er KLIFS - the kinase structures database

Browse kinase structures

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetailsFile
AAK1NAKOther4wsqAAk-252aHuman3834
AAK1NAKOther4wsqABk-252aHuman3836
AAK1NAKOther4wsqBAk-252aHuman3833
AAK1NAKOther4wsqBBk-252aHuman3835
AAK1NAKOther5l4qAA~{n}-[5-(4-cyanophenyl)-1~{h}-pyrrolo[2,3-b]pyridin-3-yl]pyridine-3-carboxamideHuman6679
AAK1NAKOther5l4qAB~{n}-[5-(4-cyanophenyl)-1~{h}-pyrrolo[2,3-b]pyridin-3-yl]pyridine-3-carboxamideHuman6677
AAK1NAKOther5l4qBA~{n}-[5-(4-cyanophenyl)-1~{h}-pyrrolo[2,3-b]pyridin-3-yl]pyridine-3-carboxamideHuman6680
AAK1NAKOther5l4qBB~{n}-[5-(4-cyanophenyl)-1~{h}-pyrrolo[2,3-b]pyridin-3-yl]pyridine-3-carboxamideHuman6678
AAK1NAKOther5te0Amethyl (3z)-3-{[(4-{methyl[(4-methylpiperazin-1-yl)acetyl]amino}phenyl)amino](phenyl)methylidene}-2-oxo-2,3-dihydro-1h-indole-6-carboxylateHuman7156
Abl1 (ABL1)AblTK1fpuAn-[4-methyl-3-[[4-(3-pyridinyl)-2-pyrimidinyl]amino]phenyl]-3-pyridinecarboxamideMouse5728
Abl1 (ABL1)AblTK1fpuBn-[4-methyl-3-[[4-(3-pyridinyl)-2-pyrimidinyl]amino]phenyl]-3-pyridinecarboxamideMouse5705
Abl1 (ABL1)AblTK1iepA4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideMouse5703
Abl1 (ABL1)AblTK1iepB4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideMouse5727
Abl1 (ABL1)AblTK1m52A6-(2,6-dichloro-phenyl)-8-methyl-2-(3-methylsulfanyl-phenylamino)-8h-pyrido[2,3-d]pyrimidin-7-oneMouse5720
Abl1 (ABL1)AblTK1m52B6-(2,6-dichloro-phenyl)-8-methyl-2-(3-methylsulfanyl-phenylamino)-8h-pyrido[2,3-d]pyrimidin-7-oneMouse5715
Abl1 (ABL1)AblTK1opjA4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideMouse5732
Abl1 (ABL1)AblTK1opjB4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideMouse5736
Abl1 (ABL1)AblTK1opkA6-(2,6-dichlorophenyl)-2-{[3-(hydroxymethyl)phenyl]amino}-8-methylpyrido[2,3-d]pyrimidin-7(8h)-oneMouse5709
Abl1 (ABL1)AblTK2hznA1-[4-(pyridin-4-yloxy)phenyl]-3-[3-(trifluoromethyl)phenyl]ureaMouse5701
Abl1 (ABL1)AblTK2qohA5-[3-(2-methoxyphenyl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylpyridine-3-carboxamideMouse5707
Abl1 (ABL1)AblTK2qohB5-[3-(2-methoxyphenyl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylpyridine-3-carboxamideMouse5716
Abl1 (ABL1)AblTK2z60A5-[3-(2-methoxyphenyl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylpyridine-3-carboxamideMouse5735
Abl1 (ABL1)AblTK3dk3AA2-amino-5-[3-(1-ethyl-1h-pyrazol-5-yl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylbenzamideMouse5726
Abl1 (ABL1)AblTK3dk3AB2-amino-5-[3-(1-ethyl-1h-pyrazol-5-yl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylbenzamideMouse5729
Abl1 (ABL1)AblTK3dk3BA2-amino-5-[3-(1-ethyl-1h-pyrazol-5-yl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylbenzamideMouse5712
Abl1 (ABL1)AblTK3dk3BB2-amino-5-[3-(1-ethyl-1h-pyrazol-5-yl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylbenzamideMouse5737
Abl1 (ABL1)AblTK3dk6A2-amino-5-[3-(1-ethyl-1h-pyrazol-5-yl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylbenzamideMouse5725
Abl1 (ABL1)AblTK3dk6B2-amino-5-[3-(1-ethyl-1h-pyrazol-5-yl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylbenzamideMouse5718
Abl1 (ABL1)AblTK3dk7A2-amino-5-[3-(1-ethyl-1h-pyrazol-5-yl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylbenzamideMouse5704
Abl1 (ABL1)AblTK3dk7B2-amino-5-[3-(1-ethyl-1h-pyrazol-5-yl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylbenzamideMouse5714
Abl1 (ABL1)AblTK3ik3A3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideMouse5731
Abl1 (ABL1)AblTK3ik3B3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideMouse5739
Abl1 (ABL1)AblTK3k5vAA4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideMouse5734
Abl1 (ABL1)AblTK3k5vAB4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideMouse5723
Abl1 (ABL1)AblTK3k5vBA4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideMouse5710
Abl1 (ABL1)AblTK3k5vBB4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideMouse5722
Abl1 (ABL1)AblTK3kf4An-[4-(dimethylphosphoryl)phenyl]-9-[(e)-2-(5-methyl-1h-indazol-4-yl)ethenyl]-9h-purin-6-amineMouse5717
Abl1 (ABL1)AblTK3kf4Bn-[4-(dimethylphosphoryl)phenyl]-9-[(e)-2-(5-methyl-1h-indazol-4-yl)ethenyl]-9h-purin-6-amineMouse5741
Abl1 (ABL1)AblTK3kfaA3-{(e)-2-[6-(cyclopropylamino)-9h-purin-9-yl]ethenyl}-4-methyl-n-[3-(4-methyl-1h-imidazol-1-yl)-5-(trifluoromethyl)phenyl]benzamideMouse5742
Abl1 (ABL1)AblTK3kfaB3-{(e)-2-[6-(cyclopropylamino)-9h-purin-9-yl]ethenyl}-4-methyl-n-[3-(4-methyl-1h-imidazol-1-yl)-5-(trifluoromethyl)phenyl]benzamideMouse5740
Abl1 (ABL1)AblTK3ms9AA4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideMouse5733
Abl1 (ABL1)AblTK3ms9AB4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideMouse5708
Abl1 (ABL1)AblTK3ms9BA4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideMouse5713
Abl1 (ABL1)AblTK3ms9BB4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideMouse5706
Abl1 (ABL1)AblTK3mssA4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideMouse5724
Abl1 (ABL1)AblTK3mssB4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideMouse5730
Abl1 (ABL1)AblTK3mssC4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideMouse5719
Abl1 (ABL1)AblTK3mssD4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideMouse5702
Abl1 (ABL1)AblTK3oxzA3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideMouse5721
Abl1 (ABL1)AblTK3oy3A5-[(5-{[4-{[4-(2-hydroxyethyl)piperazin-1-yl]methyl}-3-(trifluoromethyl)phenyl]carbamoyl}-2-methylphenyl)ethynyl]-1-methyl-1h-imidazole-2-carboxamideMouse5711
Abl1 (ABL1)AblTK3oy3B5-[(5-{[4-{[4-(2-hydroxyethyl)piperazin-1-yl]methyl}-3-(trifluoromethyl)phenyl]carbamoyl}-2-methylphenyl)ethynyl]-1-methyl-1h-imidazole-2-carboxamideMouse5738
Abl1 (ABL1)AblTK6hd4AA4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideMouse10645
Abl1 (ABL1)AblTK6hd4AB4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideMouse10647
Abl1 (ABL1)AblTK6hd4BA4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideMouse10648
Abl1 (ABL1)AblTK6hd4BB4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideMouse10646
Abl1 (ABL1)AblTK6hd6AA4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideMouse10609
Abl1 (ABL1)AblTK6hd6AB4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideMouse10608
Abl1 (ABL1)AblTK6hd6BA4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideMouse10611
Abl1 (ABL1)AblTK6hd6BB4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideMouse10610
ABL1AblTK1oplA6-(2,6-dichlorophenyl)-2-{[3-(hydroxymethyl)phenyl]amino}-8-methylpyrido[2,3-d]pyrimidin-7(8h)-oneHuman1104
ABL1AblTK1oplB6-(2,6-dichlorophenyl)-2-{[3-(hydroxymethyl)phenyl]amino}-8-methylpyrido[2,3-d]pyrimidin-7(8h)-oneHuman1086
ABL1AblTK2e2bAn-[3-(4,5'-bipyrimidin-2-ylamino)-4-methylphenyl]-4-{[(3s)-3-(dimethylamino)pyrrolidin-1-yl]methyl}-3-(trifluoromethyl)benzamideHuman1054
ABL1AblTK2e2bBn-[3-(4,5'-bipyrimidin-2-ylamino)-4-methylphenyl]-4-{[(3s)-3-(dimethylamino)pyrrolidin-1-yl]methyl}-3-(trifluoromethyl)benzamideHuman1065
ABL1AblTK2f4jAcyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amideHuman1090
ABL1AblTK2fo0A6-(2,6-dichlorophenyl)-2-{[3-(hydroxymethyl)phenyl]amino}-8-methylpyrido[2,3-d]pyrimidin-7(8h)-oneHuman1073
ABL1AblTK2g1tA-Human1045
ABL1AblTK2g1tB-Human1105
ABL1AblTK2g1tC-Human1064
ABL1AblTK2g1tD-Human1096
ABL1AblTK2g2fA-Human1097
ABL1AblTK2g2fBphosphothiophosphoric acid-adenylate esterHuman1079
ABL1AblTK2g2hA6-(2,6-dichlorophenyl)-2-{[3-(hydroxymethyl)phenyl]amino}-8-methylpyrido[2,3-d]pyrimidin-7(8h)-oneHuman1106
ABL1AblTK2g2hB6-(2,6-dichlorophenyl)-2-{[3-(hydroxymethyl)phenyl]amino}-8-methylpyrido[2,3-d]pyrimidin-7(8h)-oneHuman1089
ABL1AblTK2g2iAadenosine-5'-diphosphateHuman1111
ABL1AblTK2g2iBadenosine-5'-diphosphateHuman1075
ABL1AblTK2gqgAAn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman1060
ABL1AblTK2gqgABn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman1053
ABL1AblTK2gqgBAn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman1084
ABL1AblTK2gqgBBn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman1082
ABL1AblTK2hiwA7-amino-1-methyl-3-(2-methyl-5-{[3-(trifluoromethyl)benzoyl]amino}phenyl)-2-oxo-2,3-dihydropyrimido[4,5-d]pyrimidin-1-iumHuman1069
ABL1AblTK2hiwB7-amino-1-methyl-3-(2-methyl-5-{[3-(trifluoromethyl)benzoyl]amino}phenyl)-2-oxo-2,3-dihydropyrimido[4,5-d]pyrimidin-1-iumHuman1110
ABL1AblTK2hyyA4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman1092
ABL1AblTK2hyyB4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman1078
ABL1AblTK2hyyC4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman1048
ABL1AblTK2hyyD4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman1068
ABL1AblTK2hz0AA2-{[(6-oxo-1,6-dihydropyridin-3-yl)methyl]amino}-n-[4-propyl-3-(trifluoromethyl)phenyl]benzamideHuman1052
ABL1AblTK2hz0AB2-{[(6-oxo-1,6-dihydropyridin-3-yl)methyl]amino}-n-[4-propyl-3-(trifluoromethyl)phenyl]benzamideHuman1083
ABL1AblTK2hz0BA2-{[(6-oxo-1,6-dihydropyridin-3-yl)methyl]amino}-n-[4-propyl-3-(trifluoromethyl)phenyl]benzamideHuman1095
ABL1AblTK2hz0BB2-{[(6-oxo-1,6-dihydropyridin-3-yl)methyl]amino}-n-[4-propyl-3-(trifluoromethyl)phenyl]benzamideHuman1109
ABL1AblTK2hz4A-Human1059
ABL1AblTK2hz4B1,2,3,4-tetrahydrogen-staurosporineHuman1058
ABL1AblTK2hz4C-Human1067
ABL1AblTK2hziAA6-(2,6-dichlorophenyl)-2-[(4-fluoro-3-methylphenyl)amino]-8-methylpyrido[2,3-d]pyrimidin-7(8h)-oneHuman1102
ABL1AblTK2hziAB6-(2,6-dichlorophenyl)-2-[(4-fluoro-3-methylphenyl)amino]-8-methylpyrido[2,3-d]pyrimidin-7(8h)-oneHuman1087
ABL1AblTK2hziBA6-(2,6-dichlorophenyl)-2-[(4-fluoro-3-methylphenyl)amino]-8-methylpyrido[2,3-d]pyrimidin-7(8h)-oneHuman1108
ABL1AblTK2hziBB6-(2,6-dichlorophenyl)-2-[(4-fluoro-3-methylphenyl)amino]-8-methylpyrido[2,3-d]pyrimidin-7(8h)-oneHuman1055
ABL1AblTK2v7aAn-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamideHuman1088
ABL1AblTK2v7aBn-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamideHuman1072
ABL1AblTK3cs9AAnilotinibHuman1080
ABL1AblTK3cs9ABnilotinibHuman1107
ABL1AblTK3cs9BAnilotinibHuman1050
ABL1AblTK3cs9BBnilotinibHuman1112
ABL1AblTK3cs9CAnilotinibHuman1046
ABL1AblTK3cs9CBnilotinibHuman1093
ABL1AblTK3cs9DAnilotinibHuman1077
ABL1AblTK3cs9DBnilotinibHuman1066
ABL1AblTK3pyyAA4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman1049
ABL1AblTK3pyyAB4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman1071
ABL1AblTK3pyyBA4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman1062
ABL1AblTK3pyyBB4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman1098
ABL1AblTK3qriAA4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamideHuman1051
ABL1AblTK3qriAB4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamideHuman1047
ABL1AblTK3qriBA4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamideHuman1103
ABL1AblTK3qriBB4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamideHuman1076
ABL1AblTK3qrjAA4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamideHuman1085
ABL1AblTK3qrjAB4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamideHuman1099
ABL1AblTK3qrjBA4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamideHuman1101
ABL1AblTK3qrjBB4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamideHuman1070
ABL1AblTK3qrkA(3s)-6-(3-tert-butyl-5-{[(2,3-dichlorophenyl)carbamoyl]amino}-1h-pyrazol-1-yl)-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acidHuman1056
ABL1AblTK3ue4A4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrileHuman1057
ABL1AblTK3ue4B4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrileHuman1074
ABL1AblTK4twpAaxitinibHuman1091
ABL1AblTK4twpBaxitinibHuman1081
ABL1AblTK4wa9AaxitinibHuman1061
ABL1AblTK4wa9BaxitinibHuman1063
ABL1AblTK4xeyAn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman1094
ABL1AblTK4xeyBn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman1100
ABL1AblTK4yc8A2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-n-(4-phenoxyphenyl)-1,3-thiazole-5-carboxamideHuman6419
ABL1AblTK4yc8B2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-n-(4-phenoxyphenyl)-1,3-thiazole-5-carboxamideHuman6420
ABL1AblTK4zogAcyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amideHuman7043
ABL1AblTK4zogBcyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amideHuman7042
ABL1AblTK5hu9AA4-[(4-methylpiperazin-1-yl)methyl]-n-(4-methyl-3-{[1-(pyridin-3-ylcarbonyl)piperidin-4-yl]oxy}phenyl)-3-(trifluoromethyl)benzamideHuman6754
ABL1AblTK5hu9AB4-[(4-methylpiperazin-1-yl)methyl]-n-(4-methyl-3-{[1-(pyridin-3-ylcarbonyl)piperidin-4-yl]oxy}phenyl)-3-(trifluoromethyl)benzamideHuman6755
ABL1AblTK5mo4AAnilotinibHuman7527
ABL1AblTK5mo4ABnilotinibHuman7526
ABL1AblTK6bl8AApurvalanol bHuman9699
ABL1AblTK6bl8ABpurvalanol bHuman9698
ABL1AblTK6bl8BApurvalanol bHuman9701
ABL1AblTK6bl8BBpurvalanol bHuman9700
ABL1AblTK6npeAA4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman10946
ABL1AblTK6npeAB4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman10943
ABL1AblTK6npeBA4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman10947
ABL1AblTK6npeBB4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman10945
ABL1AblTK6npuA4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman10942
ABL1AblTK6npuB4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman10944
ABL1AblTK6npvAA4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman10948
ABL1AblTK6npvAB4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman10951
ABL1AblTK6npvBA4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman10949
ABL1AblTK6npvBB4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman10950
Abl2 (ABL2)AblTK4xliAn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideMouse5689
Abl2 (ABL2)AblTK4xliBn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideMouse5690
ABL2AblTK2xynAAcyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amideHuman110
ABL2AblTK2xynABcyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amideHuman112
ABL2AblTK2xynBAcyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amideHuman111
ABL2AblTK2xynBBcyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amideHuman113
ABL2AblTK2xynCAcyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amideHuman116
ABL2AblTK2xynCBcyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amideHuman114
ABL2AblTK3gvuAA4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman117
ABL2AblTK3gvuAB4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman109
ABL2AblTK3hmiAA5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamideHuman115
ABL2AblTK3hmiAB5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamideHuman118
ACVR1 (ALK2)STKRTKL3h9rA6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHuman1531
ACVR1 (ALK2)STKRTKL3mtfAA3-[6-amino-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenolHuman1513
ACVR1 (ALK2)STKRTKL3mtfAB3-[6-amino-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenolHuman1521
ACVR1 (ALK2)STKRTKL3mtfBA3-[6-amino-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenolHuman1515
ACVR1 (ALK2)STKRTKL3mtfBB3-[6-amino-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenolHuman1530
ACVR1 (ALK2)STKRTKL3oomAA1-{3-[6-(tetrahydro-2h-pyran-4-ylamino)imidazo[1,2-b]pyridazin-3-yl]phenyl}ethanoneHuman1517
ACVR1 (ALK2)STKRTKL3oomAB1-{3-[6-(tetrahydro-2h-pyran-4-ylamino)imidazo[1,2-b]pyridazin-3-yl]phenyl}ethanoneHuman1518
ACVR1 (ALK2)STKRTKL3q4uAA4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1527
ACVR1 (ALK2)STKRTKL3q4uAB4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1524
ACVR1 (ALK2)STKRTKL3q4uBA4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1510
ACVR1 (ALK2)STKRTKL3q4uBB4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1523
ACVR1 (ALK2)STKRTKL3q4uCA4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1516
ACVR1 (ALK2)STKRTKL3q4uCB4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1533
ACVR1 (ALK2)STKRTKL3q4uDA4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1520
ACVR1 (ALK2)STKRTKL3q4uDB4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1529
ACVR1 (ALK2)STKRTKL4bggAA1-{4-[5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl}piperazineHuman1528
ACVR1 (ALK2)STKRTKL4bggAB1-{4-[5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl}piperazineHuman1508
ACVR1 (ALK2)STKRTKL4bggBA1-{4-[5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl}piperazineHuman1514
ACVR1 (ALK2)STKRTKL4bggBB1-{4-[5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl}piperazineHuman1526
ACVR1 (ALK2)STKRTKL4bggCA1-{4-[5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl}piperazineHuman1511
ACVR1 (ALK2)STKRTKL4bggCB1-{4-[5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl}piperazineHuman1522
ACVR1 (ALK2)STKRTKL4bggDA1-{4-[5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl}piperazineHuman1519
ACVR1 (ALK2)STKRTKL4bggDB1-{4-[5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl}piperazineHuman1512
ACVR1 (ALK2)STKRTKL4c02AA6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHuman1525
ACVR1 (ALK2)STKRTKL4c02AB6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHuman1532
ACVR1 (ALK2)STKRTKL4dymA1-(3-{6-[(cyclopropylmethyl)amino]imidazo[1,2-b]pyridazin-3-yl}phenyl)ethanoneHuman1509
ACVR1 (ALK2)STKRTKL5oxgAA5-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman8514
ACVR1 (ALK2)STKRTKL5oxgAB5-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman8518
ACVR1 (ALK2)STKRTKL5oxgBA5-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman8516
ACVR1 (ALK2)STKRTKL5oxgBB5-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman8519
ACVR1 (ALK2)STKRTKL5oxgCA5-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman8517
ACVR1 (ALK2)STKRTKL5oxgCB5-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman8513
ACVR1 (ALK2)STKRTKL5oxgDA5-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman8520
ACVR1 (ALK2)STKRTKL5oxgDB5-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman8515
ACVR1 (ALK2)STKRTKL5oy6Acyclical inhibitor od36Human8532
ACVR1 (ALK2)STKRTKL5oy6Bcyclical inhibitor od36Human8531
ACVR1 (ALK2)STKRTKL5oy6Ccyclical inhibitor od36Human8529
ACVR1 (ALK2)STKRTKL5oy6Dcyclical inhibitor od36Human8534
ACVR1 (ALK2)STKRTKL6acrAn-(4-methoxyphenyl)-4-[3-(pyridin-3-yl)-1h-pyrazol-4-yl]pyrimidin-2-amineHuman10969
ACVR1 (ALK2)STKRTKL6acrBn-(4-methoxyphenyl)-4-[3-(pyridin-3-yl)-1h-pyrazol-4-yl]pyrimidin-2-amineHuman10968
ACVR1 (ALK2)STKRTKL6eixAA3-[6-amino-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenolHuman8530
ACVR1 (ALK2)STKRTKL6eixAB3-[6-amino-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenolHuman8533
ACVR1 (ALK2)STKRTKL6gi6A5-methyl-6-quinolin-5-yl-3~{h}-quinazolin-4-oneHuman9919
ACVR1 (ALK2)STKRTKL6ginAA3-(4-morpholin-4-ylphenyl)-6-quinolin-4-yl-quinazolin-4-oneHuman9914
ACVR1 (ALK2)STKRTKL6ginAB3-(4-morpholin-4-ylphenyl)-6-quinolin-4-yl-quinazolin-4-oneHuman9918
ACVR1 (ALK2)STKRTKL6ginBA3-(4-morpholin-4-ylphenyl)-6-quinolin-4-yl-quinazolin-4-oneHuman9920
ACVR1 (ALK2)STKRTKL6ginBB3-(4-morpholin-4-ylphenyl)-6-quinolin-4-yl-quinazolin-4-oneHuman9916
ACVR1 (ALK2)STKRTKL6gipAA2,5-dimethyl-6-quinolin-4-yl-3~{h}-quinazolin-4-oneHuman9915
ACVR1 (ALK2)STKRTKL6gipAB2,5-dimethyl-6-quinolin-4-yl-3~{h}-quinazolin-4-oneHuman9917
ACVR1 (ALK2)STKRTKL6i1sAA(4~{s},5~{r},6~{z},9~{s},10~{s},12~{e})-16-(ethylamino)-4,5-dimethyl-9,10,18-tris(oxidanyl)-3-oxabicyclo[12.4.0]octadeca-1(14),6,12,15,17-pentaene-2,8-dioneHuman11603
ACVR1 (ALK2)STKRTKL6i1sAB(4~{s},5~{r},6~{z},9~{s},10~{s},12~{e})-16-(ethylamino)-4,5-dimethyl-9,10,18-tris(oxidanyl)-3-oxabicyclo[12.4.0]octadeca-1(14),6,12,15,17-pentaene-2,8-dioneHuman11604
ACVR1 (ALK2)STKRTKL6juxAA4-(1-ethyl-3-pyridin-3-yl-pyrazol-4-yl)-~{n}-(4-piperazin-1-ylphenyl)pyrimidin-2-amineHuman12161
ACVR1 (ALK2)STKRTKL6juxAB4-(1-ethyl-3-pyridin-3-yl-pyrazol-4-yl)-~{n}-(4-piperazin-1-ylphenyl)pyrimidin-2-amineHuman12160
ACVR1 (ALK2)STKRTKL6srhAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman11632
ACVR1 (ALK2)STKRTKL6srhAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman11630
ACVR1 (ALK2)STKRTKL6srhBA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman11631
ACVR1 (ALK2)STKRTKL6srhBB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman11633
ACVR1 (ALK2)STKRTKL6szmAA1-[4-[4-methyl-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl]piperazineHuman11735
ACVR1 (ALK2)STKRTKL6szmAB1-[4-[4-methyl-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl]piperazineHuman11737
ACVR1 (ALK2)STKRTKL6szmBA1-[4-[4-methyl-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl]piperazineHuman11734
ACVR1 (ALK2)STKRTKL6szmBB1-[4-[4-methyl-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl]piperazineHuman11736
ACVR1 (ALK2)STKRTKL6t6dAA2-methoxy-4-[4-methyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]benzamideHuman11779
ACVR1 (ALK2)STKRTKL6t6dAB2-methoxy-4-[4-methyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]benzamideHuman11784
ACVR1 (ALK2)STKRTKL6t6dBA2-methoxy-4-[4-methyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]benzamideHuman11781
ACVR1 (ALK2)STKRTKL6t6dBB2-methoxy-4-[4-methyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]benzamideHuman11782
ACVR1 (ALK2)STKRTKL6t6dCA2-methoxy-4-[4-methyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]benzamideHuman11778
ACVR1 (ALK2)STKRTKL6t6dCB2-methoxy-4-[4-methyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]benzamideHuman11780
ACVR1 (ALK2)STKRTKL6t6dDA2-methoxy-4-[4-methyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]benzamideHuman11783
ACVR1 (ALK2)STKRTKL6t6dDB2-methoxy-4-[4-methyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]benzamideHuman11785
ACVR1 (ALK2)STKRTKL6t8nAAcyclopropyl-[4-[6-[5-(4-ethoxy-1-propan-2-yl-piperidin-4-yl)pyridin-2-yl]pyrrolo[1,2-b]pyridazin-4-yl]piperazin-1-yl]methanoneHuman11831
ACVR1 (ALK2)STKRTKL6t8nABcyclopropyl-[4-[6-[5-(4-ethoxy-1-propan-2-yl-piperidin-4-yl)pyridin-2-yl]pyrrolo[1,2-b]pyridazin-4-yl]piperazin-1-yl]methanoneHuman11830
ACVR1 (ALK2)STKRTKL6t8nBAcyclopropyl-[4-[6-[5-(4-ethoxy-1-propan-2-yl-piperidin-4-yl)pyridin-2-yl]pyrrolo[1,2-b]pyridazin-4-yl]piperazin-1-yl]methanoneHuman11828
ACVR1 (ALK2)STKRTKL6t8nBBcyclopropyl-[4-[6-[5-(4-ethoxy-1-propan-2-yl-piperidin-4-yl)pyridin-2-yl]pyrrolo[1,2-b]pyridazin-4-yl]piperazin-1-yl]methanoneHuman11829
ACVR1 (ALK2)STKRTKL6tn8AA4-[4-[(dimethylamino)methyl]-2,5-dimethoxy-phenyl]-2-methyl-2,7-naphthyridin-1-oneHuman11888
ACVR1 (ALK2)STKRTKL6tn8AB4-[4-[(dimethylamino)methyl]-2,5-dimethoxy-phenyl]-2-methyl-2,7-naphthyridin-1-oneHuman11887
ACVR1 (ALK2)STKRTKL6z36AA4-methyl-3-(4-piperidin-4-ylphenyl)-5-(3,4,5-trimethoxyphenyl)pyridineHuman12277
ACVR1 (ALK2)STKRTKL6z36AB4-methyl-3-(4-piperidin-4-ylphenyl)-5-(3,4,5-trimethoxyphenyl)pyridineHuman12278
ACVR1 (ALK2)STKRTKL6z36BA4-methyl-3-(4-piperidin-4-ylphenyl)-5-(3,4,5-trimethoxyphenyl)pyridineHuman12276
ACVR1 (ALK2)STKRTKL6z36BB4-methyl-3-(4-piperidin-4-ylphenyl)-5-(3,4,5-trimethoxyphenyl)pyridineHuman12275
ACVR1 (ALK2)STKRTKL6zgcAn-(5-chloro-1,3-benzodioxol-4-yl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]-5-(tetrahydro-2h-pyran-4-yloxy)quinazolin-4-amineHuman12638
ACVR1 (ALK2)STKRTKL6zgcBn-(5-chloro-1,3-benzodioxol-4-yl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]-5-(tetrahydro-2h-pyran-4-yloxy)quinazolin-4-amineHuman12641
ACVR1 (ALK2)STKRTKL6zgcCn-(5-chloro-1,3-benzodioxol-4-yl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]-5-(tetrahydro-2h-pyran-4-yloxy)quinazolin-4-amineHuman12640
ACVR1 (ALK2)STKRTKL6zgcDn-(5-chloro-1,3-benzodioxol-4-yl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]-5-(tetrahydro-2h-pyran-4-yloxy)quinazolin-4-amineHuman12639
ACVR1 (ALK2)STKRTKL7a21AA4-methyl-3-[4-(pyrrolidin-1-ylmethyl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman12777
ACVR1 (ALK2)STKRTKL7a21AB4-methyl-3-[4-(pyrrolidin-1-ylmethyl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman12779
ACVR1 (ALK2)STKRTKL7a21BA4-methyl-3-[4-(pyrrolidin-1-ylmethyl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman12776
ACVR1 (ALK2)STKRTKL7a21BB4-methyl-3-[4-(pyrrolidin-1-ylmethyl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman12778
ACVR2A (ACTR2)STKRTKL3q4tAA6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHuman2682
ACVR2A (ACTR2)STKRTKL3q4tAB6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHuman2686
ACVR2A (ACTR2)STKRTKL3q4tBA6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHuman2680
ACVR2A (ACTR2)STKRTKL3q4tBB6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHuman2684
ACVR2A (ACTR2)STKRTKL3socAA[4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl}imino)cyclohexa-2,5-dien-1-yl]acetonitrileHuman2675
ACVR2A (ACTR2)STKRTKL3socAB[4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl}imino)cyclohexa-2,5-dien-1-yl]acetonitrileHuman2676
ACVR2A (ACTR2)STKRTKL3socBA[4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl}imino)cyclohexa-2,5-dien-1-yl]acetonitrileHuman2677
ACVR2A (ACTR2)STKRTKL3socBB[4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl}imino)cyclohexa-2,5-dien-1-yl]acetonitrileHuman2685
ACVR2A (ACTR2)STKRTKL4asxAA7,8-bis(chloranyl)-9-methyl-3,4-dihydro-2h-pyrido[3,4-b]indol-1-oneHuman2678
ACVR2A (ACTR2)STKRTKL4asxAB7,8-bis(chloranyl)-9-methyl-3,4-dihydro-2h-pyrido[3,4-b]indol-1-oneHuman2681
ACVR2A (ACTR2)STKRTKL4asxBA7,8-bis(chloranyl)-9-methyl-3,4-dihydro-2h-pyrido[3,4-b]indol-1-oneHuman2683
ACVR2A (ACTR2)STKRTKL4asxBB7,8-bis(chloranyl)-9-methyl-3,4-dihydro-2h-pyrido[3,4-b]indol-1-oneHuman2679
ACVR2B (ACTR2B)STKRTKL2qluAadenineHuman2940
ACVRL1 (ALK1)STKRTKL3my0A4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1266
ACVRL1 (ALK1)STKRTKL3my0B4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1273
ACVRL1 (ALK1)STKRTKL3my0C4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1269
ACVRL1 (ALK1)STKRTKL3my0D4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1258
ACVRL1 (ALK1)STKRTKL3my0E4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1263
ACVRL1 (ALK1)STKRTKL3my0F4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1276
ACVRL1 (ALK1)STKRTKL3my0G4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1272
ACVRL1 (ALK1)STKRTKL3my0H4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1260
ACVRL1 (ALK1)STKRTKL3my0I4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1261
ACVRL1 (ALK1)STKRTKL3my0J4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1277
ACVRL1 (ALK1)STKRTKL3my0K4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1267
ACVRL1 (ALK1)STKRTKL3my0L4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1265
ACVRL1 (ALK1)STKRTKL3my0M4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1268
ACVRL1 (ALK1)STKRTKL3my0N4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1257
ACVRL1 (ALK1)STKRTKL3my0O4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1262
ACVRL1 (ALK1)STKRTKL3my0P4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1270
ACVRL1 (ALK1)STKRTKL3my0Q4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1274
ACVRL1 (ALK1)STKRTKL3my0R4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1256
ACVRL1 (ALK1)STKRTKL3my0S4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1259
ACVRL1 (ALK1)STKRTKL3my0T4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1264
ACVRL1 (ALK1)STKRTKL3my0U4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1278
