1U59 - chain A (model A) | Zeta chain of T cell receptor associated protein kinase 70kDa
Structure information
PDB: | 1U59 |
PubMed: | 15292186 |
Release date: | 2004-08-17 |
Resolution: | 2.3 Å |
Kinase: | ZAP70 |
Family: | Syk |
Group: | TK |
Species: | HUMAN |
Quality Score: | 8 |
Missing Residues: | 0 |
Missing Atoms: | 0 |
DFG conformation: | in |
αC-helix conformation: | in |
Salt bridge KIII.17 and EαC.24: | Yes (2.6Å) |
ASP rotation (xDFG.81) : | 342° |
PHE rotation (xDFG.82) : | 9° |
Activation loop position: | -3.5Å |
αC-helix position: | 18.6Å |
G-rich loop angle: | 60.7° |
G-rich loop distance: | 18.4Å |
G-rich loop rotation: | 52.9° |
Other models from this PDB:
2D & 3D views
Binding pocket waters
The following waters were found in the defined clusters:
I4
H-bond protein
Binding pocket sequence
Uniprot | IELGCGNFGSVRQVAIKVLEMMREAQIMHQLDPYIVRLIGVMLVMEMAGGGPLHKFLVGYLEEKNFVHRDLAARNVLLISDFGLS |
Structure: | IELGCGNFGSVRQVAIKVLEMMREAQIMHQLDPYIVRLIGVMLVMEMAGGGPLHKFLVGYLEEKNFVHRDLAARNVLLISDFGLS |
Modified residues
No modified residues identified.
Orthosteric ligand
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- LABELS
- KLIFS residue #
- Amino Acid
- None
- COLORS
- Interaction types
- KLIFS (all res.)
- KLIFS (interacting res.)
- None
- OTHER
- Show/hide non-interacting res.
- En/disable resizing interacting res.
This ligand targets the following (sub)pockets:
Main pockets | |
---|---|
Front | |
Gate | |
Back |
Subpockets | |
---|---|
FP-I | |
FP-II | |
BP-I-A | |
BP-I-B | |
BP-II-in | |
BP-II-A-in | |
BP-II-B-in | |
BP-II-out | |
BP-II-B | |
BP-III | |
BP-IV | |
BP-V |
Kinase-ligand interactions
■ Hydrophobic ♦ Aromatic face-to-face ♦ Aromatic face-to-edge ▲ H-bond donor ▲ H-bond acceptor ● Ionic positive ● Ionic negative
I | g.l | II | III | αC | |||||||||||||||
1 I 342 | 2 E 343 | 3 L 344 | 4 G 345 | 5 C 346 | 6 G 347 | 7 N 348 | 8 F 349 | 9 G 350 | 10 S 351 | 11 V 352 | 12 R 353 | 13 Q 354 | 14 V 366 | 15 A 367 | 16 I 368 | 17 K 369 | 18 V 370 | 19 L 371 | 20 E 382 |
■ | ■ | ■ | ■ | ■ | |||||||||||||||
αC | b.l | IV | |||||||||||||||||
21 M 383 | 22 M 384 | 23 R 385 | 24 E 386 | 25 A 387 | 26 Q 388 | 27 I 389 | 28 M 390 | 29 H 391 | 30 Q 392 | 31 L 393 | 32 D 394 | 33 P 396 | 34 Y 397 | 35 I 398 | 36 V 399 | 37 R 400 | 38 L 401 | 39 I 402 | 40 G 403 |
■ | |||||||||||||||||||
IV | V | GK | hinge | linker | αD | αE | |||||||||||||
41 V 404 | 42 M 411 | 43 L 412 | 44 V 413 | 45 M 414 | 46 E 415 | 47 M 416 | 48 A 417 | 49 G 418 | 50 G 419 | 51 G 420 | 52 P 421 | 53 L 422 | 54 H 423 | 55 K 424 | 56 F 425 | 57 L 426 | 58 V 427 | 59 G 428 | 60 Y 451 |
■ | ▲ | ■ | ■▲ | ■ | ■ | ■ | |||||||||||||
αE | VI | c.l | VII | VIII | x | ||||||||||||||
61 L 452 | 62 E 453 | 63 E 454 | 64 K 455 | 65 N 456 | 66 F 457 | 67 V 458 | 68 H 459 | 69 R 460 | 70 D 461 | 71 L 462 | 72 A 463 | 73 A 464 | 74 R 465 | 75 N 466 | 76 V 467 | 77 L 468 | 78 L 469 | 79 I 477 | 80 S 478 |
■▲ | ■ | ■ | ■ | ||||||||||||||||
DFG | a.l | ||||||||||||||||||
81 D 479 | 82 F 480 | 83 G 481 | 84 L 482 | 85 S 483 | |||||||||||||||
■ |
Binding affinities
ChEMBL ID:CHEMBL388978Bioaffinities: 1829 records for 404 kinase(s)
Species | Kinase (ChEMBL naming) | Median | Min | Max | Type | Records |
---|---|---|---|---|---|---|
Homo sapiens | 3-phosphoinositide dependent protein kinase-1 | 8 | 8 | 8.3 | pIC50 | 2 |
