-4-phosphate 5-kinase type-1 alpha5.75.75.7pKd2
Homo sapiensPhosphatidylinositol-4-phosphate 5-kinase type-1 gamma5.45.45.4pKd1
Homo sapiensPhosphatidylinositol-5-phosphate 4-kinase type-2 beta6.66.66.6pKd2
Homo sapiensPhosphorylase kinase gamma subunit 16.26.26.2pKd2
Homo sapiensPhosphorylase kinase gamma subunit 25.15.15.1pKd2
Homo sapiensPhosphorylase kinase gamma subunit 2666pKi1
Homo sapiensPlatelet-derived growth factor receptor alpha7.37.37.3pKd2
Homo sapiensPlatelet-derived growth factor receptor alpha6.66.66.6pKi1
Homo sapiensPlatelet-derived growth factor receptor beta7.37.37.3pEC501
Homo sapiensPlatelet-derived growth factor receptor beta8.38.39pIC502
Homo sapiensPlatelet-derived growth factor receptor beta8.47.58.4pKd3
Homo sapiensPlatelet-derived growth factor receptor beta8.28.28.2pKi1
Homo sapiensProtein kinase C delta5.75.75.7pKi1
Homo sapiensProtein kinase C nu5.95.95.9pKi1
Homo sapiensProtein kinase C theta5.55.55.5pKd2
Homo sapiensProtein kinase N16.85.16.8pKd3
Homo sapiensProtein kinase N2555pKd2
Homo sapiensProtein kinase N26.26.26.2pKi1
Homo sapiensProto-oncogene tyrosine-protein kinase MER5.85.85.8pKd2
Homo sapiensReceptor-interacting serine/threonine-protein kinase 16.56.56.5pKd2
Homo sapiensRho-associated protein kinase 16.16.16.1pKd1
Homo sapiensRho-associated protein kinase 25.55.55.5pKd1
Homo sapiensRho-associated protein kinase 25.45.45.4pKi1
Homo sapiensRhodopsin kinase5.75.75.7pKd1
Homo sapiensRibosomal protein S6 kinase 16.26.26.2pKd1
Homo sapiensRibosomal protein S6 kinase 1777pKi1
Homo sapiensRibosomal protein S6 kinase alpha 16.45.66.4pKd6
Homo sapiensRibosomal protein S6 kinase alpha 26.56.56.5pKd4
Homo sapiensRibosomal protein S6 kinase alpha 35.35.35.3pKd6
Homo sapiensRibosomal protein S6 kinase alpha 36.56.56.5pKi2
Homo sapiensRibosomal protein S6 kinase alpha 46.26.26.4pKd6
Homo sapiensRibosomal protein S6 kinase alpha 56.26.26.2pKd4
Homo sapiensRibosomal protein S6 kinase alpha 5666pKi2
Homo sapiensRibosomal protein S6 kinase alpha 65.35.35.3pKd4
Homo sapiensSerine/threonine-protein kinase 106.36.36.3pKd2
Homo sapiensSerine/threonine-protein kinase 115.45.45.4pKd2
Homo sapiensSerine/threonine-protein kinase 165.85.85.8pKd1
Homo sapiensSerine/threonine-protein kinase 17A6.16.16.1pKd2
Homo sapiensSerine/threonine-protein kinase 17B5.85.85.8pKd2
Homo sapiensSerine/threonine-protein kinase 26.56.56.5pKd2
Homo sapiensSerine/threonine-protein kinase 26.76.76.7pKi1
Homo sapiensSerine/threonine-protein kinase 246.46.46.4pKd2
Homo sapiensSerine/threonine-protein kinase 255.95.95.9pKd2
Homo sapiensSerine/threonine-protein kinase 386.26.26.2pKd1
Homo sapiensSerine/threonine-protein kinase Aurora-B6.666.6pKd3
Homo sapiensSerine/threonine-protein kinase Aurora-B7.17.17.1pKi1
Homo sapiensSerine/threonine-protein kinase Aurora-C666pKd2
Homo sapiensSerine/threonine-protein kinase Chk15.95.55.9pKd3
Homo sapiensSerine/threonine-protein kinase Chk16.86.86.8pKi1
Homo sapiensSerine/threonine-protein kinase Chk25.85.85.8pKi1
Homo sapiensSerine/threonine-protein kinase c-TAK15.555.5pKd3
Homo sapiensSerine/threonine-protein kinase c-TAK16.96.96.9pKi1
Homo sapiensSerine/threonine-protein kinase D25.75.75.7pKi1