ACVRL1 (ALK1)STKRTKL3my0V4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1271
ACVRL1 (ALK1)STKRTKL3my0W4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1255
ACVRL1 (ALK1)STKRTKL3my0X4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1275
AKT1AktAGC3cquAAn-[2-(5-methyl-4h-1,2,4-triazol-3-yl)phenyl]-7h-pyrrolo[2,3-d]pyrimidin-4-amineHuman6764
AKT1AktAGC3cquABn-[2-(5-methyl-4h-1,2,4-triazol-3-yl)phenyl]-7h-pyrrolo[2,3-d]pyrimidin-4-amineHuman6762
AKT1AktAGC3cqwAA5-(5-chloro-7h-pyrrolo[2,3-d]pyrimidin-4-yl)-4,5,6,7-tetrahydro-1h-imidazo[4,5-c]pyridineHuman6763
AKT1AktAGC3cqwAB5-(5-chloro-7h-pyrrolo[2,3-d]pyrimidin-4-yl)-4,5,6,7-tetrahydro-1h-imidazo[4,5-c]pyridineHuman6765
AKT1AktAGC3mv5AA(3r)-1-(5-methyl-7h-pyrrolo[2,3-d]pyrimidin-4-yl)pyrrolidin-3-amineHuman2537
AKT1AktAGC3mv5AB(3r)-1-(5-methyl-7h-pyrrolo[2,3-d]pyrimidin-4-yl)pyrrolidin-3-amineHuman2532
AKT1AktAGC3mvhAAn-{[(3s)-3-amino-1-(5-ethyl-7h-pyrrolo[2,3-d]pyrimidin-4-yl)pyrrolidin-3-yl]methyl}-2,4-difluorobenzamideHuman2538
AKT1AktAGC3mvhABn-{[(3s)-3-amino-1-(5-ethyl-7h-pyrrolo[2,3-d]pyrimidin-4-yl)pyrrolidin-3-yl]methyl}-2,4-difluorobenzamideHuman2531
AKT1AktAGC3o96A-Human2545
AKT1AktAGC3ocbA(2s)-2-(4-chlorobenzyl)-3-oxo-3-[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperazin-1-yl]propan-1-amineHuman2548
AKT1AktAGC3ocbB(2s)-2-(4-chlorobenzyl)-3-oxo-3-[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperazin-1-yl]propan-1-amineHuman2534
AKT1AktAGC3ow4A(2r)-3-(1h-indol-3-yl)-1-{4-[(5s)-5-methyl-5,7-dihydrothieno[3,4-d]pyrimidin-4-yl]piperazin-1-yl}-1-oxopropan-2-amineHuman2547
AKT1AktAGC3ow4B(2r)-3-(1h-indol-3-yl)-1-{4-[(5s)-5-methyl-5,7-dihydrothieno[3,4-d]pyrimidin-4-yl]piperazin-1-yl}-1-oxopropan-2-amineHuman2533
AKT1AktAGC3qkkAn-(2-ethoxyethyl)-n-{(2s)-2-hydroxy-3-[(2r)-6-hydroxy-4-oxo-3,4-dihydro-1'h-spiro[chromene-2,3'-piperidin]-1'-yl]propyl}-2,6-dimethylbenzenesulfonamideHuman2535
AKT1AktAGC3qklAn-{(2s)-3-[(3s)-8',9'-dihydro-1h,3'h-spiro[piperidine-3,7'-pyrano[3,2-e]indazol]-1-yl]-2-hydroxypropyl}-n-(2-ethoxyethyl)-2,6-dimethylbenzenesulfonamideHuman2544
AKT1AktAGC3qkmAn-(2-ethoxyethyl)-n-{(2s)-2-hydroxy-3-[(5r)-2-(quinazolin-4-yl)-2,7-diazaspiro[4.5]dec-7-yl]propyl}-2,6-dimethylbenzenesulfonamideHuman2546
AKT1AktAGC4ejnA-Human2542
AKT1AktAGC4ekkAphosphoaminophosphonic acid-adenylate esterHuman2541
AKT1AktAGC4ekkBphosphoaminophosphonic acid-adenylate esterHuman2539
AKT1AktAGC4eklA(2s)-2-(4-chlorophenyl)-1-{4-[(5r,7r)-7-hydroxy-5-methyl-6,7-dihydro-5h-cyclopenta[d]pyrimidin-4-yl]piperazin-1-yl}-3-(propan-2-ylamino)propan-1-oneHuman2540
AKT1AktAGC4gv1AA4-amino-n-[(1s)-1-(4-chlorophenyl)-3-hydroxypropyl]-1-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperidine-4-carboxamideHuman2543
AKT1AktAGC4gv1AB4-amino-n-[(1s)-1-(4-chlorophenyl)-3-hydroxypropyl]-1-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperidine-4-carboxamideHuman2536
AKT1AktAGC5kcvA3-[3-[4-(1-azanylcyclobutyl)phenyl]-5-phenyl-imidazo[4,5-b]pyridin-2-yl]pyridin-2-amineHuman6708
AKT1AktAGC6buuAA-Human10432
AKT1AktAGC6buuAB-Human10433
AKT1AktAGC6buuAC-Human10438
AKT1AktAGC6buuBA-Human10430
AKT1AktAGC6buuBB-Human10439
AKT1AktAGC6buuBC-Human10428
AKT1AktAGC6ccyAA(5r)-4-(4-{4-[4-fluoro-3-(trifluoromethyl)phenyl]-1-[2-(pyrrolidin-1-yl)ethyl]-1h-imidazol-2-yl}piperidin-1-yl)-5-methyl-5,8-dihydropyrido[2,3-d]pyrimidin-7(6h)-oneHuman9868
AKT1AktAGC6ccyAB(5r)-4-(4-{4-[4-fluoro-3-(trifluoromethyl)phenyl]-1-[2-(pyrrolidin-1-yl)ethyl]-1h-imidazol-2-yl}piperidin-1-yl)-5-methyl-5,8-dihydropyrido[2,3-d]pyrimidin-7(6h)-oneHuman9869
AKT1AktAGC6hhfAborussertibHuman10970
AKT1AktAGC6hhgA~{n}-[2-chloranyl-5-[[1-[[4-(5-oxidanylidene-3-phenyl-6~{h}-1,6-naphthyridin-2-yl)phenyl]methyl]piperidin-4-yl]carbamoylamino]phenyl]propanamideHuman10916
AKT1AktAGC6hhhA~{n}-[4-[4-[[4-(5-oxidanylidene-3-phenyl-6~{h}-1,6-naphthyridin-2-yl)phenyl]methyl]piperazin-1-yl]phenyl]propanamideHuman10915
AKT1AktAGC6hhiA~{n}-[1-[[4-(5-oxidanylidene-3-phenyl-6~{h}-1,6-naphthyridin-2-yl)phenyl]methyl]piperidin-4-yl]-3-(propanoylamino)benzamideHuman10913
AKT1AktAGC6hhjA~{n}-[1-methyl-2-oxidanylidene-3-[1-[[4-(5-oxidanylidene-3-phenyl-6~{h}-1,6-naphthyridin-2-yl)phenyl]methyl]piperidin-4-yl]benzimidazol-5-yl]propanamideHuman10914
AKT1AktAGC6npzAA-Human10880
AKT1AktAGC6npzAB-Human10882
AKT1AktAGC6npzBA-Human10881
AKT1AktAGC6npzBB-Human10879
AKT1AktAGC6s9wAA~{n}-[3-[1-[[4-(5-methyl-6-oxidanylidene-3-phenyl-1~{h}-pyrazin-2-yl)phenyl]methyl]piperidin-4-yl]-2-oxidanylidene-1~{h}-benzimidazol-5-yl]propanamideHuman11748
AKT1AktAGC6s9wAB~{n}-[3-[1-[[4-(5-methyl-6-oxidanylidene-3-phenyl-1~{h}-pyrazin-2-yl)phenyl]methyl]piperidin-4-yl]-2-oxidanylidene-1~{h}-benzimidazol-5-yl]propanamideHuman11747
AKT1AktAGC6s9xA~{n}-[3-[1-[[4-[5-[(4-hydroxyphenyl)methyl]-6-oxidanylidene-2-phenyl-1~{h}-pyrazin-3-yl]phenyl]methyl]piperidin-4-yl]-2-oxidanylidene-1~{h}-benzimidazol-5-yl]propanamideHuman11746
AKT2AktAGC1gzkA-Human1916
AKT2AktAGC1gznA-Human1915
AKT2AktAGC1gzoA-Human1914
AKT2AktAGC1mrvA-Human1917
AKT2AktAGC1mryA-Human1907
AKT2AktAGC1o6kAphosphoaminophosphonic acid-adenylate esterHuman1923
AKT2AktAGC1o6lAphosphoaminophosphonic acid-adenylate esterHuman1906
AKT2AktAGC2jdoAisoquinoline-5-sulfonic acid (2-(2-(4-chlorobenzyloxy)ethylamino)ethyl)amideHuman1922
AKT2AktAGC2jdrA(2s)-1-(1h-indol-3-yl)-3-{[5-(3-methyl-1h-indazol-5-yl)pyridin-3-yl]oxy}propan-2-amineHuman1918
AKT2AktAGC2uw9A4-(4-chlorophenyl)-4-[4-(1h-pyrazol-4-yl)phenyl]piperidineHuman1919
AKT2AktAGC2x39A4-amino-n-(4-chlorobenzyl)-1-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperidine-4-carboxamideHuman1913
AKT2AktAGC2xh5A4-(4-tert-butylbenzyl)-1-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperidin-4-aminiumHuman1924
AKT2AktAGC3d0eA4-{2-(4-amino-1,2,5-oxadiazol-3-yl)-1-ethyl-7-[(3s)-piperidin-3-ylmethoxy]-1h-imidazo[4,5-c]pyridin-4-yl}-2-methylbut-3-yn-2-olHuman1912
AKT2AktAGC3d0eB4-{2-(4-amino-1,2,5-oxadiazol-3-yl)-1-ethyl-7-[(3s)-piperidin-3-ylmethoxy]-1h-imidazo[4,5-c]pyridin-4-yl}-2-methylbut-3-yn-2-olHuman1920
AKT2AktAGC3e87AAn-[(1s)-2-amino-1-phenylethyl]-5-(1h-pyrrolo[2,3-b]pyridin-4-yl)thiophene-2-carboxamideHuman1910
AKT2AktAGC3e87ABn-[(1s)-2-amino-1-phenylethyl]-5-(1h-pyrrolo[2,3-b]pyridin-4-yl)thiophene-2-carboxamideHuman1911
AKT2AktAGC3e87BAn-[(1s)-2-amino-1-phenylethyl]-5-(1h-pyrrolo[2,3-b]pyridin-4-yl)thiophene-2-carboxamideHuman1909
AKT2AktAGC3e87BBn-[(1s)-2-amino-1-phenylethyl]-5-(1h-pyrrolo[2,3-b]pyridin-4-yl)thiophene-2-carboxamideHuman1903
AKT2AktAGC3e88A4-[2-(4-amino-1,2,5-oxadiazol-3-yl)-6-{[(2r)-2-amino-3-phenylpropyl]oxy}-1-ethyl-1h-imidazo[4,5-c]pyridin-4-yl]-2-methylbut-3-yn-2-olHuman1908
AKT2AktAGC3e88B4-[2-(4-amino-1,2,5-oxadiazol-3-yl)-6-{[(2r)-2-amino-3-phenylpropyl]oxy}-1-ethyl-1h-imidazo[4,5-c]pyridin-4-yl]-2-methylbut-3-yn-2-olHuman1905
AKT2AktAGC3e8dAA4-[2-(4-amino-2,5-dihydro-1,2,5-oxadiazol-3-yl)-6-{[(1s)-3-amino-1-phenylpropyl]oxy}-1-ethyl-1h-imidazo[4,5-c]pyridin-4-yl]-2-methylbut-3-yn-2-olHuman1921
AKT2AktAGC3e8dAB4-[2-(4-amino-2,5-dihydro-1,2,5-oxadiazol-3-yl)-6-{[(1s)-3-amino-1-phenylpropyl]oxy}-1-ethyl-1h-imidazo[4,5-c]pyridin-4-yl]-2-methylbut-3-yn-2-olHuman1926
AKT2AktAGC3e8dBA4-[2-(4-amino-2,5-dihydro-1,2,5-oxadiazol-3-yl)-6-{[(1s)-3-amino-1-phenylpropyl]oxy}-1-ethyl-1h-imidazo[4,5-c]pyridin-4-yl]-2-methylbut-3-yn-2-olHuman1925
AKT2AktAGC3e8dBB4-[2-(4-amino-2,5-dihydro-1,2,5-oxadiazol-3-yl)-6-{[(1s)-3-amino-1-phenylpropyl]oxy}-1-ethyl-1h-imidazo[4,5-c]pyridin-4-yl]-2-methylbut-3-yn-2-olHuman1904
ALKALKTK2xb7A5-chloro-n-[2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]-n'-(2-propan-2-ylsulfonylphenyl)pyrimidine-2,4-diamineHuman5365
ALKALKTK2xbaA5-[(2r)-2-hydroxy-2-phenylacetyl]-3-({[4-(4-methylpiperazin-1-yl)phenyl]carbonyl}amino)-1,6-dihydropyrrolo[3,4-c]pyrazol-5-ium Human5408
ALKALKTK2xp2A3-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-5-(1-piperidin-4-yl-1h-pyrazol-4-yl)pyridin-2-amineHuman5394
ALKALKTK2yfxA3-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-5-(1-piperidin-4-yl-1h-pyrazol-4-yl)pyridin-2-amineHuman5402
ALKALKTK2yhvA-Human5384
ALKALKTK2yjrAA-Human5399
ALKALKTK2yjrAB-Human5380
ALKALKTK2yjsA-Human5373
ALKALKTK3aoxAA9-ethyl-6,6-dimethyl-8-[4-(morpholin-4-yl)piperidin-1-yl]-11-oxo-6,11-dihydro-5h-benzo[b]carbazole-3-carbonitrileHuman5387
ALKALKTK3aoxAB9-ethyl-6,6-dimethyl-8-[4-(morpholin-4-yl)piperidin-1-yl]-11-oxo-6,11-dihydro-5h-benzo[b]carbazole-3-carbonitrileHuman5370
ALKALKTK3l9pAA-Human5363
ALKALKTK3l9pAB-Human5375
ALKALKTK3lcsAAstaurosporineHuman5381
ALKALKTK3lcsABstaurosporineHuman5376
ALKALKTK3lctAAadenosine-5'-diphosphateHuman5393
ALKALKTK3lctABadenosine-5'-diphosphateHuman5400
ALKALKTK4anlA-Human5385
ALKALKTK4anqA3-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-5-(1-piperidin-4-yl-1h-pyrazol-4-yl)pyridin-2-amineHuman5368
ALKALKTK4ansA3-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-5-(1-piperidin-4-yl-1h-pyrazol-4-yl)pyridin-2-amineHuman5374
ALKALKTK4ccbA3-[(1r)-1-[5-fluoranyl-2-(1,2,3-triazol-2-yl)phenyl]ethoxy]-5-(3-methyl-1h-pyrazol-4-yl)pyridin-2-amineHuman5390
ALKALKTK4ccuA2-(5-(6-amino-5-((r)-1-(5-fluoro-2-(2h-1,2,3-triazol-2-yl)phenyl)ethoxy)pyridin-3-yl)-4-methylthiazol-2-yl)propan-2-olHuman5396
ALKALKTK4cd0A(2r)-2-[5-(6-amino-5-{(1r)-1-[2-(1,3-dihydro-2h-1,2,3-triazol-2-yl)-5-fluorophenyl]ethoxy}pyridin-3-yl)-4-methyl-1,3-thiazol-2-yl]propane-1,2-diolHuman5407
ALKALKTK4cliA(10r)-7-amino-12-fluoro-2,10,16-trimethyl-15-oxo-10,15,16,17-tetrahydro-2h-8,4-(metheno)pyrazolo[4,3-h][2,5,11]benzoxadiazacyclotetradecine-3-carbonitrileHuman5405
ALKALKTK4cljA(10r)-7-amino-12-fluoro-2,10,16-trimethyl-15-oxo-10,15,16,17-tetrahydro-2h-8,4-(metheno)pyrazolo[4,3-h][2,5,11]benzoxadiazacyclotetradecine-3-carbonitrileHuman5369
ALKALKTK4cmoA2-[(1r)-1-{[3-amino-6-(2-methoxypyridin-3-yl)pyrazin-2-yl]oxy}ethyl]-4-fluoro-n-methylbenzamideHuman5391
ALKALKTK4cmtA3-{(1r)-1-[2-(1,3-dihydro-2h-1,2,3-triazol-2-yl)-5-fluorophenyl]ethoxy}-5-[3-(methylsulfonyl)phenyl]pyridin-2-amineHuman5371
ALKALKTK4cmuA(10r)-7-amino-12-fluoro-1,3,10,16-tetramethyl-16,17-dihydro-1h-8,4-(metheno)pyrazolo[4,3-h][2,5,11]benzoxadiazacyclotetradecin-15(10h)-oneHuman5398
ALKALKTK4cnhA3-[(1r)-1-(5-fluoro-2-methoxyphenyl)ethoxy]-5-(1-methyl-1h-1,2,3-triazol-5-yl)pyridin-2-amineHuman5388
ALKALKTK4cnhB3-[(1r)-1-(5-fluoro-2-methoxyphenyl)ethoxy]-5-(1-methyl-1h-1,2,3-triazol-5-yl)pyridin-2-amineHuman5378
ALKALKTK4ctbA(5r)-8-amino-3-fluoro-5,19-dimethyl-20-oxo-5,18,19,20-tetrahydro-11,7-(azeno)pyrido[2',1':2,3]imidazo[4,5-h][2,5,11]benzoxadiazacyclotetradecine-14-carbonitrileHuman5395
ALKALKTK4ctcA(10r)-7-amino-3-cyclopropyl-12-fluoro-1,10,16-trimethyl-16,17-dihydro-1h-8,4-(metheno)pyrazolo[4,3-h][2,5,11]benzoxadiazacyclotetradecin-15(10h)-oneHuman5364
ALKALKTK4dceA(3s)-n-(4-methylbenzyl)-1-{2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}piperidine-3-carboxamideHuman5379
ALKALKTK4dceB(3s)-n-(4-methylbenzyl)-1-{2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}piperidine-3-carboxamideHuman5372
ALKALKTK4fnwA-Human5403
ALKALKTK4fnxA-Human5366
ALKALKTK4fnyAn-(4-chlorophenyl)-5-[(6,7-dimethoxyquinolin-4-yl)oxy]-1,3-benzoxazol-2-amineHuman5367
ALKALKTK4fnzA(3s)-n-[3-(trifluoromethoxy)benzyl]-1-{2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}piperidine-3-carboxamideHuman5397
ALKALKTK4fobAn-{1-[cis-4-(hydroxymethyl)cyclohexyl]-5-(piperidin-1-ylmethyl)-1h-benzimidazol-2-yl}-3-(prop-2-en-1-ylsulfamoyl)benzamideHuman5377
ALKALKTK4focAmethyl cis-4-[2-(benzoylamino)-6-(piperidin-1-ylmethyl)-1h-benzimidazol-1-yl]cyclohexanecarboxylateHuman5392
ALKALKTK4fodAA4-fluoro-n-{(2e)-6-{[4-(2-hydroxypropan-2-yl)piperidin-1-yl]methyl}-1-[cis-4-(propan-2-ylcarbamoyl)cyclohexyl]-1,3-dihydro-2h-benzimidazol-2-ylidene}benzamideHuman5383
ALKALKTK4fodAB4-fluoro-n-{(2e)-6-{[4-(2-hydroxypropan-2-yl)piperidin-1-yl]methyl}-1-[cis-4-(propan-2-ylcarbamoyl)cyclohexyl]-1,3-dihydro-2h-benzimidazol-2-ylidene}benzamideHuman5404
ALKALKTK4joaAA3-[1-(2,5-difluorobenzyl)-1h-pyrazol-4-yl]-5-(1-methyl-1h-pyrazol-4-yl)-1h-pyrrolo[2,3-b]pyridineHuman5389
ALKALKTK4mkcAA5-chloro-n~2~-[5-methyl-4-(piperidin-4-yl)-2-(propan-2-yloxy)phenyl]-n~4~-[2-(propan-2-ylsulfonyl)phenyl]pyrimidine-2,4-diamineHuman5401
ALKALKTK4mkcAB5-chloro-n~2~-[5-methyl-4-(piperidin-4-yl)-2-(propan-2-yloxy)phenyl]-n~4~-[2-(propan-2-ylsulfonyl)phenyl]pyrimidine-2,4-diamineHuman5386
ALKALKTK4tt7AA-Human5406
ALKALKTK4tt7AB-Human5382
ALKALKTK4z55AAn~6~-[5-methyl-4-(1-methylpiperidin-4-yl)-2-(propan-2-yloxy)phenyl]-n~4~-[2-(propan-2-ylsulfonyl)phenyl]-2h-pyrazolo[3,4-d]pyrimidine-4,6-diamineHuman6393
ALKALKTK4z55ABn~6~-[5-methyl-4-(1-methylpiperidin-4-yl)-2-(propan-2-yloxy)phenyl]-n~4~-[2-(propan-2-ylsulfonyl)phenyl]-2h-pyrazolo[3,4-d]pyrimidine-4,6-diamineHuman6392
ALKALKTK5a9uAA(10r)-7-amino-12-fluoro-2,10,16-trimethyl-15-oxo-10,15,16,17-tetrahydro-2h-8,4-(metheno)pyrazolo[4,3-h][2,5,11]benzoxadiazacyclotetradecine-3-carbonitrileHuman6692
ALKALKTK5a9uAB(10r)-7-amino-12-fluoro-2,10,16-trimethyl-15-oxo-10,15,16,17-tetrahydro-2h-8,4-(metheno)pyrazolo[4,3-h][2,5,11]benzoxadiazacyclotetradecine-3-carbonitrileHuman6685
ALKALKTK5aa8AA(10r)-7-amino-12-fluoro-2,10,16-trimethyl-15-oxo-10,15,16,17-tetrahydro-2h-8,4-(metheno)pyrazolo[4,3-h][2,5,11]benzoxadiazacyclotetradecine-3-carbonitrileHuman6688
ALKALKTK5aa8AB(10r)-7-amino-12-fluoro-2,10,16-trimethyl-15-oxo-10,15,16,17-tetrahydro-2h-8,4-(metheno)pyrazolo[4,3-h][2,5,11]benzoxadiazacyclotetradecine-3-carbonitrileHuman6684
ALKALKTK5aa9AA(10r)-7-amino-12-fluoro-2,10,16-trimethyl-15-oxo-10,15,16,17-tetrahydro-2h-8,4-(metheno)pyrazolo[4,3-h][2,5,11]benzoxadiazacyclotetradecine-3-carbonitrileHuman6682
ALKALKTK5aa9AB(10r)-7-amino-12-fluoro-2,10,16-trimethyl-15-oxo-10,15,16,17-tetrahydro-2h-8,4-(metheno)pyrazolo[4,3-h][2,5,11]benzoxadiazacyclotetradecine-3-carbonitrileHuman6687
ALKALKTK5aaaAA3-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-5-(1-piperidin-4-yl-1h-pyrazol-4-yl)pyridin-2-amineHuman6691
ALKALKTK5aaaAB3-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-5-(1-piperidin-4-yl-1h-pyrazol-4-yl)pyridin-2-amineHuman6683
ALKALKTK5aabAA3-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-5-(1-piperidin-4-yl-1h-pyrazol-4-yl)pyridin-2-amineHuman6689
ALKALKTK5aabAB3-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-5-(1-piperidin-4-yl-1h-pyrazol-4-yl)pyridin-2-amineHuman6681
ALKALKTK5aacAA3-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-5-(1-piperidin-4-yl-1h-pyrazol-4-yl)pyridin-2-amineHuman6690
ALKALKTK5aacAB3-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-5-(1-piperidin-4-yl-1h-pyrazol-4-yl)pyridin-2-amineHuman6686
ALKALKTK5ftoAAentrectinibHuman6520
ALKALKTK5ftoABentrectinibHuman6521
ALKALKTK5ftqAAn-[5-(3,5-difluorobenzyl)-1h-indazol-3-yl]-2-[(4-hydroxycyclohexyl)amino]-4-(4-methylpiperazin-1-yl) benzamideHuman6519
ALKALKTK5ftqABn-[5-(3,5-difluorobenzyl)-1h-indazol-3-yl]-2-[(4-hydroxycyclohexyl)amino]-4-(4-methylpiperazin-1-yl) benzamideHuman6518
ALKALKTK5imxA5-chloro-n~2~-{5-methyl-4-(1-methylpiperidin-4-yl)-2-[(propan-2-yl)oxy]phenyl}-n~4~-{1-methyl-3-[(propan-2-yl)sulfonyl]-1h-pyrazol-4-yl}pyrimidine-2,4-diamineHuman6604
ALKALKTK5iugAAn-[3-(4-{[(5-tert-butyl-1,2-oxazol-3-yl)carbamoyl]amino}-3-methylphenyl)-1h-pyrazol-5-yl]-4-[(4-methylpiperazin-1-yl)methyl]benzamideHuman6640
ALKALKTK5iugABn-[3-(4-{[(5-tert-butyl-1,2-oxazol-3-yl)carbamoyl]amino}-3-methylphenyl)-1h-pyrazol-5-yl]-4-[(4-methylpiperazin-1-yl)methyl]benzamideHuman6639
ALKALKTK5iuhA4-[(4-methylpiperazin-1-yl)methyl]-n-{3-[3-methyl-4-({[5-(propan-2-yl)-1,2-oxazol-3-yl]carbamoyl}amino)phenyl]-1h-pyrazol-5-yl}benzamideHuman6638
ALKALKTK5iuiAAn-[3-(4-amino-3-methylphenyl)-1h-pyrazol-5-yl]-4-[(4-methylpiperazin-1-yl)methyl]benzamideHuman6641
ALKALKTK5iuiABn-[3-(4-amino-3-methylphenyl)-1h-pyrazol-5-yl]-4-[(4-methylpiperazin-1-yl)methyl]benzamideHuman6642
ALKALKTK5kz0A2-[(1~{r})-1-[2-azanyl-5-(1,3-dimethylpyrazol-4-yl)pyridin-3-yl]oxyethyl]-4-fluoranyl-~{n},~{n}-dimethyl-benzamideHuman6970
ALKALKTK6cdtA-Human11263
ALKALKTK6e0rAAn-[(1s)-1-(5-fluoropyridin-2-yl)ethyl]-1-(5-methyl-1h-pyrazol-3-yl)-3-[(oxetan-3-yl)sulfonyl]-1h-pyrrolo[2,3-b]pyridin-6-amineHuman11268
ALKALKTK6e0rABn-[(1s)-1-(5-fluoropyridin-2-yl)ethyl]-1-(5-methyl-1h-pyrazol-3-yl)-3-[(oxetan-3-yl)sulfonyl]-1h-pyrrolo[2,3-b]pyridin-6-amineHuman11266
ALKALKTK6ebwAA[6-{[(1s)-1-(5-fluoropyridin-2-yl)ethyl]amino}-1-(5-methyl-1h-pyrazol-3-yl)-1h-pyrrolo[2,3-b]pyridin-3-yl](morpholin-4-yl)methanoneHuman11269
ALKALKTK6ebwAB[6-{[(1s)-1-(5-fluoropyridin-2-yl)ethyl]amino}-1-(5-methyl-1h-pyrazol-3-yl)-1h-pyrrolo[2,3-b]pyridin-3-yl](morpholin-4-yl)methanoneHuman11264
ALKALKTK6edlAAn-[(1s)-1-(2,4-difluorophenyl)ethyl]-3-(5-methyl-1h-pyrazol-3-yl)imidazo[1,2-b]pyridazin-6-amineHuman11267
ALKALKTK6edlABn-[(1s)-1-(2,4-difluorophenyl)ethyl]-3-(5-methyl-1h-pyrazol-3-yl)imidazo[1,2-b]pyridazin-6-amineHuman11265
ALKALKTK6mx8AA5-chloro-n~4~-[2-(dimethylphosphoryl)phenyl]-n~2~-{2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl}pyrimidine-2,4-diamineHuman10798
ALKALKTK6mx8AB5-chloro-n~4~-[2-(dimethylphosphoryl)phenyl]-n~2~-{2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl}pyrimidine-2,4-diamineHuman10799
ANTXR1 (DNAPK)PIKKAtypical5luqA-Human9321
ANTXR1 (DNAPK)PIKKAtypical5luqB-Human9319
ANTXR1 (DNAPK)PIKKAtypical5w1rA-Human9320
ANTXR1 (DNAPK)PIKKAtypical5y3rC-Human9318
ATMPIKKAtypical5np0A-Human9267
ATMPIKKAtypical5np0B-Human9266
ATMPIKKAtypical5np1A-Human9268
ATMPIKKAtypical6k9kA-Human11897
ATMPIKKAtypical6k9lA-Human11896
ATMPIKKAtypical6k9lB-Human11895
ATRPIKKAtypical5yz0A-Human9523
ATRPIKKAtypical5yz0B-Human9524
Aurka (AurA)AUROther3d14AA1-{5-[2-(thieno[3,2-d]pyrimidin-4-ylamino)ethyl]-1,3-thiazol-2-yl}-3-[3-(trifluoromethyl)phenyl]ureaMouse5781
Aurka (AurA)AUROther3d14AB1-{5-[2-(thieno[3,2-d]pyrimidin-4-ylamino)ethyl]-1,3-thiazol-2-yl}-3-[3-(trifluoromethyl)phenyl]ureaMouse5775
Aurka (AurA)AUROther3d15AA1-(3-chlorophenyl)-3-{5-[2-(thieno[3,2-d]pyrimidin-4-ylamino)ethyl]-1,3-thiazol-2-yl}ureaMouse5777
Aurka (AurA)AUROther3d2iA1-(5-{2-[(1-methyl-1h-pyrazolo[4,3-d]pyrimidin-7-yl)amino]ethyl}-1,3-thiazol-2-yl)-3-[3-(trifluoromethyl)phenyl]ureaMouse5782
Aurka (AurA)AUROther3d2kA(7-{[2-(2-{[(3-chlorophenyl)carbamoyl]amino}-1,3-thiazol-5-yl)ethyl]amino}-1h-pyrazolo[4,3-d]pyrimidin-1-yl)acetic acidMouse5776
Aurka (AurA)AUROther3dajAn-butyl-3-{[6-(9h-purin-6-ylamino)hexanoyl]amino}benzamideMouse5779
Aurka (AurA)AUROther3dj5A3-({3-[(6-amino-5-bromopyrimidin-4-yl)sulfanyl]propanoyl}amino)-4-methoxy-n-phenylbenzamideMouse5783
Aurka (AurA)AUROther3dj6A4-methoxy-n-phenyl-3-({3-[(1h-pyrrolo[2,3-b]pyridin-5-ylmethyl)sulfanyl]propanoyl}amino)benzamideMouse5778
Aurka (AurA)AUROther3dj7AA1-(5-{2-[(6-amino-5-bromopyrimidin-4-yl)amino]ethyl}-1,3-thiazol-2-yl)-3-[3-(trifluoromethyl)phenyl]ureaMouse5780
AURKA (AurA)AurOther1mq4Aadenosine-5'-diphosphateHuman1977
AURKA (AurA)AurOther1muoAadenosineHuman2062
AURKA (AurA)AurOther1ol5Aadenosine-5'-diphosphateHuman2080
AURKA (AurA)AurOther1ol6Aadenosine-5'-triphosphateHuman2081
AURKA (AurA)AurOther1ol7Aadenosine-5'-diphosphateHuman2014
AURKA (AurA)AurOther2bmcA(3e)-n-(2,6-diethylphenyl)-3-{[4-(4-methylpiperazin-1-yl)benzoyl]imino}pyrrolo[3,4-c]pyrazole-5(3h)-carboxamideHuman2015
AURKA (AurA)AurOther2bmcB(3e)-n-(2,6-diethylphenyl)-3-{[4-(4-methylpiperazin-1-yl)benzoyl]imino}pyrrolo[3,4-c]pyrazole-5(3h)-carboxamideHuman2008
AURKA (AurA)AurOther2bmcC(3e)-n-(2,6-diethylphenyl)-3-{[4-(4-methylpiperazin-1-yl)benzoyl]imino}pyrrolo[3,4-c]pyrazole-5(3h)-carboxamideHuman2060
AURKA (AurA)AurOther2bmcD(3e)-n-(2,6-diethylphenyl)-3-{[4-(4-methylpiperazin-1-yl)benzoyl]imino}pyrrolo[3,4-c]pyrazole-5(3h)-carboxamideHuman1984
AURKA (AurA)AurOther2bmcE(3e)-n-(2,6-diethylphenyl)-3-{[4-(4-methylpiperazin-1-yl)benzoyl]imino}pyrrolo[3,4-c]pyrazole-5(3h)-carboxamideHuman2069
AURKA (AurA)AurOther2bmcF(3e)-n-(2,6-diethylphenyl)-3-{[4-(4-methylpiperazin-1-yl)benzoyl]imino}pyrrolo[3,4-c]pyrazole-5(3h)-carboxamideHuman1993
AURKA (AurA)AurOther2c6dAAphosphoaminophosphonic acid-adenylate esterHuman2019
AURKA (AurA)AurOther2c6dABphosphoaminophosphonic acid-adenylate esterHuman1981
AURKA (AurA)AurOther2c6eAn-{5-[(7-{[(2s)-2-hydroxy-3-piperidin-1-ylpropyl]oxy}-6-methoxyquinazolin-4-yl)amino]pyrimidin-2-yl}benzamideHuman1989
AURKA (AurA)AurOther2c6eBn-{5-[(7-{[(2s)-2-hydroxy-3-piperidin-1-ylpropyl]oxy}-6-methoxyquinazolin-4-yl)amino]pyrimidin-2-yl}benzamideHuman2046
AURKA (AurA)AurOther2dwbAphosphoaminophosphonic acid-adenylate esterHuman2035
AURKA (AurA)AurOther2j4zA4-(4-methylpiperazin-1-yl)-n-[5-(2-thienylacetyl)-1,5-dihydropyrrolo[3,4-c]pyrazol-3-yl]benzamideHuman2053
AURKA (AurA)AurOther2j4zB4-(4-methylpiperazin-1-yl)-n-[5-(2-thienylacetyl)-1,5-dihydropyrrolo[3,4-c]pyrazol-3-yl]benzamideHuman1990
AURKA (AurA)AurOther2j50An-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamideHuman2001
AURKA (AurA)AurOther2j50Bn-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamideHuman2050
AURKA (AurA)AurOther2np8An-{3-[(4-{[3-(trifluoromethyl)phenyl]amino}pyrimidin-2-yl)amino]phenyl}cyclopropanecarboxamideHuman2075
AURKA (AurA)AurOther2w1cA4-{[2-(4-{[(4-fluorophenyl)carbonyl]amino}-1h-pyrazol-3-yl)-1h-benzimidazol-6-yl]methyl}morpholin-4-iumHuman2027
AURKA (AurA)AurOther2w1dA2-(1h-pyrazol-3-yl)-1h-benzimidazoleHuman2011
AURKA (AurA)AurOther2w1eA4-[(2-{4-[(phenylcarbamoyl)amino]-1h-pyrazol-3-yl}-1h-benzimidazol-5-yl)methyl]morpholin-4-iumHuman2038
AURKA (AurA)AurOther2w1fAn-[3-(1h-benzimidazol-2-yl)-1h-pyrazol-4-yl]benzamideHuman2055
AURKA (AurA)AurOther2w1gA2-{4-[(cyclopropylcarbamoyl)amino]-1h-pyrazol-3-yl}-6-(morpholin-4-ium-4-ylmethyl)-1h-3,1-benzimidazol-3-iumHuman1962
AURKA (AurA)AurOther2wqeAadenosine-5'-diphosphateHuman2071
AURKA (AurA)AurOther2wtvAA4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acidHuman2056
AURKA (AurA)AurOther2wtvAB4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acidHuman1997
AURKA (AurA)AurOther2wtvBA4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acidHuman2037
AURKA (AurA)AurOther2wtvBB4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acidHuman2057
AURKA (AurA)AurOther2wtvCA4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acidHuman2017
AURKA (AurA)AurOther2wtvCB4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acidHuman2016
AURKA (AurA)AurOther2wtvDA4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acidHuman2078
AURKA (AurA)AurOther2wtvDB4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acidHuman2076
AURKA (AurA)AurOther2wtwA4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acidHuman1956
AURKA (AurA)AurOther2x6dAA6-bromo-7-[4-(4-chlorobenzyl)piperazin-1-yl]-2-[4-(morpholin-4-ylmethyl)phenyl]-3h-imidazo[4,5-b]pyridineHuman1978
AURKA (AurA)AurOther2x6dAB6-bromo-7-[4-(4-chlorobenzyl)piperazin-1-yl]-2-[4-(morpholin-4-ylmethyl)phenyl]-3h-imidazo[4,5-b]pyridineHuman1975
AURKA (AurA)AurOther2x6eA6-bromo-7-{4-[(5-methylisoxazol-3-yl)methyl]piperazin-1-yl}-2-[4-(4-methylpiperazin-1-yl)phenyl]-1h-imidazo[4,5-b]pyridineHuman2079
AURKA (AurA)AurOther2x81A4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acidHuman1966
AURKA (AurA)AurOther2xneA3-chloro-n-(4-morpholin-4-ylphenyl)-6-pyridin-3-ylimidazo[1,2-a]pyrazin-8-amineHuman7221
AURKA (AurA)AurOther2xngAAn-(3-{3-chloro-8-[(4-morpholin-4-ylphenyl)amino]imidazo[1,2-a]pyrazin-6-yl}benzyl)methanesulfonamideHuman1994
AURKA (AurA)AurOther2xngABn-(3-{3-chloro-8-[(4-morpholin-4-ylphenyl)amino]imidazo[1,2-a]pyrazin-6-yl}benzyl)methanesulfonamideHuman2083
AURKA (AurA)AurOther2xruA3-({[4-(4-methylpiperazin-1-yl)phenyl]carbonyl}amino)-n-[(1r)-1-phenylpropyl]-1h-thieno[3,2-c]pyrazole-5-carboxamideHuman1954
AURKA (AurA)AurOther3cohA8-ethyl-3,10,10-trimethyl-4,5,6,8,10,12-hexahydropyrazolo[4',3':6,7]cyclohepta[1,2-b]pyrrolo[2,3-f]indol-9(1h)-oneHuman1963
AURKA (AurA)AurOther3cohB8-ethyl-3,10,10-trimethyl-4,5,6,8,10,12-hexahydropyrazolo[4',3':6,7]cyclohepta[1,2-b]pyrrolo[2,3-f]indol-9(1h)-oneHuman2024
AURKA (AurA)AurOther3e5aAcyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amideHuman2006
AURKA (AurA)AurOther3efwA1-[3-methyl-4-({3-[2-(methylamino)pyrimidin-4-yl]pyridin-2-yl}oxy)phenyl]-3-[3-(trifluoromethyl)phenyl]ureaHuman2010
AURKA (AurA)AurOther3efwB1-[3-methyl-4-({3-[2-(methylamino)pyrimidin-4-yl]pyridin-2-yl}oxy)phenyl]-3-[3-(trifluoromethyl)phenyl]ureaHuman2074
AURKA (AurA)AurOther3fdnAn-[3-(acetylamino)phenyl]-5-{(2e)-2-[(4-methoxyphenyl)methylidene]hydrazino}-3-methyl-1h-pyrazole-4-carboxamideHuman1973
AURKA (AurA)AurOther3h0yA2-chloro-n-[4-({5-fluoro-2-[(4-hydroxyphenyl)amino]pyrimidin-4-yl}amino)phenyl]benzamideHuman1965
AURKA (AurA)AurOther3h0zA4-{[2-({4-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]phenyl}amino)-5-fluoropyrimidin-4-yl]amino}-n-(2-chlorophenyl)benzamideHuman1970
AURKA (AurA)AurOther3h0zB4-{[2-({4-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]phenyl}amino)-5-fluoropyrimidin-4-yl]amino}-n-(2-chlorophenyl)benzamideHuman1986
AURKA (AurA)AurOther3h0zC4-{[2-({4-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]phenyl}amino)-5-fluoropyrimidin-4-yl]amino}-n-(2-chlorophenyl)benzamideHuman2063
AURKA (AurA)AurOther3h10A9-chloro-7-(2,6-difluorophenyl)-n-{4-[(4-methylpiperazin-1-yl)carbonyl]phenyl}-5h-pyrimido[5,4-d][2]benzazepin-2-amineHuman2009
AURKA (AurA)AurOther3h10B9-chloro-7-(2,6-difluorophenyl)-n-{4-[(4-methylpiperazin-1-yl)carbonyl]phenyl}-5h-pyrimido[5,4-d][2]benzazepin-2-amineHuman1988
AURKA (AurA)AurOther3h10D9-chloro-7-(2,6-difluorophenyl)-n-{4-[(4-methylpiperazin-1-yl)carbonyl]phenyl}-5h-pyrimido[5,4-d][2]benzazepin-2-amineHuman2059
AURKA (AurA)AurOther3ha6An~2~-(3,4-dimethoxyphenyl)-n~4~-[2-(2-fluorophenyl)ethyl]-n~6~-quinolin-6-yl-1,3,5-triazine-2,4,6-triamineHuman2048
AURKA (AurA)AurOther3k5uA2-[(5,6-diphenylfuro[2,3-d]pyrimidin-4-yl)amino]ethanolHuman2031
AURKA (AurA)AurOther3lauAn-[6-(4-hydroxyphenyl)-1h-indazol-3-yl]butanamideHuman1971
AURKA (AurA)AurOther3m11A1-(4-{2-[(5,6-diphenylfuro[2,3-d]pyrimidin-4-yl)amino]ethyl}phenyl)-3-phenylureaHuman2036
AURKA (AurA)AurOther3mygA2-{ethyl[(5-{[6-methyl-3-(1h-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-yl]amino}isothiazol-3-yl)methyl]amino}-2-methylpropan-1-olHuman2065
AURKA (AurA)AurOther3nrmAn-(3-methylisothiazol-5-yl)-3-(1h-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-amineHuman2052
AURKA (AurA)AurOther3o50An-{3-methyl-4-[(3-pyrimidin-4-ylpyridin-2-yl)oxy]phenyl}-3-(trifluoromethyl)benzamideHuman1958
AURKA (AurA)AurOther3o50Bn-{3-methyl-4-[(3-pyrimidin-4-ylpyridin-2-yl)oxy]phenyl}-3-(trifluoromethyl)benzamideHuman2067
AURKA (AurA)AurOther3o51An-[4-({3-[5-fluoro-2-(methylideneamino)pyrimidin-4-yl]pyridin-2-yl}oxy)phenyl]-2-(phenylamino)benzamideHuman1974
AURKA (AurA)AurOther3p9jA4-[(5-methyl-1h-pyrazol-3-yl)amino]-2-phenylphthalazin-1(2h)-oneHuman2003
AURKA (AurA)AurOther3qbnA5-chloro-n~4~-cyclopropyl-n~2~-[4-(2-methoxyethoxy)phenyl]pyrimidine-2,4-diamineHuman2032
AURKA (AurA)AurOther3r21AAn-(2-aminoethyl)-n-{5-[(1-cycloheptyl-1h-pyrazolo[3,4-d]pyrimidin-6-yl)amino]pyridin-2-yl}methanesulfonamideHuman1991
