1MRV - chain A | V-akt murine thymoma viral oncogene homolog 2
Structure information
PDB:1MRV
PubMed:12517337
Release date:2003-09-23
Resolution:2.8 Å
 
Kinase:AKT2
Family:Akt
Group:AGC
Species:HUMAN
 
Quality Score:4
Missing Residues:10
Missing Atoms:26
DFG conformation:out
αC-helix conformation:na
Salt bridge KIII.17 and EαC.24:NA
 
 
ASP rotation (xDFG.81) :183°
PHE rotation (xDFG.82) :230°
Activation loop position:1.6Å
αC-helix position:0Å
 
G-rich loop angle:61.5°
G-rich loop distance:18.3Å
G-rich loop rotation:60.9°
2D & 3D views

The orthosteric binding pocket
Binding pocket waters
The following waters were found in the defined clusters:
I5
H-bond protein
Binding pocket sequence
UniprotKLLGKGTFGKVILYAMKILHTVTESRVLQNTRPFLTALKYACFVMEYANGGELFFHLSRYLHSRDVVYRDIKLENLMLITDFGLC
Structure:KLLGKGTFGKVILYAMKIL_______VLQNTRPFLTALKYACFVMEYANGGELFFHLSRYLHSRDVVYRDIKLENLMLITDF___


Modified residues
No modified residues identified.