Homo sapiensSerine/threonine-protein kinase DCLK35.95.95.9pKd2
Homo sapiensSerine/threonine-protein kinase GAK6.35.76.3pKd3
Homo sapiensSerine/threonine-protein kinase LATS15.85.86pKd3
Homo sapiensSerine/threonine-protein kinase LATS26.36.36.3pKd2
Homo sapiensSerine/threonine-protein kinase MARK15.65.65.6pKd2
Homo sapiensSerine/threonine-protein kinase MST16.766.7pKd3
Homo sapiensSerine/threonine-protein kinase MST26.35.76.3pKd3
Homo sapiensSerine/threonine-protein kinase MST26.76.76.7pKi1
Homo sapiensSerine/threonine-protein kinase MST46.36.36.3pKd2
Homo sapiensSerine/threonine-protein kinase NEK25.75.75.7pKd2
Homo sapiensSerine/threonine-protein kinase NEK26.36.36.3pKi1
Homo sapiensSerine/threonine-protein kinase Nek45.65.65.6pKd1
Homo sapiensSerine/threonine-protein kinase Nek45.35.35.3pKi1
Homo sapiensSerine/threonine-protein kinase Nek55.65.65.6pKd2
Homo sapiensSerine/threonine-protein kinase NEK65.85.85.8pKd2
Homo sapiensSerine/threonine-protein kinase NEK75.35.35.3pKd2
Homo sapiensSerine/threonine-protein kinase NEK9555.7pKd3
Homo sapiensSerine/threonine-protein kinase NIM16.16.16.1pKd1
Homo sapiensSerine/threonine-protein kinase PAK 36.16.16.1pKd1
Homo sapiensSerine/threonine-protein kinase PAK 45.75.75.7pKi1
Homo sapiensSerine/threonine-protein kinase PCTAIRE-16.46.46.4pKd2
Homo sapiensSerine/threonine-protein kinase PCTAIRE-25.55.55.5pKd2
Homo sapiensSerine/threonine-protein kinase PCTAIRE-35.15.15.1pKd1
Homo sapiensSerine/threonine-protein kinase PIM25.95.95.9pKi1
Mycobacterium tuberculosisSerine/threonine-protein kinase pknB6.56.56.5pKd1
Homo sapiensSerine/threonine-protein kinase PLK26.26.26.2pKd1
Homo sapiensSerine/threonine-protein kinase PLK45.95.95.9pKi1
Homo sapiensSerine/threonine-protein kinase PRKX5.85.85.8pKi1
Homo sapiensSerine/threonine-protein kinase PRP4 homolog6.36.36.3pKd1
Homo sapiensSerine/threonine-protein kinase RIO16.46.46.4pKd2
Homo sapiensSerine/threonine-protein kinase RIO26.66.66.6pKd1
Homo sapiensSerine/threonine-protein kinase RIO36.26.26.2pKd2
Homo sapiensSerine/threonine-protein kinase SBK15.85.85.8pKd1
Homo sapiensSerine/threonine-protein kinase Sgk25.95.95.9pKi1
Homo sapiensSerine/threonine-protein kinase Sgk3666pKd1
Homo sapiensSerine/threonine-protein kinase SIK25.45.45.4pKd2
Homo sapiensSerine/threonine-protein kinase SIK2777pKi1
Homo sapiensSerine/threonine-protein kinase SRPK16.46.46.4pKd2
Homo sapiensSerine/threonine-protein kinase SRPK15.35.35.3pKi1
Homo sapiensSerine/threonine-protein kinase SRPK26.56.56.5pKd2
Homo sapiensSerine/threonine-protein kinase SRPK36.66.66.6pKd1
Homo sapiensSerine/threonine-protein kinase TBK1666.9pKd2
Homo sapiensSerine/threonine-protein kinase tousled-like 25.65.65.6pKd2
Homo sapiensSerine/threonine-protein kinase ULK16.16.17.3pKd2
Homo sapiensSerine/threonine-protein kinase ULK27.37.37.3pKd1
Homo sapiensSerine/threonine-protein kinase ULK3666.8pKd2
Homo sapiensSerine/threonine-protein kinase WEE15.95.15.9pKd3
Homo sapiensSPS1/STE20-related protein kinase YSK47.97.97.9pKd1
Homo sapiensSTE20/SPS1-related proline-alanine-rich protein kinase6.36.36.3pKd1
Homo sapiensStem cell growth factor receptor8.57.39pIC504
Homo sapiensStem cell growth factor receptor8.15.98.8pKd15