AURKA (AurA)AurOther3r21ABn-(2-aminoethyl)-n-{5-[(1-cycloheptyl-1h-pyrazolo[3,4-d]pyrimidin-6-yl)amino]pyridin-2-yl}methanesulfonamideHuman2033
AURKA (AurA)AurOther3r22An-{5-[(1-cycloheptyl-1h-pyrazolo[3,4-d]pyrimidin-6-yl)amino]pyridin-2-yl}methanesulfonamideHuman2034
AURKA (AurA)AurOther3unzA4-({4-[(2-fluorophenyl)amino]pyrimidin-2-yl}amino)benzoic acidHuman1972
AURKA (AurA)AurOther3unzB4-({4-[(2-fluorophenyl)amino]pyrimidin-2-yl}amino)benzoic acidHuman2049
AURKA (AurA)AurOther3uo4A4-{[4-(biphenyl-2-ylamino)pyrimidin-2-yl]amino}benzoic acidHuman1976
AURKA (AurA)AurOther3uo5A4-{[4-(phenylamino)pyrimidin-2-yl]amino}benzoic acidHuman2045
AURKA (AurA)AurOther3uo6A4-({4-[(2-chlorophenyl)amino]pyrimidin-2-yl}amino)benzoic acidHuman1985
AURKA (AurA)AurOther3uo6B4-({4-[(2-chlorophenyl)amino]pyrimidin-2-yl}amino)benzoic acidHuman1960
AURKA (AurA)AurOther3uodA4-[(4-{[2-(trifluoromethyl)phenyl]amino}pyrimidin-2-yl)amino]benzoic acidHuman1980
AURKA (AurA)AurOther3uohA4-({4-[(2-bromophenyl)amino]pyrimidin-2-yl}amino)benzoic acidHuman2077
AURKA (AurA)AurOther3uohB4-({4-[(2-bromophenyl)amino]pyrimidin-2-yl}amino)benzoic acidHuman2000
AURKA (AurA)AurOther3uojA4-({4-[(2-cyanophenyl)amino]pyrimidin-2-yl}amino)benzoic acidHuman2042
AURKA (AurA)AurOther3uojB4-({4-[(2-cyanophenyl)amino]pyrimidin-2-yl}amino)benzoic acidHuman1979
AURKA (AurA)AurOther3uokA4-({4-[(2-chlorophenyl)amino]-5-fluoropyrimidin-2-yl}amino)benzoic acidHuman2054
AURKA (AurA)AurOther3uokB4-({4-[(2-chlorophenyl)amino]-5-fluoropyrimidin-2-yl}amino)benzoic acidHuman2047
AURKA (AurA)AurOther3uolAn~4~-(2-chlorophenyl)-n~2~-[4-(1h-tetrazol-5-yl)phenyl]pyrimidine-2,4-diamineHuman2004
AURKA (AurA)AurOther3uolBn~4~-(2-chlorophenyl)-n~2~-[4-(1h-tetrazol-5-yl)phenyl]pyrimidine-2,4-diamineHuman2051
AURKA (AurA)AurOther3up2A4-[(4-{[2-(trifluoromethoxy)phenyl]amino}pyrimidin-2-yl)amino]benzoic acidHuman2005
AURKA (AurA)AurOther3up7A2-({2-[(4-carboxyphenyl)amino]pyrimidin-4-yl}amino)benzoic acidHuman2025
AURKA (AurA)AurOther3vapA3-(1-{2-[(3-fluoropyridinium-4-yl)amino]-2-oxoethyl}-1h-pyrazol-4-yl)-6-methyl-8-[(3-{[(1r,3r)-3-methylpiperidinium-1-yl]methyl}-1,2-thiazol-5-yl)amino]imidazo[1,2-a]pyrazin-1-iumHuman2029
AURKA (AurA)AurOther3w10A1-(3-methoxyphenyl)-n-(5-methyl-1h-pyrazol-3-yl)isoquinolin-3-amineHuman2068
AURKA (AurA)AurOther3w16A4-[(5-methyl-1h-pyrazol-3-yl)amino]-2-phenylphthalazin-1(2h)-oneHuman2012
AURKA (AurA)AurOther3w18A2-{3-[3-(1h-benzimidazol-2-yl)-1h-indazol-6-yl]-1h-pyrazol-5-yl}-n-(3-fluorophenyl)acetamideHuman1961
AURKA (AurA)AurOther3w18B2-{3-[3-(1h-benzimidazol-2-yl)-1h-indazol-6-yl]-1h-pyrazol-5-yl}-n-(3-fluorophenyl)acetamideHuman1967
AURKA (AurA)AurOther3w2cA2-{4-[3-(1h-benzimidazol-2-yl)-1h-indazol-6-yl]-1h-pyrazol-1-yl}-n-(3-methylbutyl)acetamideHuman2066
AURKA (AurA)AurOther3w2cC2-{4-[3-(1h-benzimidazol-2-yl)-1h-indazol-6-yl]-1h-pyrazol-1-yl}-n-(3-methylbutyl)acetamideHuman2021
AURKA (AurA)AurOther3w2cE2-{4-[3-(1h-benzimidazol-2-yl)-1h-indazol-6-yl]-1h-pyrazol-1-yl}-n-(3-methylbutyl)acetamideHuman1953
AURKA (AurA)AurOther3w2cG2-{4-[3-(1h-benzimidazol-2-yl)-1h-indazol-6-yl]-1h-pyrazol-1-yl}-n-(3-methylbutyl)acetamideHuman2026
AURKA (AurA)AurOther4b0gAA6-bromo-2-(1-methyl-1h-imidazol-5-yl)-7-{4-[(5-methyl-1,2-oxazol-3-yl)methyl]piperazin-1-yl}-1h-imidazo[4,5-b]pyridineHuman2082
AURKA (AurA)AurOther4b0gAB6-bromo-2-(1-methyl-1h-imidazol-5-yl)-7-{4-[(5-methyl-1,2-oxazol-3-yl)methyl]piperazin-1-yl}-1h-imidazo[4,5-b]pyridineHuman2070
AURKA (AurA)AurOther4bn1AAadenosine-5'-diphosphateHuman1955
AURKA (AurA)AurOther4bn1ABadenosine-5'-diphosphateHuman1983
AURKA (AurA)AurOther4byiA(s)-n-((1-(6-chloro-2-(1,3-dimethyl-1h-pyrazol-4-yl)-3h-imidazo[4,5-b]pyridin-7-yl)pyrrolidin-3-yl)methyl)acetamideHuman1992
AURKA (AurA)AurOther4byjA(s)-n-(1-(6-chloro-2-(1,3-dimethyl-1h-pyrazol-4-yl)-3h-imidazo[4,5-b]pyridin-7-yl)pyrrolidin-3-yl)acetamideHuman1969
AURKA (AurA)AurOther4c3pAphosphomethylphosphonic acid adenylate esterHuman2018
AURKA (AurA)AurOther4c3pDphosphomethylphosphonic acid adenylate esterHuman2030
AURKA (AurA)AurOther4c3rAphosphomethylphosphonic acid adenylate esterHuman2058
AURKA (AurA)AurOther4cegAadenosine-5'-diphosphateHuman2073
AURKA (AurA)AurOther4deaA4,4'-(pyrimidine-2,4-diyldiimino)dibenzoic acidHuman2064
AURKA (AurA)AurOther4debA4-[(4-{[3-(trifluoromethyl)phenyl]amino}pyrimidin-2-yl)amino]benzamideHuman1996
AURKA (AurA)AurOther4dedA2-({2-[(4-carbamoylphenyl)amino]pyrimidin-4-yl}amino)benzamideHuman2043
AURKA (AurA)AurOther4deeAadenosine-5'-diphosphateHuman1952
AURKA (AurA)AurOther4dhfA7-cyclopentyl-2-({1-methyl-5-[(4-methylpiperazin-1-yl)carbonyl]-1h-pyrrol-3-yl}amino)-7h-pyrrolo[2,3-d]pyrimidine-6-carboxamideHuman1964
AURKA (AurA)AurOther4dhfB7-cyclopentyl-2-({1-methyl-5-[(4-methylpiperazin-1-yl)carbonyl]-1h-pyrrol-3-yl}amino)-7h-pyrrolo[2,3-d]pyrimidine-6-carboxamideHuman1982
AURKA (AurA)AurOther4j8mA1-[4-[[4-[(5-cyclopentyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl]amino]phenyl]-3-[3-(trifluoromethyl)phenyl]ureaHuman2020
AURKA (AurA)AurOther4j8nA-Human2028
AURKA (AurA)AurOther4j8nB-Human2061
AURKA (AurA)AurOther4j8nC-Human2007
AURKA (AurA)AurOther4j8nD-Human1995
AURKA (AurA)AurOther4jaiAn-{4-[(6-oxo-5,6-dihydrobenzo[c][1,8]naphthyridin-1-yl)amino]phenyl}benzamideHuman1999
AURKA (AurA)AurOther4jajAbenzo[c][1,8]naphthyridin-6(5h)-oneHuman2040
AURKA (AurA)AurOther4jboA1-(4-{2-[(6-{4-[2-(dimethylamino)ethoxy]phenyl}furo[2,3-d]pyrimidin-4-yl)amino]ethyl}phenyl)-3-phenylureaHuman2072
AURKA (AurA)AurOther4jbpA1-(4-{2-[(6-{4-[2-(4-hydroxypiperidin-1-yl)ethoxy]phenyl}furo[2,3-d]pyrimidin-4-yl)amino]ethyl}phenyl)-3-phenylureaHuman2041
AURKA (AurA)AurOther4jbqAcyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amideHuman1957
AURKA (AurA)AurOther4o0sAadenosineHuman2039
AURKA (AurA)AurOther4o0uAadenosineHuman2022
AURKA (AurA)AurOther4o0wAadenosineHuman1959
AURKA (AurA)AurOther4prjAn-[1-(3-cyanobenzyl)-1h-pyrazol-4-yl]-6-(1h-pyrazol-4-yl)-1h-indazole-3-carboxamideHuman2023
AURKA (AurA)AurOther4uynAethyl (9s)-9-[5-(1h-benzimidazol-2-ylsulfanyl)furan-2-yl]-8-hydroxy-5,6,7,9-tetrahydro-2h-pyrrolo[3,4-b]quinoline-3-carboxylateHuman2002
AURKA (AurA)AurOther4uzdAethyl (9s)-9-[3-(1h-benzimidazol-2-yloxy)phenyl]-8-oxo-4,5,6,7,8,9-hexahydro-2h-pyrrolo[3,4-b]quinoline-3-carboxylateHuman2013
AURKA (AurA)AurOther4uzdBethyl (9s)-9-[3-(1h-benzimidazol-2-yloxy)phenyl]-8-oxo-4,5,6,7,8,9-hexahydro-2h-pyrrolo[3,4-b]quinoline-3-carboxylateHuman1968
AURKA (AurA)AurOther4uzhA(4s)-4-(2-fluorophenyl)-2,4,6,7,8,9-hexahydro-5h-pyrazolo[3,4-b][1,7]naphthyridin-5-oneHuman1998
AURKA (AurA)AurOther4zs0A5-hydroxy-1'h-1,2'-bibenzimidazol-2(3h)-oneHuman6801
AURKA (AurA)AurOther4ztqA(2z,5z)-2-[(4-ethylphenyl)imino]-3-(2-methoxyethyl)-5-(pyridin-4-ylmethylidene)-1,3-thiazolidin-4-oneHuman6804
AURKA (AurA)AurOther4ztrA6-({4-[(z)-{(2z)-2-[(4-ethylphenyl)imino]-3-methyl-4-oxo-1,3-thiazolidin-5-ylidene}methyl]pyridin-2-yl}amino)pyridine-3-carboxylic acidHuman6817
AURKA (AurA)AurOther4ztsA(2z,5z)-2-[(4-ethylphenyl)imino]-3-methyl-5-[(2-{[4-(1h-tetrazol-5-yl)phenyl]amino}pyridin-4-yl)methylidene]-1,3-thiazolidin-4-oneHuman6814
AURKA (AurA)AurOther5aadA7-(1-benzyl-1h-pyrazol-4-yl)-6-chloro-2-(1,3-dimethyl-1h-pyrazol-4-yl)-3h-imidazo[4,5-b]pyridineHuman6011
AURKA (AurA)AurOther5aaeA3-((4-(6-chloro-2-(1,3-dimethyl-1h-pyrazol-4-yl)-3h-imidazo[4,5-b]pyridin-7-yl)-1h-pyrazol-1-yl)methyl)-5-methylisoxazoleHuman6012
AURKA (AurA)AurOther5aafA3-((4-(6-chloro-2-(1,3-dimethyl-1h-pyrazol-4-yl)-3h-imidazo[4,5-b]pyridin-7-yl)-1h-pyrazol-1-yl)methyl)-n,n-dimethylbenzamideHuman6013
AURKA (AurA)AurOther5aagA[3-[[4-[6-chloranyl-2-(1,3-dimethylpyrazol-4-yl)-3h-imidazo[4,5-b]pyridin-7-yl]pyrazol-1-yl]methyl]phenyl]-(4-methylpiperazin-1-yl)methanoneHuman6010
AURKA (AurA)AurOther5dn3AAadenosine-5'-triphosphateHuman6802
AURKA (AurA)AurOther5dn3ABadenosine-5'-triphosphateHuman6818
AURKA (AurA)AurOther5dnrAAadenosine-5'-triphosphateHuman6810
AURKA (AurA)AurOther5dnrABadenosine-5'-triphosphateHuman6809
AURKA (AurA)AurOther5dosAadenosine-5'-triphosphateHuman6807
AURKA (AurA)AurOther5dpvAA4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHuman6808
AURKA (AurA)AurOther5dpvAB4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHuman6826
AURKA (AurA)AurOther5dr2Aadenosine-5'-triphosphateHuman6825
AURKA (AurA)AurOther5dr6AA4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHuman6811
AURKA (AurA)AurOther5dr6AB4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHuman6805
AURKA (AurA)AurOther5dr9A4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHuman6821
AURKA (AurA)AurOther5drdAadenosine-5'-triphosphateHuman6823
AURKA (AurA)AurOther5dt0AA4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHuman6806
AURKA (AurA)AurOther5dt0AB4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHuman6803
AURKA (AurA)AurOther5dt3Aadenosine-5'-triphosphateHuman6816
AURKA (AurA)AurOther5dt4Aadenosine-5'-triphosphateHuman6815
AURKA (AurA)AurOther5ew9AA4-(3-chloranyl-2-fluoranyl-phenoxy)-1-[[6-(1,3-thiazol-2-ylamino)pyridin-2-yl]methyl]cyclohexane-1-carboxylic acidHuman6359
AURKA (AurA)AurOther5ew9AB4-(3-chloranyl-2-fluoranyl-phenoxy)-1-[[6-(1,3-thiazol-2-ylamino)pyridin-2-yl]methyl]cyclohexane-1-carboxylic acidHuman6360
AURKA (AurA)AurOther5g15AAphosphomethylphosphonic acid adenylate esterHuman9737
AURKA (AurA)AurOther5g15ABphosphomethylphosphonic acid adenylate esterHuman9739
AURKA (AurA)AurOther5g1xAAadenosine-5'-diphosphateHuman7267
AURKA (AurA)AurOther5g1xABadenosine-5'-diphosphateHuman7266
AURKA (AurA)AurOther5l8jAAadenosine-5'-diphosphateHuman6820
AURKA (AurA)AurOther5l8jABadenosine-5'-diphosphateHuman6812
AURKA (AurA)AurOther5l8kAAadenosine-5'-diphosphateHuman6819
AURKA (AurA)AurOther5l8kABadenosine-5'-diphosphateHuman6813
AURKA (AurA)AurOther5l8lAAadenosine-5'-diphosphateHuman6822
AURKA (AurA)AurOther5l8lABadenosine-5'-diphosphateHuman6824
AURKA (AurA)AurOther5lxmAAadenosine-5'-diphosphateHuman7142
AURKA (AurA)AurOther5lxmABadenosine-5'-diphosphateHuman7141
AURKA (AurA)AurOther5objAadenosine-5'-triphosphateHuman8305
AURKA (AurA)AurOther5obrA4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHuman8304
AURKA (AurA)AurOther5odtAAadenosine-5'-diphosphateHuman9738
AURKA (AurA)AurOther5odtABadenosine-5'-diphosphateHuman9736
AURKA (AurA)AurOther5oneAA4-(propanoylamino)-~{n}-[4-[(5,8,11-trimethyl-6-oxidanylidene-pyrimido[4,5-b][1,4]benzodiazepin-2-yl)amino]phenyl]benzamideHuman8371
AURKA (AurA)AurOther5oneAB4-(propanoylamino)-~{n}-[4-[(5,8,11-trimethyl-6-oxidanylidene-pyrimido[4,5-b][1,4]benzodiazepin-2-yl)amino]phenyl]benzamideHuman8370
AURKA (AurA)AurOther5orlAadenosine-5'-diphosphateHuman8642
AURKA (AurA)AurOther5ornAadenosine-5'-diphosphateHuman8649
AURKA (AurA)AurOther5oroAadenosine-5'-diphosphateHuman8641
AURKA (AurA)AurOther5orpAadenosine-5'-diphosphateHuman8648
AURKA (AurA)AurOther5orrAadenosine-5'-diphosphateHuman8636
AURKA (AurA)AurOther5orsAadenosine-5'-diphosphateHuman8646
AURKA (AurA)AurOther5ortAadenosine-5'-diphosphateHuman8638
AURKA (AurA)AurOther5orvAadenosine-5'-diphosphateHuman8643
AURKA (AurA)AurOther5orwAadenosine-5'-diphosphateHuman8631
AURKA (AurA)AurOther5orxAadenosine-5'-diphosphateHuman8644
AURKA (AurA)AurOther5oryAadenosine-5'-diphosphateHuman8627
AURKA (AurA)AurOther5orzAAadenosine-5'-diphosphateHuman8639
AURKA (AurA)AurOther5orzABadenosine-5'-diphosphateHuman8650
AURKA (AurA)AurOther5os0Aadenosine-5'-diphosphateHuman8632
AURKA (AurA)AurOther5os1AAadenosine-5'-diphosphateHuman8628
AURKA (AurA)AurOther5os1ABadenosine-5'-diphosphateHuman8630
AURKA (AurA)AurOther5os2AAadenosine-5'-diphosphateHuman8635
AURKA (AurA)AurOther5os2ABadenosine-5'-diphosphateHuman8633
AURKA (AurA)AurOther5os3Aadenosine-5'-diphosphateHuman8637
AURKA (AurA)AurOther5os4Aadenosine-5'-diphosphateHuman8652
AURKA (AurA)AurOther5os5AAadenosine-5'-diphosphateHuman8647
AURKA (AurA)AurOther5os5ABadenosine-5'-diphosphateHuman8629
AURKA (AurA)AurOther5os6Aadenosine-5'-diphosphateHuman8651
AURKA (AurA)AurOther5osdAadenosine-5'-diphosphateHuman8634
AURKA (AurA)AurOther5oseAadenosine-5'-diphosphateHuman8645
AURKA (AurA)AurOther5osfAadenosine-5'-diphosphateHuman8640
AURKA (AurA)AurOther5zanA7-(4-methylpiperazin-1-yl)-n-(5-methyl-1h-pyrazol-3-yl)-2-[(e)-2-phenylethenyl]quinazolin-4-amineHuman10898
AURKA (AurA)AurOther6c2rAA(2r,4r)-1-[(3-chloro-2-fluorophenyl)methyl]-4-({3-fluoro-6-[(5-methyl-1h-pyrazol-3-yl)amino]pyridin-2-yl}methyl)-2-methylpiperidine-4-carboxylic acidHuman10864
AURKA (AurA)AurOther6c2rAB(2r,4r)-1-[(3-chloro-2-fluorophenyl)methyl]-4-({3-fluoro-6-[(5-methyl-1h-pyrazol-3-yl)amino]pyridin-2-yl}methyl)-2-methylpiperidine-4-carboxylic acidHuman10865
AURKA (AurA)AurOther6c2tAA(2s,4r)-1-[(3-chloro-2-fluorophenyl)methyl]-2-methyl-4-({3-[(1,3-thiazol-2-yl)amino]isoquinolin-1-yl}methyl)piperidine-4-carboxylic acidHuman10866
AURKA (AurA)AurOther6c2tAB(2s,4r)-1-[(3-chloro-2-fluorophenyl)methyl]-2-methyl-4-({3-[(1,3-thiazol-2-yl)amino]isoquinolin-1-yl}methyl)piperidine-4-carboxylic acidHuman10863
AURKA (AurA)AurOther6c83Aphosphomethylphosphonic acid adenylate esterHuman10934
AURKA (AurA)AurOther6c83Bphosphomethylphosphonic acid adenylate esterHuman10935
AURKA (AurA)AurOther6cpeAA-Human10036
AURKA (AurA)AurOther6cpeAB-Human10035
AURKA (AurA)AurOther6cpfAphosphomethylphosphonic acid adenylate esterHuman10033
AURKA (AurA)AurOther6cpgA1-cyclopropyl-3-{3-[5-(morpholin-4-ylmethyl)-1h-benzimidazol-2-yl]-1h-pyrazol-4-yl}ureaHuman10032
AURKA (AurA)AurOther6cpgD1-cyclopropyl-3-{3-[5-(morpholin-4-ylmethyl)-1h-benzimidazol-2-yl]-1h-pyrazol-4-yl}ureaHuman10034
AURKA (AurA)AurOther6graA1-[(2~{r},3~{s})-2-[[1,3-benzodioxol-5-ylmethyl(methyl)amino]methyl]-3-methyl-6-oxidanylidene-5-[(2~{s})-1-oxidanylpropan-2-yl]-3,4-dihydro-2~{h}-1,5-benzoxazocin-8-yl]-3-(4-methoxyphenyl)ureaHuman11130
AURKA (AurA)AurOther6hjjAA~{n}-[4-(4-azanyl-1-propan-2-yl-pyrazolo[3,4-d]pyrimidin-3-yl)-3-methyl-phenyl]-4-[4-fluoranyl-3-(trifluoromethyl)phenyl]-4-oxidanylidene-butanamideHuman10410
AURKA (AurA)AurOther6hjjAB~{n}-[4-(4-azanyl-1-propan-2-yl-pyrazolo[3,4-d]pyrimidin-3-yl)-3-methyl-phenyl]-4-[4-fluoranyl-3-(trifluoromethyl)phenyl]-4-oxidanylidene-butanamideHuman10412
AURKA (AurA)AurOther6hjkA(~{e})-~{n}-[4-(4-azanyl-1-propan-2-yl-pyrazolo[3,4-d]pyrimidin-3-yl)phenyl]-4-[4-fluoranyl-3-(trifluoromethyl)phenyl]-4-oxidanylidene-but-2-enamideHuman10411
AURKA (AurA)AurOther6i2uA-Human11652
AURKA (AurA)AurOther6r49Aadenosine-5'-diphosphateHuman11131
AURKA (AurA)AurOther6r4aAadenosine-5'-diphosphateHuman11134
AURKA (AurA)AurOther6r4bABadenosine-5'-diphosphateHuman11133
AURKA (AurA)AurOther6r4cAadenosine-5'-diphosphateHuman11135
AURKA (AurA)AurOther6r4dAadenosine-5'-diphosphateHuman11132
AURKA (AurA)AurOther6vpgAAphosphoaminophosphonic acid-adenylate esterHuman12659
AURKA (AurA)AurOther6vpgABphosphoaminophosphonic acid-adenylate esterHuman12667
AURKA (AurA)AurOther6vphAAdithiane diolHuman12666
AURKA (AurA)AurOther6vphABdithiane diolHuman12655
AURKA (AurA)AurOther6vpiAAphosphoaminophosphonic acid-adenylate esterHuman12656
AURKA (AurA)AurOther6vpiABphosphoaminophosphonic acid-adenylate esterHuman12669
AURKA (AurA)AurOther6vpjAAphosphoaminophosphonic acid-adenylate esterHuman12657
AURKA (AurA)AurOther6vpjABphosphoaminophosphonic acid-adenylate esterHuman12654
AURKA (AurA)AurOther6vplAAphosphoaminophosphonic acid-adenylate esterHuman12662
AURKA (AurA)AurOther6vplABphosphoaminophosphonic acid-adenylate esterHuman12670
AURKA (AurA)AurOther6vplBAphosphoaminophosphonic acid-adenylate esterHuman12664
AURKA (AurA)AurOther6vplBBphosphoaminophosphonic acid-adenylate esterHuman12668
AURKA (AurA)AurOther6vpmAAadenosine monophosphateHuman12661
AURKA (AurA)AurOther6vpmABadenosine monophosphateHuman12658
AURKA (AurA)AurOther6vpmBAadenosine monophosphateHuman12660
AURKA (AurA)AurOther6vpmBBadenosine monophosphateHuman12663
AURKA (AurA)AurOther6xkaA-Human12665
AURKA (AurA)AurOther6z4yAA6-(2-methoxyethoxy)-11-methyl-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one Human12306
AURKA (AurA)AurOther6z4yAB6-(2-methoxyethoxy)-11-methyl-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one Human12307
AURKB (AurB)AurOther4af3Acyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amideHuman407
AURKC (AurC)AurOther6gr8AA1-[(2~{r},3~{s})-2-[[1,3-benzodioxol-5-ylmethyl(methyl)amino]methyl]-3-methyl-6-oxidanylidene-5-[(2~{s})-1-oxidanylpropan-2-yl]-3,4-dihydro-2~{h}-1,5-benzoxazocin-8-yl]-3-(4-methoxyphenyl)ureaHuman11122
AURKC (AurC)AurOther6gr8AB1-[(2~{r},3~{s})-2-[[1,3-benzodioxol-5-ylmethyl(methyl)amino]methyl]-3-methyl-6-oxidanylidene-5-[(2~{s})-1-oxidanylpropan-2-yl]-3,4-dihydro-2~{h}-1,5-benzoxazocin-8-yl]-3-(4-methoxyphenyl)ureaHuman11125
AURKC (AurC)AurOther6gr9AAcyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amideHuman11123
AURKC (AurC)AurOther6gr9ABcyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amideHuman11124
AXLAxlTK5u6bA(10r)-7-amino-11-chloro-12-fluoro-1-(2-hydroxyethyl)-3,10,16-trimethyl-16,17-dihydro-1h-8,4-(azeno)pyrazolo[4,3-h][2,5,11]benzoxadiazacyclotetradecin-15(10h)-oneHuman8258
AXLAxlTK5u6bB(10r)-7-amino-11-chloro-12-fluoro-1-(2-hydroxyethyl)-3,10,16-trimethyl-16,17-dihydro-1h-8,4-(azeno)pyrazolo[4,3-h][2,5,11]benzoxadiazacyclotetradecin-15(10h)-oneHuman8260
AXLAxlTK5u6bC(10r)-7-amino-11-chloro-12-fluoro-1-(2-hydroxyethyl)-3,10,16-trimethyl-16,17-dihydro-1h-8,4-(azeno)pyrazolo[4,3-h][2,5,11]benzoxadiazacyclotetradecin-15(10h)-oneHuman8257
AXLAxlTK5u6bD(10r)-7-amino-11-chloro-12-fluoro-1-(2-hydroxyethyl)-3,10,16-trimethyl-16,17-dihydro-1h-8,4-(azeno)pyrazolo[4,3-h][2,5,11]benzoxadiazacyclotetradecin-15(10h)-oneHuman8259
BMP2K (BIKE)NAKOther4w9wAA5-(3-fluorophenyl)-n-[(3s)-3-piperidyl]-3-ureido-thiophene-2-carboxamideHuman3274
BMP2K (BIKE)NAKOther4w9wAB5-(3-fluorophenyl)-n-[(3s)-3-piperidyl]-3-ureido-thiophene-2-carboxamideHuman3272
BMP2K (BIKE)NAKOther4w9xAbaricitinibHuman3273
BMP2K (BIKE)NAKOther5i3oAn-(6-{3-[(dimethylsulfamoyl)amino]phenyl}-1h-indazol-3-yl)cyclopropanecarboxamideHuman6437
BMP2K (BIKE)NAKOther5i3oBn-(6-{3-[(dimethylsulfamoyl)amino]phenyl}-1h-indazol-3-yl)cyclopropanecarboxamideHuman6434
BMP2K (BIKE)NAKOther5i3rAn-[6-(3-{[(cyclopropylmethyl)sulfonyl]amino}phenyl)-1h-indazol-3-yl]cyclopropanecarboxamideHuman6435
BMP2K (BIKE)NAKOther5i3rBn-[6-(3-{[(cyclopropylmethyl)sulfonyl]amino}phenyl)-1h-indazol-3-yl]cyclopropanecarboxamideHuman6436
BMP2K (BIKE)NAKOther5ikwAn-(6-{3-[(cyclopropylsulfonyl)amino]phenyl}-1h-indazol-3-yl)cyclopropanecarboxamideHuman6709
BMPR1BSTKRTKL3mdyAA4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1502
BMPR1BSTKRTKL3mdyAB4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1501
BMPR1BSTKRTKL3mdyCA4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1503
BMPR1BSTKRTKL3mdyCB4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1500
BMPR2STKRTKL3g2fAAadenosine-5'-diphosphateHuman6870
BMPR2STKRTKL3g2fABadenosine-5'-diphosphateHuman6868
BMPR2STKRTKL3g2fBAadenosine-5'-diphosphateHuman6867
BMPR2STKRTKL3g2fBBadenosine-5'-diphosphateHuman6869
BMXTecTK3sxrAn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman3482
BMXTecTK3sxrBn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman3481
BMXTecTK3sxsA1-tert-butyl-3-(4-chloro-phenyl)-1h-pyrazolo[3,4-d]pyrimidin-4-ylamineHuman3483
BMXTecTK6i99A~{n}-[2-methyl-5-[8-[4-(methylsulfonylamino)phenyl]-2-oxidanylidene-benzo[h][1,6]naphthyridin-1-yl]phenyl]-3-oxidanyl-propanamideHuman12348
BMXTecTK6i99B~{n}-[2-methyl-5-[8-[4-(methylsulfonylamino)phenyl]-2-oxidanylidene-benzo[h][1,6]naphthyridin-1-yl]phenyl]-3-oxidanyl-propanamideHuman12349
BRAFRAFTKL1uwhA4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamideHuman3127
BRAFRAFTKL1uwhB4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamideHuman3109
BRAFRAFTKL1uwjA4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamideHuman3135
BRAFRAFTKL1uwjB4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamideHuman3105
BRAFRAFTKL2fb8A(1z)-5-(2-{4-[2-(dimethylamino)ethoxy]phenyl}-5-pyridin-4-yl-1h-imidazol-4-yl)indan-1-one oximeHuman3062
BRAFRAFTKL2fb8B(1z)-5-(2-{4-[2-(dimethylamino)ethoxy]phenyl}-5-pyridin-4-yl-1h-imidazol-4-yl)indan-1-one oximeHuman3086
BRAFRAFTKL3c4cAn-{3-[(5-chloro-1h-pyrrolo[2,3-b]pyridin-3-yl)carbonyl]-2,4-difluorophenyl}propane-1-sulfonamideHuman3115
BRAFRAFTKL3c4cBn-{3-[(5-chloro-1h-pyrrolo[2,3-b]pyridin-3-yl)carbonyl]-2,4-difluorophenyl}propane-1-sulfonamideHuman3063
BRAFRAFTKL3d4qA(1e)-5-(1-piperidin-4-yl-3-pyridin-4-yl-1h-pyrazol-4-yl)-2,3-dihydro-1h-inden-1-one oximeHuman3095
BRAFRAFTKL3d4qB(1e)-5-(1-piperidin-4-yl-3-pyridin-4-yl-1h-pyrazol-4-yl)-2,3-dihydro-1h-inden-1-one oximeHuman3060
BRAFRAFTKL3idpAn~1~-(4-chlorophenyl)-6-methyl-n~5~-[3-(7h-purin-6-yl)pyridin-2-yl]isoquinoline-1,5-diamineHuman3077
BRAFRAFTKL3idpBn~1~-(4-chlorophenyl)-6-methyl-n~5~-[3-(7h-purin-6-yl)pyridin-2-yl]isoquinoline-1,5-diamineHuman3121
BRAFRAFTKL3ii5An-[3-(3-{4-[(dimethylamino)methyl]phenyl}pyrazolo[1,5-a]pyrimidin-7-yl)phenyl]-3-(trifluoromethyl)benzamideHuman3116
BRAFRAFTKL3ii5Bn-[3-(3-{4-[(dimethylamino)methyl]phenyl}pyrazolo[1,5-a]pyrimidin-7-yl)phenyl]-3-(trifluoromethyl)benzamideHuman3076
BRAFRAFTKL3og7An-(3-{[5-(4-chlorophenyl)-1h-pyrrolo[2,3-b]pyridin-3-yl]carbonyl}-2,4-difluorophenyl)propane-1-sulfonamideHuman3113
BRAFRAFTKL3og7B-Human3140
BRAFRAFTKL3ppjAmethyl 3-{[(5s)-1-(hydroxyamino)-5h-inden-5-yl]amino}furo[2,3-c]pyridine-2-carboxylateHuman3091
BRAFRAFTKL3ppjBmethyl 3-{[(5s)-1-(hydroxyamino)-5h-inden-5-yl]amino}furo[2,3-c]pyridine-2-carboxylateHuman3087
BRAFRAFTKL3ppkA3-[(5-hydroxynaphthalen-2-yl)amino]-n-(pyrimidin-4-yl)furo[2,3-c]pyridine-2-carboxamideHuman3106
BRAFRAFTKL3ppkB3-[(5-hydroxynaphthalen-2-yl)amino]-n-(pyrimidin-4-yl)furo[2,3-c]pyridine-2-carboxamideHuman3092
BRAFRAFTKL3prfA2-chloro-5-{[2-(pyrimidin-2-yl)furo[2,3-c]pyridin-3-yl]amino}phenolHuman3129
BRAFRAFTKL3prfB2-chloro-5-{[2-(pyrimidin-2-yl)furo[2,3-c]pyridin-3-yl]amino}phenolHuman3139
BRAFRAFTKL3priA3-(4-{[2-(pyrimidin-2-yl)furo[2,3-c]pyridin-3-yl]amino}-1h-indazol-3-yl)propan-1-olHuman3093
BRAFRAFTKL3priB3-(4-{[2-(pyrimidin-2-yl)furo[2,3-c]pyridin-3-yl]amino}-1h-indazol-3-yl)propan-1-olHuman3103
BRAFRAFTKL3psbAethyl 3-{[1-(hydroxyamino)-2h-inden-5-yl]amino}thieno[2,3-c]pyridine-2-carboxylateHuman3111
BRAFRAFTKL3psbBethyl 3-{[1-(hydroxyamino)-2h-inden-5-yl]amino}thieno[2,3-c]pyridine-2-carboxylateHuman3125
BRAFRAFTKL3psdA6-[1-(piperidin-4-yl)-3-(pyridin-4-yl)-1h-pyrazol-4-yl]indeno[1,2-c]pyrazoleHuman3142
BRAFRAFTKL3psdB6-[1-(piperidin-4-yl)-3-(pyridin-4-yl)-1h-pyrazol-4-yl]indeno[1,2-c]pyrazoleHuman3083
BRAFRAFTKL3q4cA[(1,2,3,4,5,6-eta)-(1s,2r,3r,4r,5s,6s)-1-carboxycyclohexane-1,2,3,4,5,6-hexayl](chloro)(3-methyl-5,7-dioxo-6,7-dihydro-5h-pyrido[2,3-a]pyrrolo[3,4-c]carbazol-12-ide-kappa~2~n~1~,n~12~)ruthenium(1+)Human7251
BRAFRAFTKL3q4cB-Human7250
BRAFRAFTKL3q96A(2s)-n-[3-(2-aminopropan-2-yl)-5-(trifluoromethyl)phenyl]-7-[(7-oxo-5,6,7,8-tetrahydro-1,8-naphthyridin-4-yl)oxy]-1,2,3,4-tetrahydronaphthalene-2-carboxamideHuman3072
BRAFRAFTKL3q96B(2s)-n-[3-(2-aminopropan-2-yl)-5-(trifluoromethyl)phenyl]-7-[(7-oxo-5,6,7,8-tetrahydro-1,8-naphthyridin-4-yl)oxy]-1,2,3,4-tetrahydronaphthalene-2-carboxamideHuman3089
BRAFRAFTKL3skcA2,6-difluoro-n-[(5s)-3-methoxy-5h-pyrazolo[3,4-b]pyridin-5-yl]-3-[(phenylsulfonyl)amino]benzamideHuman3100
BRAFRAFTKL3skcB2,6-difluoro-n-[(5s)-3-methoxy-5h-pyrazolo[3,4-b]pyridin-5-yl]-3-[(phenylsulfonyl)amino]benzamideHuman3128
BRAFRAFTKL3tv4An-(6-amino-5-bromopyridin-3-yl)-2,6-difluoro-3-[(propylsulfonyl)amino]benzamideHuman3054
BRAFRAFTKL3tv4Bn-(6-amino-5-bromopyridin-3-yl)-2,6-difluoro-3-[(propylsulfonyl)amino]benzamideHuman3133
BRAFRAFTKL3tv6A2,6-difluoro-n-(3-methoxy-2h-pyrazolo[3,4-b]pyridin-5-yl)-3-[(propylsulfonyl)amino]benzamideHuman3080
BRAFRAFTKL3tv6B2,6-difluoro-n-(3-methoxy-2h-pyrazolo[3,4-b]pyridin-5-yl)-3-[(propylsulfonyl)amino]benzamideHuman3136
BRAFRAFTKL4cqeAn-{4-[2-(1-cyclopropylpiperidin-4-yl)-4-(3-{[(2,5-difluorophenyl)sulfonyl]amino}-2-fluorophenyl)-1,3-thiazol-5-yl]pyridin-2-yl}acetamideHuman3088
BRAFRAFTKL4cqeBn-{4-[2-(1-cyclopropylpiperidin-4-yl)-4-(3-{[(2,5-difluorophenyl)sulfonyl]amino}-2-fluorophenyl)-1,3-thiazol-5-yl]pyridin-2-yl}acetamideHuman3107
BRAFRAFTKL4dbnA2-chloro-3-(1-cyanocyclopropyl)-n-[5-({2-[(cyclopropylcarbonyl)amino][1,3]thiazolo[5,4-b]pyridin-5-yl}oxy)-2-fluorophenyl]benzamideHuman3052
BRAFRAFTKL4dbnB2-chloro-3-(1-cyanocyclopropyl)-n-[5-({2-[(cyclopropylcarbonyl)amino][1,3]thiazolo[5,4-b]pyridin-5-yl}oxy)-2-fluorophenyl]benzamideHuman3070
BRAFRAFTKL4e26A5-chloro-7-[(r)-furan-2-yl(pyridin-2-ylamino)methyl]quinolin-8-olHuman3108
BRAFRAFTKL4e26B5-chloro-7-[(r)-furan-2-yl(pyridin-2-ylamino)methyl]quinolin-8-olHuman3102
BRAFRAFTKL4e4xAn-(2,4-difluoro-3-{2-[(3-hydroxypropyl)amino]-8-methyl-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl}phenyl)propane-1-sulfonamideHuman3051
BRAFRAFTKL4e4xBn-(2,4-difluoro-3-{2-[(3-hydroxypropyl)amino]-8-methyl-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl}phenyl)propane-1-sulfonamideHuman3104
BRAFRAFTKL4eheA4-amino-n-{2,6-difluoro-3-[(propylsulfonyl)amino]phenyl}thieno[3,2-d]pyrimidine-7-carboxamideHuman3112
BRAFRAFTKL4eheB4-amino-n-{2,6-difluoro-3-[(propylsulfonyl)amino]phenyl}thieno[3,2-d]pyrimidine-7-carboxamideHuman3082
BRAFRAFTKL4ehgAn-{2,4-difluoro-3-[({6-[(2-hydroxyethyl)amino]pyrimidin-4-yl}carbamoyl)amino]phenyl}propane-1-sulfonamideHuman3064
BRAFRAFTKL4ehgBn-{2,4-difluoro-3-[({6-[(2-hydroxyethyl)amino]pyrimidin-4-yl}carbamoyl)amino]phenyl}propane-1-sulfonamideHuman3078
BRAFRAFTKL4fc0A2-chloro-3-[(2-cyanopropan-2-yl)oxy]-n-{5-[{2-[(cyclopropylcarbonyl)amino][1,3]thiazolo[5,4-b]pyridin-5-yl}(methyl)amino]-2-fluorophenyl}benzamideHuman3131
BRAFRAFTKL4fc0B2-chloro-3-[(2-cyanopropan-2-yl)oxy]-n-{5-[{2-[(cyclopropylcarbonyl)amino][1,3]thiazolo[5,4-b]pyridin-5-yl}(methyl)amino]-2-fluorophenyl}benzamideHuman3069
BRAFRAFTKL4fk3An-{2,4-difluoro-3-[(5-pyridin-3-yl-1h-pyrrolo[2,3-b]pyridin-3-yl)carbonyl]phenyl}ethanesulfonamideHuman3118
BRAFRAFTKL4fk3B-Human3068
BRAFRAFTKL4g9cA3-{[3-(2-cyanopropan-2-yl)benzoyl]amino}-2,6-difluoro-n-(3-methoxy-2h-pyrazolo[3,4-b]pyridin-5-yl)benzamideHuman3084
BRAFRAFTKL4g9cB3-{[3-(2-cyanopropan-2-yl)benzoyl]amino}-2,6-difluoro-n-(3-methoxy-2h-pyrazolo[3,4-b]pyridin-5-yl)benzamideHuman3067
BRAFRAFTKL4g9rA3-(2-cyanopropan-2-yl)-n-{4-methyl-3-[(3-methyl-4-oxo-3,4-dihydroquinazolin-6-yl)amino]phenyl}benzamideHuman3130
BRAFRAFTKL4g9rB3-(2-cyanopropan-2-yl)-n-{4-methyl-3-[(3-methyl-4-oxo-3,4-dihydroquinazolin-6-yl)amino]phenyl}benzamideHuman3101
BRAFRAFTKL4h58AAn-(4-{[(2-methoxyethyl)amino]methyl}phenyl)-6-(pyridin-4-yl)quinazolin-2-amineHuman3137
BRAFRAFTKL4h58ABn-(4-{[(2-methoxyethyl)amino]methyl}phenyl)-6-(pyridin-4-yl)quinazolin-2-amineHuman3110
BRAFRAFTKL4h58BA-Human3097
BRAFRAFTKL4h58BB-Human3120
BRAFRAFTKL4h58CA-Human3056
BRAFRAFTKL4h58CB-Human3114
BRAFRAFTKL4jvgA1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-ureaHuman3134
BRAFRAFTKL4jvgB1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-ureaHuman3085
BRAFRAFTKL4jvgC1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-ureaHuman3050
BRAFRAFTKL4jvgD1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-ureaHuman3059
BRAFRAFTKL4kspAn-{7-cyano-6-[4-fluoro-3-({[3-(trifluoromethyl)phenyl]acetyl}amino)phenoxy]-1,3-benzothiazol-2-yl}cyclopropanecarboxamideHuman3081
BRAFRAFTKL4kspBn-{7-cyano-6-[4-fluoro-3-({[3-(trifluoromethyl)phenyl]acetyl}amino)phenoxy]-1,3-benzothiazol-2-yl}cyclopropanecarboxamideHuman3066
BRAFRAFTKL4ksqAn-{7-cyano-6-[4-fluoro-3-({[3-(trifluoromethyl)phenyl]carbamoyl}amino)phenoxy]-1,3-benzothiazol-2-yl}cyclopropanecarboxamideHuman3065
BRAFRAFTKL4ksqBn-{7-cyano-6-[4-fluoro-3-({[3-(trifluoromethyl)phenyl]carbamoyl}amino)phenoxy]-1,3-benzothiazol-2-yl}cyclopropanecarboxamideHuman3055
BRAFRAFTKL4mbjA2,6-difluoro-n-(1h-imidazo[4,5-b]pyridin-6-yl)-3-[(propylsulfonyl)amino]benzamideHuman3090
BRAFRAFTKL4mbjB2,6-difluoro-n-(1h-imidazo[4,5-b]pyridin-6-yl)-3-[(propylsulfonyl)amino]benzamideHuman3057
BRAFRAFTKL4mneBA-Human3075
BRAFRAFTKL4mneBB-Human3061
BRAFRAFTKL4mneCA-Human3122
BRAFRAFTKL4mneCB-Human3058
BRAFRAFTKL4mneFA-Human3099
BRAFRAFTKL4mneFB-Human3117
BRAFRAFTKL4mneGA-Human3071
BRAFRAFTKL4mneGB-Human3073
BRAFRAFTKL4mnfAA2-{4-[(1e)-1-(hydroxyimino)-2,3-dihydro-1h-inden-5-yl]-3-(pyridin-4-yl)-1h-pyrazol-1-yl}ethanolHuman3096
BRAFRAFTKL4mnfAB2-{4-[(1e)-1-(hydroxyimino)-2,3-dihydro-1h-inden-5-yl]-3-(pyridin-4-yl)-1h-pyrazol-1-yl}ethanolHuman3141
BRAFRAFTKL4mnfBA2-{4-[(1e)-1-(hydroxyimino)-2,3-dihydro-1h-inden-5-yl]-3-(pyridin-4-yl)-1h-pyrazol-1-yl}ethanolHuman3124
BRAFRAFTKL4mnfBB2-{4-[(1e)-1-(hydroxyimino)-2,3-dihydro-1h-inden-5-yl]-3-(pyridin-4-yl)-1h-pyrazol-1-yl}ethanolHuman3098
BRAFRAFTKL4pp7An-{2,4-difluoro-3-[methyl(3-methyl-4-oxo-3,4-dihydroquinazolin-6-yl)amino]phenyl}propane-1-sulfonamideHuman3094
BRAFRAFTKL4pp7Bn-{2,4-difluoro-3-[methyl(3-methyl-4-oxo-3,4-dihydroquinazolin-6-yl)amino]phenyl}propane-1-sulfonamideHuman3126
BRAFRAFTKL4r5yA5-({(1r,1as,6br)-1-[5-(trifluoromethyl)-1h-benzimidazol-2-yl]-1a,6b-dihydro-1h-cyclopropa[b][1]benzofuran-5-yl}oxy)-3,4-dihydro-1,8-naphthyridin-2(1h)-oneHuman6414
BRAFRAFTKL4r5yB5-({(1r,1as,6br)-1-[5-(trifluoromethyl)-1h-benzimidazol-2-yl]-1a,6b-dihydro-1h-cyclopropa[b][1]benzofuran-5-yl}oxy)-3,4-dihydro-1,8-naphthyridin-2(1h)-oneHuman6413
BRAFRAFTKL4rzvAn-(3-{[5-(4-chlorophenyl)-1h-pyrrolo[2,3-b]pyridin-3-yl]carbonyl}-2,4-difluorophenyl)propane-1-sulfonamideHuman6944
BRAFRAFTKL4rzvBn-(3-{[5-(4-chlorophenyl)-1h-pyrrolo[2,3-b]pyridin-3-yl]carbonyl}-2,4-difluorophenyl)propane-1-sulfonamideHuman6941
BRAFRAFTKL4rzwA3-(2-cyanopropan-2-yl)-n-{4-methyl-3-[(3-methyl-4-oxo-3,4-dihydroquinazolin-6-yl)amino]phenyl}benzamideHuman6939
BRAFRAFTKL4rzwB3-(2-cyanopropan-2-yl)-n-{4-methyl-3-[(3-methyl-4-oxo-3,4-dihydroquinazolin-6-yl)amino]phenyl}benzamideHuman6942
BRAFRAFTKL4wo5An-{3-[(5-chloro-1h-pyrrolo[2,3-b]pyridin-3-yl)carbonyl]-2,4-difluorophenyl}propane-1-sulfonamideHuman3079
BRAFRAFTKL4wo5Bn-{3-[(5-chloro-1h-pyrrolo[2,3-b]pyridin-3-yl)carbonyl]-2,4-difluorophenyl}propane-1-sulfonamideHuman3143
BRAFRAFTKL4xv1An'-(3-{[5-(2-cyclopropylpyrimidin-5-yl)-1h-pyrrolo[2,3-b]pyridin-3-yl]carbonyl}-2,4-difluorophenyl)-n-ethyl-n-methylsulfuric diamideHuman6214
BRAFRAFTKL4xv1B-Human6216
BRAFRAFTKL4xv2AdabrafenibHuman6213
BRAFRAFTKL4xv2BdabrafenibHuman6219
BRAFRAFTKL4xv3An'-{3-[5-(2-aminopyrimidin-4-yl)-2-tert-butyl-1,3-thiazol-4-yl]-2-fluorophenyl}-n-ethyl-n-methylsulfuric diamideHuman6217
BRAFRAFTKL4xv3B-Human6218
BRAFRAFTKL4xv9AAn-{3-[(5-chloro-1h-pyrrolo[2,3-b]pyridin-3-yl)carbonyl]-2,4-difluorophenyl}-4-(trifluoromethyl)benzenesulfonamideHuman6220
BRAFRAFTKL4xv9ABn-{3-[(5-chloro-1h-pyrrolo[2,3-b]pyridin-3-yl)carbonyl]-2,4-difluorophenyl}-4-(trifluoromethyl)benzenesulfonamideHuman6215
BRAFRAFTKL4yhtA3-[(5-chloro-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamideHuman6442
BRAFRAFTKL4yhtB3-[(5-chloro-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamideHuman6443
BRAFRAFTKL5c9cAA1-(3,3-dimethylbutyl)-3-{2-fluoro-4-methyl-5-[7-methyl-2-(methylamino)pyrido[2,3-d]pyrimidin-6-yl]phenyl}ureaHuman3123
BRAFRAFTKL5c9cAB1-(3,3-dimethylbutyl)-3-{2-fluoro-4-methyl-5-[7-methyl-2-(methylamino)pyrido[2,3-d]pyrimidin-6-yl]phenyl}ureaHuman3074
BRAFRAFTKL5c9cBA1-(3,3-dimethylbutyl)-3-{2-fluoro-4-methyl-5-[7-methyl-2-(methylamino)pyrido[2,3-d]pyrimidin-6-yl]phenyl}ureaHuman3138
BRAFRAFTKL5c9cBB1-(3,3-dimethylbutyl)-3-{2-fluoro-4-methyl-5-[7-methyl-2-(methylamino)pyrido[2,3-d]pyrimidin-6-yl]phenyl}ureaHuman3119
BRAFRAFTKL5cswAdabrafenibHuman6433
BRAFRAFTKL5cswBdabrafenibHuman6431
BRAFRAFTKL5csxAn-(3-{5-[(1-ethylpiperidin-4-yl)(methyl)amino]-3-(pyrimidin-5-yl)-1h-pyrrolo[3,2-b]pyridin-1-yl}-2,4-difluorophenyl)propane-1-sulfonamideHuman6432
BRAFRAFTKL5ct7A1-methyl-5-({2-[5-(trifluoromethyl)-1h-imidazol-2-yl]pyridin-4-yl}oxy)-n-[4-(trifluoromethyl)phenyl]-1h-benzimidazol-2-amineHuman6032
BRAFRAFTKL5ct7B1-methyl-5-({2-[5-(trifluoromethyl)-1h-imidazol-2-yl]pyridin-4-yl}oxy)-n-[4-(trifluoromethyl)phenyl]-1h-benzimidazol-2-amineHuman6033
BRAFRAFTKL5fd2A6-[2-[[3-(dimethylsulfamoylamino)-2,6-bis(fluoranyl)phenyl]amino]pyridin-3-yl]-7~{h}-purineHuman6603
BRAFRAFTKL5fd2B6-[2-[[3-(dimethylsulfamoylamino)-2,6-bis(fluoranyl)phenyl]amino]pyridin-3-yl]-7~{h}-purineHuman6602
BRAFRAFTKL5hi2A4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamideHuman6515
BRAFRAFTKL5hidAA3-(2-cyanopropan-2-yl)-n-{4-methyl-3-[(3-methyl-4-oxo-3,4-dihydroquinazolin-6-yl)amino]phenyl}benzamideHuman6506
BRAFRAFTKL5hidAB3-(2-cyanopropan-2-yl)-n-{4-methyl-3-[(3-methyl-4-oxo-3,4-dihydroquinazolin-6-yl)amino]phenyl}benzamideHuman6512
BRAFRAFTKL5hidBA3-(2-cyanopropan-2-yl)-n-{4-methyl-3-[(3-methyl-4-oxo-3,4-dihydroquinazolin-6-yl)amino]phenyl}benzamideHuman6511
BRAFRAFTKL5hidBB3-(2-cyanopropan-2-yl)-n-{4-methyl-3-[(3-methyl-4-oxo-3,4-dihydroquinazolin-6-yl)amino]phenyl}benzamideHuman6517
BRAFRAFTKL5hieAAdabrafenibHuman6516
BRAFRAFTKL5hieABdabrafenibHuman6508
BRAFRAFTKL5hieBAdabrafenibHuman6509
BRAFRAFTKL5hieBBdabrafenibHuman6505
BRAFRAFTKL5hieCAdabrafenibHuman6513
BRAFRAFTKL5hieCBdabrafenibHuman6507
BRAFRAFTKL5hieDAdabrafenibHuman6510
BRAFRAFTKL5hieDBdabrafenibHuman6514
BRAFRAFTKL5itaAn-{2-cyano-3-[(3-methyl-4-oxo-3,4-dihydroquinazolin-6-yl)amino]phenyl}propane-1-sulfonamideHuman6940
BRAFRAFTKL5itaBn-{2-cyano-3-[(3-methyl-4-oxo-3,4-dihydroquinazolin-6-yl)amino]phenyl}propane-1-sulfonamideHuman6943
BRAFRAFTKL5jrqA(3-{[dihydroxy(propyl)-lambda~4~-sulfanyl]amino}-2,6-difluorophenyl)[5-(4-methoxyphenyl)-1h-pyrrolo[2,3-b]pyridin-3-yl]methanoneHuman7061
BRAFRAFTKL5jrqB(3-{[dihydroxy(propyl)-lambda~4~-sulfanyl]amino}-2,6-difluorophenyl)[5-(4-methoxyphenyl)-1h-pyrrolo[2,3-b]pyridin-3-yl]methanoneHuman7054
BRAFRAFTKL5jsmAA-Human7056
BRAFRAFTKL5jsmAB-Human7058
BRAFRAFTKL5jsmBAn,n'-{ethane-1,2-diylbis[oxyethane-2,1-diyloxy-4,1-phenylene-1h-pyrrolo[2,3-b]pyridine-5,3-diylcarbonyl(2,4-difluoro-3,1-phenylene)]}di(propane-1-sulfonamide)Human7060
BRAFRAFTKL5jsmBBn,n'-{ethane-1,2-diylbis[oxyethane-2,1-diyloxy-4,1-phenylene-1h-pyrrolo[2,3-b]pyridine-5,3-diylcarbonyl(2,4-difluoro-3,1-phenylene)]}di(propane-1-sulfonamide)Human7062
BRAFRAFTKL5jsmCAn,n'-{ethane-1,2-diylbis[oxyethane-2,1-diyloxy-4,1-phenylene-1h-pyrrolo[2,3-b]pyridine-5,3-diylcarbonyl(2,4-difluoro-3,1-phenylene)]}di(propane-1-sulfonamide)Human7059
BRAFRAFTKL5jsmCBn,n'-{ethane-1,2-diylbis[oxyethane-2,1-diyloxy-4,1-phenylene-1h-pyrrolo[2,3-b]pyridine-5,3-diylcarbonyl(2,4-difluoro-3,1-phenylene)]}di(propane-1-sulfonamide)Human7063
BRAFRAFTKL5jsmDA-Human7055
BRAFRAFTKL5jsmDB-Human7053
BRAFRAFTKL5jt2A2,2'-oxybis[n-({4-[3-(3-{[dihydroxy(propyl)-lambda~4~-sulfanyl]amino}-2,6-difluorobenzene-1-carbonyl)-1h-pyrrolo[2,3-b]pyridin-5-yl]phenyl}methyl)acetamide]Human7065
BRAFRAFTKL5jt2B-Human7057
BRAFRAFTKL5jt2C2,2'-oxybis[n-({4-[3-(3-{[dihydroxy(propyl)-lambda~4~-sulfanyl]amino}-2,6-difluorobenzene-1-carbonyl)-1h-pyrrolo[2,3-b]pyridin-5-yl]phenyl}methyl)acetamide]Human7064
BRAFRAFTKL5jt2D-Human7066
BRAFRAFTKL5valAn-(3-tert-butylphenyl)-4-methyl-3-[6-(morpholin-4-yl)pyrimidin-4-yl]benzamideHuman8190
BRAFRAFTKL5valBn-(3-tert-butylphenyl)-4-methyl-3-[6-(morpholin-4-yl)pyrimidin-4-yl]benzamideHuman8188
BRAFRAFTKL5vamAAn-{2-methyl-5'-(morpholin-4-yl)-6'-[(oxan-4-yl)oxy][3,3'-bipyridin]-5-yl}-3-(trifluoromethyl)benzamideHuman8185
BRAFRAFTKL5vamABn-{2-methyl-5'-(morpholin-4-yl)-6'-[(oxan-4-yl)oxy][3,3'-bipyridin]-5-yl}-3-(trifluoromethyl)benzamideHuman8189
BRAFRAFTKL5vamBAn-{2-methyl-5'-(morpholin-4-yl)-6'-[(oxan-4-yl)oxy][3,3'-bipyridin]-5-yl}-3-(trifluoromethyl)benzamideHuman8186
BRAFRAFTKL5vamBBn-{2-methyl-5'-(morpholin-4-yl)-6'-[(oxan-4-yl)oxy][3,3'-bipyridin]-5-yl}-3-(trifluoromethyl)benzamideHuman8187
BRAFRAFTKL6b8uA~{n}-[3-(2-acetamidoimidazo[1,2-a]pyridin-6-yl)-4-methyl-phenyl]-3-(trifluoromethyl)benzamideHuman8679
BRAFRAFTKL6b8uB~{n}-[3-(2-acetamidoimidazo[1,2-a]pyridin-6-yl)-4-methyl-phenyl]-3-(trifluoromethyl)benzamideHuman8678
BRAFRAFTKL6cadA1-(propan-2-yl)-3-({3-[3-(trifluoromethyl)phenyl]isoquinolin-8-yl}ethynyl)-1h-pyrazolo[3,4-d]pyrimidin-4-amineHuman9576
BRAFRAFTKL6cadB1-(propan-2-yl)-3-({3-[3-(trifluoromethyl)phenyl]isoquinolin-8-yl}ethynyl)-1h-pyrazolo[3,4-d]pyrimidin-4-amineHuman9575
BRAFRAFTKL6n0pAAn-{3-[2-(2-hydroxyethoxy)-6-(morpholin-4-yl)pyridin-4-yl]-4-methylphenyl}-2-(trifluoromethyl)pyridine-4-carboxamideHuman11597
BRAFRAFTKL6n0pABn-{3-[2-(2-hydroxyethoxy)-6-(morpholin-4-yl)pyridin-4-yl]-4-methylphenyl}-2-(trifluoromethyl)pyridine-4-carboxamideHuman11596
BRAFRAFTKL6n0pBAn-{3-[2-(2-hydroxyethoxy)-6-(morpholin-4-yl)pyridin-4-yl]-4-methylphenyl}-2-(trifluoromethyl)pyridine-4-carboxamideHuman11594
BRAFRAFTKL6n0pBBn-{3-[2-(2-hydroxyethoxy)-6-(morpholin-4-yl)pyridin-4-yl]-4-methylphenyl}-2-(trifluoromethyl)pyridine-4-carboxamideHuman11595
BRAFRAFTKL6n0qAAn-[4-methyl-3-(1-methyl-2-oxo-2,3-dihydro-1h-benzimidazol-5-yl)phenyl]-3-(trifluoromethyl)benzamideHuman11771
BRAFRAFTKL6n0qABn-[4-methyl-3-(1-methyl-2-oxo-2,3-dihydro-1h-benzimidazol-5-yl)phenyl]-3-(trifluoromethyl)benzamideHuman11768
BRAFRAFTKL6n0qBAn-[4-methyl-3-(1-methyl-2-oxo-2,3-dihydro-1h-benzimidazol-5-yl)phenyl]-3-(trifluoromethyl)benzamideHuman11770
BRAFRAFTKL6n0qBBn-[4-methyl-3-(1-methyl-2-oxo-2,3-dihydro-1h-benzimidazol-5-yl)phenyl]-3-(trifluoromethyl)benzamideHuman11769
BRAFRAFTKL6nsqA5-[(4-amino-1-ethyl-1h-pyrazolo[3,4-d]pyrimidin-3-yl)ethynyl]-n-(4-chlorophenyl)-6-methylisoquinolin-1-amineHuman11328
BRAFRAFTKL6nsqB5-[(4-amino-1-ethyl-1h-pyrazolo[3,4-d]pyrimidin-3-yl)ethynyl]-n-(4-chlorophenyl)-6-methylisoquinolin-1-amineHuman11329
BRAFRAFTKL6nybAphosphothiophosphoric acid-adenylate esterHuman11708
BRAFRAFTKL6p3dA3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHuman12809
BRAFRAFTKL6p7gA3-[(imidazo[1,2-b]pyridazin-3-yl)ethynyl]-4-methyl-n-[4-({[2-(morpholin-4-yl)ethyl]amino}methyl)-3-(trifluoromethyl)phenyl]benzamideHuman12810
BRAFRAFTKL6p7gB3-[(imidazo[1,2-b]pyridazin-3-yl)ethynyl]-4-methyl-n-[4-({[2-(morpholin-4-yl)ethyl]amino}methyl)-3-(trifluoromethyl)phenyl]benzamideHuman12806
BRAFRAFTKL6p7gC3-[(imidazo[1,2-b]pyridazin-3-yl)ethynyl]-4-methyl-n-[4-({[2-(morpholin-4-yl)ethyl]amino}methyl)-3-(trifluoromethyl)phenyl]benzamideHuman12807
BRAFRAFTKL6p7gD3-[(imidazo[1,2-b]pyridazin-3-yl)ethynyl]-4-methyl-n-[4-({[2-(morpholin-4-yl)ethyl]amino}methyl)-3-(trifluoromethyl)phenyl]benzamideHuman12808
BRAFRAFTKL6pp9AAphosphoaminophosphonic acid-adenylate esterHuman11711
BRAFRAFTKL6pp9ABphosphoaminophosphonic acid-adenylate esterHuman11709
BRAFRAFTKL6q0jAA-Human11704
BRAFRAFTKL6q0jAB-Human11701
BRAFRAFTKL6q0jBA-Human11703
BRAFRAFTKL6q0jBB-Human11712
BRAFRAFTKL6q0kA-Human11706
BRAFRAFTKL6q0kB-Human11710
BRAFRAFTKL6q0tAA-Human11705
BRAFRAFTKL6q0tAB-Human11707
BRAFRAFTKL6q0tBA-Human11702
BRAFRAFTKL6q0tBB-Human11700
BRAFRAFTKL6u2gBphosphomethylphosphonic acid adenylate esterHuman11567
BRAFRAFTKL6u2hCA2-{4-[(1e)-1-(hydroxyimino)-2,3-dihydro-1h-inden-5-yl]-3-(pyridin-4-yl)-1h-pyrazol-1-yl}ethanolHuman11568
BRAFRAFTKL6u2hDA2-{4-[(1e)-1-(hydroxyimino)-2,3-dihydro-1h-inden-5-yl]-3-(pyridin-4-yl)-1h-pyrazol-1-yl}ethanolHuman11569
BRAFRAFTKL6uanB-Human11641
BRAFRAFTKL6uanC-Human11642
BRAFRAFTKL6uuoA1-[4-{[1-(3-{[dihydroxy(propyl)-lambda~4~-sulfanyl]amino}-2,6-difluorophenyl)-3-(pyrimidin-5-yl)-1h-pyrrolo[3,2-b]pyridin-5-yl](methyl)amino}pyridin-1(4h)-yl]ethan-1-oneHuman12347
BRAFRAFTKL6uuoB1-[4-{[1-(3-{[dihydroxy(propyl)-lambda~4~-sulfanyl]amino}-2,6-difluorophenyl)-3-(pyrimidin-5-yl)-1h-pyrrolo[3,2-b]pyridin-5-yl](methyl)amino}pyridin-1(4h)-yl]ethan-1-oneHuman12346
Brsk2 (BRSK2)CAMKLCAMK4ynzA-Mouse6293
Brsk2 (BRSK2)CAMKLCAMK4ynzB-Mouse6291
Brsk2 (BRSK2)CAMKLCAMK4yomB-Mouse6292
Btk (BTK)TecTK4xi2A-Mouse5815
Btk (BTK)TecTK6mnyAA5-amino-1-[(3r)-1-cyanopiperidin-3-yl]-3-[4-(2,4-difluorophenoxy)phenyl]-1h-pyrazole-4-carboxamideMouse11307
Btk (BTK)TecTK6mnyAB5-amino-1-[(3r)-1-cyanopiperidin-3-yl]-3-[4-(2,4-difluorophenoxy)phenyl]-1h-pyrazole-4-carboxamideMouse11308
Btk (BTK)TecTK6mnyBA-Mouse11306
Btk (BTK)TecTK6mnyBB-Mouse11309
BTKTecTK1k2pA-Human2918
BTKTecTK1k2pB-Human2919
BTKTecTK3genAA4-amino-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-7-yl-cyclopentaneHuman2928
BTKTecTK3genAB4-amino-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-7-yl-cyclopentaneHuman2900
BTKTecTK3k54AAn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman2932
BTKTecTK3k54ABn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman2906
BTKTecTK3ocsA4-tert-butyl-n-[2-methyl-3-(4-methyl-6-{[4-(morpholin-4-ylcarbonyl)phenyl]amino}-5-oxo-4,5-dihydropyrazin-2-yl)phenyl]benzamideHuman2907
BTKTecTK3octAAn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman2899
BTKTecTK3octABn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman2908
BTKTecTK3p08A-Human2905
BTKTecTK3p08B-Human2894
BTKTecTK3pixA7-(4-methylpiperazin-1-yl)-4-[(5-methyl-1h-pyrazol-3-yl)amino]-2-(propan-2-yl)phthalazin-1(2h)-oneHuman2927
BTKTecTK3piyA6-({5-fluoro-2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}amino)-2,2-dimethyl-2h-pyrido[3,2-b][1,4]oxazin-3(4h)-oneHuman2909
BTKTecTK3pizA[5-amino-1-(2-methylphenyl)-1h-pyrazol-4-yl]{3-[1-(methylsulfonyl)piperidin-4-yl]phenyl}methanoneHuman2922
BTKTecTK3pj1A3-(2,6-dichlorophenyl)-7-({4-[2-(diethylamino)ethoxy]phenyl}amino)-1-methyl-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman2904
BTKTecTK3pj2A2-({4-[2-(diethylamino)ethoxy]phenyl}amino)-6-(4-fluorophenoxy)-8-methylpyrido[2,3-d]pyrimidin-7(8h)-oneHuman2911
BTKTecTK3pj3A2-methyl-n-(2-phenyl-3h-imidazo[4,5-b]pyridin-6-yl)-5-{[(2e)-3-phenylprop-2-enoyl]amino}benzamideHuman2910
BTKTecTK4nwmAA4-tert-butyl-n-[2-methyl-3-(6-{[4-(morpholin-4-ylcarbonyl)phenyl]amino}-7h-purin-2-yl)phenyl]benzamideHuman2930
BTKTecTK4nwmAB4-tert-butyl-n-[2-methyl-3-(6-{[4-(morpholin-4-ylcarbonyl)phenyl]amino}-7h-purin-2-yl)phenyl]benzamideHuman2917
BTKTecTK4nwmBA4-tert-butyl-n-[2-methyl-3-(6-{[4-(morpholin-4-ylcarbonyl)phenyl]amino}-7h-purin-2-yl)phenyl]benzamideHuman2898
BTKTecTK4nwmBB4-tert-butyl-n-[2-methyl-3-(6-{[4-(morpholin-4-ylcarbonyl)phenyl]amino}-7h-purin-2-yl)phenyl]benzamideHuman2903
BTKTecTK4ot5A4-tert-butyl-n-{3-[8-({4-[(4-methylpiperazin-1-yl)carbonyl]phenyl}amino)imidazo[1,2-a]pyrazin-6-yl]phenyl}benzamideHuman2913
BTKTecTK4ot6A4-(methylsulfonyl)-n-[3-(8-{[4-(morpholin-4-ylcarbonyl)phenyl]amino}imidazo[1,2-a]pyrazin-6-yl)phenyl]benzamideHuman2931
BTKTecTK4otfAAn-{3-[6-({4-[(2r)-1,4-dimethyl-3-oxopiperazin-2-yl]phenyl}amino)-4-methyl-5-oxo-4,5-dihydropyrazin-2-yl]-2-methylphenyl}-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamideHuman2901
BTKTecTK4otfABn-{3-[6-({4-[(2r)-1,4-dimethyl-3-oxopiperazin-2-yl]phenyl}amino)-4-methyl-5-oxo-4,5-dihydropyrazin-2-yl]-2-methylphenyl}-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamideHuman2921
BTKTecTK4otqA1-{5-[3-(7-tert-butyl-4-oxoquinazolin-3(4h)-yl)-2-methylphenyl]-1-methyl-2-oxo-1,2-dihydropyridin-3-yl}-3-methylureaHuman2895
BTKTecTK4otrA6-cyclopropyl-2-[3-(5-{[5-(4-ethylpiperazin-1-yl)pyridin-2-yl]amino}-1-methyl-6-oxo-1,6-dihydropyridin-3-yl)-2-(hydroxymethyl)phenyl]-8-fluoroisoquinolin-1(2h)-oneHuman2896
BTKTecTK4rfyAA6-(dimethylamino)-2-[2-(hydroxymethyl)-3-(1-methyl-5-{[5-(morpholin-4-ylcarbonyl)pyridin-2-yl]amino}-6-oxo-1,6-dihydropyridin-3-yl)phenyl]-3,4-dihydroisoquinolin-1(2h)-oneHuman2935
BTKTecTK4rfyAB6-(dimethylamino)-2-[2-(hydroxymethyl)-3-(1-methyl-5-{[5-(morpholin-4-ylcarbonyl)pyridin-2-yl]amino}-6-oxo-1,6-dihydropyridin-3-yl)phenyl]-3,4-dihydroisoquinolin-1(2h)-oneHuman2933
BTKTecTK4rfzA6-(dimethylamino)-8-fluoro-2-[2-(hydroxymethyl)-3-(1-methyl-5-{[5-(morpholin-4-ylcarbonyl)pyridin-2-yl]amino}-6-oxo-1,6-dihydropyridin-3-yl)phenyl]isoquinolin-1(2h)-oneHuman2925
BTKTecTK4rg0A2-{8-fluoro-2-[2-(hydroxymethyl)-3-(1-methyl-5-{[5-(4-methylpiperazin-1-yl)pyridin-2-yl]amino}-6-oxo-1,6-dihydropyridin-3-yl)phenyl]-1-oxo-1,2,3,4-tetrahydroisoquinolin-6-yl}-2-methylpropanenitrileHuman2929
BTKTecTK4rx5AAn-(6-fluoro-2-methyl-3-{5-[(5-methyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl)amino]-6-oxo-1,6-dihydropyridazin-3-yl}phenyl)-1-benzothiophene-2-carboxamideHuman6259
BTKTecTK4rx5ABn-(6-fluoro-2-methyl-3-{5-[(5-methyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl)amino]-6-oxo-1,6-dihydropyridazin-3-yl}phenyl)-1-benzothiophene-2-carboxamideHuman6258
BTKTecTK4yhfAA(2s)-2-({(3r)-3-[4-amino-3-(4-phenoxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl}carbonyl)-4,4-dimethylpentanenitrileHuman2916
BTKTecTK4yhfAB(2s)-2-({(3r)-3-[4-amino-3-(4-phenoxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl}carbonyl)-4,4-dimethylpentanenitrileHuman2902
BTKTecTK4yhfBA(2s)-2-({(3r)-3-[4-amino-3-(4-phenoxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl}carbonyl)-4,4-dimethylpentanenitrileHuman2897
BTKTecTK4yhfBB(2s)-2-({(3r)-3-[4-amino-3-(4-phenoxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl}carbonyl)-4,4-dimethylpentanenitrileHuman2912
BTKTecTK4z3vAA4-amino-8-(5-methyl-1h-indazol-6-yl)cinnoline-3-carboxamideHuman2934
BTKTecTK4z3vAB4-amino-8-(5-methyl-1h-indazol-6-yl)cinnoline-3-carboxamideHuman2914
BTKTecTK4zlyAA4-aminocinnoline-3-carboxamideHuman2926
BTKTecTK4zlyAB4-aminocinnoline-3-carboxamideHuman2920
BTKTecTK4zlyAC4-aminocinnoline-3-carboxamideHuman2915
BTKTecTK4zlzAA4-amino-8-(4-methylpyridin-3-yl)cinnoline-3-carboxamideHuman2923
BTKTecTK4zlzAB4-amino-8-(4-methylpyridin-3-yl)cinnoline-3-carboxamideHuman2924
BTKTecTK5bpyA6-{(3r)-3-[(4-tert-butylbenzoyl)amino]piperidin-1-yl}-2-{[4-(morpholin-4-ylcarbonyl)phenyl]amino}pyridine-3-carboxamideHuman6095
BTKTecTK5bpyB6-{(3r)-3-[(4-tert-butylbenzoyl)amino]piperidin-1-yl}-2-{[4-(morpholin-4-ylcarbonyl)phenyl]amino}pyridine-3-carboxamideHuman6094
BTKTecTK5bq0AA4-(2-chlorophenyl)-7-[(4-methylpiperazin-1-yl)carbonyl]-9h-carbazole-1-carboxamideHuman6871
BTKTecTK5bq0AB4-(2-chlorophenyl)-7-[(4-methylpiperazin-1-yl)carbonyl]-9h-carbazole-1-carboxamideHuman6872
BTKTecTK5fbnCA4-[8-azanyl-3-[(3~{r})-1-(3-methyloxetan-3-yl)carbonylpiperidin-3-yl]imidazo[1,5-a]pyrazin-1-yl]-~{n}-[4-(trifluoromethyl)pyridin-2-yl]benzamideHuman6381
BTKTecTK5fbnCB4-[8-azanyl-3-[(3~{r})-1-(3-methyloxetan-3-yl)carbonylpiperidin-3-yl]imidazo[1,5-a]pyrazin-1-yl]-~{n}-[4-(trifluoromethyl)pyridin-2-yl]benzamideHuman6382
BTKTecTK5fbnDA4-[8-azanyl-3-[(3~{r})-1-(3-methyloxetan-3-yl)carbonylpiperidin-3-yl]imidazo[1,5-a]pyrazin-1-yl]-~{n}-[4-(trifluoromethyl)pyridin-2-yl]benzamideHuman6384
BTKTecTK5fbnDB4-[8-azanyl-3-[(3~{r})-1-(3-methyloxetan-3-yl)carbonylpiperidin-3-yl]imidazo[1,5-a]pyrazin-1-yl]-~{n}-[4-(trifluoromethyl)pyridin-2-yl]benzamideHuman6383
BTKTecTK5fboAA4-[8-azanyl-3-[(3~{r},6~{s})-1-cyclopropylcarbonyl-6-methyl-piperidin-3-yl]imidazo[1,5-a]pyrazin-1-yl]-3-fluoranyl-~{n}-[4-(trifluoromethyl)pyridin-2-yl]benzamideHuman6455
BTKTecTK5fboAB4-[8-azanyl-3-[(3~{r},6~{s})-1-cyclopropylcarbonyl-6-methyl-piperidin-3-yl]imidazo[1,5-a]pyrazin-1-yl]-3-fluoranyl-~{n}-[4-(trifluoromethyl)pyridin-2-yl]benzamideHuman6456
BTKTecTK5j87AAn-[3-(5-{[3-(acryloylamino)-4-(morpholine-4-carbonyl)phenyl]amino}-1-methyl-6-oxo-1,6-dihydropyridin-3-yl)-2-methylphenyl]-4-tert-butylbenzamideHuman8002
BTKTecTK5j87ABn-[3-(5-{[3-(acryloylamino)-4-(morpholine-4-carbonyl)phenyl]amino}-1-methyl-6-oxo-1,6-dihydropyridin-3-yl)-2-methylphenyl]-4-tert-butylbenzamideHuman8003
BTKTecTK5j87BAn-[3-(5-{[3-(acryloylamino)-4-(morpholine-4-carbonyl)phenyl]amino}-1-methyl-6-oxo-1,6-dihydropyridin-3-yl)-2-methylphenyl]-4-tert-butylbenzamideHuman8005
BTKTecTK5j87BBn-[3-(5-{[3-(acryloylamino)-4-(morpholine-4-carbonyl)phenyl]amino}-1-methyl-6-oxo-1,6-dihydropyridin-3-yl)-2-methylphenyl]-4-tert-butylbenzamideHuman8007
BTKTecTK5j87CAn-[3-(5-{[3-(acryloylamino)-4-(morpholine-4-carbonyl)phenyl]amino}-1-methyl-6-oxo-1,6-dihydropyridin-3-yl)-2-methylphenyl]-4-tert-butylbenzamideHuman8004
BTKTecTK5j87CBn-[3-(5-{[3-(acryloylamino)-4-(morpholine-4-carbonyl)phenyl]amino}-1-methyl-6-oxo-1,6-dihydropyridin-3-yl)-2-methylphenyl]-4-tert-butylbenzamideHuman8006
BTKTecTK5j87DAn-[3-(5-{[3-(acryloylamino)-4-(morpholine-4-carbonyl)phenyl]amino}-1-methyl-6-oxo-1,6-dihydropyridin-3-yl)-2-methylphenyl]-4-tert-butylbenzamideHuman8008
BTKTecTK5j87DBn-[3-(5-{[3-(acryloylamino)-4-(morpholine-4-carbonyl)phenyl]amino}-1-methyl-6-oxo-1,6-dihydropyridin-3-yl)-2-methylphenyl]-4-tert-butylbenzamideHuman8001
BTKTecTK5jrsA4-[2-fluoro-3-(4-oxoquinazolin-3(4h)-yl)phenyl]-7-(2-hydroxypropan-2-yl)-9h-carbazole-1-carboxamideHuman7032
BTKTecTK5jrsB4-[2-fluoro-3-(4-oxoquinazolin-3(4h)-yl)phenyl]-7-(2-hydroxypropan-2-yl)-9h-carbazole-1-carboxamideHuman7033
BTKTecTK5kupAA6-~{tert}-butyl-8-fluoranyl-2-[3-(hydroxymethyl)-4-[1-methyl-6-oxidanylidene-5-(pyrimidin-4-ylamino)pyridin-3-yl]pyridin-2-yl]phthalazin-1-oneHuman7051
BTKTecTK5kupAB6-~{tert}-butyl-8-fluoranyl-2-[3-(hydroxymethyl)-4-[1-methyl-6-oxidanylidene-5-(pyrimidin-4-ylamino)pyridin-3-yl]pyridin-2-yl]phthalazin-1-oneHuman7052
BTKTecTK5p9fAAn-{3-[6-({4-[(2r)-1,4-dimethyl-3-oxopiperazin-2-yl]phenyl}amino)-4-methyl-5-oxo-4,5-dihydropyrazin-2-yl]-2-methylphenyl}-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamideHuman7632
BTKTecTK5p9fABn-{3-[6-({4-[(2r)-1,4-dimethyl-3-oxopiperazin-2-yl]phenyl}amino)-4-methyl-5-oxo-4,5-dihydropyrazin-2-yl]-2-methylphenyl}-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamideHuman7629
BTKTecTK5p9gAA6-cyclopropyl-8-fluoranyl-2-[2-(hydroxymethyl)-3-[1-methyl-5-[[5-(4-methylpiperazin-1-yl)pyridin-2-yl]amino]-6-oxidanylidene-pyridin-3-yl]phenyl]isoquinolin-1-oneHuman7635
BTKTecTK5p9gAB6-cyclopropyl-8-fluoranyl-2-[2-(hydroxymethyl)-3-[1-methyl-5-[[5-(4-methylpiperazin-1-yl)pyridin-2-yl]amino]-6-oxidanylidene-pyridin-3-yl]phenyl]isoquinolin-1-oneHuman7644
BTKTecTK5p9hAA6-~{tert}-butyl-8-fluoranyl-2-[3-(hydroxymethyl)-4-[1-methyl-5-[[5-(1-methylpiperidin-4-yl)pyridin-2-yl]amino]-6-oxidanylidene-pyridazin-3-yl]pyridin-2-yl]phthalazin-1-oneHuman7631
BTKTecTK5p9hAB6-~{tert}-butyl-8-fluoranyl-2-[3-(hydroxymethyl)-4-[1-methyl-5-[[5-(1-methylpiperidin-4-yl)pyridin-2-yl]amino]-6-oxidanylidene-pyridazin-3-yl]pyridin-2-yl]phthalazin-1-oneHuman7643
BTKTecTK5p9iAA1-{(3r)-3-[4-amino-3-(4-phenoxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl}prop-2-en-1-oneHuman7627
BTKTecTK5p9iAB1-{(3r)-3-[4-amino-3-(4-phenoxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl}prop-2-en-1-oneHuman7642
BTKTecTK5p9iAC1-{(3r)-3-[4-amino-3-(4-phenoxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl}prop-2-en-1-oneHuman7638
BTKTecTK5p9jAA1-[(3~{r})-3-[4-azanyl-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-oneHuman7637
BTKTecTK5p9jAB1-[(3~{r})-3-[4-azanyl-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-oneHuman7628
BTKTecTK5p9jAC1-[(3~{r})-3-[4-azanyl-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-oneHuman7640
BTKTecTK5p9kAA4-[4-[[5-fluoranyl-4-[[3-(propanoylamino)phenyl]amino]pyrimidin-2-yl]amino]phenoxy]-~{n}-methyl-pyridine-2-carboxamideHuman7633
BTKTecTK5p9kAB4-[4-[[5-fluoranyl-4-[[3-(propanoylamino)phenyl]amino]pyrimidin-2-yl]amino]phenoxy]-~{n}-methyl-pyridine-2-carboxamideHuman7636
BTKTecTK5p9kAC4-[4-[[5-fluoranyl-4-[[3-(propanoylamino)phenyl]amino]pyrimidin-2-yl]amino]phenoxy]-~{n}-methyl-pyridine-2-carboxamideHuman7626
BTKTecTK5p9lAA~{n}-[3-[[5-fluoranyl-2-[[4-(2-methoxyethoxy)phenyl]amino]pyrimidin-4-yl]amino]phenyl]propanamideHuman7625
BTKTecTK5p9lAB~{n}-[3-[[5-fluoranyl-2-[[4-(2-methoxyethoxy)phenyl]amino]pyrimidin-4-yl]amino]phenyl]propanamideHuman7630
BTKTecTK5p9mAA6-azanyl-9-[(3~{r})-1-[(~{e})-but-2-enoyl]pyrrolidin-3-yl]-7-(4-phenoxyphenyl)purin-8-oneHuman7634
BTKTecTK5p9mAB6-azanyl-9-[(3~{r})-1-[(~{e})-but-2-enoyl]pyrrolidin-3-yl]-7-(4-phenoxyphenyl)purin-8-oneHuman7639
BTKTecTK5p9mAC6-azanyl-9-[(3~{r})-1-[(~{e})-but-2-enoyl]pyrrolidin-3-yl]-7-(4-phenoxyphenyl)purin-8-oneHuman7641
BTKTecTK5t18AA6-fluoro-5-(r)-(3-(s)-(8-fluoro-1-methyl-2,4-dioxo-1,2-dihydroquinazolin-3(4h)-yl)-2-methylphenyl)-2-(s)-(2-hydroxypropan-2-yl)-2,3,4,9-tetrahydro-1h-carbazole-8-carboxamideHuman7508
BTKTecTK5t18AB6-fluoro-5-(r)-(3-(s)-(8-fluoro-1-methyl-2,4-dioxo-1,2-dihydroquinazolin-3(4h)-yl)-2-methylphenyl)-2-(s)-(2-hydroxypropan-2-yl)-2,3,4,9-tetrahydro-1h-carbazole-8-carboxamideHuman7507
BTKTecTK5u9dAA(r)-n-methyl-2-(3-((quinoxalin-6-ylamino)methyl)furan-2-carbonyl)-2,3,4,9-tetrahydro-1h-pyrido[3,4-b]indole-3-carboxamideHuman7393
BTKTecTK5u9dAB(r)-n-methyl-2-(3-((quinoxalin-6-ylamino)methyl)furan-2-carbonyl)-2,3,4,9-tetrahydro-1h-pyrido[3,4-b]indole-3-carboxamideHuman7392
BTKTecTK5vfiAA2-[3'-(hydroxymethyl)-1-methyl-5-({5-[(2s)-2-methyl-4-(oxetan-3-yl)piperazin-1-yl]pyridin-2-yl}amino)-6-oxo[1,6-dihydro[3,4'-bipyridine]]-2'-yl]-7,7-dimethyl-3,4,7,8-tetrahydro-2h-cyclopenta[4,5]pyrrolo[1,2-a]pyrazin-1(6h)-oneHuman9602
BTKTecTK5vfiAB2-[3'-(hydroxymethyl)-1-methyl-5-({5-[(2s)-2-methyl-4-(oxetan-3-yl)piperazin-1-yl]pyridin-2-yl}amino)-6-oxo[1,6-dihydro[3,4'-bipyridine]]-2'-yl]-7,7-dimethyl-3,4,7,8-tetrahydro-2h-cyclopenta[4,5]pyrrolo[1,2-a]pyrazin-1(6h)-oneHuman9601
BTKTecTK5vgoAA2-(2-methoxyethoxy)ethanolHuman8218
BTKTecTK5vgoAB2-(2-methoxyethoxy)ethanolHuman8219
BTKTecTK5xyzAAn-[3-(5-{[(2-chloro-6-fluorophenyl)methyl]amino}-1h-1,2,4-triazol-3-yl)phenyl]propanamideHuman9929
BTKTecTK5xyzABn-[3-(5-{[(2-chloro-6-fluorophenyl)methyl]amino}-1h-1,2,4-triazol-3-yl)phenyl]propanamideHuman9932
BTKTecTK5xyzBAn-[3-(5-{[(2-chloro-6-fluorophenyl)methyl]amino}-1h-1,2,4-triazol-3-yl)phenyl]propanamideHuman9931
BTKTecTK5xyzBBn-[3-(5-{[(2-chloro-6-fluorophenyl)methyl]amino}-1h-1,2,4-triazol-3-yl)phenyl]propanamideHuman9930
BTKTecTK5zz4An-[3-(4-amino-6-{[4-(morpholine-4-carbonyl)phenyl]amino}-1,3,5-triazin-2-yl)-2-methylphenyl]-4-tert-butylbenzamideHuman10479
BTKTecTK5zz4Bn-[3-(4-amino-6-{[4-(morpholine-4-carbonyl)phenyl]amino}-1,3,5-triazin-2-yl)-2-methylphenyl]-4-tert-butylbenzamideHuman10468
BTKTecTK5zz4Cn-[3-(4-amino-6-{[4-(morpholine-4-carbonyl)phenyl]amino}-1,3,5-triazin-2-yl)-2-methylphenyl]-4-tert-butylbenzamideHuman10464
BTKTecTK5zz4Dn-[3-(4-amino-6-{[4-(morpholine-4-carbonyl)phenyl]amino}-1,3,5-triazin-2-yl)-2-methylphenyl]-4-tert-butylbenzamideHuman10478
BTKTecTK5zz4En-[3-(4-amino-6-{[4-(morpholine-4-carbonyl)phenyl]amino}-1,3,5-triazin-2-yl)-2-methylphenyl]-4-tert-butylbenzamideHuman10470