Homo sapiensStem cell growth factor receptor7.77.77.7pKi1
Homo sapiensTestis-specific serine/threonine-protein kinase 16.36.36.3pKi1
Homo sapiensTRAF2- and NCK-interacting kinase8.17.28.7pIC503
Homo sapiensTRAF2- and NCK-interacting kinase7.67.67.6pKd3
Homo sapiensTyrosine-protein kinase ABL6.46.46.6pIC502
Homo sapiensTyrosine-protein kinase ABL6.25.27.5pKd22
Homo sapiensTyrosine-protein kinase ABL777pKi1
Homo sapiensTyrosine-protein kinase ABL2666pKd1
Homo sapiensTyrosine-protein kinase BLK6.76.76.7pKd2
Homo sapiensTyrosine-protein kinase BLK7.97.97.9pKi1
Homo sapiensTyrosine-protein kinase BTK5.75.75.7pKi1
Homo sapiensTyrosine-protein kinase FGR6.76.76.7pKd2
Homo sapiensTyrosine-protein kinase FRK5.65.65.6pKd2
Homo sapiensTyrosine-protein kinase FYN6.46.16.4pKd3
Homo sapiensTyrosine-protein kinase FYN7.27.27.2pKi1
Homo sapiensTyrosine-protein kinase HCK5.55.56pKd3
Homo sapiensTyrosine-protein kinase HCK6.86.86.8pKi1
Homo sapiensTyrosine-protein kinase ITK/TSK6.36.36.3pKd2
Homo sapiensTyrosine-protein kinase ITK/TSK7.37.37.3pKi1
Homo sapiensTyrosine-protein kinase JAK16.46.46.4pKd6
Homo sapiensTyrosine-protein kinase JAK25.25.26.9pKd4
Homo sapiensTyrosine-protein kinase JAK2666pKi2
Homo sapiensTyrosine-protein kinase JAK35.15.16.4pKd4
Homo sapiensTyrosine-protein kinase LCK6.66.26.6pKd3
Homo sapiensTyrosine-protein kinase LCK7.77.77.7pKi1
Homo sapiensTyrosine-protein kinase Lyn6.16.16.1pKd3
Homo sapiensTyrosine-protein kinase Lyn7.27.27.2pKi1
Homo sapiensTyrosine-protein kinase receptor FLT38.58.59pIC502
Homo sapiensTyrosine-protein kinase receptor FLT38.38.19.5pKd13
Homo sapiensTyrosine-protein kinase receptor FLT38.58.58.5pKi1
Homo sapiensTyrosine-protein kinase receptor RET7.37.27.6pKd7
Homo sapiensTyrosine-protein kinase receptor RET8.38.38.3pKi1
Homo sapiensTyrosine-protein kinase receptor Tie-15.45.45.4pKd2
Homo sapiensTyrosine-protein kinase receptor TYRO3555pKd2
Homo sapiensTyrosine-protein kinase receptor TYRO37.37.37.3pKi1
Homo sapiensTyrosine-protein kinase receptor UFO5.45.45.4pKd2
Homo sapiensTyrosine-protein kinase receptor UFO6.66.66.6pKi1
Gallus gallusTyrosine-protein kinase SRC7.17.17.1pIC501
Homo sapiensTyrosine-protein kinase SRC5.85.86.2pKd3
Homo sapiensTyrosine-protein kinase SRC7.27.27.2pKi1
Homo sapiensTyrosine-protein kinase TYK25.75.76.8pKd4
Homo sapiensTyrosine-protein kinase TYK26.76.76.7pKi2
Homo sapiensTyrosine-protein kinase YES7.57.58.9pIC502
Homo sapiensTyrosine-protein kinase YES6.26.26.2pKd3
Homo sapiensVascular endothelial growth factor receptor 1888.5pIC502
Homo sapiensVascular endothelial growth factor receptor 17.27.27.2pKd2
Homo sapiensVascular endothelial growth factor receptor 17.47.47.4pKi1
Homo sapiensVascular endothelial growth factor receptor 27.37.37.3pEC501
Homo sapiensVascular endothelial growth factor receptor 27.97.27.9pIC503
Homo sapiensVascular endothelial growth factor receptor 27.27.27.2pKd2
Homo sapiensVascular endothelial growth factor receptor 27.77.77.7pKi1
Homo sapiensVascular endothelial growth factor receptor 38.58.18.6pIC503
Homo sapiensVascular endothelial growth factor receptor 36.26.26.2pKd2
Homo sapiensVascular endothelial growth factor receptor 3777pKi1