BTKTecTK5zz4Fn-[3-(4-amino-6-{[4-(morpholine-4-carbonyl)phenyl]amino}-1,3,5-triazin-2-yl)-2-methylphenyl]-4-tert-butylbenzamideHuman10469
BTKTecTK6auaAAn-{3-[(2r)-6-{[3-amino-4-(morpholine-4-carbonyl)phenyl]amino}-5-oxo-2,5-dihydropyrazin-2-yl]-2-methylphenyl}-4-(piperidin-1-yl)benzamideHuman10472
BTKTecTK6auaABn-{3-[(2r)-6-{[3-amino-4-(morpholine-4-carbonyl)phenyl]amino}-5-oxo-2,5-dihydropyrazin-2-yl]-2-methylphenyl}-4-(piperidin-1-yl)benzamideHuman10473
BTKTecTK6aubAA4-tert-butyl-n-[2-methyl-3-(1-methyl-5-{[5-(morpholine-4-carbonyl)pyridin-2-yl]amino}-6-oxo-1,6-dihydropyridin-3-yl)phenyl]benzamideHuman10466
BTKTecTK6aubAB4-tert-butyl-n-[2-methyl-3-(1-methyl-5-{[5-(morpholine-4-carbonyl)pyridin-2-yl]amino}-6-oxo-1,6-dihydropyridin-3-yl)phenyl]benzamideHuman10475
BTKTecTK6bikAA4-tert-butyl-n-[2-(hydroxymethyl)-3-(1-methyl-5-{[5-(morpholine-4-carbonyl)pyridin-2-yl]amino}-6-oxo-1,6-dihydropyridazin-3-yl)phenyl]benzamideHuman10680
BTKTecTK6bikAB4-tert-butyl-n-[2-(hydroxymethyl)-3-(1-methyl-5-{[5-(morpholine-4-carbonyl)pyridin-2-yl]amino}-6-oxo-1,6-dihydropyridazin-3-yl)phenyl]benzamideHuman10678
BTKTecTK6bkeAAn-[2-(2-hydroxyethyl)-3-{5-[(5-methyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl)amino]-6-oxo-1,6-dihydropyridazin-3-yl}phenyl]-1-benzothiophene-2-carboxamideHuman10681
BTKTecTK6bkeABn-[2-(2-hydroxyethyl)-3-{5-[(5-methyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl)amino]-6-oxo-1,6-dihydropyridazin-3-yl}phenyl]-1-benzothiophene-2-carboxamideHuman10683
BTKTecTK6bkhAAn-[2-(hydroxymethyl)-3-{5-[(5-methyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl)amino]-6-oxo-1,6-dihydropyridazin-3-yl}phenyl]-1-benzothiophene-2-carboxamideHuman10682
BTKTecTK6bkhABn-[2-(hydroxymethyl)-3-{5-[(5-methyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl)amino]-6-oxo-1,6-dihydropyridazin-3-yl}phenyl]-1-benzothiophene-2-carboxamideHuman10677
BTKTecTK6bkwAAn-(3-{5-[(1,5-dimethyl-1h-pyrazol-3-yl)amino]-1-methyl-6-oxo-1,6-dihydropyridazin-3-yl}-2,6-difluorophenyl)-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamideHuman10686
BTKTecTK6bkwABn-(3-{5-[(1,5-dimethyl-1h-pyrazol-3-yl)amino]-1-methyl-6-oxo-1,6-dihydropyridazin-3-yl}-2,6-difluorophenyl)-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamideHuman10679
BTKTecTK6blnAAn-(3-{5-[(1,5-dimethyl-1h-pyrazol-3-yl)amino]-6-oxo-1,6-dihydropyridazin-3-yl}-2,6-difluorophenyl)-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamideHuman10685
BTKTecTK6blnABn-(3-{5-[(1,5-dimethyl-1h-pyrazol-3-yl)amino]-6-oxo-1,6-dihydropyridazin-3-yl}-2,6-difluorophenyl)-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamideHuman10684
BTKTecTK6di0AA6-(cyclohexylamino)pyridine-3-carboxamideHuman10629
BTKTecTK6di0AB6-(cyclohexylamino)pyridine-3-carboxamideHuman10626
BTKTecTK6di0AC6-(cyclohexylamino)pyridine-3-carboxamideHuman10628
BTKTecTK6di1AA4-amino-2-[(3s)-3-(propanoylamino)pyrrolidin-1-yl]pyrimidine-5-carboxamideHuman10630
BTKTecTK6di1AB4-amino-2-[(3s)-3-(propanoylamino)pyrrolidin-1-yl]pyrimidine-5-carboxamideHuman10627
BTKTecTK6di3A6-[(3s)-3-(acryloylamino)pyrrolidin-1-yl]-2-(4-phenoxyphenoxy)pyridine-3-carboxamideHuman10474
BTKTecTK6di5AA2-(4-phenoxyphenoxy)-6-[(1s,4s)-5-propanoyl-2,5-diazabicyclo[2.2.1]heptan-2-yl]pyridine-3-carboxamideHuman10471
BTKTecTK6di5AB2-(4-phenoxyphenoxy)-6-[(1s,4s)-5-propanoyl-2,5-diazabicyclo[2.2.1]heptan-2-yl]pyridine-3-carboxamideHuman10481
BTKTecTK6di9AA6-[(3s)-3-(acryloylamino)pyrrolidin-1-yl]-2-{[4-(tert-butylcarbamoyl)phenyl]amino}pyridine-3-carboxamideHuman10465
BTKTecTK6di9AB6-[(3s)-3-(acryloylamino)pyrrolidin-1-yl]-2-{[4-(tert-butylcarbamoyl)phenyl]amino}pyridine-3-carboxamideHuman10476
BTKTecTK6e4fAA1,5-anhydro-2-{[5-(2-chloro-4-phenoxybenzene-1-carbonyl)-7h-pyrrolo[2,3-d]pyrimidin-4-yl]amino}-2,3,4-trideoxy-d-erythro-hexitolHuman10477
BTKTecTK6e4fAB1,5-anhydro-2-{[5-(2-chloro-4-phenoxybenzene-1-carbonyl)-7h-pyrrolo[2,3-d]pyrimidin-4-yl]amino}-2,3,4-trideoxy-d-erythro-hexitolHuman10480
BTKTecTK6ep9An-[2-methyl-3-[4-methyl-6-[4-(4-methylpiperazine-1-carbonyl)anilino]-5-oxo-pyrazin-2-yl]phenyl]-4-(1-piperidyl)benzamideHuman10467
BTKTecTK6hrpA6-~{tert}-butyl-8-fluoranyl-2-[2-(hydroxymethyl)-3-[1-methyl-5-[(5-morpholin-4-ylcarbonylpyridin-2-yl)amino]-6-oxidanylidene-pyridazin-3-yl]phenyl]phthalazin-1-oneHuman10971
BTKTecTK6hrtA(9~{s})-12-(6-~{tert}-butyl-8-fluoranyl-1-oxidanylidene-phthalazin-2-yl)-6-methyl-4-[(5-morpholin-4-ylcarbonylpyridin-2-yl)amino]-9-oxidanyl-6-azatricyclo[9.4.0.0^{2,7}]pentadeca-1(15),2(7),3,11,13-pentaen-5-oneHuman10972
BTKTecTK6j6mAA(7s)-2-(4-phenoxyphenyl)-7-(1-propanoylpiperidin-4-yl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11767
BTKTecTK6j6mAB(7s)-2-(4-phenoxyphenyl)-7-(1-propanoylpiperidin-4-yl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11766
BTKTecTK6n9pAAn-(3-{[2-amino-3-(4-phenoxyphenyl)pyridin-4-yl]oxy}phenyl)propanamideHuman10886
BTKTecTK6n9pABn-(3-{[2-amino-3-(4-phenoxyphenyl)pyridin-4-yl]oxy}phenyl)propanamideHuman10887
BTKTecTK6n9pACn-(3-{[2-amino-3-(4-phenoxyphenyl)pyridin-4-yl]oxy}phenyl)propanamideHuman10888
BTKTecTK6nfhAA8-(2,3-dihydro-1h-inden-5-yl)-2-({4-[(2s)-3-(dimethylamino)-2-hydroxypropoxy]phenyl}amino)-5,8-dihydropteridine-6,7-dioneHuman10964
BTKTecTK6nfhAB8-(2,3-dihydro-1h-inden-5-yl)-2-({4-[(2s)-3-(dimethylamino)-2-hydroxypropoxy]phenyl}amino)-5,8-dihydropteridine-6,7-dioneHuman10965
BTKTecTK6nfiAAn-(3-{[(2,6-dimethylphenyl)methyl]amino}-7-methoxyindeno[1,2-c]pyrazol-6-yl)methanesulfonamideHuman10962
BTKTecTK6nfiABn-(3-{[(2,6-dimethylphenyl)methyl]amino}-7-methoxyindeno[1,2-c]pyrazol-6-yl)methanesulfonamideHuman10963
BTKTecTK6nzmAAn-[2-fluoro-6-(pyrrolidin-1-yl)phenyl]-n'-{3-[(2r)-1-(2-hydroxyethyl)-4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperazin-2-yl]phenyl}ureaHuman11144
BTKTecTK6nzmABn-[2-fluoro-6-(pyrrolidin-1-yl)phenyl]-n'-{3-[(2r)-1-(2-hydroxyethyl)-4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperazin-2-yl]phenyl}ureaHuman11143
BTKTecTK6nzmDAn-[2-fluoro-6-(pyrrolidin-1-yl)phenyl]-n'-{3-[(2r)-1-(2-hydroxyethyl)-4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperazin-2-yl]phenyl}ureaHuman11141
BTKTecTK6nzmDBn-[2-fluoro-6-(pyrrolidin-1-yl)phenyl]-n'-{3-[(2r)-1-(2-hydroxyethyl)-4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperazin-2-yl]phenyl}ureaHuman11142
BTKTecTK6o8iAA4-[(3s)-3-{[(2e)-but-2-enoyl]amino}piperidin-1-yl]-5-fluoro-2,3-dimethyl-1h-indole-7-carboxamideHuman11002
BTKTecTK6o8iAB4-[(3s)-3-{[(2e)-but-2-enoyl]amino}piperidin-1-yl]-5-fluoro-2,3-dimethyl-1h-indole-7-carboxamideHuman11001
BTKTecTK6omuAA1-[4-({[6-amino-5-(4-phenoxyphenyl)pyrimidin-4-yl]amino}methyl)piperidin-1-yl]prop-2-en-1-oneHuman11529
BTKTecTK6omuAB1-[4-({[6-amino-5-(4-phenoxyphenyl)pyrimidin-4-yl]amino}methyl)piperidin-1-yl]prop-2-en-1-oneHuman11530
BTKTecTK6omuAC-Human11528
BTKTecTK6s90A4-~{tert}-butyl-~{n}-[2-methyl-3-[6-[4-(4-methylpiperazin-1-yl)carbonylphenyl]-7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl]phenyl]benzamideHuman11636
BTKTecTK6s90B4-~{tert}-butyl-~{n}-[2-methyl-3-[6-[4-(4-methylpiperazin-1-yl)carbonylphenyl]-7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl]phenyl]benzamideHuman11635
BTKTecTK6tfpA~{n}-[3-[6-azanyl-5-[2-[methyl(propanoyl)amino]ethoxy]pyrimidin-4-yl]-5-fluoranyl-2-methyl-phenyl]-4-cyclopropyl-2-fluoranyl-benzamideHuman12024
BTKTecTK6tfpB~{n}-[3-[6-azanyl-5-[2-[methyl(propanoyl)amino]ethoxy]pyrimidin-4-yl]-5-fluoranyl-2-methyl-phenyl]-4-cyclopropyl-2-fluoranyl-benzamideHuman12020
BTKTecTK6tfpC~{n}-[3-[6-azanyl-5-[2-[methyl(propanoyl)amino]ethoxy]pyrimidin-4-yl]-5-fluoranyl-2-methyl-phenyl]-4-cyclopropyl-2-fluoranyl-benzamideHuman12023
BTKTecTK6tfpD~{n}-[3-[6-azanyl-5-[2-[methyl(propanoyl)amino]ethoxy]pyrimidin-4-yl]-5-fluoranyl-2-methyl-phenyl]-4-cyclopropyl-2-fluoranyl-benzamideHuman12021
BTKTecTK6tfpE~{n}-[3-[6-azanyl-5-[2-[methyl(propanoyl)amino]ethoxy]pyrimidin-4-yl]-5-fluoranyl-2-methyl-phenyl]-4-cyclopropyl-2-fluoranyl-benzamideHuman12022
BTKTecTK6x3nAA4-{8-amino-3-[(6r,8as)-3-oxohexahydro-3h-[1,3]oxazolo[3,4-a]pyridin-6-yl]imidazo[1,5-a]pyrazin-1-yl}-n-[4-(trifluoromethyl)pyridin-2-yl]benzamideHuman12514
BTKTecTK6x3nAB4-{8-amino-3-[(6r,8as)-3-oxohexahydro-3h-[1,3]oxazolo[3,4-a]pyridin-6-yl]imidazo[1,5-a]pyrazin-1-yl}-n-[4-(trifluoromethyl)pyridin-2-yl]benzamideHuman12510
BTKTecTK6x3oAA4-{8-amino-3-[(6r,8as)-3-oxo-3,5,6,7,8,8a-hexahydroindolizin-6-yl]imidazo[1,5-a]pyrazin-1-yl}-3-methoxy-n-[4-(trifluoromethyl)pyridin-2-yl]benzamideHuman12513
BTKTecTK6x3oAB4-{8-amino-3-[(6r,8as)-3-oxo-3,5,6,7,8,8a-hexahydroindolizin-6-yl]imidazo[1,5-a]pyrazin-1-yl}-3-methoxy-n-[4-(trifluoromethyl)pyridin-2-yl]benzamideHuman12512
BTKTecTK6x3oBA4-{8-amino-3-[(6r,8as)-3-oxo-3,5,6,7,8,8a-hexahydroindolizin-6-yl]imidazo[1,5-a]pyrazin-1-yl}-3-methoxy-n-[4-(trifluoromethyl)pyridin-2-yl]benzamideHuman12508
BTKTecTK6x3oBB4-{8-amino-3-[(6r,8as)-3-oxo-3,5,6,7,8,8a-hexahydroindolizin-6-yl]imidazo[1,5-a]pyrazin-1-yl}-3-methoxy-n-[4-(trifluoromethyl)pyridin-2-yl]benzamideHuman12511
BTKTecTK6x3pAA4-{8-amino-3-[(6r,8as)-3-oxooctahydroindolizin-6-yl]imidazo[1,5-a]pyrazin-1-yl}-3-(cyclopropyloxy)-n-[4-(trifluoromethyl)pyridin-2-yl]benzamideHuman12516
BTKTecTK6x3pAB4-{8-amino-3-[(6r,8as)-3-oxooctahydroindolizin-6-yl]imidazo[1,5-a]pyrazin-1-yl}-3-(cyclopropyloxy)-n-[4-(trifluoromethyl)pyridin-2-yl]benzamideHuman12517
BTKTecTK6xe4AA(1s,2s)-n-[2'-(6-tert-butyl-8-fluoro-1-oxophthalazin-2(1h)-yl)-3'-(hydroxymethyl)-1-methyl-6-oxo[1,6-dihydro[3,4'-bipyridine]]-5-yl]-2-fluorocyclopropane-1-carboxamideHuman12515
BTKTecTK6xe4AB(1s,2s)-n-[2'-(6-tert-butyl-8-fluoro-1-oxophthalazin-2(1h)-yl)-3'-(hydroxymethyl)-1-methyl-6-oxo[1,6-dihydro[3,4'-bipyridine]]-5-yl]-2-fluorocyclopropane-1-carboxamideHuman12509
BUB1BUBOther4qpmAadenosine-5'-diphosphateHuman1843
BUB1BUBOther4qpmBadenosine-5'-diphosphateHuman1844
BUB1BUBOther4r8qAadenosine-5'-diphosphateHuman1842
BUB1BUBOther5dmzAadenosine-5'-diphosphateHuman6287
BUB1BUBOther5dmzBadenosine-5'-diphosphateHuman6286
BUB1BUBOther6f7bAA2-[3,5-bis(fluoranyl)-4-[[3-[5-methoxy-4-[(3-methoxypyridin-4-yl)amino]pyrimidin-2-yl]indazol-1-yl]methyl]phenoxy]ethanolHuman10808
BUB1BUBOther6f7bAB2-[3,5-bis(fluoranyl)-4-[[3-[5-methoxy-4-[(3-methoxypyridin-4-yl)amino]pyrimidin-2-yl]indazol-1-yl]methyl]phenoxy]ethanolHuman10807
BUB1B (BUBR1)BUBOther6tljS-Human11992
CAMK1 (CaMK1a)CAMK1CAMK4fg7Aadenosine-5'-triphosphateHuman4848
CAMK1 (CaMK1a)CAMK1CAMK4fg8Aadenosine-5'-triphosphateHuman4850
CAMK1 (CaMK1a)CAMK1CAMK4fg8Badenosine-5'-triphosphateHuman4849
CAMK1 (CaMK1a)CAMK1CAMK4fg9Aadenosine-5'-triphosphateHuman4846
CAMK1 (CaMK1a)CAMK1CAMK4fg9Badenosine-5'-triphosphateHuman4845
CAMK1 (CaMK1a)CAMK1CAMK4fgbA-Human4847
CAMK1D (CaMK1d)CAMK1CAMK2jc6AAn-(5-methyl-1h-pyrazol-3-yl)-2-phenylquinazolin-4-amineHuman4829
CAMK1D (CaMK1d)CAMK1CAMK2jc6ABn-(5-methyl-1h-pyrazol-3-yl)-2-phenylquinazolin-4-amineHuman4830
CAMK1D (CaMK1d)CAMK1CAMK2jc6CAn-(5-methyl-1h-pyrazol-3-yl)-2-phenylquinazolin-4-amineHuman4832
CAMK1D (CaMK1d)CAMK1CAMK2jc6CBn-(5-methyl-1h-pyrazol-3-yl)-2-phenylquinazolin-4-amineHuman4831
CAMK1D (CaMK1d)CAMK1CAMK6qp5AA-Human12028
CAMK1D (CaMK1d)CAMK1CAMK6qp5AB-Human12029
CAMK1D (CaMK1d)CAMK1CAMK6t6fAA2-[(3~{s})-3-azanylpiperidin-1-yl]-4-[[3-(trifluoromethyl)phenyl]amino]pyrimidine-5-carboxamideHuman11939
CAMK1D (CaMK1d)CAMK1CAMK6t6fAB2-[(3~{s})-3-azanylpiperidin-1-yl]-4-[[3-(trifluoromethyl)phenyl]amino]pyrimidine-5-carboxamideHuman11940
CAMK1D (CaMK1d)CAMK1CAMK6t6fBA2-[(3~{s})-3-azanylpiperidin-1-yl]-4-[[3-(trifluoromethyl)phenyl]amino]pyrimidine-5-carboxamideHuman11941
CAMK1D (CaMK1d)CAMK1CAMK6t6fBB2-[(3~{s})-3-azanylpiperidin-1-yl]-4-[[3-(trifluoromethyl)phenyl]amino]pyrimidine-5-carboxamideHuman11942
CAMK1G (CaMK1g)CAMK1CAMK2jamAA5-[(e)-(5-chloro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-n-[2-(diethylamino)ethyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman1218
CAMK1G (CaMK1g)CAMK1CAMK2jamAB5-[(e)-(5-chloro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-n-[2-(diethylamino)ethyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman1221
CAMK1G (CaMK1g)CAMK1CAMK2jamBA5-[(e)-(5-chloro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-n-[2-(diethylamino)ethyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman1220
CAMK1G (CaMK1g)CAMK1CAMK2jamBB5-[(e)-(5-chloro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-n-[2-(diethylamino)ethyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman1219
CAMK2A (CaMK2a)CAMK2CAMK2vz6AA(2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime}Human2472
CAMK2A (CaMK2a)CAMK2CAMK2vz6AB(2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime}Human2471
CAMK2A (CaMK2a)CAMK2CAMK2vz6BA(2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime}Human2474
CAMK2A (CaMK2a)CAMK2CAMK2vz6BB(2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime}Human2470
CAMK2A (CaMK2a)CAMK2CAMK3soaA4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrileHuman2473
CAMK2A (CaMK2a)CAMK2CAMK6vzkA4'-hydroxycinnamic acidHuman12165
CAMK2A (CaMK2a)CAMK2CAMK6w4oO-Human12485
CAMK2A (CaMK2a)CAMK2CAMK6w4pH-Human12484
CAMK2B (CaMK2b)CAMK2CAMK3bhhA[4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]-6-(methylamino)pyrimidin-2-yl}amino)phenyl]acetonitrileHuman1507
CAMK2B (CaMK2b)CAMK2CAMK3bhhB[4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]-6-(methylamino)pyrimidin-2-yl}amino)phenyl]acetonitrileHuman1506
CAMK2B (CaMK2b)CAMK2CAMK3bhhC-Human1505
CAMK2B (CaMK2b)CAMK2CAMK3bhhD-Human1504
Camk2d (CaMK2d)CAMK2CAMK6babAAn-[(2s)-2-(diethylamino)propyl]-2-(3-hydroxyazetidin-1-yl)-6-[5-(thiophen-2-yl)pyrazolo[1,5-a]pyrimidin-3-yl]pyridine-4-carboxamideMouse8694
Camk2d (CaMK2d)CAMK2CAMK6babABn-[(2s)-2-(diethylamino)propyl]-2-(3-hydroxyazetidin-1-yl)-6-[5-(thiophen-2-yl)pyrazolo[1,5-a]pyrimidin-3-yl]pyridine-4-carboxamideMouse8691
Camk2d (CaMK2d)CAMK2CAMK6babBAn-[(2s)-2-(diethylamino)propyl]-2-(3-hydroxyazetidin-1-yl)-6-[5-(thiophen-2-yl)pyrazolo[1,5-a]pyrimidin-3-yl]pyridine-4-carboxamideMouse8690
Camk2d (CaMK2d)CAMK2CAMK6babBBn-[(2s)-2-(diethylamino)propyl]-2-(3-hydroxyazetidin-1-yl)-6-[5-(thiophen-2-yl)pyrazolo[1,5-a]pyrimidin-3-yl]pyridine-4-carboxamideMouse8693
Camk2d (CaMK2d)CAMK2CAMK6babCAn-[(2s)-2-(diethylamino)propyl]-2-(3-hydroxyazetidin-1-yl)-6-[5-(thiophen-2-yl)pyrazolo[1,5-a]pyrimidin-3-yl]pyridine-4-carboxamideMouse8697
Camk2d (CaMK2d)CAMK2CAMK6babCBn-[(2s)-2-(diethylamino)propyl]-2-(3-hydroxyazetidin-1-yl)-6-[5-(thiophen-2-yl)pyrazolo[1,5-a]pyrimidin-3-yl]pyridine-4-carboxamideMouse8692
Camk2d (CaMK2d)CAMK2CAMK6babDAn-[(2s)-2-(diethylamino)propyl]-2-(3-hydroxyazetidin-1-yl)-6-[5-(thiophen-2-yl)pyrazolo[1,5-a]pyrimidin-3-yl]pyridine-4-carboxamideMouse8695
Camk2d (CaMK2d)CAMK2CAMK6babDBn-[(2s)-2-(diethylamino)propyl]-2-(3-hydroxyazetidin-1-yl)-6-[5-(thiophen-2-yl)pyrazolo[1,5-a]pyrimidin-3-yl]pyridine-4-carboxamideMouse8696
CAMK2D (CaMK2d)CAMK2CAMK2vn9A[4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl}imino)cyclohexa-2,5-dien-1-yl]acetonitrileHuman2140
CAMK2D (CaMK2d)CAMK2CAMK2vn9B[4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl}imino)cyclohexa-2,5-dien-1-yl]acetonitrileHuman2139
CAMK2D (CaMK2d)CAMK2CAMK2welAA(3z)-n,n-dimethyl-2-oxo-3-(4,5,6,7-tetrahydro-1h-indol-2-ylmethylidene)-2,3-dihydro-1h-indole-5-sulfonamideHuman2138
CAMK2D (CaMK2d)CAMK2CAMK2welAB(3z)-n,n-dimethyl-2-oxo-3-(4,5,6,7-tetrahydro-1h-indol-2-ylmethylidene)-2,3-dihydro-1h-indole-5-sulfonamideHuman2137
CAMK2D (CaMK2d)CAMK2CAMK2welAC(3z)-n,n-dimethyl-2-oxo-3-(4,5,6,7-tetrahydro-1h-indol-2-ylmethylidene)-2,3-dihydro-1h-indole-5-sulfonamideHuman2136
CAMK2D (CaMK2d)CAMK2CAMK5vloAn-[(2s)-2-(diethylamino)propyl]-2-[(2s)-2-(methylcarbamoyl)azetidin-1-yl]-6-[5-(thiophen-2-yl)pyrazolo[1,5-a]pyrimidin-3-yl]pyridine-4-carboxamideHuman8348
CAMK2D (CaMK2d)CAMK2CAMK5vloBn-[(2s)-2-(diethylamino)propyl]-2-[(2s)-2-(methylcarbamoyl)azetidin-1-yl]-6-[5-(thiophen-2-yl)pyrazolo[1,5-a]pyrimidin-3-yl]pyridine-4-carboxamideHuman8347
CAMK2D (CaMK2d)CAMK2CAMK6aywAn-[2-(dimethylamino)ethyl]-3-[6-(thiophen-2-yl)imidazo[1,2-b]pyridazin-3-yl]benzamideHuman8666
CAMK2D (CaMK2d)CAMK2CAMK6aywBn-[2-(dimethylamino)ethyl]-3-[6-(thiophen-2-yl)imidazo[1,2-b]pyridazin-3-yl]benzamideHuman8665
CAMK2G (CaMK2g)CAMK2CAMK2v7oAA-Human7239
CAMK2G (CaMK2g)CAMK2CAMK2v7oAB-Human7238
CAMK4 (CaMK4)CAMK1CAMK2w4oA5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamideHuman2687
CAMKK1 (CaMKK1)CAMKKOther6ccfAn-[2-oxo-3-((e)-phenyl{[4-(piperidin-1-ylmethyl)phenyl]imino}methyl)-2,6-dihydro-1h-indol-5-yl]ethanesulfonamideHuman9712
CAMKK1 (CaMKK1)CAMKKOther6ccfBn-[2-oxo-3-((e)-phenyl{[4-(piperidin-1-ylmethyl)phenyl]imino}methyl)-2,6-dihydro-1h-indol-5-yl]ethanesulfonamideHuman9717
CAMKK1 (CaMKK1)CAMKKOther6cd6AA2-cyclopentyl-4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acidHuman9716
CAMKK1 (CaMKK1)CAMKKOther6cd6AB2-cyclopentyl-4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acidHuman9714
CAMKK1 (CaMKK1)CAMKKOther6cd6BA2-cyclopentyl-4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acidHuman9709
CAMKK1 (CaMKK1)CAMKKOther6cd6BB2-cyclopentyl-4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acidHuman9713
CAMKK1 (CaMKK1)CAMKKOther6cd6CA2-cyclopentyl-4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acidHuman9711
CAMKK1 (CaMKK1)CAMKKOther6cd6CB2-cyclopentyl-4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acidHuman9715
CAMKK1 (CaMKK1)CAMKKOther6cd6DA2-cyclopentyl-4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acidHuman9710
CAMKK1 (CaMKK1)CAMKKOther6cd6DB2-cyclopentyl-4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acidHuman9708
CAMKK2 (CaMKK2)CAMKKOther2zv2A7-oxo-7h-benzimidazo[2,1-a]benz[de]isoquinoline-3-carboxylic acidHuman406
CAMKK2 (CaMKK2)CAMKKOther5uy6A2-cyclopentyl-4-(5-phenylfuro[2,3-b]pyridin-3-yl)benzoic acidHuman7982
CAMKK2 (CaMKK2)CAMKKOther5uyjAA2-cyclopentyl-4-(7-methoxyquinolin-4-yl)benzoic acidHuman7560
CAMKK2 (CaMKK2)CAMKKOther5uyjAB2-cyclopentyl-4-(7-methoxyquinolin-4-yl)benzoic acidHuman7559
CAMKK2 (CaMKK2)CAMKKOther5vt1A4-({5-[(3-hydroxy-4-methylphenyl)amino]-4-oxo-4h-1,2,6-thiadiazin-3-yl}amino)benzamideHuman7591
CAMKK2 (CaMKK2)CAMKKOther5yv8AA1-amino-4-hydroxy-9,10-dioxo-9,10-dihydroanthracene-2-carboxylic acidHuman10753
CAMKK2 (CaMKK2)CAMKKOther5yv8AB1-amino-4-hydroxy-9,10-dioxo-9,10-dihydroanthracene-2-carboxylic acidHuman10755
CAMKK2 (CaMKK2)CAMKKOther5yv9A5-chloro-2-methoxy-4[(1z)-3-(4-methoxyphenyl)-3-oxoprop-1-en-1-yl]aminobenzoic acidHuman10752
CAMKK2 (CaMKK2)CAMKKOther5yvaA3-(1h-tetrazol-5-yl)-10lambda~6~-thioxanthene-9,10,10-trioneHuman10750
CAMKK2 (CaMKK2)CAMKKOther5yvbA(3z)-5-chloro-3-[(1-methyl-1h-pyrazol-4-yl)methylidene]-1,3-dihydro-2h-indol-2-oneHuman10751
CAMKK2 (CaMKK2)CAMKKOther5yvcA3-{2,4-dimethyl-5-[(z)-(2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-1h-pyrrol-3-yl}propanoic acidHuman10754
CAMKK2 (CaMKK2)CAMKKOther6bkuA2-cyclopentyl-4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acidHuman8687
CAMKK2 (CaMKK2)CAMKKOther6bleAA1-{2-[5-(2-methoxyethoxy)-1h-benzimidazol-1-yl]quinolin-8-yl}piperidin-4-amineHuman8688
CAMKK2 (CaMKK2)CAMKKOther6bleAB1-{2-[5-(2-methoxyethoxy)-1h-benzimidazol-1-yl]quinolin-8-yl}piperidin-4-amineHuman8689
CAMKK2 (CaMKK2)CAMKKOther6bqlA2-({5-chloro-2-[(2-methoxy-4-morpholin-4-ylphenyl)amino]pyrimidin-4-yl}amino)-n-methylbenzamideHuman9061
CAMKK2 (CaMKK2)CAMKKOther6bqpA1-(2-{5-[(3-methyloxetan-3-yl)methoxy]-1h-benzimidazol-1-yl}quinolin-8-yl)piperidin-4-amineHuman9064
CAMKK2 (CaMKK2)CAMKKOther6bqqA4-{[(7r)-8-cyclopentyl-7-ethyl-5-methyl-6-oxo-5,6,7,8-tetrahydropteridin-2-yl]amino}-3-methoxy-n-(1-methylpiperidin-4-yl)benzamideHuman9063
CAMKK2 (CaMKK2)CAMKKOther6brcA5-chloro-n~2~-{4-[4-(dimethylamino)piperidin-1-yl]-2-methoxyphenyl}-n~4~-[2-(dimethylphosphoryl)phenyl]pyrimidine-2,4-diamineHuman9062
CAMKK2 (CaMKK2)CAMKKOther6brcB5-chloro-n~2~-{4-[4-(dimethylamino)piperidin-1-yl]-2-methoxyphenyl}-n~4~-[2-(dimethylphosphoryl)phenyl]pyrimidine-2,4-diamineHuman9060
CAMKK2 (CaMKK2)CAMKKOther6cmjAA2-(2-methylpropyl)-4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acidHuman9784
CAMKK2 (CaMKK2)CAMKKOther6cmjAB2-(2-methylpropyl)-4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acidHuman9783
CAMKK2 (CaMKK2)CAMKKOther6cmjBA2-(2-methylpropyl)-4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acidHuman9786
CAMKK2 (CaMKK2)CAMKKOther6cmjBB2-(2-methylpropyl)-4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acidHuman9785
CASKCASKCAMK3c0gAA[(2r,3s,4r,5r)-5-(6-aminopurin-9-yl)-4-hydroxy-2-(hydroxymethyl)oxolan-3-yl] dihydrogen phosphateHuman3828
CASKCASKCAMK3c0gAB[(2r,3s,4r,5r)-5-(6-aminopurin-9-yl)-4-hydroxy-2-(hydroxymethyl)oxolan-3-yl] dihydrogen phosphateHuman3827
CASKCASKCAMK3c0gBA[(2r,3s,4r,5r)-5-(6-aminopurin-9-yl)-4-hydroxy-2-(hydroxymethyl)oxolan-3-yl] dihydrogen phosphateHuman3824
CASKCASKCAMK3c0gBB[(2r,3s,4r,5r)-5-(6-aminopurin-9-yl)-4-hydroxy-2-(hydroxymethyl)oxolan-3-yl] dihydrogen phosphateHuman3826
CASKCASKCAMK3c0hAadenosine monophosphateHuman3825
CASKCASKCAMK3c0hBadenosine monophosphateHuman3817
CASKCASKCAMK3c0iAA[(2r,3s,4r,5r)-5-(6-aminopurin-9-yl)-4-hydroxy-2-(hydroxymethyl)oxolan-3-yl] dihydrogen phosphateHuman3830
CASKCASKCAMK3c0iAB[(2r,3s,4r,5r)-5-(6-aminopurin-9-yl)-4-hydroxy-2-(hydroxymethyl)oxolan-3-yl] dihydrogen phosphateHuman3819
CASKCASKCAMK3mfrAAphosphoaminophosphonic acid-adenylate esterHuman3822
CASKCASKCAMK3mfrABphosphoaminophosphonic acid-adenylate esterHuman3831
CASKCASKCAMK3mfsAAphosphoaminophosphonic acid-adenylate esterHuman3818
CASKCASKCAMK3mfsABphosphoaminophosphonic acid-adenylate esterHuman3829
CASKCASKCAMK3mftAA-Human3823
CASKCASKCAMK3mftAB-Human3821
CASKCASKCAMK3mfuAAphosphoaminophosphonic acid-adenylate esterHuman3816
CASKCASKCAMK3mfuABphosphoaminophosphonic acid-adenylate esterHuman3832
CASKCASKCAMK3tacA-Human3820
CASKCASKCAMK6kmhA-Human12672
CASKCASKCAMK6kmhB-Human12671
CDC42BPB (MRCKb)DMPKAGC3qfvA2-(carbamoylamino)-5-(4-fluorophenyl)thiophene-3-carboxamideHuman4860
CDC42BPB (MRCKb)DMPKAGC3qfvB2-(carbamoylamino)-5-(4-fluorophenyl)thiophene-3-carboxamideHuman4857
CDC42BPB (MRCKb)DMPKAGC3tkuA5-(1,4-diazepan-1-sulfonyl)isoquinolineHuman4862
CDC42BPB (MRCKb)DMPKAGC3tkuB5-(1,4-diazepan-1-sulfonyl)isoquinolineHuman4859
CDC42BPB (MRCKb)DMPKAGC4uakAAadenosine-5'-diphosphateHuman4864
CDC42BPB (MRCKb)DMPKAGC4uakABadenosine-5'-diphosphateHuman4863
CDC42BPB (MRCKb)DMPKAGC4ualAA4-chloro-1-(piperidin-4-yl)-n-[3-(pyridin-2-yl)-1h-pyrazol-4-yl]-1h-pyrazole-3-carboxamideHuman4861
CDC42BPB (MRCKb)DMPKAGC4ualAB4-chloro-1-(piperidin-4-yl)-n-[3-(pyridin-2-yl)-1h-pyrazol-4-yl]-1h-pyrazole-3-carboxamideHuman4858
CDC42BPB (MRCKb)DMPKAGC5oteA2-[4-[(6~{s})-1,8-diazaspiro[5.5]undecan-8-yl]-1~{h}-pyrrolo[2,3-b]pyridin-3-yl]-1,3-thiazoleHuman9578
CDC42BPB (MRCKb)DMPKAGC5otfA(6~{s})-8-(3-pyrimidin-4-yl-1~{h}-pyrrolo[2,3-b]pyridin-4-yl)-1,8-diazaspiro[5.5]undecaneHuman9577
CDC7CDC7Other4f99Aadenosine-5'-diphosphateHuman4824
CDC7CDC7Other4f9aAadenosine-5'-diphosphateHuman4825
CDC7CDC7Other4f9aCadenosine-5'-diphosphateHuman4826
CDC7CDC7Other4f9bA2-(pyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman4828
CDC7CDC7Other4f9bC2-(pyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman4827
CDC7CDC7Other4f9cA8-chloro-2-[(2s)-pyrrolidin-2-yl][1]benzofuro[3,2-d]pyrimidin-4(3h)-oneHuman4823
CDK1 (CDC2)CDKCMGC4y72AA{[(2,6-difluorophenyl)carbonyl]amino}-n-(4-fluorophenyl)-1h-pyrazole-3-carboxamideHuman4610
CDK1 (CDC2)CDKCMGC4y72AB{[(2,6-difluorophenyl)carbonyl]amino}-n-(4-fluorophenyl)-1h-pyrazole-3-carboxamideHuman4609
CDK1 (CDC2)CDKCMGC4yc3AA-Human6555
CDK1 (CDC2)CDKCMGC4yc3AB-Human6554
CDK1 (CDC2)CDKCMGC4yc6AA-Human4607
CDK1 (CDC2)CDKCMGC4yc6AB-Human4616
CDK1 (CDC2)CDKCMGC4yc6CA-Human4608
CDK1 (CDC2)CDKCMGC4yc6CB-Human4611
CDK1 (CDC2)CDKCMGC4yc6EA-Human4612
CDK1 (CDC2)CDKCMGC4yc6EB-Human4614
CDK1 (CDC2)CDKCMGC4yc6GA-Human4613
CDK1 (CDC2)CDKCMGC4yc6GB-Human4615
CDK1 (CDC2)CDKCMGC5hq0AA{[(2,6-difluorophenyl)carbonyl]amino}-n-(4-fluorophenyl)-1h-pyrazole-3-carboxamideHuman6422
CDK1 (CDC2)CDKCMGC5hq0AB{[(2,6-difluorophenyl)carbonyl]amino}-n-(4-fluorophenyl)-1h-pyrazole-3-carboxamideHuman6421
CDK1 (CDC2)CDKCMGC5lqfAAo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman7364
CDK1 (CDC2)CDKCMGC5lqfABo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman7366
CDK1 (CDC2)CDKCMGC5lqfDAo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman7365
CDK1 (CDC2)CDKCMGC5lqfDBo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman7367
CDK1 (CDC2)CDKCMGC6gu2AA2-(2-chlorophenyl)-8-[(3~{r},4~{r})-1-methyl-3-oxidanyl-piperidin-4-yl]-5,7-bis(oxidanyl)chromen-4-oneHuman10780
CDK1 (CDC2)CDKCMGC6gu2AB2-(2-chlorophenyl)-8-[(3~{r},4~{r})-1-methyl-3-oxidanyl-piperidin-4-yl]-5,7-bis(oxidanyl)chromen-4-oneHuman10776
CDK1 (CDC2)CDKCMGC6gu3A4-(2-methyl-3-propan-2-yl-imidazol-4-yl)-~{n}-(4-methylsulfonylphenyl)pyrimidin-2-amineHuman10778
CDK1 (CDC2)CDKCMGC6gu4A~{n}2-[(1~{r},2~{s})-2-azanylcyclohexyl]-~{n}6-(3-chlorophenyl)-9-ethyl-purine-2,6-diamineHuman10777
CDK1 (CDC2)CDKCMGC6gu6A3-[({3-ethyl-5-[(2s)-2-(2-hydroxyethyl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1-hydroxypyridiniumHuman10774
CDK1 (CDC2)CDKCMGC6gu7A4-(2-methyl-3-propan-2-yl-imidazol-4-yl)-~{n}-(4-methylsulfonylphenyl)pyrimidin-2-amineHuman10781
CDK1 (CDC2)CDKCMGC6gu7C-Human10775
CDK1 (CDC2)CDKCMGC6gu7E-Human10782
CDK1 (CDC2)CDKCMGC6gu7G-Human10779
CDK12 (CRK7)CDKCMGC4cxaAphosphoaminophosphonic acid-adenylate esterHuman4856
CDK12 (CRK7)CDKCMGC4cxaC-Human4853
CDK12 (CRK7)CDKCMGC4nstAadenosine-5'-diphosphateHuman4852
CDK12 (CRK7)CDKCMGC4nstCadenosine-5'-diphosphateHuman4851
CDK12 (CRK7)CDKCMGC4un0C-Human4854
CDK12 (CRK7)CDKCMGC4un0D-Human4855
CDK12 (CRK7)CDKCMGC5acbCn-[4-[(3r)-3-[[5-chloranyl-4-(1h-indol-3-yl)pyrimidin-2-yl]amino]piperidin-1-yl]carbonylphenyl]-4-(dimethylamino)butanamideHuman6701
CDK12 (CRK7)CDKCMGC5acbDn-[4-[(3r)-3-[[5-chloranyl-4-(1h-indol-3-yl)pyrimidin-2-yl]amino]piperidin-1-yl]carbonylphenyl]-4-(dimethylamino)butanamideHuman6702
CDK12 (CRK7)CDKCMGC6b3eA2-[(2s)-1-(6-{[(4,5-difluoro-1h-benzimidazol-2-yl)methyl]amino}-9-ethyl-9h-purin-2-yl)piperidin-2-yl]ethan-1-olHuman9452
CDK12 (CRK7)CDKCMGC6b3eC2-[(2s)-1-(6-{[(4,5-difluoro-1h-benzimidazol-2-yl)methyl]amino}-9-ethyl-9h-purin-2-yl)piperidin-2-yl]ethan-1-olHuman9453
CDK12 (CRK7)CDKCMGC6ckxAn-[4-(1-methyl-1h-pyrazol-4-yl)phenyl]-n-{trans-4-[(quinazolin-2-yl)amino]cyclohexyl}acetamideHuman10578
CDK12 (CRK7)CDKCMGC6ckxCn-[4-(1-methyl-1h-pyrazol-4-yl)phenyl]-n-{trans-4-[(quinazolin-2-yl)amino]cyclohexyl}acetamideHuman10579
CDK12 (CRK7)CDKCMGC6td3B(2r)-2-({9-(1-methylethyl)-6-[(4-pyridin-2-ylbenzyl)amino]-9h-purin-2-yl}amino)butan-1-olHuman12371
CDK12 (CRK7)CDKCMGC6td3E(2r)-2-({9-(1-methylethyl)-6-[(4-pyridin-2-ylbenzyl)amino]-9h-purin-2-yl}amino)butan-1-olHuman12369
CDK12 (CRK7)CDKCMGC6td3H(2r)-2-({9-(1-methylethyl)-6-[(4-pyridin-2-ylbenzyl)amino]-9h-purin-2-yl}amino)butan-1-olHuman12370
CDK13 (CHED)CDKCMGC5efqAadenosine-5'-diphosphateHuman6323
CDK13 (CHED)CDKCMGC5efqCadenosine-5'-diphosphateHuman6324
CDK16 (PCTAIRE1)CDKCMGC3mtlAA(2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime}Human1701
CDK16 (PCTAIRE1)CDKCMGC3mtlAB(2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime}Human1702
CDK16 (PCTAIRE1)CDKCMGC5g6vA4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamideHuman7273
CDK16 (PCTAIRE1)CDKCMGC5g6vB4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamideHuman7274
CDK2CDKCMGC1aq1AstaurosporineHuman4267
CDK2CDKCMGC1b38Aadenosine-5'-triphosphateHuman4483
CDK2CDKCMGC1b39Aadenosine-5'-triphosphateHuman4407
CDK2CDKCMGC1buhA-Human4178
CDK2CDKCMGC1ckpAApurvalanol bHuman4066
CDK2CDKCMGC1ckpABpurvalanol bHuman4214
CDK2CDKCMGC1di8A4-[3-hydroxyanilino]-6,7-dimethoxyquinazolineHuman4577
CDK2CDKCMGC1dm2AA4-(5-amino-4-oxo-4h-pyrazol-3-yl)-2-bromo-4,5,6,7-tetrahydro-3ah-pyrrolo[2,3-c]azepin-8-oneHuman4104
CDK2CDKCMGC1dm2AB4-(5-amino-4-oxo-4h-pyrazol-3-yl)-2-bromo-4,5,6,7-tetrahydro-3ah-pyrrolo[2,3-c]azepin-8-oneHuman4024
CDK2CDKCMGC1e1vA6-o-cyclohexylmethyl guanineHuman3886
CDK2CDKCMGC1e1xA6-cyclohexylmethyloxy-5-nitroso-pyrimidine-2,4-diamineHuman4114
CDK2CDKCMGC1e9hA2',3-dioxo-1,1',2',3-tetrahydro-2,3'-biindole-5'-sulfonic acidHuman4302
CDK2CDKCMGC1e9hC2',3-dioxo-1,1',2',3-tetrahydro-2,3'-biindole-5'-sulfonic acidHuman4570
CDK2CDKCMGC1f5qAA-Human4194
CDK2CDKCMGC1f5qAB-Human4517
CDK2CDKCMGC1f5qCA-Human4281
CDK2CDKCMGC1f5qCB-Human3952
CDK2CDKCMGC1finAadenosine-5'-triphosphateHuman4367
CDK2CDKCMGC1finCadenosine-5'-triphosphateHuman4479
CDK2CDKCMGC1fq1Badenosine-5'-triphosphateHuman4266
CDK2CDKCMGC1fvtA4-(5-bromo-2-oxo-2h-indol-3-ylazo)-benzenesulfonamideHuman4480
CDK2CDKCMGC1fvvA4-[(7-oxo-7h-thiazolo[5,4-e]indol-8-ylmethyl)-amino]-n-pyridin-2-yl-benzenesulfonamideHuman4065
CDK2CDKCMGC1fvvC4-[(7-oxo-7h-thiazolo[5,4-e]indol-8-ylmethyl)-amino]-n-pyridin-2-yl-benzenesulfonamideHuman4461
CDK2CDKCMGC1g5sA2-[trans-(4-aminocyclohexyl)amino]-6-(benzyl-amino)-9-cyclopentylpurineHuman3888
CDK2CDKCMGC1gihA1-(5-oxo-2,3,5,9b-tetrahydro-1h-pyrrolo[2,1-a]isoindol-9-yl)-3-pyridin-2-yl-ureaHuman3922
CDK2CDKCMGC1giiA1-(5-oxo-2,3,5,9b-tetrahydro-1h-pyrrolo[2,1-a]isoindol-9-yl)-3-pyridin-2-yl-ureaHuman4448
CDK2CDKCMGC1gijA1-(5-oxo-2,3,5,9b-tetrahydro-1h-pyrrolo[2,1-a]isoindol-9-yl)-3-(5-pyrrolidin-2-yl-1h-pyrazol-3-yl)-ureaHuman4542
CDK2CDKCMGC1gy3Aadenosine-5'-triphosphateHuman3978
CDK2CDKCMGC1gy3Cadenosine-5'-triphosphateHuman4445
CDK2CDKCMGC1gz8AA1-[(2-amino-6,9-dihydro-1h-purin-6-yl)oxy]-3-methyl-2-butanolHuman3981
CDK2CDKCMGC1gz8AB1-[(2-amino-6,9-dihydro-1h-purin-6-yl)oxy]-3-methyl-2-butanolHuman3956
CDK2CDKCMGC1h00AA(2s)-1-[4-({6-[(2,6-difluorophenyl)amino]pyrimidin-4-yl}amino)phenoxy]-3-(dimethylamino)propan-2-olHuman4484
CDK2CDKCMGC1h00AB(2r)-1-[4-({6-[(2,6-difluorophenyl)amino]pyrimidin-4-yl}amino)phenoxy]-3-(dimethylamino)propan-2-olHuman4428
CDK2CDKCMGC1h01AA(2r)-1-[4-({4-[(2,5-dichlorophenyl)amino]pyrimidin-2-yl}amino)phenoxy]-3-(dimethylamino)propan-2-olHuman3974
CDK2CDKCMGC1h01AB(2s)-1-[4-({4-[(2,5-dichlorophenyl)amino]pyrimidin-2-yl}amino)phenoxy]-3-(dimethylamino)propan-2-olHuman4561
CDK2CDKCMGC1h07AA((2-bromo-4-methylphenyl){6-[(4-{[(2r)-3-(dimethylamino)-2-hydroxypropyl]oxy}phenyl)amino]pyrimidin-4-yl}amino)acetonitrileHuman3918
CDK2CDKCMGC1h07AB((2-bromo-4-methylphenyl){6-[(4-{[(2s)-3-(dimethylamino)-2-hydroxypropyl]oxy}phenyl)amino]pyrimidin-4-yl}amino)acetonitrileHuman3908
CDK2CDKCMGC1h08AA(2r)-1-{4-[(4-anilino-5-bromopyrimidin-2-yl)amino]phenoxy}-3-(dimethylamino)propan-2-olHuman4220
CDK2CDKCMGC1h08AB(2s)-1-{4-[(4-anilino-5-bromopyrimidin-2-yl)amino]phenoxy}-3-(dimethylamino)propan-2-olHuman4411
CDK2CDKCMGC1h0vAA5-{[(2-amino-9h-purin-6-yl)oxy]methyl}-2-pyrrolidinoneHuman4368
CDK2CDKCMGC1h0vAB5-{[(2-amino-9h-purin-6-yl)oxy]methyl}-2-pyrrolidinoneHuman3933
CDK2CDKCMGC1h0wAA1-amino-6-cyclohex-3-enylmethyloxypurineHuman3987
CDK2CDKCMGC1h0wAB1-amino-6-cyclohex-3-enylmethyloxypurineHuman4016
CDK2CDKCMGC1h1pA6-o-cyclohexylmethyl guanineHuman4309
CDK2CDKCMGC1h1pC6-o-cyclohexylmethyl guanineHuman4581
CDK2CDKCMGC1h1qA2-anilino-6-cyclohexylmethoxypurineHuman4195
CDK2CDKCMGC1h1qC2-anilino-6-cyclohexylmethoxypurineHuman4053
CDK2CDKCMGC1h1rAA6-cyclohexylmethoxy-2-(3'-chloroanilino) purineHuman3906
CDK2CDKCMGC1h1rAB6-cyclohexylmethoxy-2-(3'-chloroanilino) purineHuman4494
CDK2CDKCMGC1h1rCA6-cyclohexylmethoxy-2-(3'-chloroanilino) purineHuman3920
CDK2CDKCMGC1h1rCB6-cyclohexylmethoxy-2-(3'-chloroanilino) purineHuman4081
CDK2CDKCMGC1h1sAo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman4400
CDK2CDKCMGC1h1sCo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman4572
CDK2CDKCMGC1h24A-Human4199
CDK2CDKCMGC1h24C-Human4296
CDK2CDKCMGC1h25A-Human4273
CDK2CDKCMGC1h25C-Human4112
CDK2CDKCMGC1h26A-Human4122
CDK2CDKCMGC1h26C-Human4179
CDK2CDKCMGC1h27A-Human4116
CDK2CDKCMGC1h27C-Human4030
CDK2CDKCMGC1h28A-Human4169
CDK2CDKCMGC1h28C-Human4351
CDK2CDKCMGC1hckAAadenosine-5'-triphosphateHuman3878
CDK2CDKCMGC1hckABadenosine-5'-triphosphateHuman4416
CDK2CDKCMGC1hclAA-Human4545
CDK2CDKCMGC1hclAB-Human4540
CDK2CDKCMGC1jstAadenosine-5'-triphosphateHuman4455
CDK2CDKCMGC1jstCadenosine-5'-triphosphateHuman4356
CDK2CDKCMGC1jsuA-Human4146
CDK2CDKCMGC1jsvA4-[(6-amino-4-pyrimidinyl)amino]benzenesulfonamideHuman4171
CDK2CDKCMGC1jvpP13-pyridin-4-yl-2,4-dihydro-indeno[1,2-.c.]pyrazoleHuman3919
CDK2CDKCMGC1jvpP23-pyridin-4-yl-2,4-dihydro-indeno[1,2-.c.]pyrazoleHuman4097
CDK2CDKCMGC1ke5An-methyl-4-{[(2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]amino}benzenesulfonamideHuman4376
CDK2CDKCMGC1ke6An-methyl-{4-[2-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)hydrazino]phenyl}methanesulfonamideHuman4219
CDK2CDKCMGC1ke7A3-{[(2,2-dioxido-1,3-dihydro-2-benzothien-5-yl)amino]methylene}-5-(1,3-oxazol-5-yl)-1,3-dihydro-2h-indol-2-oneHuman4295
CDK2CDKCMGC1ke8A4-{[(2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]amino}-n-(1,3-thiazol-2-yl)benzenesulfonamideHuman4048
CDK2CDKCMGC1ke9A3-{[4-([amino(imino)methyl]aminosulfonyl)anilino]methylene}-2-oxo-2,3-dihydro-1h-indoleHuman4250
CDK2CDKCMGC1oguAA4-{[4-amino-6-(cyclohexylmethoxy)-5-nitrosopyrimidin-2-yl]amino}benzamideHuman3965
CDK2CDKCMGC1oguAB4-{[4-amino-6-(cyclohexylmethoxy)-5-nitrosopyrimidin-2-yl]amino}benzamideHuman3935
CDK2CDKCMGC1oguCA4-{[4-amino-6-(cyclohexylmethoxy)-5-nitrosopyrimidin-2-yl]amino}benzamideHuman3964
CDK2CDKCMGC1oguCB4-{[4-amino-6-(cyclohexylmethoxy)-5-nitrosopyrimidin-2-yl]amino}benzamideHuman4560
CDK2CDKCMGC1oi9AA6-cyclohexylmethyloxy-2-(4'-hydroxyanilino)purineHuman4033
CDK2CDKCMGC1oi9AB6-cyclohexylmethyloxy-2-(4'-hydroxyanilino)purineHuman4492
CDK2CDKCMGC1oi9CA6-cyclohexylmethyloxy-2-(4'-hydroxyanilino)purineHuman4571
CDK2CDKCMGC1oi9CB6-cyclohexylmethyloxy-2-(4'-hydroxyanilino)purineHuman4036
CDK2CDKCMGC1oiqAn-[4-(2-methylimidazo[1,2-a]pyridin-3-yl)-2-pyrimidinyl]acetamideHuman4379
CDK2CDKCMGC1oirA1-(dimethylamino)-3-(4-{{4-(2-methylimidazo[1,2-a]pyridin-3-yl)pyrimidin-2-yl]amino}phenoxy)propan-2-olHuman4389
CDK2CDKCMGC1oitA4-[(4-imidazo[1,2-a]pyridin-3-ylpyrimidin-2-yl)amino]benzenesulfonamideHuman4025
CDK2CDKCMGC1oiuAA3-(6-cyclohexylmethoxy-9h-purin-2-ylamino)-benzenesulfonamideHuman4110
CDK2CDKCMGC1oiuAB3-(6-cyclohexylmethoxy-9h-purin-2-ylamino)-benzenesulfonamideHuman4556
CDK2CDKCMGC1oiuCA3-(6-cyclohexylmethoxy-9h-purin-2-ylamino)-benzenesulfonamideHuman4524
CDK2CDKCMGC1oiuCB3-(6-cyclohexylmethoxy-9h-purin-2-ylamino)-benzenesulfonamideHuman4049
CDK2CDKCMGC1oiyAA4-(6-cyclohexylmethoxy-9h-purin-2-ylamino)--benzamideHuman4225
CDK2CDKCMGC1oiyAB4-(6-cyclohexylmethoxy-9h-purin-2-ylamino)--benzamideHuman3945
CDK2CDKCMGC1oiyCA4-(6-cyclohexylmethoxy-9h-purin-2-ylamino)--benzamideHuman4465
CDK2CDKCMGC1oiyCB4-(6-cyclohexylmethoxy-9h-purin-2-ylamino)--benzamideHuman4245
CDK2CDKCMGC1okvA-Human3921
CDK2CDKCMGC1okvC-Human4093
CDK2CDKCMGC1okwA-Human4314
CDK2CDKCMGC1okwC-Human3896
CDK2CDKCMGC1ol1A-Human4429
CDK2CDKCMGC1ol1C-Human3951
CDK2CDKCMGC1ol2A-Human4305
CDK2CDKCMGC1ol2C-Human4497
CDK2CDKCMGC1p2aA5-[(2-aminoethyl)amino]-6-fluoro-3-(1h-pyrrol-2-yl)benzo[cd]indol-2(1h)-oneHuman4422
CDK2CDKCMGC1p5eA4,5,6,7-tetrabromobenzotriazoleHuman4090
CDK2CDKCMGC1p5eC4,5,6,7-tetrabromobenzotriazoleHuman4434
CDK2CDKCMGC1pf8A(3z)-3-(1h-imidazol-5-ylmethylene)-5-methoxy-1h-indol-2(3h)-oneHuman3861
CDK2CDKCMGC1pkdA7-hydroxystaurosporineHuman4170
CDK2CDKCMGC1pkdC7-hydroxystaurosporineHuman3973
CDK2CDKCMGC1pw2A-Human4432
CDK2CDKCMGC1pxiAA4-(2,5-dichlorothien-3-yl)pyrimidin-2-amineHuman4381
CDK2CDKCMGC1pxiAB-Human3924
CDK2CDKCMGC1pxjAA4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-amineHuman3927
CDK2CDKCMGC1pxjAB-Human3911
CDK2CDKCMGC1pxkAAn-[4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-yl]-n'-hydroxyimidoformamideHuman3915
CDK2CDKCMGC1pxkAB-Human3980
CDK2CDKCMGC1pxlAA4-(2,4-dimethyl-1,3-thiazol-5-yl)-n-[4-(trifluoromethyl)phenyl]pyrimidin-2-amineHuman4233
CDK2CDKCMGC1pxlAB-Human4074
CDK2CDKCMGC1pxmAA3-[4-(2,4-dimethyl-thiazol-5-yl)-pyrimidin-2-ylamino]-phenolHuman3944
CDK2CDKCMGC1pxmAB-Human3936
CDK2CDKCMGC1pxnAA4-[4-(4-methyl-2-methylamino-thiazol-5-yl)-pyrimidin-2-ylamino]-phenolHuman4383
CDK2CDKCMGC1pxnAB-Human4172
CDK2CDKCMGC1pxoAA[4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amineHuman4512
CDK2CDKCMGC1pxoAB-Human3860
CDK2CDKCMGC1pxoAC[4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amineHuman4546
CDK2CDKCMGC1pxoAD[4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amineHuman4167
CDK2CDKCMGC1pxpAAn-[4-(2,4-dimethyl-thiazol-5-yl)-pyrimidin-2-yl]-n',n'-dimethyl-benzene-1,4-diamineHuman4316
CDK2CDKCMGC1pxpAB-Human3943
CDK2CDKCMGC1pyeA[2-amino-6-(2,6-difluoro-benzoyl)-imidazo[1,2-a]pyridin-3-yl]-phenyl-methanoneHuman4284
CDK2CDKCMGC1qmzAadenosine-5'-triphosphateHuman4242
CDK2CDKCMGC1qmzCadenosine-5'-triphosphateHuman4527
CDK2CDKCMGC1r78AA4-((3r,4s,5r)-4-amino-3,5-dihydroxy-hex-1-ynyl)-5-fluoro-3-[1-(3-methoxy-1h-pyrrol-2-yl)-meth-(z)-ylidene]-1,3-dihydro-indol-2-oneHuman4253
CDK2CDKCMGC1r78AB4-((3r,4s,5r)-4-amino-3,5-dihydroxy-hex-1-ynyl)-5-fluoro-3-[1-(3-methoxy-1h-pyrrol-2-yl)-meth-(z)-ylidene]-1,3-dihydro-indol-2-oneHuman4249
CDK2CDKCMGC1urcAA-Human4334
CDK2CDKCMGC1urcAB-Human4010
CDK2CDKCMGC1urcCA-Human4006
CDK2CDKCMGC1urcCB-Human3937
CDK2CDKCMGC1urwAA2-[4-(n-(3-dimethylaminopropyl)sulphamoyl)anilino]-Human4054
CDK2CDKCMGC1urwAB2-[4-(n-(3-dimethylaminopropyl)sulphamoyl)anilino]-Human4196
CDK2CDKCMGC1v1kAA(2r)-1-(dimethylamino)-3-{4-[(6-{[2-fluoro-5-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]phenoxy}propan-2-olHuman4189
CDK2CDKCMGC1v1kAB(2r)-1-(dimethylamino)-3-{4-[(6-{[2-fluoro-5-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]phenoxy}propan-2-olHuman3928
CDK2CDKCMGC1vywAn-(3-cyclopropyl-1h-pyrazol-5-yl)-2-(2-naphthyl)acetamideHuman3992
CDK2CDKCMGC1vywCn-(3-cyclopropyl-1h-pyrazol-5-yl)-2-(2-naphthyl)acetamideHuman4133
CDK2CDKCMGC1vyzAn-(5-cyclopropyl-1h-pyrazol-3-yl)benzamideHuman4325
CDK2CDKCMGC1w0xCAolomoucineHuman4537
CDK2CDKCMGC1w0xCBolomoucineHuman4478
CDK2CDKCMGC1w8cAA6-(cyclohexylmethoxy)-8-isopropyl-9h-purin-2-amineHuman4332
CDK2CDKCMGC1w8cAB6-(cyclohexylmethoxy)-8-isopropyl-9h-purin-2-amineHuman4197
CDK2CDKCMGC1w98A-Human4013
CDK2CDKCMGC1wccAA2-amino-6-chloropyrazineHuman4394
CDK2CDKCMGC1wccAB2-amino-6-chloropyrazineHuman3897
CDK2CDKCMGC1y8yA(5-chloropyrazolo[1,5-a]pyrimidin-7-yl)-(4-methanesulfonylphenyl)amineHuman3914
CDK2CDKCMGC1y91A4-[5-(trans-4-aminocyclohexylamino)-3-isopropylpyrazolo[1,5-a]pyrimidin-7-ylamino]-n,n-dimethylbenzenesulfonamideHuman4505
CDK2CDKCMGC1ykrA4-{[6-(2,6-dichlorobenzoyl)imidazo[1,2-a]pyridin-2-yl]amino}benzenesulfonamideHuman4578
CDK2CDKCMGC2a0cXA2-{[(2-{[(1r)-1-(hydroxymethyl)propyl]amino}-9-isopropyl-9h-purin-6-yl)amino]methyl}phenolHuman4157
CDK2CDKCMGC2a0cXB2-{[(2-{[(1r)-1-(hydroxymethyl)propyl]amino}-9-isopropyl-9h-purin-6-yl)amino]methyl}phenolHuman3868
CDK2CDKCMGC2a4lAr-roscovitineHuman4238
CDK2CDKCMGC2b52A1-(3-(2,4-dimethylthiazol-5-yl)-4-oxo-2,4-dihydroindeno[1,2-c]pyrazol-5-yl)-3-(4-methylpiperazin-1-yl)ureaHuman3997
CDK2CDKCMGC2b53A6-(3-aminophenyl)-n-(tert-butyl)-2-(trifluoromethyl)quinazolin-4-amineHuman3875
CDK2CDKCMGC2b54A6-(3,4-dihydroxybenzyl)-3-ethyl-1-(2,4,6-trichlorophenyl)-1h-pyrazolo[3,4-d]pyrimidin-4(5h)-oneHuman4292
CDK2CDKCMGC2b55A2-(4-(aminomethyl)piperidin-1-yl)-n-(3_cyclohexyl-4-oxo-2,4-dihydroindeno[1,2-c]pyrazol-5-yl)acetamideHuman4216
CDK2CDKCMGC2bheA(2z)-5'-bromo-2,3'-biindole-2',3(1h,1'h)-dione ammoniateHuman4184
CDK2CDKCMGC2bhhA(2e,3s)-3-hydroxy-5'-[(4-hydroxypiperidin-1-yl)sulfonyl]-3-methyl-1,3-dihydro-2,3'-biindol-2'(1'h)-oneHuman4417
CDK2CDKCMGC2bkzA1-[4-(aminosulfonyl)phenyl]-1,6-dihydropyrazolo[3,4-e]indazole-3-carboxamideHuman3942
CDK2CDKCMGC2bkzC1-[4-(aminosulfonyl)phenyl]-1,6-dihydropyrazolo[3,4-e]indazole-3-carboxamideHuman4555
CDK2CDKCMGC2bpmA(2s)-n-[(3z)-5-cyclopropyl-3h-pyrazol-3-ylidene]-2-[4-(2-oxoimidazolidin-1-yl)phenyl]propanamideHuman4042
CDK2CDKCMGC2bpmC(2s)-n-[(3z)-5-cyclopropyl-3h-pyrazol-3-ylidene]-2-[4-(2-oxoimidazolidin-1-yl)phenyl]propanamideHuman4128
CDK2CDKCMGC2btrAn-(5-isopropyl-thiazol-2-yl)-2-pyridin-3-yl-acetamideHuman3998
CDK2CDKCMGC2btsA4-[(5-isopropyl-1,3-thiazol-2-yl)amino]benzenesulfonamideHuman4443
CDK2CDKCMGC2c4gA(3z)-5-acetyl-3-(benzoylimino)-3,6-dihydropyrrolo[3,4-c]pyrazol-5-iumHuman4088
CDK2CDKCMGC2c4gC(3z)-5-acetyl-3-(benzoylimino)-3,6-dihydropyrrolo[3,4-c]pyrazol-5-iumHuman4453
CDK2CDKCMGC2c5nAAn-[4-(2,4-dimethyl-thiazol-5-yl)-pyrimidin-2-yl]-n',n'-dimethyl-benzene-1,4-diamineHuman4063
CDK2CDKCMGC2c5nABn-[4-(2,4-dimethyl-thiazol-5-yl)-pyrimidin-2-yl]-n',n'-dimethyl-benzene-1,4-diamineHuman4223
CDK2CDKCMGC2c5nCAn-[4-(2,4-dimethyl-thiazol-5-yl)-pyrimidin-2-yl]-n',n'-dimethyl-benzene-1,4-diamineHuman4161
CDK2CDKCMGC2c5nCBn-[4-(2,4-dimethyl-thiazol-5-yl)-pyrimidin-2-yl]-n',n'-dimethyl-benzene-1,4-diamineHuman3903
CDK2CDKCMGC2c5oAA4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-amineHuman4388
CDK2CDKCMGC2c5oAB4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-amineHuman4440
CDK2CDKCMGC2c5oCA4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-amineHuman4414
CDK2CDKCMGC2c5oCB4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-amineHuman4050
CDK2CDKCMGC2c5vAA4-(2,4-dimethyl-1,3-thiazol-5-yl)-n-[4-(trifluoromethyl)phenyl]pyrimidin-2-amineHuman4012
CDK2CDKCMGC2c5vAB4-(2,4-dimethyl-1,3-thiazol-5-yl)-n-[4-(trifluoromethyl)phenyl]pyrimidin-2-amineHuman4338
CDK2CDKCMGC2c5vCA4-(2,4-dimethyl-1,3-thiazol-5-yl)-n-[4-(trifluoromethyl)phenyl]pyrimidin-2-amineHuman4384
CDK2CDKCMGC2c5vCB4-(2,4-dimethyl-1,3-thiazol-5-yl)-n-[4-(trifluoromethyl)phenyl]pyrimidin-2-amineHuman4209
CDK2CDKCMGC2c5xAAhydroxy(oxo)(3-{[(2z)-4-[3-(1h-1,2,4-triazol-1-ylmethyl)phenyl]pyrimidin-2(5h)-ylidene]amino}phenyl)ammoniumHuman4312
CDK2CDKCMGC2c5xABhydroxy(oxo)(3-{[(2z)-4-[3-(1h-1,2,4-triazol-1-ylmethyl)phenyl]pyrimidin-2(5h)-ylidene]amino}phenyl)ammoniumHuman3892
CDK2CDKCMGC2c5xCAhydroxy(oxo)(3-{[(2z)-4-[3-(1h-1,2,4-triazol-1-ylmethyl)phenyl]pyrimidin-2(5h)-ylidene]amino}phenyl)ammoniumHuman4466
CDK2CDKCMGC2c5xCBhydroxy(oxo)(3-{[(2z)-4-[3-(1h-1,2,4-triazol-1-ylmethyl)phenyl]pyrimidin-2(5h)-ylidene]amino}phenyl)ammoniumHuman4418
CDK2CDKCMGC2c5yAAhydroxy(oxo)(3-{[(2z)-4-[3-(1h-1,2,4-triazol-1-ylmethyl)phenyl]pyrimidin-2(5h)-ylidene]amino}phenyl)ammoniumHuman6785
CDK2CDKCMGC2c5yABhydroxy(oxo)(3-{[(2z)-4-[3-(1h-1,2,4-triazol-1-ylmethyl)phenyl]pyrimidin-2(5h)-ylidene]amino}phenyl)ammoniumHuman6777
CDK2CDKCMGC2c68A(5z)-5-(3-bromocyclohexa-2,5-dien-1-ylidene)-n-(pyridin-4-ylmethyl)-1,5-dihydropyrazolo[1,5-a]pyrimidin-7-amineHuman6776
CDK2CDKCMGC2c69A(5z)-5-(3-bromocyclohexa-2,5-dien-1-ylidene)-n-(pyridin-4-ylmethyl)-1,5-dihydro[1,2,4]triazolo[1,5-a]pyrimidin-7-amineHuman6775
CDK2CDKCMGC2c6iA4-{[5-(cyclohexylmethoxy)[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]amino}benzenesulfonamideHuman6774
CDK2CDKCMGC2c6kA4-{[5-(cyclohexylamino)[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]amino}benzenesulfonamideHuman6773
CDK2CDKCMGC2c6lA4-({5-[(4-aminocyclohexyl)amino][1,2,4]triazolo[1,5-a]pyrimidin-7-yl}amino)benzenesulfonamideHuman6779
CDK2CDKCMGC2c6mA4-{[5-(cyclohexyloxy)[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]amino}benzenesulfonamideHuman6782
CDK2CDKCMGC2c6oAo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman6783
CDK2CDKCMGC2c6tA4-{[5-(cyclohexyloxy)[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]amino}benzenesulfonamideHuman4371
CDK2CDKCMGC2c6tC4-{[5-(cyclohexyloxy)[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]amino}benzenesulfonamideHuman3994
CDK2CDKCMGC2cchAAadenosine-5'-triphosphateHuman4303
CDK2CDKCMGC2cchABadenosine-5'-triphosphateHuman4553
CDK2CDKCMGC2cchAC-Human4566
CDK2CDKCMGC2cchCAadenosine-5'-triphosphateHuman3932
CDK2CDKCMGC2cchCBadenosine-5'-triphosphateHuman4000
CDK2CDKCMGC2cchCC-Human4431
CDK2CDKCMGC2cciAadenosine-5'-triphosphateHuman4373
CDK2CDKCMGC2cciCadenosine-5'-triphosphateHuman4532
CDK2CDKCMGC2cjmAadenosine-5'-triphosphateHuman4406
CDK2CDKCMGC2cjmCadenosine-5'-triphosphateHuman4126
CDK2CDKCMGC2clxAA4-[(e)-(3,5-diamino-1h-pyrazol-4-yl)diazenyl]phenolHuman3909
CDK2CDKCMGC2clxAB4-[(e)-(3,5-diamino-1h-pyrazol-4-yl)diazenyl]phenolHuman3880
CDK2CDKCMGC2ds1A(13r,15s)-13-methyl-16-oxa-8,9,12,22,24-pentaazahexacyclo[15.6.2.16,9.1,12,15.0,2,7.0,21,25]heptacosa-1(24),2,4,6,17(25),18,20-heptaene-23,26-dioneHuman4513
CDK2CDKCMGC2duvA2-(3,4-dihydroxyphenyl)-8-(1,1-dioxidoisothiazolidin-2-yl)-3-hydroxy-6-methyl-4h-chromen-4-oneHuman4193
CDK2CDKCMGC2exmAn-(3-methylbut-2-en-1-yl)-9h-purin-6-amineHuman4055
CDK2CDKCMGC2fvdA(4-amino-2-{[1-(methylsulfonyl)piperidin-4-yl]amino}pyrimidin-5-yl)(2,3-difluoro-6-methoxyphenyl)methanoneHuman4408
CDK2CDKCMGC2g9xA3-({2-[(4-{[6-(cyclohexylmethoxy)-9h-purin-2-yl]amino}phenyl)sulfonyl]ethyl}amino)propan-1-olHuman3883
CDK2CDKCMGC2g9xC3-({2-[(4-{[6-(cyclohexylmethoxy)-9h-purin-2-yl]amino}phenyl)sulfonyl]ethyl}amino)propan-1-olHuman4082
CDK2CDKCMGC2i40AA5-[5,6-bis(methyloxy)-1h-benzimidazol-1-yl]-3-{[1-(2-chlorophenyl)ethyl]oxy}-2-thiophenecarboxamideHuman4363
CDK2CDKCMGC2i40AB5-[5,6-bis(methyloxy)-1h-benzimidazol-1-yl]-3-{[1-(2-chlorophenyl)ethyl]oxy}-2-thiophenecarboxamideHuman4470
CDK2CDKCMGC2i40CA5-[5,6-bis(methyloxy)-1h-benzimidazol-1-yl]-3-{[1-(2-chlorophenyl)ethyl]oxy}-2-thiophenecarboxamideHuman4222
CDK2CDKCMGC2i40CB5-[5,6-bis(methyloxy)-1h-benzimidazol-1-yl]-3-{[1-(2-chlorophenyl)ethyl]oxy}-2-thiophenecarboxamideHuman4043
CDK2CDKCMGC2iw6A[(2-chloro-5-methylphenyl){6-[(4-{[(2r)-3-(dimethylamino)-2-hydroxypropyl]oxy}phenyl)amino]pyrimidin-4-yl}amino]acetonitrileHuman4019
CDK2CDKCMGC2iw6C[(2-chloro-5-methylphenyl){6-[(4-{[(2r)-3-(dimethylamino)-2-hydroxypropyl]oxy}phenyl)amino]pyrimidin-4-yl}amino]acetonitrileHuman4108
CDK2CDKCMGC2iw8AAo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman4142
CDK2CDKCMGC2iw8ABo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman4377
CDK2CDKCMGC2iw8CAo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman4294
CDK2CDKCMGC2iw8CBo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman4350
CDK2CDKCMGC2iw9AAo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman4174
CDK2CDKCMGC2iw9ABo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman3955
CDK2CDKCMGC2iw9CAo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman4218
CDK2CDKCMGC2iw9CBo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman3858
CDK2CDKCMGC2j9mAA6-bromo-13-thia-2,4,8,12,19-pentaazatricyclo[12.3.1.1~3,7~]nonadeca-1(18),3(19),4,6,14,16-hexaene 13,13-dioxideHuman4154
CDK2CDKCMGC2j9mAB6-bromo-13-thia-2,4,8,12,19-pentaazatricyclo[12.3.1.1~3,7~]nonadeca-1(18),3(19),4,6,14,16-hexaene 13,13-dioxideHuman4246
CDK2CDKCMGC2jgzA-Human4117
CDK2CDKCMGC2r3fAA5-(2,3-dichlorophenyl)-n-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amineHuman4175
CDK2CDKCMGC2r3fAB5-(2,3-dichlorophenyl)-n-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amineHuman4291
CDK2CDKCMGC2r3gAA6-(2-fluorophenyl)-n-(pyridin-3-ylmethyl)imidazo[1,2-a]pyrazin-8-amineHuman4276
CDK2CDKCMGC2r3gAB6-(2-fluorophenyl)-n-(pyridin-3-ylmethyl)imidazo[1,2-a]pyrazin-8-amineHuman3923
CDK2CDKCMGC2r3hAA3-methyl-n-(pyridin-4-ylmethyl)imidazo[1,2-a]pyrazin-8-amineHuman4152
CDK2CDKCMGC2r3hAB3-methyl-n-(pyridin-4-ylmethyl)imidazo[1,2-a]pyrazin-8-amineHuman3970
CDK2CDKCMGC2r3iAA5-(2-fluorophenyl)-n-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amineHuman4135
CDK2CDKCMGC2r3iAB5-(2-fluorophenyl)-n-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amineHuman4059
CDK2CDKCMGC2r3iAC-Human4317
CDK2CDKCMGC2r3jAA3-bromo-5-phenyl-n-(pyridin-3-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amineHuman4185
CDK2CDKCMGC2r3jAB3-bromo-5-phenyl-n-(pyridin-3-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amineHuman4544
CDK2CDKCMGC2r3kAA3-bromo-5-phenyl-n-(pyrimidin-5-ylmethyl)pyrazolo[1,5-a]pyridin-7-amineHuman3953
CDK2CDKCMGC2r3kAB3-bromo-5-phenyl-n-(pyrimidin-5-ylmethyl)pyrazolo[1,5-a]pyridin-7-amineHuman3876
CDK2CDKCMGC2r3kAC3-bromo-5-phenyl-n-(pyrimidin-5-ylmethyl)pyrazolo[1,5-a]pyridin-7-amineHuman4022
CDK2CDKCMGC2r3lAA3-bromo-6-phenyl-n-(pyrimidin-5-ylmethyl)imidazo[1,2-a]pyridin-8-amineHuman4200
CDK2CDKCMGC2r3lAB3-bromo-6-phenyl-n-(pyrimidin-5-ylmethyl)imidazo[1,2-a]pyridin-8-amineHuman4085
CDK2CDKCMGC2r3lAC3-bromo-6-phenyl-n-(pyrimidin-5-ylmethyl)imidazo[1,2-a]pyridin-8-amineHuman4496
CDK2CDKCMGC2r3mAAn-((2-aminopyrimidin-5-yl)methyl)-5-(2,6-difluorophenyl)-3-ethylpyrazolo[1,5-a]pyrimidin-7-amineHuman4286
CDK2CDKCMGC2r3mABn-((2-aminopyrimidin-5-yl)methyl)-5-(2,6-difluorophenyl)-3-ethylpyrazolo[1,5-a]pyrimidin-7-amineHuman4576
CDK2CDKCMGC2r3nAA3-cyclopropyl-5-phenyl-n-(pyridin-3-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amineHuman4101
CDK2CDKCMGC2r3nAB3-cyclopropyl-5-phenyl-n-(pyridin-3-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amineHuman4046
CDK2CDKCMGC2r3oAA(5-phenyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-3-yl)methanolHuman4147
CDK2CDKCMGC2r3oAB(5-phenyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-3-yl)methanolHuman4354
CDK2CDKCMGC2r3oAC(5-phenyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-3-yl)methanolHuman4229
CDK2CDKCMGC2r3pAA5-(2,3-dichlorophenyl)-n-(pyridin-4-ylmethyl)-3-thiocyanatopyrazolo[1,5-a]pyrimidin-7-amineHuman4176
CDK2CDKCMGC2r3pAB5-(2,3-dichlorophenyl)-n-(pyridin-4-ylmethyl)-3-thiocyanatopyrazolo[1,5-a]pyrimidin-7-amineHuman4392
CDK2CDKCMGC2r3qAA3-((3-bromo-5-o-tolylpyrazolo[1,5-a]pyrimidin-7-ylamino)methyl)pyridine 1-oxideHuman4038
CDK2CDKCMGC2r3qAB3-((3-bromo-5-o-tolylpyrazolo[1,5-a]pyrimidin-7-ylamino)methyl)pyridine 1-oxideHuman4459
CDK2CDKCMGC2r3qAC3-((3-bromo-5-o-tolylpyrazolo[1,5-a]pyrimidin-7-ylamino)methyl)pyridine 1-oxideHuman3976
CDK2CDKCMGC2r3rAA3-bromo-5-phenyl-n-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amineHuman4040
CDK2CDKCMGC2r3rAB3-bromo-5-phenyl-n-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amineHuman4215
CDK2CDKCMGC2r64An-[5-(1,1-dioxidoisothiazolidin-2-yl)-1h-indazol-3-yl]-2-(4-piperidin-1-ylphenyl)acetamideHuman4425
CDK2CDKCMGC2uueA4-methyl-5-{(2e)-2-[(4-morpholin-4-ylphenyl)imino]-2,5-dihydropyrimidin-4-yl}-1,3-thiazol-2-amineHuman4515
CDK2CDKCMGC2uueC4-methyl-5-{(2e)-2-[(4-morpholin-4-ylphenyl)imino]-2,5-dihydropyrimidin-4-yl}-1,3-thiazol-2-amineHuman4321
CDK2CDKCMGC2uzbAC4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]-2-furyl}-n-methylbenzenesulfonamideHuman4099
CDK2CDKCMGC2uzbAD4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]-2-furyl}-n-methylbenzenesulfonamideHuman3866
CDK2CDKCMGC2uzbCC4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]-2-furyl}-n-methylbenzenesulfonamideHuman4045
CDK2CDKCMGC2uzbCD4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]-2-furyl}-n-methylbenzenesulfonamideHuman4502
CDK2CDKCMGC2uzdA4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}benzenesulfonamideHuman3877
CDK2CDKCMGC2uzdC4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}benzenesulfonamideHuman3900
CDK2CDKCMGC2uzeA4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}benzoic acidHuman3949
CDK2CDKCMGC2uzeC4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}benzoic acidHuman4071
CDK2CDKCMGC2uzlA4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}-2-(trifluoromethyl)benzenesulfonamideHuman3917
CDK2CDKCMGC2uzlC4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}-2-(trifluoromethyl)benzenesulfonamideHuman4106
CDK2CDKCMGC2uznA4-{5-[(1z)-1-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)ethyl]-2-furyl}benzenesulfonamideHuman4064
CDK2CDKCMGC2uzoA4-{5-[(z)-(2,4-dioxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}benzenesulfonamideHuman3862
CDK2CDKCMGC2v0dA2-imino-5-(1-pyridin-2-yl-meth-(e)-ylidene)-1,3-thiazolidin-4-oneHuman4327
CDK2CDKCMGC2v22A-Human4077
CDK2CDKCMGC2v22C-Human4255
CDK2CDKCMGC2vtaA1h-indazoleHuman4118
CDK2CDKCMGC2vthA5-hydroxynaphthalene-1-sulfonamideHuman4274
CDK2CDKCMGC2vtiAn-(4-sulfamoylphenyl)-1h-indazole-3-carboxamideHuman4177
CDK2CDKCMGC2vtjA4-[(6-chloropyrazin-2-yl)amino]benzenesulfonamideHuman3959
CDK2CDKCMGC2vtlAn-phenyl-1h-pyrazole-3-carboxamideHuman3870
CDK2CDKCMGC2vtmApyrazolo[1,5-a]pyrimidine-3-carbonitrileHuman4283
CDK2CDKCMGC2vtnA4-(acetylamino)-n-(4-fluorophenyl)-1h-pyrazole-3-carboxamideHuman4027
CDK2CDKCMGC2vtoAAn-(4-fluorophenyl)-4-[(phenylcarbonyl)amino]-1h-pyrazole-3-carboxamideHuman4421
CDK2CDKCMGC2vtoABn-(4-fluorophenyl)-4-[(phenylcarbonyl)amino]-1h-pyrazole-3-carboxamideHuman3946
CDK2CDKCMGC2vtpAA{[(2,6-difluorophenyl)carbonyl]amino}-n-(4-fluorophenyl)-1h-pyrazole-3-carboxamideHuman4511
CDK2CDKCMGC2vtpAB{[(2,6-difluorophenyl)carbonyl]amino}-n-(4-fluorophenyl)-1h-pyrazole-3-carboxamideHuman4401
CDK2CDKCMGC2vtqA{[(2,6-difluorophenyl)carbonyl]amino}-n-piperidin-4-yl-1h-pyrazole-3-carboxamideHuman3891
CDK2CDKCMGC2vtrAA5-chloro-7-[(1-methylethyl)amino]pyrazolo[1,5-a]pyrimidine-3-carbonitrileHuman4391
CDK2CDKCMGC2vtrAB5-chloro-7-[(1-methylethyl)amino]pyrazolo[1,5-a]pyrimidine-3-carbonitrileHuman3907
CDK2CDKCMGC2vtsA5-[(4-aminocyclohexyl)amino]-7-(propan-2-ylamino)pyrazolo[1,5-a]pyrimidine-3-carbonitrileHuman4300
CDK2CDKCMGC2vttA4-{[(2,6-difluorophenyl)carbonyl]amino}-n-[(3s)-piperidin-3-yl]-1h-pyrazole-3-carboxamideHuman4100
CDK2CDKCMGC2vu3AA4-{[(2,6-dichlorophenyl)carbonyl]amino}-n-piperidin-4-yl-1h-pyrazole-3-carboxamideHuman4582
CDK2CDKCMGC2vu3AB4-{[(2,6-dichlorophenyl)carbonyl]amino}-n-piperidin-4-yl-1h-pyrazole-3-carboxamideHuman3884
CDK2CDKCMGC2vv9AA2-{4-[4-({4-[2-methyl-1-(1-methylethyl)-1h-imidazol-5-yl]pyrimidin-2-yl}amino)phenyl]piperazin-1-yl}-2-oxoethanolHuman3989
CDK2CDKCMGC2vv9AB2-{4-[4-({4-[2-methyl-1-(1-methylethyl)-1h-imidazol-5-yl]pyrimidin-2-yl}amino)phenyl]piperazin-1-yl}-2-oxoethanolHuman3881
CDK2CDKCMGC2w05AAn-(2-methoxyethyl)-4-({4-[2-methyl-1-(1-methylethyl)-1h-imidazol-5-yl]pyrimidin-2-yl}amino)benzenesulfonamideHuman4547
CDK2CDKCMGC2w05ABn-(2-methoxyethyl)-4-({4-[2-methyl-1-(1-methylethyl)-1h-imidazol-5-yl]pyrimidin-2-yl}amino)benzenesulfonamideHuman4256
CDK2CDKCMGC2w06A4-{[4-(1-cyclopropyl-2-methyl-1h-imidazol-5-yl)pyrimidin-2-yl]amino}-n-methylbenzenesulfonamideHuman3982
CDK2CDKCMGC2w17AAn-(4-{[(3s)-3-(dimethylamino)pyrrolidin-1-yl]carbonyl}phenyl)-5-fluoro-4-[2-methyl-1-(1-methylethyl)-1h-imidazol-5-yl]pyrimidin-2-amineHuman3968
CDK2CDKCMGC2w17ABn-(4-{[(3s)-3-(dimethylamino)pyrrolidin-1-yl]carbonyl}phenyl)-5-fluoro-4-[2-methyl-1-(1-methylethyl)-1h-imidazol-5-yl]pyrimidin-2-amineHuman4165
CDK2CDKCMGC2w1hAn-[3-(1h-benzimidazol-2-yl)-1h-pyrazol-4-yl]benzamideHuman4228
CDK2CDKCMGC2wevAA[4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amineHuman4067
CDK2CDKCMGC2wevAB[4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amineHuman4580
CDK2CDKCMGC2wevAC[4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amineHuman4007
CDK2CDKCMGC2wevCA[4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amineHuman4503
CDK2CDKCMGC2wevCB[4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amineHuman3859
CDK2CDKCMGC2wevCC[4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amineHuman4288
CDK2CDKCMGC2wfyAA-Human4324
CDK2CDKCMGC2wfyAB-Human4426
CDK2CDKCMGC2wfyCA-Human4329
CDK2CDKCMGC2wfyCB-Human4096
CDK2CDKCMGC2whbAA-Human4471
CDK2CDKCMGC2whbAB-Human4457
CDK2CDKCMGC2whbCA-Human4132
CDK2CDKCMGC2whbCB-Human4352
CDK2CDKCMGC2wihAn,1,4,4-tetramethyl-8-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxamideHuman4163
CDK2CDKCMGC2wihCn,1,4,4-tetramethyl-8-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxamideHuman4119
CDK2CDKCMGC2wipA1-methyl-8-(phenylamino)-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxylic acidHuman4520
CDK2CDKCMGC2wipC1-methyl-8-(phenylamino)-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxylic acidHuman4190
CDK2CDKCMGC2wmaA-Human4435
CDK2CDKCMGC2wmaC-Human4410
CDK2CDKCMGC2wmbA-Human4060
CDK2CDKCMGC2wmbC-Human4474
CDK2CDKCMGC2wpaAn-{6,6-dimethyl-5-[(1-methylpiperidin-4-yl)carbonyl]-1,4,5,6-tetrahydropyrrolo[3,4-c]pyrazol-3-yl}-3-methylbutanamideHuman4399
CDK2CDKCMGC2wpaCn-{6,6-dimethyl-5-[(1-methylpiperidin-4-yl)carbonyl]-1,4,5,6-tetrahydropyrrolo[3,4-c]pyrazol-3-yl}-3-methylbutanamideHuman4162
CDK2CDKCMGC2wxvAn,1-dimethyl-8-{[1-(methylsulfonyl)piperidin-4-yl]amino}-1h-pyrazolo[4,3-h]quinazoline-3-carboxamideHuman4318
CDK2CDKCMGC2wxvCn,1-dimethyl-8-{[1-(methylsulfonyl)piperidin-4-yl]amino}-1h-pyrazolo[4,3-h]quinazoline-3-carboxamideHuman4504
CDK2CDKCMGC2x1nAA2-methyl-n-[(1z)-3-nitrocyclohexa-2,4-dien-1-ylidene]-4,5-dihydro[1,3]thiazolo[4,5-h]quinazolin-8-amineHuman4579
CDK2CDKCMGC2x1nAB2-methyl-n-[(1z)-3-nitrocyclohexa-2,4-dien-1-ylidene]-4,5-dihydro[1,3]thiazolo[4,5-h]quinazolin-8-amineHuman4078
CDK2CDKCMGC2x1nCA2-methyl-n-[(1z)-3-nitrocyclohexa-2,4-dien-1-ylidene]-4,5-dihydro[1,3]thiazolo[4,5-h]quinazolin-8-amineHuman3991
CDK2CDKCMGC2x1nCB2-methyl-n-[(1z)-3-nitrocyclohexa-2,4-dien-1-ylidene]-4,5-dihydro[1,3]thiazolo[4,5-h]quinazolin-8-amineHuman4062
CDK2CDKCMGC2xmyAA4-[4-(3,4-dimethyl-2-oxo-2,3-dihydro-thiazol-5-yl)-pyrimidin-2-ylamino]-n-(2-methoxy-ethyl)-benzenesulfonamideHuman4526
CDK2CDKCMGC2xmyAB4-[4-(3,4-dimethyl-2-oxo-2,3-dihydro-thiazol-5-yl)-pyrimidin-2-ylamino]-n-(2-methoxy-ethyl)-benzenesulfonamideHuman3985
CDK2CDKCMGC2xnbAA3,4-dimethyl-5-(2-{[(1z)-4-piperazin-1-ylcyclohexa-2,4-dien-1-ylidene]amino}pyrimidin-4-yl)-1,3-thiazol-2(3h)-oneHuman4217
CDK2CDKCMGC2xnbAB3,4-dimethyl-5-(2-{[(1z)-4-piperazin-1-ylcyclohexa-2,4-dien-1-ylidene]amino}pyrimidin-4-yl)-1,3-thiazol-2(3h)-oneHuman4034
CDK2CDKCMGC3bhtAA4-(4-methoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHuman3950
CDK2CDKCMGC3bhtAB4-(4-methoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHuman4491
CDK2CDKCMGC3bhtCA4-(4-methoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHuman4151
CDK2CDKCMGC3bhtCB4-(4-methoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHuman3889
CDK2CDKCMGC3bhuAA4-(4-propoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHuman4105
CDK2CDKCMGC3bhuAB4-(4-propoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHuman4446
CDK2CDKCMGC3bhuCA4-(4-propoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHuman4087
CDK2CDKCMGC3bhuCB4-(4-propoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHuman4464
CDK2CDKCMGC3bhvAA9-amino-5-(2-aminopyrimidin-4-yl)pyrido[3',2':4,5]pyrrolo[1,2-c]pyrimidin-4-olHuman4531
CDK2CDKCMGC3bhvAB9-amino-5-(2-aminopyrimidin-4-yl)pyrido[3',2':4,5]pyrrolo[1,2-c]pyrimidin-4-olHuman4001
CDK2CDKCMGC3bhvCA9-amino-5-(2-aminopyrimidin-4-yl)pyrido[3',2':4,5]pyrrolo[1,2-c]pyrimidin-4-olHuman4353
CDK2CDKCMGC3bhvCB9-amino-5-(2-aminopyrimidin-4-yl)pyrido[3',2':4,5]pyrrolo[1,2-c]pyrimidin-4-olHuman4529
CDK2CDKCMGC3ddpAA(2r)-2-({9-(1-methylethyl)-6-[(4-pyridin-2-ylbenzyl)amino]-9h-purin-2-yl}amino)butan-1-olHuman6781
CDK2CDKCMGC3ddpAB(2r)-2-({9-(1-methylethyl)-6-[(4-pyridin-2-ylbenzyl)amino]-9h-purin-2-yl}amino)butan-1-olHuman6780
CDK2CDKCMGC3ddpCA(2r)-2-({9-(1-methylethyl)-6-[(4-pyridin-2-ylbenzyl)amino]-9h-purin-2-yl}amino)butan-1-olHuman6784
CDK2CDKCMGC3ddpCB(2r)-2-({9-(1-methylethyl)-6-[(4-pyridin-2-ylbenzyl)amino]-9h-purin-2-yl}amino)butan-1-olHuman6778
CDK2CDKCMGC3ddqAAr-roscovitineHuman4477
CDK2CDKCMGC3ddqABr-roscovitineHuman4269
CDK2CDKCMGC3ddqCAr-roscovitineHuman4364
CDK2CDKCMGC3ddqCBr-roscovitineHuman4289
CDK2CDKCMGC3dogAA(2r)-2-{[4-(benzylamino)-8-(1-methylethyl)pyrazolo[1,5-a][1,3,5]triazin-2-yl]amino}butan-1-olHuman4541
CDK2CDKCMGC3dogAB(2r)-2-{[4-(benzylamino)-8-(1-methylethyl)pyrazolo[1,5-a][1,3,5]triazin-2-yl]amino}butan-1-olHuman4365
CDK2CDKCMGC3dogCA(2r)-2-{[4-(benzylamino)-8-(1-methylethyl)pyrazolo[1,5-a][1,3,5]triazin-2-yl]amino}butan-1-olHuman4382
CDK2CDKCMGC3dogCB(2r)-2-{[4-(benzylamino)-8-(1-methylethyl)pyrazolo[1,5-a][1,3,5]triazin-2-yl]amino}butan-1-olHuman4121
CDK2CDKCMGC3eidAA(2s)-1-(dimethylamino)-3-(4-{[4-(6-morpholin-4-ylpyrazolo[1,5-b]pyridazin-3-yl)pyrimidin-2-yl]amino}phenoxy)propan-2-olHuman4386
CDK2CDKCMGC3eidAB(2s)-1-(dimethylamino)-3-(4-{[4-(6-morpholin-4-ylpyrazolo[1,5-b]pyridazin-3-yl)pyrimidin-2-yl]amino}phenoxy)propan-2-olHuman4424
CDK2CDKCMGC3eidCA-Human4072
CDK2CDKCMGC3eidCB-Human4467
CDK2CDKCMGC3ej1An-cyclopropyl-4-pyrazolo[1,5-b]pyridazin-3-ylpyrimidin-2-amineHuman4168
CDK2CDKCMGC3ej1Cn-cyclopropyl-4-pyrazolo[1,5-b]pyridazin-3-ylpyrimidin-2-amineHuman4092
CDK2CDKCMGC3eocA5-methyl-7-phenyl-n-(3,4,5-trimethoxyphenyl)imidazo[5,1-f][1,2,4]triazin-2-amineHuman4390
CDK2CDKCMGC3eocC5-methyl-7-phenyl-n-(3,4,5-trimethoxyphenyl)imidazo[5,1-f][1,2,4]triazin-2-amineHuman3969
CDK2CDKCMGC3ezrA3-methoxy-4-{3-[4-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]-1h-indazol-6-yl}anilineHuman4475
CDK2CDKCMGC3ezvA4-{3-[7-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]-1h-indazol-6-yl}anilineHuman4083
CDK2CDKCMGC3f5xA4-{3-[7-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]-1h-indazol-6-yl}anilineHuman3882
CDK2CDKCMGC3f5xC4-{3-[7-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]-1h-indazol-6-yl}anilineHuman3894
CDK2CDKCMGC3fz1A(3r)-3-(aminomethyl)-9-methoxy-1,2,3,4-tetrahydro-5h-[1]benzothieno[3,2-e][1,4]diazepin-5-oneHuman4335
CDK2CDKCMGC3ig7An-{1-[cis-3-(acetylamino)cyclobutyl]-1h-imidazol-4-yl}-2-(4-methoxyphenyl)acetamideHuman4021
CDK2CDKCMGC3iggAn-[1-(cis-3-hydroxycyclobutyl)-1h-imidazol-4-yl]-2-(4-methoxyphenyl)acetamideHuman4360
CDK2CDKCMGC3le6A5-(2-chlorophenyl)-3-methyl-7-nitropyrazolo[3,4-b][1,4]benzodiazepineHuman4125
CDK2CDKCMGC3lfnAn-[6-(4-hydroxyphenyl)-5-phenyl-1h-indazol-3-yl]butanamideHuman4330
CDK2CDKCMGC3lfqAn-(6,7-difluoro-5-phenyl-1h-indazol-3-yl)butanamideHuman4320
CDK2CDKCMGC3lfsAn-(6-chloro-5-phenyl-1h-indazol-3-yl)butanamideHuman4069
CDK2CDKCMGC3my5AA5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazoleHuman4554
CDK2CDKCMGC3my5AB5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazoleHuman3887
CDK2CDKCMGC3my5AC5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazoleHuman3910
CDK2CDKCMGC3my5CA5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazoleHuman4473
CDK2CDKCMGC3my5CB5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazoleHuman4003
CDK2CDKCMGC3my5CC5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazoleHuman3929
CDK2CDKCMGC3ns9A(2s,3s)-3-{[7-(benzylamino)-3-(1-methylethyl)pyrazolo[1,5-a]pyrimidin-5-yl]amino}butane-1,2,4-triolHuman4575
CDK2CDKCMGC3pj8AA(2r)-2-{[7-(benzylamino)-3-(propan-2-yl)-1h-pyrazolo[4,3-d]pyrimidin-5-yl]amino}butan-1-olHuman4375
CDK2CDKCMGC3pj8AB(2r)-2-{[7-(benzylamino)-3-(propan-2-yl)-1h-pyrazolo[4,3-d]pyrimidin-5-yl]amino}butan-1-olHuman4454
CDK2CDKCMGC3pxfAA8-anilino-1-naphthalene sulfonateHuman4047
CDK2CDKCMGC3pxfAB8-anilino-1-naphthalene sulfonateHuman4301
CDK2CDKCMGC3pxqA8-anilino-1-naphthalene sulfonateHuman3947
CDK2CDKCMGC3pxrAA-Human3941
CDK2CDKCMGC3pxrAB-Human4173
CDK2CDKCMGC3pxyAA2-(4,6-diamino-1,3,5-triazin-2-yl)-4-methoxyphenolHuman4057
CDK2CDKCMGC3pxyAB2-(4,6-diamino-1,3,5-triazin-2-yl)-4-methoxyphenolHuman3904
CDK2CDKCMGC3pxzA8-anilino-1-naphthalene sulfonateHuman4251
CDK2CDKCMGC3py0AA(3z)-3-(1h-imidazol-5-ylmethylene)-5-methoxy-1h-indol-2(3h)-oneHuman3995
CDK2CDKCMGC3py0AB(3z)-3-(1h-imidazol-5-ylmethylene)-5-methoxy-1h-indol-2(3h)-oneHuman3869
CDK2CDKCMGC3py1AA(3z)-3-(1h-imidazol-5-ylmethylene)-5-methoxy-1h-indol-2(3h)-oneHuman4361
CDK2CDKCMGC3py1AB(3z)-3-(1h-imidazol-5-ylmethylene)-5-methoxy-1h-indol-2(3h)-oneHuman4444
CDK2CDKCMGC3qhrAadenosine-5'-diphosphateHuman4458
CDK2CDKCMGC3qhrCadenosine-5'-diphosphateHuman3879
CDK2CDKCMGC3qhwAAadenosine-5'-diphosphateHuman4346
CDK2CDKCMGC3qhwABadenosine-5'-diphosphateHuman4156
CDK2CDKCMGC3qhwCAadenosine-5'-diphosphateHuman4129
CDK2CDKCMGC3qhwCBadenosine-5'-diphosphateHuman4143
CDK2CDKCMGC3ql8AA3-(4-amino-1,3,5-triazin-2-yl)-4-hydroxybenzonitrileHuman3916
CDK2CDKCMGC3ql8AB3-(4-amino-1,3,5-triazin-2-yl)-4-hydroxybenzonitrileHuman4306
CDK2CDKCMGC3qqfAA5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman4211
CDK2CDKCMGC3qqfAB5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman4287
CDK2CDKCMGC3qqgAA4-chloro-2-(4,6-diamino-1,3,5-triazin-2-yl)phenolHuman4130
CDK2CDKCMGC3qqgAB4-chloro-2-(4,6-diamino-1,3,5-triazin-2-yl)phenolHuman4310
CDK2CDKCMGC3qqhAA2-[4-amino-6-(phenylamino)-1,3,5-triazin-2-yl]-4-chlorophenolHuman4393
CDK2CDKCMGC3qqhAB2-[4-amino-6-(phenylamino)-1,3,5-triazin-2-yl]-4-chlorophenolHuman4533
CDK2CDKCMGC3qqjAA2-(4,6-diamino-1,3,5-triazin-2-yl)phenolHuman4113
CDK2CDKCMGC3qqjAB2-(4,6-diamino-1,3,5-triazin-2-yl)phenolHuman4204
CDK2CDKCMGC3qqkAA[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](phenyl)methanoneHuman4568
CDK2CDKCMGC3qqkAB[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](phenyl)methanoneHuman4514
CDK2CDKCMGC3qqlAA(5r)-5-(2-methylbutan-2-yl)-4,5,6,7-tetrahydro-1h-indazole-3-carbohydrazideHuman4341
CDK2CDKCMGC3qqlAB(5r)-5-(2-methylbutan-2-yl)-4,5,6,7-tetrahydro-1h-indazole-3-carbohydrazideHuman4378
CDK2CDKCMGC3qrtAA(5r)-5-(2-methylbutan-2-yl)-n-(4-sulfamoylbenzyl)-4,5,6,7-tetrahydro-2h-indazole-3-carboxamideHuman4586
CDK2CDKCMGC3qrtAB(5r)-5-(2-methylbutan-2-yl)-n-(4-sulfamoylbenzyl)-4,5,6,7-tetrahydro-2h-indazole-3-carboxamideHuman4536
CDK2CDKCMGC3qruAA(5s)-n-methyl-5-(2-methylbutan-2-yl)-4,5,6,7-tetrahydro-2h-indazole-3-carboxamideHuman4237
CDK2CDKCMGC3qruAB(5s)-n-methyl-5-(2-methylbutan-2-yl)-4,5,6,7-tetrahydro-2h-indazole-3-carboxamideHuman4516
CDK2CDKCMGC3qtqAA[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](pyridin-3-yl)methanoneHuman4210
CDK2CDKCMGC3qtqAB[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](pyridin-3-yl)methanoneHuman4103
CDK2CDKCMGC3qtrAA[4-amino-2-(phenylamino)-1,3-thiazol-5-yl](phenyl)methanoneHuman3874
CDK2CDKCMGC3qtrAB[4-amino-2-(phenylamino)-1,3-thiazol-5-yl](phenyl)methanoneHuman4243
CDK2CDKCMGC3qtsAA[4-amino-2-(phenylamino)-1,3-thiazol-5-yl](3-methoxyphenyl)methanoneHuman4275
CDK2CDKCMGC3qtsAB[4-amino-2-(phenylamino)-1,3-thiazol-5-yl](3-methoxyphenyl)methanoneHuman4564
CDK2CDKCMGC3qtuAA4-{[4-amino-5-(4-sulfamoylbenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4009
CDK2CDKCMGC3qtuAB4-{[4-amino-5-(4-sulfamoylbenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4323
CDK2CDKCMGC3qtwAA[4-amino-2-(phenylamino)-1,3-thiazol-5-yl](pyridin-3-yl)methanoneHuman4397
CDK2CDKCMGC3qtwAB[4-amino-2-(phenylamino)-1,3-thiazol-5-yl](pyridin-3-yl)methanoneHuman3890
CDK2CDKCMGC3qtxAA4-{[4-amino-5-(3-nitrobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4339
CDK2CDKCMGC3qtxAB4-{[4-amino-5-(3-nitrobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4419
CDK2CDKCMGC3qtzAA4-{[4-amino-5-(3-fluorobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4109
CDK2CDKCMGC3qtzAB4-{[4-amino-5-(3-fluorobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4337
CDK2CDKCMGC3qu0AA4-{[4-amino-5-(pyridin-3-ylcarbonyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4427
CDK2CDKCMGC3qu0AB4-{[4-amino-5-(pyridin-3-ylcarbonyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4558
CDK2CDKCMGC3qwjAA2-{[(2-aminopyrimidin-5-yl)methyl]amino}-4-chloro-5-nitrobenzamideHuman4265
CDK2CDKCMGC3qwjAB2-{[(2-aminopyrimidin-5-yl)methyl]amino}-4-chloro-5-nitrobenzamideHuman4182
CDK2CDKCMGC3qwkAA4-chloro-2-{[(2-chloropyrimidin-5-yl)methyl]amino}-5-nitrobenzamideHuman4091
CDK2CDKCMGC3qwkAB4-chloro-2-{[(2-chloropyrimidin-5-yl)methyl]amino}-5-nitrobenzamideHuman4155
CDK2CDKCMGC3qx2AA2-{[(2-aminopyrimidin-5-yl)methyl]amino}-4-[(2-hydroxyethyl)amino]-5-nitrobenzamideHuman4031
CDK2CDKCMGC3qx2AB2-{[(2-aminopyrimidin-5-yl)methyl]amino}-4-[(2-hydroxyethyl)amino]-5-nitrobenzamideHuman4297
CDK2CDKCMGC3qx4AA4-chloro-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman4409
CDK2CDKCMGC3qx4AB4-chloro-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman3990
CDK2CDKCMGC3qxoA5-nitro-2-[(4-sulfamoylbenzyl)amino]benzamideHuman4282
CDK2CDKCMGC3qxpAA4-{[4-amino-5-(2-nitrobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4343
CDK2CDKCMGC3qxpAB4-{[4-amino-5-(2-nitrobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4482
CDK2CDKCMGC3qzfA2-(4,6-diamino-1,3,5-triazin-2-yl)benzene-1,4-diolHuman4569
CDK2CDKCMGC3qzgAA2-(4,6-diamino-1,3,5-triazin-2-yl)-4-fluorophenolHuman4144
CDK2CDKCMGC3qzgAB2-(4,6-diamino-1,3,5-triazin-2-yl)-4-fluorophenolHuman4347
CDK2CDKCMGC3qzhA4-methoxy-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman3954
CDK2CDKCMGC3qziAA4-chloro-5-nitro-2-[(pyrimidin-5-ylmethyl)amino]benzamideHuman4094
CDK2CDKCMGC3qziAB4-chloro-5-nitro-2-[(pyrimidin-5-ylmethyl)amino]benzamideHuman4500
CDK2CDKCMGC3r1qAA4-chloro-2-{[(6-chloropyridin-3-yl)methyl]amino}-5-nitrobenzamideHuman4224
CDK2CDKCMGC3r1qAB4-chloro-2-{[(6-chloropyridin-3-yl)methyl]amino}-5-nitrobenzamideHuman4507
CDK2CDKCMGC3r1sAA2-{[(6-chloropyridin-3-yl)methyl]amino}-5-nitrobenzamideHuman4263
CDK2CDKCMGC3r1sAB2-{[(6-chloropyridin-3-yl)methyl]amino}-5-nitrobenzamideHuman4358
CDK2CDKCMGC3r1yAA2-[(pyridin-3-ylmethyl)amino]benzamideHuman4319
CDK2CDKCMGC3r1yAB2-[(pyridin-3-ylmethyl)amino]benzamideHuman4405
CDK2CDKCMGC3r28AA4-chloro-5-nitro-2-[(3,4,5-trifluorobenzyl)amino]benzamideHuman4052
CDK2CDKCMGC3r28AB4-chloro-5-nitro-2-[(3,4,5-trifluorobenzyl)amino]benzamideHuman4293
CDK2CDKCMGC3r6xAA4-[(3-hydroxypropyl)amino]-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman4398
CDK2CDKCMGC3r6xAB4-[(3-hydroxypropyl)amino]-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman4107
CDK2CDKCMGC3r71AA4-[(3-methoxypropyl)amino]-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman3962
CDK2CDKCMGC3r71AB4-[(3-methoxypropyl)amino]-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman4345
CDK2CDKCMGC3r73AA4-[(3-aminopropyl)amino]-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman4187
CDK2CDKCMGC3r73AB4-[(3-aminopropyl)amino]-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman3899
CDK2CDKCMGC3r7eAA5-nitro-2-[(pyrazin-2-ylmethyl)amino]benzamideHuman4159
CDK2CDKCMGC3r7eAB5-nitro-2-[(pyrazin-2-ylmethyl)amino]benzamideHuman4447
CDK2CDKCMGC3r7iAA4-{[(2-carbamoyl-4-nitrophenyl)amino]methyl}benzoic acidHuman4450
CDK2CDKCMGC3r7iAB4-{[(2-carbamoyl-4-nitrophenyl)amino]methyl}benzoic acidHuman4070
CDK2CDKCMGC3r7uAA2-{[4-(aminomethyl)benzyl]amino}-5-nitrobenzamideHuman4510
CDK2CDKCMGC3r7uAB2-{[4-(aminomethyl)benzyl]amino}-5-nitrobenzamideHuman4023
CDK2CDKCMGC3r7vAA5-nitro-2-[(pyridin-2-ylmethyl)amino]benzamideHuman4380
CDK2CDKCMGC3r7vAB5-nitro-2-[(pyridin-2-ylmethyl)amino]benzamideHuman4183
CDK2CDKCMGC3r7yAA2-{[(2-aminopyrimidin-5-yl)methyl]amino}-4-(morpholin-4-yl)-5-nitrobenzamideHuman4476
CDK2CDKCMGC3r7yAB2-{[(2-aminopyrimidin-5-yl)methyl]amino}-4-(morpholin-4-yl)-5-nitrobenzamideHuman3975
CDK2CDKCMGC3r83AA4-(4-aminopiperidin-1-yl)-2-{[(2-aminopyrimidin-5-yl)methyl]amino}-5-nitrobenzamideHuman4234
CDK2CDKCMGC3r83AB4-(4-aminopiperidin-1-yl)-2-{[(2-aminopyrimidin-5-yl)methyl]amino}-5-nitrobenzamideHuman4543
CDK2CDKCMGC3r8lAA(5r)-5-tert-butyl-4,5,6,7-tetrahydro-1h-indazole-3-carbohydrazideHuman4186
CDK2CDKCMGC3r8lAB(5r)-5-tert-butyl-4,5,6,7-tetrahydro-1h-indazole-3-carbohydrazideHuman4523
CDK2CDKCMGC3r8mAA1h-indazole-3-carbohydrazideHuman4111
CDK2CDKCMGC3r8mAB1h-indazole-3-carbohydrazideHuman4451
CDK2CDKCMGC3r8pAA(5r)-5-propyl-4,5,6,7-tetrahydro-1h-indazole-3-carbohydrazideHuman4232
CDK2CDKCMGC3r8pAB(5r)-5-propyl-4,5,6,7-tetrahydro-1h-indazole-3-carbohydrazideHuman4538
CDK2CDKCMGC3r8uAA[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](naphthalen-2-yl)methanoneHuman3926
CDK2CDKCMGC3r8uAB[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](naphthalen-2-yl)methanoneHuman3864
CDK2CDKCMGC3r8vAA[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](3-nitrophenyl)methanoneHuman3938
CDK2CDKCMGC3r8vAB[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](3-nitrophenyl)methanoneHuman4191
CDK2CDKCMGC3r8zAA[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](pyridin-4-yl)methanoneHuman4137
CDK2CDKCMGC3r8zAB[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](pyridin-4-yl)methanoneHuman4140
CDK2CDKCMGC3r9dAA4-amino-n-(3-fluorophenyl)-2-[(4-sulfamoylphenyl)amino]-1,3-thiazole-5-carboxamideHuman4562
CDK2CDKCMGC3r9dAB4-amino-n-(3-fluorophenyl)-2-[(4-sulfamoylphenyl)amino]-1,3-thiazole-5-carboxamideHuman4565
CDK2CDKCMGC3r9hAA4-amino-n-(2,6-difluorophenyl)-2-[(4-sulfamoylphenyl)amino]-1,3-thiazole-5-carboxamideHuman3958
CDK2CDKCMGC3r9hAB4-amino-n-(2,6-difluorophenyl)-2-[(4-sulfamoylphenyl)amino]-1,3-thiazole-5-carboxamideHuman4336
CDK2CDKCMGC3r9nAA[4-amino-2-(cyclohexylamino)-1,3-thiazol-5-yl](3-nitrophenyl)methanoneHuman3885
CDK2CDKCMGC3r9nAB[4-amino-2-(cyclohexylamino)-1,3-thiazol-5-yl](3-nitrophenyl)methanoneHuman3867
CDK2CDKCMGC3r9oA4-amino-n-(3,5-difluorophenyl)-2-[(4-sulfamoylphenyl)amino]-1,3-thiazole-5-carboxamideHuman4279
CDK2CDKCMGC3rahAA[4-amino-2-(cyclohexylamino)-1,3-thiazol-5-yl](naphthalen-2-yl)methanoneHuman4438
CDK2CDKCMGC3rahAB[4-amino-2-(cyclohexylamino)-1,3-thiazol-5-yl](naphthalen-2-yl)methanoneHuman4206
CDK2CDKCMGC3raiAA4-{[3-(morpholin-4-yl)propyl]amino}-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman4441
CDK2CDKCMGC3raiAB4-{[3-(morpholin-4-yl)propyl]amino}-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman4002
CDK2CDKCMGC3rakAA4-[(4-amino-5-benzoyl-1,3-thiazol-2-yl)amino]benzenesulfonamideHuman4574
CDK2CDKCMGC3rakAB4-[(4-amino-5-benzoyl-1,3-thiazol-2-yl)amino]benzenesulfonamideHuman4331
CDK2CDKCMGC3ralAA4-{[4-amino-5-(3-methoxybenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4017
CDK2CDKCMGC3ralAB4-{[4-amino-5-(3-methoxybenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman3984
CDK2CDKCMGC3rjcAA{4-amino-2-[(3-fluorophenyl)amino]-1,3-thiazol-5-yl}(phenyl)methanoneHuman4032
CDK2CDKCMGC3rjcAB{4-amino-2-[(3-fluorophenyl)amino]-1,3-thiazol-5-yl}(phenyl)methanoneHuman4469
CDK2CDKCMGC3rk5A4-{[4-amino-5-(pyridin-3-ylcarbonyl)-1,3-thiazol-2-yl]amino}benzoic acidHuman4160
CDK2CDKCMGC3rk7A4-{[4-amino-5-(pyridin-3-ylcarbonyl)-1,3-thiazol-2-yl]amino}benzamideHuman4236
CDK2CDKCMGC3rk9AA[4-amino-2-(propan-2-ylamino)-1,3-thiazol-5-yl](pyridin-3-yl)methanoneHuman4158
CDK2CDKCMGC3rk9AB[4-amino-2-(propan-2-ylamino)-1,3-thiazol-5-yl](pyridin-3-yl)methanoneHuman4259
CDK2CDKCMGC3rkbAA[4-amino-2-(cyclohexylamino)-1,3-thiazol-5-yl](pyridin-3-yl)methanoneHuman4460
CDK2CDKCMGC3rkbAB[4-amino-2-(cyclohexylamino)-1,3-thiazol-5-yl](pyridin-3-yl)methanoneHuman4039
CDK2CDKCMGC3rm6AA2-{[(2-aminopyrimidin-5-yl)methyl]amino}-5-nitro-4-{[2-(piperazin-1-yl)ethyl]amino}benzamideHuman4262
CDK2CDKCMGC3rm6AB2-{[(2-aminopyrimidin-5-yl)methyl]amino}-5-nitro-4-{[2-(piperazin-1-yl)ethyl]amino}benzamideHuman4357
CDK2CDKCMGC3rm7AA2-[(4-hydroxybenzyl)amino]-5-nitrobenzamideHuman3893
CDK2CDKCMGC3rm7AB2-[(4-hydroxybenzyl)amino]-5-nitrobenzamideHuman4499
CDK2CDKCMGC3rmfAA4-{[4-amino-5-(naphthalen-2-ylcarbonyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman3873
CDK2CDKCMGC3rmfAB4-{[4-amino-5-(naphthalen-2-ylcarbonyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4014
CDK2CDKCMGC3rniAA3-[(4-amino-5-benzoyl-1,3-thiazol-2-yl)amino]benzenesulfonamideHuman3993
CDK2CDKCMGC3rniAB3-[(4-amino-5-benzoyl-1,3-thiazol-2-yl)amino]benzenesulfonamideHuman4420
CDK2CDKCMGC3royAA4-(hexylamino)-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman4131
CDK2CDKCMGC3royAB4-(hexylamino)-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman4239
CDK2CDKCMGC3rpoAA4-({4-carbamoyl-2-nitro-5-[(pyridin-3-ylmethyl)amino]phenyl}amino)butanoic acidHuman3966
CDK2CDKCMGC3rpoAB4-({4-carbamoyl-2-nitro-5-[(pyridin-3-ylmethyl)amino]phenyl}amino)butanoic acidHuman4098
CDK2CDKCMGC3rprAA[4-amino-2-(phenylamino)-1,3-thiazol-5-yl][3-(trifluoromethyl)phenyl]methanoneHuman4452
CDK2CDKCMGC3rprAB[4-amino-2-(phenylamino)-1,3-thiazol-5-yl][3-(trifluoromethyl)phenyl]methanoneHuman4241
CDK2CDKCMGC3rpvAA4-{[4-amino-5-(3-aminobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4348
CDK2CDKCMGC3rpvAB4-{[4-amino-5-(3-aminobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4372
CDK2CDKCMGC3rpyAA4-amino-2-[(4-sulfamoylphenyl)amino]-1,3-thiazole-5-carboxamideHuman4261
CDK2CDKCMGC3rpyAB4-amino-2-[(4-sulfamoylphenyl)amino]-1,3-thiazole-5-carboxamideHuman4519
CDK2CDKCMGC3rzbAA4-amino-2-(phenylamino)-1,3-thiazole-5-carboxamideHuman4264
CDK2CDKCMGC3rzbAB4-amino-2-(phenylamino)-1,3-thiazole-5-carboxamideHuman4395
CDK2CDKCMGC3s00AA[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](5-chlorothiophen-2-yl)methanoneHuman4208
CDK2CDKCMGC3s00AB[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](5-chlorothiophen-2-yl)methanoneHuman4248
CDK2CDKCMGC3s0oAA[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](pyridin-2-yl)methanoneHuman3898
CDK2CDKCMGC3s0oAB[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](pyridin-2-yl)methanoneHuman4123
CDK2CDKCMGC3s1hAA4-{[4-amino-5-(4-methoxybenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4068
CDK2CDKCMGC3s1hAB4-{[4-amino-5-(4-methoxybenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4226
CDK2CDKCMGC3s2pA(3s,4s)-1-{3-[2-amino-6-(propan-2-yl)pyrimidin-4-yl]-4-hydroxyphenyl}pyrrolidine-3,4-diolHuman4404
CDK2CDKCMGC3sqqAA4-{[4-amino-5-(2-methylbenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4231
CDK2CDKCMGC3sqqAB4-{[4-amino-5-(2-methylbenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman3925
CDK2CDKCMGC3sw4AAn'-[4-(2-amino-4-methyl-1,3-thiazol-5-yl)pyrimidin-2-yl]-n,n-dimethylbenzene-1,4-diamineHuman4076
CDK2CDKCMGC3sw4ABn'-[4-(2-amino-4-methyl-1,3-thiazol-5-yl)pyrimidin-2-yl]-n,n-dimethylbenzene-1,4-diamineHuman4439
CDK2CDKCMGC3sw7AAn~4~-[4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-yl]-n~1~,n~1~-dimethyl-2-nitrobenzene-1,4-diamineHuman4198
CDK2CDKCMGC3sw7ABn~4~-[4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-yl]-n~1~,n~1~-dimethyl-2-nitrobenzene-1,4-diamineHuman4584
CDK2CDKCMGC3ti1AAn-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman4201
CDK2CDKCMGC3ti1ABn-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman4213
CDK2CDKCMGC3tiyAA2,3,4,6-tetrahydroxy-5h-benzo[7]annulen-5-oneHuman4413
CDK2CDKCMGC3tiyAB2,3,4,6-tetrahydroxy-5h-benzo[7]annulen-5-oneHuman4488
CDK2CDKCMGC3tizA1-{(e)-[(4-hydroxyphenyl)imino]methyl}naphthalen-2-olHuman4136
CDK2CDKCMGC3tnwAA4-[(e)-(3,5-diamino-1h-pyrazol-4-yl)diazenyl]phenolHuman4254
CDK2CDKCMGC3tnwAB4-[(e)-(3,5-diamino-1h-pyrazol-4-yl)diazenyl]phenolHuman3948
CDK2CDKCMGC3tnwCA4-[(e)-(3,5-diamino-1h-pyrazol-4-yl)diazenyl]phenolHuman3940
CDK2CDKCMGC3tnwCB4-[(e)-(3,5-diamino-1h-pyrazol-4-yl)diazenyl]phenolHuman4493
CDK2CDKCMGC3uliAA1-(aminomethyl)-n-(3-{[6-bromo-2-(4-methoxyphenyl)-3h-imidazo[4,5-b]pyridin-7-yl]amino}propyl)cyclopropanecarboxamideHuman4115
CDK2CDKCMGC3unjA4-{[4-(phenylamino)pyrimidin-2-yl]amino}benzoic acidHuman4498
CDK2CDKCMGC3unkA4-({4-[(2-chlorophenyl)amino]pyrimidin-2-yl}amino)benzoic acidHuman4374
CDK2CDKCMGC3wblAn~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamineHuman3895
CDK2CDKCMGC4acmAA3-amino-6-(4-{[2-(dimethylamino)ethyl]sulfamoyl}phenyl)-n-pyridin-3-ylpyrazine-2-carboxamideHuman4247
CDK2CDKCMGC4acmAB3-amino-6-(4-{[2-(dimethylamino)ethyl]sulfamoyl}phenyl)-n-pyridin-3-ylpyrazine-2-carboxamideHuman3983
CDK2CDKCMGC4bckAA3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamideHuman4095
CDK2CDKCMGC4bckAB3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamideHuman3960
CDK2CDKCMGC4bckAC3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamideHuman4433
CDK2CDKCMGC4bckAD3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamideHuman4563
CDK2CDKCMGC4bckCA3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamideHuman4268
CDK2CDKCMGC4bckCB3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamideHuman4506
CDK2CDKCMGC4bckCC3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamideHuman4029
CDK2CDKCMGC4bckCD3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamideHuman4080
CDK2CDKCMGC4bcmAA4-(4-methyl-2-methylimino-3h-1,3-thiazol-5-yl)-2-[(4-methyl-3-morpholin-4-ylsulfonyl-phenyl)amino]pyrimidine-5-carbonitrileHuman4290
CDK2CDKCMGC4bcmAB4-(4-methyl-2-methylimino-3h-1,3-thiazol-5-yl)-2-[(4-methyl-3-morpholin-4-ylsulfonyl-phenyl)amino]pyrimidine-5-carbonitrileHuman4203
CDK2CDKCMGC4bcmCA4-(4-methyl-2-methylimino-3h-1,3-thiazol-5-yl)-2-[(4-methyl-3-morpholin-4-ylsulfonyl-phenyl)amino]pyrimidine-5-carbonitrileHuman4227
CDK2CDKCMGC4bcmCB4-(4-methyl-2-methylimino-3h-1,3-thiazol-5-yl)-2-[(4-methyl-3-morpholin-4-ylsulfonyl-phenyl)amino]pyrimidine-5-carbonitrileHuman4124
CDK2CDKCMGC4bcnAA2-[(3-hydroxyphenyl)amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman4084
CDK2CDKCMGC4bcnAB2-[(3-hydroxyphenyl)amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman4298
CDK2CDKCMGC4bcnCA2-[(3-hydroxyphenyl)amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman4436
CDK2CDKCMGC4bcnCB2-[(3-hydroxyphenyl)amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman4150
CDK2CDKCMGC4bcoAA2-[[3-(4-ethanoyl-1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman3988
CDK2CDKCMGC4bcoAB2-[[3-(4-ethanoyl-1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman4051
CDK2CDKCMGC4bcoCA2-[[3-(4-ethanoyl-1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman4333
CDK2CDKCMGC4bcoCB2-[[3-(4-ethanoyl-1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman4018
CDK2CDKCMGC4bcpAA2-[[3-(1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman4552
CDK2CDKCMGC4bcpAB2-[[3-(1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman4304
CDK2CDKCMGC4bcpCA2-[[3-(1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman3872
CDK2CDKCMGC4bcpCB2-[[3-(1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman4501
CDK2CDKCMGC4bcqAA4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]-2-{[3-(morpholin-4-ylcarbonyl)phenyl]amino}pyrimidine-5-carbonitrileHuman4396
CDK2CDKCMGC4bcqAB4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]-2-{[3-(morpholin-4-ylcarbonyl)phenyl]amino}pyrimidine-5-carbonitrileHuman4415
CDK2CDKCMGC4bcqCA4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]-2-{[3-(morpholin-4-ylcarbonyl)phenyl]amino}pyrimidine-5-carbonitrileHuman3996
CDK2CDKCMGC4bcqCB4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]-2-{[3-(morpholin-4-ylcarbonyl)phenyl]amino}pyrimidine-5-carbonitrileHuman4120
CDK2CDKCMGC4bghAA4-((5-bromo-4-(prop-2-yn-1-ylamino)pyrimidin-2-yl)amino)benzenesulfonamideHuman4073
CDK2CDKCMGC4bghAB4-((5-bromo-4-(prop-2-yn-1-ylamino)pyrimidin-2-yl)amino)benzenesulfonamideHuman4509
CDK2CDKCMGC4bzdAA6-(benzimidazol-1-yl)-n-[5-[3-(dimethylamino)propoxy]pyridin-2-yl]pyrimidin-4-amineHuman3865
CDK2CDKCMGC4bzdAB6-(benzimidazol-1-yl)-n-[5-[3-(dimethylamino)propoxy]pyridin-2-yl]pyrimidin-4-amineHuman4490
CDK2CDKCMGC4cfmAA6-(cyclohexylmethoxy)-8-(2-methylphenyl)-9h-purin-2-amineHuman4207
CDK2CDKCMGC4cfmAB6-(cyclohexylmethoxy)-8-(2-methylphenyl)-9h-purin-2-amineHuman3986
CDK2CDKCMGC4cfmCA6-(cyclohexylmethoxy)-8-(2-methylphenyl)-9h-purin-2-amineHuman4260
CDK2CDKCMGC4cfmCB6-(cyclohexylmethoxy)-8-(2-methylphenyl)-9h-purin-2-amineHuman4005
CDK2CDKCMGC4cfnAA6-(cyclohexylmethoxy)-8-(trifluoromethyl)-9h-purin-2-amineHuman4285
CDK2CDKCMGC4cfnAB6-(cyclohexylmethoxy)-8-(trifluoromethyl)-9h-purin-2-amineHuman4437
CDK2CDKCMGC4cfnCA6-(cyclohexylmethoxy)-8-(trifluoromethyl)-9h-purin-2-amineHuman4355
CDK2CDKCMGC4cfnCB6-(cyclohexylmethoxy)-8-(trifluoromethyl)-9h-purin-2-amineHuman4567
CDK2CDKCMGC4cfuAA3-[2-azanyl-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methyl-benzoic acidHuman3905
CDK2CDKCMGC4cfuAB3-[2-azanyl-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methyl-benzoic acidHuman4308
CDK2CDKCMGC4cfuCA3-[2-azanyl-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methyl-benzoic acidHuman3967
CDK2CDKCMGC4cfuCB3-[2-azanyl-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methyl-benzoic acidHuman4539
CDK2CDKCMGC4cfvAA3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylphenolHuman4180
CDK2CDKCMGC4cfvAB3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylphenolHuman4328
CDK2CDKCMGC4cfvCA3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylphenolHuman3999
CDK2CDKCMGC4cfvCB3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylphenolHuman3979
CDK2CDKCMGC4cfwAA3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylbenzenesulfonamideHuman4280
CDK2CDKCMGC4cfwAB3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylbenzenesulfonamideHuman4557
CDK2CDKCMGC4cfwAC3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylbenzenesulfonamideHuman4141
CDK2CDKCMGC4cfwCA3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylbenzenesulfonamideHuman4549
CDK2CDKCMGC4cfwCB3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylbenzenesulfonamideHuman4508
CDK2CDKCMGC4cfwCC3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylbenzenesulfonamideHuman4102
CDK2CDKCMGC4cfxAA3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]benzenesulfonamideHuman4485
CDK2CDKCMGC4cfxAB3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]benzenesulfonamideHuman4086
CDK2CDKCMGC4cfxAC3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]benzenesulfonamideHuman3963
CDK2CDKCMGC4cfxCA3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]benzenesulfonamideHuman4166
CDK2CDKCMGC4cfxCB3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]benzenesulfonamideHuman4257
CDK2CDKCMGC4cfxCC3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]benzenesulfonamideHuman4442
CDK2CDKCMGC4d1xA(4s)-2-(6-hydroxy-1,3-benzothiazol-2-yl)-4,5-dihydro-1,3-thiazole-4-carboxylic acidHuman4344
CDK2CDKCMGC4d1zA(4s)-2-(8-hydroxyquinolin-2-yl)-4,5-dihydro-1,3-thiazole-4-carboxylic acidHuman4486
CDK2CDKCMGC4ek3AA-Human3971
CDK2CDKCMGC4ek3AB-Human4202
CDK2CDKCMGC4ek4AA4-bromo-n-(5-methyl-1h-pyrazol-3-yl)benzamideHuman4212
CDK2CDKCMGC4ek4AB4-bromo-n-(5-methyl-1h-pyrazol-3-yl)benzamideHuman3957
CDK2CDKCMGC4ek4AC4-bromo-n-(5-methyl-1h-pyrazol-3-yl)benzamideHuman4369
CDK2CDKCMGC4ek5AAn-(5-cyclopropyl-1h-pyrazol-3-yl)benzene-1,4-dicarboxamideHuman4037
CDK2CDKCMGC4ek5ABn-(5-cyclopropyl-1h-pyrazol-3-yl)benzene-1,4-dicarboxamideHuman4145
CDK2CDKCMGC4ek6AAn-(3-cyclopropyl-1h-pyrazol-5-yl)-2-[4-(thiophen-2-yl)phenyl]acetamideHuman4359
CDK2CDKCMGC4ek6ABn-(3-cyclopropyl-1h-pyrazol-5-yl)-2-[4-(thiophen-2-yl)phenyl]acetamideHuman4056
CDK2CDKCMGC4ek8AA4-(2,4-dimethyl-1,3-thiazol-5-yl)-n-(3-nitrophenyl)pyrimidin-2-amineHuman4079
CDK2CDKCMGC4ek8AB4-(2,4-dimethyl-1,3-thiazol-5-yl)-n-(3-nitrophenyl)pyrimidin-2-amineHuman3871
CDK2CDKCMGC4eoiAA(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4307
CDK2CDKCMGC4eoiAB(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4342
CDK2CDKCMGC4eoiCA(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4522
CDK2CDKCMGC4eoiCB(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4011
CDK2CDKCMGC4eojAAadenosine-5'-triphosphateHuman4271
CDK2CDKCMGC4eojABadenosine-5'-triphosphateHuman4015
CDK2CDKCMGC4eojCAadenosine-5'-triphosphateHuman4041
CDK2CDKCMGC4eojCBadenosine-5'-triphosphateHuman4311
CDK2CDKCMGC4eokAo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman3913
CDK2CDKCMGC4eokCo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman4385
CDK2CDKCMGC4eolAA(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4089
CDK2CDKCMGC4eolAB(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4270
CDK2CDKCMGC4eolCA(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4235
CDK2CDKCMGC4eolCB(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4521
CDK2CDKCMGC4eomAAadenosine-5'-triphosphateHuman4528
CDK2CDKCMGC4eomABadenosine-5'-triphosphateHuman4472
CDK2CDKCMGC4eomCAadenosine-5'-triphosphateHuman4481
CDK2CDKCMGC4eomCBadenosine-5'-triphosphateHuman4423
CDK2CDKCMGC4eonAA(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman3902
CDK2CDKCMGC4eonAB(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4326
CDK2CDKCMGC4eonCA(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4153
CDK2CDKCMGC4eonCB(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4192
CDK2CDKCMGC4eooAAadenosine-5'-triphosphateHuman4403
CDK2CDKCMGC4eooABadenosine-5'-triphosphateHuman4278
CDK2CDKCMGC4eooCAadenosine-5'-triphosphateHuman4188
CDK2CDKCMGC4eooCBadenosine-5'-triphosphateHuman4139
CDK2CDKCMGC4eopAA(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4258
CDK2CDKCMGC4eopAB(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4044
CDK2CDKCMGC4eopCA(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4061
CDK2CDKCMGC4eopCB(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4463
CDK2CDKCMGC4eoqAAadenosine-5'-triphosphateHuman4402
CDK2CDKCMGC4eoqABadenosine-5'-triphosphateHuman4230
CDK2CDKCMGC4eoqCAadenosine-5'-triphosphateHuman4004
CDK2CDKCMGC4eoqCBadenosine-5'-triphosphateHuman3912
CDK2CDKCMGC4eorAAo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman4205
CDK2CDKCMGC4eorABo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman3934
CDK2CDKCMGC4eorCAo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman4221
CDK2CDKCMGC4eorCBo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman4487
CDK2CDKCMGC4eosAA(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4340
CDK2CDKCMGC4eosAB(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4028
CDK2CDKCMGC4eosCA(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4008
CDK2CDKCMGC4eosCB(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4181
CDK2CDKCMGC4erwAstaurosporineHuman4370
CDK2CDKCMGC4ez3A4-[(e)-(6-hydroxy-2-oxo-1,2-dihydropyridin-3-yl)diazenyl]benzenesulfonamideHuman4551
CDK2CDKCMGC4ez7AstaurosporineHuman4240
CDK2CDKCMGC4fkgAA4-[(5-cyclopropyl-1h-pyrazol-3-yl)carbamoyl]benzoic acidHuman4020
CDK2CDKCMGC4fkgAB4-[(5-cyclopropyl-1h-pyrazol-3-yl)carbamoyl]benzoic acidHuman4559
CDK2CDKCMGC4fkiAAn-(5-cyclopropyl-1h-pyrazol-3-yl)-2-[4-(trifluoromethoxy)phenyl]acetamideHuman4430
CDK2CDKCMGC4fkiABn-(5-cyclopropyl-1h-pyrazol-3-yl)-2-[4-(trifluoromethoxy)phenyl]acetamideHuman4272
CDK2CDKCMGC4fkjAAn-(3-cyclopropyl-1h-pyrazol-5-yl)-2-[4-(2-pyrrolidin-1-ylethoxy)phenyl]acetamideHuman4387
CDK2CDKCMGC4fkjABn-(3-cyclopropyl-1h-pyrazol-5-yl)-2-[4-(2-pyrrolidin-1-ylethoxy)phenyl]acetamideHuman4164
CDK2CDKCMGC4fklAA4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-amineHuman4583
CDK2CDKCMGC4fklAB4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-amineHuman4134
CDK2CDKCMGC4fkoAA2-chloro-n~4~-[4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-yl]-n~1~,n~1~-dimethylbenzene-1,4-diamineHuman4449
CDK2CDKCMGC4fkoAB2-chloro-n~4~-[4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-yl]-n~1~,n~1~-dimethylbenzene-1,4-diamineHuman4534
CDK2CDKCMGC4fkpAA3-{[4-([amino(imino)methyl]aminosulfonyl)anilino]methylene}-2-oxo-2,3-dihydro-1h-indoleHuman4035
CDK2CDKCMGC4fkpAB3-{[4-([amino(imino)methyl]aminosulfonyl)anilino]methylene}-2-oxo-2,3-dihydro-1h-indoleHuman4313
CDK2CDKCMGC4fkpAC3-{[4-([amino(imino)methyl]aminosulfonyl)anilino]methylene}-2-oxo-2,3-dihydro-1h-indoleHuman4468
CDK2CDKCMGC4fkqAA4-[(2z)-2-(7-oxidanylidene-3,6-dihydropyrrolo[3,2-e]benzotriazol-8-ylidene)hydrazinyl]benzenesulfonamideHuman3972
CDK2CDKCMGC4fkqAB4-[(2z)-2-(7-oxidanylidene-3,6-dihydropyrrolo[3,2-e]benzotriazol-8-ylidene)hydrazinyl]benzenesulfonamideHuman4026
CDK2CDKCMGC4fkrAA(8z)-8-{[(2,2-dioxido-1,3-dihydro-2-benzothiophen-5-yl)amino]methylidene}-6,8-dihydro-7h-[1,3]thiazolo[5,4-e]indol-7-oneHuman4149
CDK2CDKCMGC4fkrAB(8z)-8-{[(2,2-dioxido-1,3-dihydro-2-benzothiophen-5-yl)amino]methylidene}-6,8-dihydro-7h-[1,3]thiazolo[5,4-e]indol-7-oneHuman4535
CDK2CDKCMGC4fksAAn-[(4-{[(z)-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}phenyl)sulfonyl]acetamideHuman4412
CDK2CDKCMGC4fksABn-[(4-{[(z)-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}phenyl)sulfonyl]acetamideHuman4489
CDK2CDKCMGC4fksACn-[(4-{[(z)-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}phenyl)sulfonyl]acetamideHuman4315
CDK2CDKCMGC4fktAAn-[2-(dimethylamino)ethyl]-4-{[(z)-(2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]amino}benzenesulfonamideHuman4548
CDK2CDKCMGC4fktABn-[2-(dimethylamino)ethyl]-4-{[(z)-(2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]amino}benzenesulfonamideHuman4322
CDK2CDKCMGC4fkuAA(3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylic acidHuman3863
CDK2CDKCMGC4fkuAB(3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylic acidHuman4573
CDK2CDKCMGC4fkvAA(3z)-n-[2-(1h-imidazol-4-yl)ethyl]-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxamideHuman4299
CDK2CDKCMGC4fkvAB(3z)-n-[2-(1h-imidazol-4-yl)ethyl]-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxamideHuman3939
CDK2CDKCMGC4fkwAA2-methylpropyl (3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylateHuman4252
CDK2CDKCMGC4fkwAB2-methylpropyl (3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylateHuman4277
CDK2CDKCMGC4fx3AA(3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylic acidHuman4518
CDK2CDKCMGC4fx3AB(3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylic acidHuman3931
CDK2CDKCMGC4fx3CA(3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylic acidHuman4349
CDK2CDKCMGC4fx3CB(3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylic acidHuman4495
CDK2CDKCMGC4gcjAA4-{[4-amino-5-(2-nitrobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4138
CDK2CDKCMGC4gcjAB4-{[4-amino-5-(2-nitrobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4362
CDK2CDKCMGC4i3zAadenosine-5'-diphosphateHuman4148
CDK2CDKCMGC4i3zCadenosine-5'-diphosphateHuman3961
CDK2CDKCMGC4ii5AAadenosine-5'-diphosphateHuman3930
CDK2CDKCMGC4ii5ABadenosine-5'-diphosphateHuman4456
CDK2CDKCMGC4ii5CAadenosine-5'-diphosphateHuman4530
CDK2CDKCMGC4ii5CBadenosine-5'-diphosphateHuman4462
CDK2CDKCMGC4kd1AA3-[({3-ethyl-5-[(2s)-2-(2-hydroxyethyl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1-hydroxypyridiniumHuman4585
CDK2CDKCMGC4kd1AB3-[({3-ethyl-5-[(2s)-2-(2-hydroxyethyl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1-hydroxypyridiniumHuman4525
CDK2CDKCMGC4lynA(2s)-n-(5-{[(5-tert-butyl-1,3-oxazol-2-yl)methyl]sulfanyl}-1,3-thiazol-2-yl)-2-phenylpropanamideHuman4550
CDK2CDKCMGC4nj3AA6-(3-chlorophenyl)-2-{[(2s)-3-(4-hydroxyphenyl)-1-methoxy-1-oxopropan-2-yl]carbamoyl}quinoline-4-carboxylic acidHuman4075
CDK2CDKCMGC4nj3AB6-(3-chlorophenyl)-2-{[(2s)-3-(4-hydroxyphenyl)-1-methoxy-1-oxopropan-2-yl]carbamoyl}quinoline-4-carboxylic acidHuman4366
CDK2CDKCMGC4rj3AA1-cyclopentyl-n-[2-(4-methoxypiperidin-1-yl)pyrimidin-4-yl]-1h-pyrrolo[3,2-c]pyridin-6-amineHuman4244
CDK2CDKCMGC4rj3AB1-cyclopentyl-n-[2-(4-methoxypiperidin-1-yl)pyrimidin-4-yl]-1h-pyrrolo[3,2-c]pyridin-6-amineHuman4127
CDK2CDKCMGC5a14AA1-[4-(2-azanylpyrimidin-4-yl)oxyphenyl]-3-[4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]ureaHuman3977
CDK2CDKCMGC5a14AB1-[4-(2-azanylpyrimidin-4-yl)oxyphenyl]-3-[4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]ureaHuman3901
CDK2CDKCMGC5andA2-imidazol-1-yl-1h-benzimidazoleHuman6543
CDK2CDKCMGC5aneA6-methoxy-9h-purineHuman6542
CDK2CDKCMGC5angA7-hydroxy-4-(morpholinomethyl)chromen-2-oneHuman6540
CDK2CDKCMGC5aniA6-chloro-9h-purineHuman6539
CDK2CDKCMGC5anjAn-(9h-purin-6-yl)thiophene-2-carboxamideHuman6541
CDK2CDKCMGC5ankA2,4,6-trioxo-1-phenyl-hexahydropyrimidine-5-carboxamideHuman6538
CDK2CDKCMGC5anoA-Human6537
CDK2CDKCMGC5cyiAA6-(cyclohexylmethoxy)-n-[4-(ethylsulfonyl)phenyl]-9h-purin-2-amineHuman6052
CDK2CDKCMGC5cyiAB6-(cyclohexylmethoxy)-n-[4-(ethylsulfonyl)phenyl]-9h-purin-2-amineHuman6054
CDK2CDKCMGC5cyiCA6-(cyclohexylmethoxy)-n-[4-(ethylsulfonyl)phenyl]-9h-purin-2-amineHuman6055
CDK2CDKCMGC5cyiCB6-(cyclohexylmethoxy)-n-[4-(ethylsulfonyl)phenyl]-9h-purin-2-amineHuman6053
CDK2CDKCMGC5d1jAn-(5-{[(5-tert-butyl-1,3-oxazol-2-yl)methyl]sulfanyl}-1,3-thiazol-2-yl)piperidine-4-carboxamideHuman4058
CDK2CDKCMGC5fp5A4-fluorobenzoic acidHuman6285
CDK2CDKCMGC5fp6AA3-(4,7-dichloro-1h-indol-3-yl)prop-2-yn-1-olHuman6302
CDK2CDKCMGC5fp6AB3-(4,7-dichloro-1h-indol-3-yl)prop-2-yn-1-olHuman6301
CDK2CDKCMGC5ievAAroniciclibHuman6567
CDK2CDKCMGC5ievABroniciclibHuman6570
CDK2CDKCMGC5iexAA(2r,3r)-3-[(5-bromo-2-{[4-(s-cyclopropylsulfonimidoyl)phenyl]amino}pyrimidin-4-yl)oxy]butan-2-olHuman6565
CDK2CDKCMGC5iexAB(2r,3r)-3-[(5-bromo-2-{[4-(s-cyclopropylsulfonimidoyl)phenyl]amino}pyrimidin-4-yl)oxy]butan-2-olHuman6572
CDK2CDKCMGC5ieyAA4-[(4-{[(2r,3r)-3-hydroxybutan-2-yl]amino}pyrimidin-2-yl)amino]benzene-1-sulfonamideHuman6566
CDK2CDKCMGC5ieyAB4-[(4-{[(2r,3r)-3-hydroxybutan-2-yl]amino}pyrimidin-2-yl)amino]benzene-1-sulfonamideHuman6573
CDK2CDKCMGC5if1AA-Human6568
CDK2CDKCMGC5if1AB-Human6569
CDK2CDKCMGC5if1CA-Human6564
CDK2CDKCMGC5if1CB-Human6571
CDK2CDKCMGC5jq5A(3r,4r)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-olHuman7416
CDK2CDKCMGC5jq8A(3s,4s)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-olHuman7417
CDK2CDKCMGC5k4jAA1-[(1~{s})-1-(4-chloranyl-3-fluoranyl-phenyl)-2-oxidanyl-ethyl]-4-[2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]pyridin-2-oneHuman6751
CDK2CDKCMGC5k4jAB1-[(1~{s})-1-(4-chloranyl-3-fluoranyl-phenyl)-2-oxidanyl-ethyl]-4-[2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]pyridin-2-oneHuman6750
CDK2CDKCMGC5l2wA3-[({3-ethyl-5-[(2s)-2-(2-hydroxyethyl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1-hydroxypyridiniumHuman6993
CDK2CDKCMGC5lmkAA4-[4-[3-bromanyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-5-yl]phenyl]benzamideHuman7399
CDK2CDKCMGC5lmkAB4-[4-[3-bromanyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-5-yl]phenyl]benzamideHuman7398
CDK2CDKCMGC5lmkCA4-[4-[3-bromanyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-5-yl]phenyl]benzamideHuman7396
CDK2CDKCMGC5lmkCB4-[4-[3-bromanyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-5-yl]phenyl]benzamideHuman7397
CDK2CDKCMGC5mhqAA(2~{r},3~{s})-3-[[9-propan-2-yl-6-(pyridin-3-ylmethylamino)purin-2-yl]amino]pentan-2-olHuman9409
CDK2CDKCMGC5mhqAB(2~{r},3~{s})-3-[[9-propan-2-yl-6-(pyridin-3-ylmethylamino)purin-2-yl]amino]pentan-2-olHuman9408
CDK2CDKCMGC5nevA4-[[6-(3-phenylphenyl)-7~{h}-purin-2-yl]amino]benzenesulfonamideHuman8020
CDK2CDKCMGC5nevC4-[[6-(3-phenylphenyl)-7~{h}-purin-2-yl]amino]benzenesulfonamideHuman8019
CDK2CDKCMGC5oo0AA-Human9744
CDK2CDKCMGC5oo0AC-Human9745
CDK2CDKCMGC5oo1A~{n}-(4-pyrimidin-2-ylphenyl)propanamideHuman10566
CDK2CDKCMGC5oo3AA1-(4-ethyl-2,3-dihydroquinoxalin-1-yl)propan-1-oneHuman10569
CDK2CDKCMGC5oo3AB1-(4-ethyl-2,3-dihydroquinoxalin-1-yl)propan-1-oneHuman10568
CDK2CDKCMGC5osjAA-Human9743
CDK2CDKCMGC5osjAB-Human9742
CDK2CDKCMGC5osmAAmethyl 1-propanoyl-3,4-dihydro-2~{h}-quinoline-6-carboxylateHuman9741
CDK2CDKCMGC5osmABmethyl 1-propanoyl-3,4-dihydro-2~{h}-quinoline-6-carboxylateHuman9740
CDK2CDKCMGC5uq1A-Human8220
CDK2CDKCMGC5uq1C-Human8223
CDK2CDKCMGC5uq2A-Human8221
CDK2CDKCMGC5uq3A-Human8222
CDK2CDKCMGC6athAA-Human10567
CDK2CDKCMGC6athAB-Human10570
CDK2CDKCMGC6gubA2-(2-chlorophenyl)-8-[(3~{r},4~{r})-1-methyl-3-oxidanyl-piperidin-4-yl]-5,7-bis(oxidanyl)chromen-4-oneHuman10764
CDK2CDKCMGC6gubC2-(2-chlorophenyl)-8-[(3~{r},4~{r})-1-methyl-3-oxidanyl-piperidin-4-yl]-5,7-bis(oxidanyl)chromen-4-oneHuman10763
CDK2CDKCMGC6gucA(3z)-3-(1h-imidazol-5-ylmethylene)-5-methoxy-1h-indol-2(3h)-oneHuman10767
CDK2CDKCMGC6gucC(3z)-3-(1h-imidazol-5-ylmethylene)-5-methoxy-1h-indol-2(3h)-oneHuman10766
CDK2CDKCMGC6gueA4-(2-methyl-3-propan-2-yl-imidazol-4-yl)-~{n}-(4-methylsulfonylphenyl)pyrimidin-2-amineHuman10771
CDK2CDKCMGC6gueC4-(2-methyl-3-propan-2-yl-imidazol-4-yl)-~{n}-(4-methylsulfonylphenyl)pyrimidin-2-amineHuman10772
CDK2CDKCMGC6gufAn2-[(1r,2s)-2-aminocyclohexyl]-n6-(3-chlorophenyl)-9-ethyl-9h-purine-2,6-diamineHuman10770
CDK2CDKCMGC6gufCn2-[(1r,2s)-2-aminocyclohexyl]-n6-(3-chlorophenyl)-9-ethyl-9h-purine-2,6-diamineHuman10762
CDK2CDKCMGC6guhAA4-(2-methyl-3-propan-2-yl-imidazol-4-yl)-~{n}-(4-methylsulfonylphenyl)pyrimidin-2-amineHuman10765
CDK2CDKCMGC6guhAB4-(2-methyl-3-propan-2-yl-imidazol-4-yl)-~{n}-(4-methylsulfonylphenyl)pyrimidin-2-amineHuman10769
CDK2CDKCMGC6gukAA~{n}2-[(1~{r},2~{s})-2-azanylcyclohexyl]-~{n}6-(3-chlorophenyl)-9-ethyl-purine-2,6-diamineHuman10773
CDK2CDKCMGC6gukAB~{n}2-[(1~{r},2~{s})-2-azanylcyclohexyl]-~{n}6-(3-chlorophenyl)-9-ethyl-purine-2,6-diamineHuman10768
CDK2CDKCMGC6gvaAA5-(2-azanylethylsulfanyl)-3-propan-2-yl-~{n}-[(4-pyridin-2-ylphenyl)methyl]-2~{h}-pyrazolo[4,3-d]pyrimidin-7-amineHuman11206
CDK2CDKCMGC6gvaAB5-(2-azanylethylsulfanyl)-3-propan-2-yl-~{n}-[(4-pyridin-2-ylphenyl)methyl]-2~{h}-pyrazolo[4,3-d]pyrimidin-7-amineHuman11204
CDK2CDKCMGC6inlA2,2'-{[6-{[(4-methoxyphenyl)methyl]amino}-9-(propan-2-yl)-9h-purin-2-yl]azanediyl}di(ethan-1-ol)Human11794
CDK2CDKCMGC6jgmA4-{[6-(cyclohexylmethoxy)-7h-purin-2-yl]amino}-n,n-diethylbenzamideHuman12008
CDK2CDKCMGC6oqiA5-fluoro-n-[5-(4-methylpiperazin-1-yl)pyridin-2-yl]-4-[(4s)-4-methyl-5,6,7,8-tetrahydro-4h-pyrazolo[1,5-a]azepin-3-yl]pyrimidin-2-amineHuman12648
CDK2CDKCMGC6p3wAA-Human11515
CDK2CDKCMGC6p3wAB-Human11517
CDK2CDKCMGC6p3wCA-Human11514
CDK2CDKCMGC6p3wCB-Human11516
CDK2CDKCMGC6q3bAA4-iodopyrazoleHuman11177
CDK2CDKCMGC6q3bAB4-iodopyrazoleHuman11208
CDK2CDKCMGC6q3cAA4-bromo-1h-pyrazoleHuman11191
CDK2CDKCMGC6q3cAB4-bromo-1h-pyrazoleHuman11203
CDK2CDKCMGC6q3cAC-Human11178
CDK2CDKCMGC6q3fAA-Human11181
CDK2CDKCMGC6q3fAB-Human11187
CDK2CDKCMGC6q48AA4-iodanyl-3~{h}-pyridin-2-oneHuman11192
CDK2CDKCMGC6q48AB4-iodanyl-3~{h}-pyridin-2-oneHuman11218
CDK2CDKCMGC6q48AC4-iodanyl-3~{h}-pyridin-2-oneHuman11196
CDK2CDKCMGC6q49AA-Human11185
CDK2CDKCMGC6q49AB-Human11220
CDK2CDKCMGC6q49AC-Human11193
CDK2CDKCMGC6q4aAA5-iodanylpyrimidineHuman11195
CDK2CDKCMGC6q4aAB5-iodanylpyrimidineHuman11200
CDK2CDKCMGC6q4aAC5-iodanylpyrimidineHuman11216
CDK2CDKCMGC6q4bAA5-bromanylpyrimidineHuman11198
CDK2CDKCMGC6q4bAB5-bromanylpyrimidineHuman11210
CDK2CDKCMGC6q4bAC5-bromanylpyrimidineHuman11180
CDK2CDKCMGC6q4cAA4-bromanyl-1,8-naphthyridineHuman11182
CDK2CDKCMGC6q4cAB4-bromanyl-1,8-naphthyridineHuman11207
CDK2CDKCMGC6q4cAC4-bromanyl-1,8-naphthyridineHuman11201
CDK2CDKCMGC6q4dAA2-(4-bromanyl-2-methoxy-phenyl)ethanoic acidHuman11184
CDK2CDKCMGC6q4dAB2-(4-bromanyl-2-methoxy-phenyl)ethanoic acidHuman11215
CDK2CDKCMGC6q4dAC2-(4-bromanyl-2-methoxy-phenyl)ethanoic acidHuman11188
CDK2CDKCMGC6q4eAA6-iodanyl-7~{h}-purin-2-amineHuman11199
CDK2CDKCMGC6q4eAB6-iodanyl-7~{h}-purin-2-amineHuman11205
CDK2CDKCMGC6q4eAC6-iodanyl-7~{h}-purin-2-amineHuman11219
CDK2CDKCMGC6q4fAApyridine-2,6-diamineHuman11202
CDK2CDKCMGC6q4fABpyridine-2,6-diamineHuman11211
CDK2CDKCMGC6q4fACpyridine-2,6-diamineHuman11212
CDK2CDKCMGC6q4gAA2-[3-(2-azanyl-9~{h}-purin-6-yl)phenyl]ethanoic acidHuman11214
CDK2CDKCMGC6q4gAB2-[3-(2-azanyl-9~{h}-purin-6-yl)phenyl]ethanoic acidHuman11217
CDK2CDKCMGC6q4hAA2-[3-[(2-azanyl-9~{h}-purin-6-yl)oxy]phenyl]ethanoic acidHuman11194
CDK2CDKCMGC6q4hAB2-[3-[(2-azanyl-9~{h}-purin-6-yl)oxy]phenyl]ethanoic acidHuman11190
CDK2CDKCMGC6q4iAA2-[4-[(2-oxidanylidene-3~{h}-pyridin-4-yl)oxy]phenyl]ethanoic acidHuman11183
CDK2CDKCMGC6q4iAB2-[4-[(2-oxidanylidene-3~{h}-pyridin-4-yl)oxy]phenyl]ethanoic acidHuman11197
CDK2CDKCMGC6q4jAA2-[3-(pyrimidin-4-ylamino)phenyl]ethanoic acidHuman11209
CDK2CDKCMGC6q4jAB2-[3-(pyrimidin-4-ylamino)phenyl]ethanoic acidHuman11213
CDK2CDKCMGC6q4kAA-Human11179
CDK2CDKCMGC6q4kAB-Human11186
CDK2CDKCMGC6q4kAC-Human11189
CDK2CDKCMGC6rijAA4-[[[5-nitroso-2-[[(2~{r})-1-oxidanylbutan-2-yl]amino]-6-(propan-2-ylamino)pyrimidin-4-yl]amino]methyl]phenolHuman12623
CDK2CDKCMGC6rijAB4-[[[5-nitroso-2-[[(2~{r})-1-oxidanylbutan-2-yl]amino]-6-(propan-2-ylamino)pyrimidin-4-yl]amino]methyl]phenolHuman12624
CDK2CDKCMGC6rijCA4-[[[5-nitroso-2-[[(2~{r})-1-oxidanylbutan-2-yl]amino]-6-(propan-2-ylamino)pyrimidin-4-yl]amino]methyl]phenolHuman12625
CDK2CDKCMGC6rijCB4-[[[5-nitroso-2-[[(2~{r})-1-oxidanylbutan-2-yl]amino]-6-(propan-2-ylamino)pyrimidin-4-yl]amino]methyl]phenolHuman12622
CDK2CDKCMGC6yl1AAmethyl 4-(cyclopropylmethyl)-1-prop-2-enoyl-2,3-dihydroquinoxaline-6-carboxylateHuman12497
CDK2CDKCMGC6yl1ABmethyl 4-(cyclopropylmethyl)-1-prop-2-enoyl-2,3-dihydroquinoxaline-6-carboxylateHuman12496
CDK2CDKCMGC6yl6AA-Human12498
CDK2CDKCMGC6yl6AB-Human12495
CDK2CDKCMGC6ylkAAmethyl 4-ethyl-1-propanoyl-2,3-dihydroquinoxaline-6-carboxylateHuman12499
CDK2CDKCMGC6ylkABmethyl 4-ethyl-1-propanoyl-2,3-dihydroquinoxaline-6-carboxylateHuman12494
CDK4CDKCMGC2w96BA-Human3390
CDK4CDKCMGC2w96BB-Human3389
CDK4CDKCMGC2w99B-Human3385
CDK4CDKCMGC2w9fB-Human3386
CDK4CDKCMGC2w9zBA-Human3388
CDK4CDKCMGC2w9zBB-Human3383
CDK4CDKCMGC3g33A-Human3387
CDK4CDKCMGC3g33C-Human3384
CDK4CDKCMGC5fwkK-Human6747
CDK4CDKCMGC5fwlK-Human6748
CDK4CDKCMGC5fwmK-Human6749
CDK4CDKCMGC5fwpK-Human7132
CDK4CDKCMGC6p8eB-Human11891
CDK4CDKCMGC6p8fB-Human11892
CDK4CDKCMGC6p8gB-Human11893
CDK4CDKCMGC6p8hB-Human11894
CDK5CDKCMGC1h4lA-Human2788
CDK5CDKCMGC1h4lB-Human2779
CDK5CDKCMGC1ungA6-phenyl[5h]pyrrolo[2,3-b]pyrazineHuman2792
CDK5CDKCMGC1ungB6-phenyl[5h]pyrrolo[2,3-b]pyrazineHuman2789
CDK5CDKCMGC1unhA(z)-1h,1'h-[2,3']biindolylidene-3,2'-dione-3-oximeHuman2780
CDK5CDKCMGC1unhB(z)-1h,1'h-[2,3']biindolylidene-3,2'-dione-3-oximeHuman2787
CDK5CDKCMGC1unlAr-roscovitineHuman2785
CDK5CDKCMGC1unlB-Human2790
CDK5CDKCMGC3o0gA-Human2782
CDK5CDKCMGC3o0gB{4-amino-2-[(4-chlorophenyl)amino]-1,3-thiazol-5-yl}(3-nitrophenyl)methanoneHuman2783
CDK5CDKCMGC4au8AA4-(1,3-benzothiazol-2-yl)thiophene-2-sulfonamideHuman2784
CDK5CDKCMGC4au8AB4-(1,3-benzothiazol-2-yl)thiophene-2-sulfonamideHuman2786
CDK5CDKCMGC4au8BA4-(1,3-benzothiazol-2-yl)thiophene-2-sulfonamideHuman2791
CDK5CDKCMGC4au8BB4-(1,3-benzothiazol-2-yl)thiophene-2-sulfonamideHuman2781
CDK6CDKCMGC1bi7A-Human2798
CDK6CDKCMGC1bi8A-Human2796
CDK6CDKCMGC1bi8C-Human2799
CDK6CDKCMGC1blxA-Human2802
CDK6CDKCMGC1g3nA-Human2806
CDK6CDKCMGC1g3nE-Human2805
CDK6CDKCMGC1jowB-Human2793
CDK6CDKCMGC1xo2B3,7,3',4'-tetrahydroxyflavoneHuman2794
CDK6CDKCMGC2eufB6-acetyl-8-cyclopentyl-5-methyl-2-[(5-piperazin-1-ylpyridin-2-yl)amino]pyrido[2,3-d]pyrimidin-7(8h)-oneHuman2804
CDK6CDKCMGC2f2cB(2s)-2-({6-[(3-amino-5-chlorophenyl)amino]-9-isopropyl-9h-purin-2-yl}amino)-3-methylbutan-1-olHuman2795
CDK6CDKCMGC3nupA4-[3-(1-methylethyl)-1h-pyrazol-4-yl]-n-(1-methylpiperidin-4-yl)pyrimidin-2-amineHuman2797
CDK6CDKCMGC3nuxA4-[5-chloro-3-(1-methylethyl)-1h-pyrazol-4-yl]-n-(5-piperazin-1-ylpyridin-2-yl)pyrimidin-2-amineHuman2807
CDK6CDKCMGC4auaA1h-benzimidazol-2-yl(1h-pyrrol-2-yl)methanoneHuman2801
CDK6CDKCMGC4ez5A{5-[4-(dimethylamino)piperidin-1-yl]-1h-imidazo[4,5-b]pyridin-2-yl}[2-(isoquinolin-4-yl)pyridin-4-yl]methanoneHuman2800
CDK6CDKCMGC4tthB9-cyclopentyl-n-(5-piperazin-1-ylpyridin-2-yl)pyrido[4,5]pyrrolo[1,2-d]pyrimidin-2-amineHuman2803
CDK6CDKCMGC5l2iA6-acetyl-8-cyclopentyl-5-methyl-2-[(5-piperazin-1-ylpyridin-2-yl)amino]pyrido[2,3-d]pyrimidin-7(8h)-oneHuman6991
CDK6CDKCMGC5l2sAn-{5-[(4-ethylpiperazin-1-yl)methyl]pyridin-2-yl}-5-fluoro-4-[4-fluoro-2-methyl-1-(propan-2-yl)-1h-benzimidazol-6-yl]pyrimidin-2-amineHuman6990
CDK6CDKCMGC5l2tA7-cyclopentyl-n,n-dimethyl-2-{[5-(piperazin-1-yl)pyridin-2-yl]amino}-7h-pyrrolo[2,3-d]pyrimidine-6-carboxamideHuman6992
CDK6CDKCMGC6oqlA5-fluoro-n-[5-(4-methylpiperazin-1-yl)pyridin-2-yl]-4-[(4r)-4-methyl-5,6,7,8-tetrahydro-4h-pyrazolo[1,5-a]azepin-3-yl]pyrimidin-2-amineHuman12647
CDK6CDKCMGC6oqoAn-[5-(6-ethyl-2,6-diazaspiro[3.3]heptan-2-yl)pyridin-2-yl]-5-fluoro-4-[(4r)-4-methyl-5,6,7,8-tetrahydro-4h-pyrazolo[1,5-a]azepin-3-yl]pyrimidin-2-amineHuman12646
CDK7CDKCMGC1ua2Aadenosine-5'-triphosphateHuman540
CDK7CDKCMGC1ua2Badenosine-5'-triphosphateHuman541
CDK7CDKCMGC1ua2Cadenosine-5'-triphosphateHuman542
CDK7CDKCMGC1ua2Dadenosine-5'-triphosphateHuman543
CDK7CDKCMGC6o9l8-Human11055
CDK7CDKCMGC6xbzJphosphothiophosphoric acid-adenylate esterHuman12773
CDK7CDKCMGC6xd3Jn-(3-{[5-chloro-4-(1h-indol-3-yl)pyrimidin-2-yl]amino}phenyl)-4-{[4-(dimethylamino)butanoyl]amino}benzamideHuman12772
CDK8CDKCMGC3rgfAA4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamideHuman3841
CDK8CDKCMGC3rgfAB4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamideHuman3846
CDK8CDKCMGC4crlAcortistatin aHuman6096
CDK8CDKCMGC4f6sA1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]ureaHuman3848
CDK8CDKCMGC4f6uAA1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-[3-(morpholin-4-yl)propyl]ureaHuman3849
CDK8CDKCMGC4f6uAB1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-[3-(morpholin-4-yl)propyl]ureaHuman3844
CDK8CDKCMGC4f6wAn-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-4-[2-({[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]carbamoyl}amino)ethyl]piperazine-1-carboxamideHuman3845
CDK8CDKCMGC4f70A1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-[2-(morpholin-4-yl)ethyl]ureaHuman3852
CDK8CDKCMGC4f7jAA1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-(2-hydroxyethyl)ureaHuman3842
CDK8CDKCMGC4f7jAB1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-(2-hydroxyethyl)ureaHuman3843