Homo sapiens | 3-phosphoinositide dependent protein kinase-1 | 8.8 | 8.8 | 8.8 | pKd | 2 |
Homo sapiens | Activin receptor type-1 | 5 | 5 | 5 | pIC50 | 1 |
Homo sapiens | Activin receptor type-1 | 6.3 | 6.3 | 6.3 | pKd | 2 |
Homo sapiens | Activin receptor type-1B | 5 | 5 | 5 | pIC50 | 1 |
Homo sapiens | Activin receptor type-1B | 6.2 | 6.2 | 6.2 | pKd | 2 |
Homo sapiens | Activin receptor type-2A | 5.1 | 5.1 | 5.1 | pKd | 1 |
Homo sapiens | Activin receptor type-2B | 5.3 | 5.3 | 5.3 | pKd | 2 |
Homo sapiens | Adaptor-associated kinase | 8.9 | 8.9 | 8.9 | pKd | 3 |
Homo sapiens | ALK tyrosine kinase receptor | 8.5 | 7.5 | 9.2 | pIC50 | 15 |
Homo sapiens | ALK tyrosine kinase receptor | 7.5 | 7.5 | 7.5 | pKd | 2 |
Homo sapiens | AMP-activated protein kinase, alpha-1 subunit | 8.4 | 8.1 | 8.4 | pKd | 3 |
Homo sapiens | AMP-activated protein kinase, alpha-2 subunit | 7.9 | 7.9 | 7.9 | pKd | 2 |
Homo sapiens | Ankyrin repeat and protein kinase domain-containing protein 1 | 6.6 | 6.6 | 6.6 | pKd | 2 |
Homo sapiens | Beta-adrenergic receptor kinase 2 | 6.1 | 6.1 | 6.1 | pIC50 | 1 |
Homo sapiens | BMP-2-inducible protein kinase | 8.3 | 8.3 | 8.4 | pKd | 3 |
Homo sapiens | Bone morphogenetic protein receptor type-1A | 5.4 | 5.4 | 5.4 | pIC50 | 1 |
Homo sapiens | Bone morphogenetic protein receptor type-1A | 5.4 | 5.4 | 5.4 | pKd | 2 |
Homo sapiens | Bone morphogenetic protein receptor type-1B | 6.8 | 6.8 | 6.8 | pKd | 1 |
Homo sapiens | Bone morphogenetic protein receptor type-2 | 6 | 6 | 6 | pIC50 | 1 |
Homo sapiens | Bone morphogenetic protein receptor type-2 | 5.6 | 5.6 | 5.6 | pKd | 1 |
Homo sapiens | BR serine/threonine-protein kinase 1 | 9.1 | 9.1 | 9.1 | pIC50 | 1 |
Homo sapiens | BR serine/threonine-protein kinase 1 | 7.6 | 7.6 | 7.6 | pKd | 2 |
Homo sapiens | BR serine/threonine-protein kinase 2 | 8.6 | 8.6 | 8.6 | pIC50 | 1 |
Homo sapiens | BR serine/threonine-protein kinase 2 | 8.5 | 8.5 | 8.5 | pKd | 2 |
Homo sapiens | Calcium/calmodulin-dependent protein kinase type 1B | 8.3 | 8.3 | 8.3 | pIC50 | 1 |
Plasmodium falciparum | Calcium-dependent protein kinase 1 | 9.6 | 9.6 | 9.6 | pKd | 1 |
Homo sapiens | CaM kinase I alpha | 8.5 | 8.5 | 8.5 | pIC50 | 1 |
Homo sapiens | CaM kinase I alpha | 7.6 | 7.5 | 7.6 | pKd | 3 |
Homo sapiens | CaM kinase I delta | 9.5 | 9.5 | 9.5 | pIC50 | 1 |
Homo sapiens | CaM kinase I delta | 9 | 8.7 | 9 | pKd | 3 |
Homo sapiens | CaM kinase I gamma | 8.3 | 8.3 | 8.3 | pIC50 | 1 |
Homo sapiens | CaM kinase I gamma | 7.6 | 7.3 | 7.6 | pKd | 3 |
Homo sapiens | CaM kinase II alpha | 10.2 | 10.2 | 10.2 | pIC50 | 1 |
Homo sapiens | CaM kinase II alpha | 9.8 | 9.8 | 10 | pKd | 3 |
Homo sapiens | CaM kinase II beta | 10 | 10 | 10.2 | pIC50 | 2 |
Homo sapiens | CaM kinase II beta | 8.9 | 8.5 | 8.9 | pKd | 3 |
Homo sapiens | CaM kinase II delta | 10.5 | 10.5 | 10.5 | pIC50 | 1 |
Homo sapiens | CaM kinase II delta | 9.5 | 9.3 | 9.5 | pKd | 3 |
Homo sapiens | CaM kinase II gamma | 9.4 | 9.4 | 9.4 | pIC50 | 1 |
Homo sapiens | CaM kinase II gamma | 9.3 | 9.3 | 9.3 | pKd | 3 |
Homo sapiens | CaM kinase IV | 6.8 | 6.8 | 6.8 | pIC50 | 1 |
Homo sapiens | CaM kinase IV | 7.4 | 7.4 | 7.4 | pKd | 2 |
Homo sapiens | CaM-kinase kinase alpha | 7.4 | 7.4 | 7.4 | pIC50 | 1 |
Homo sapiens | CaM-kinase kinase alpha | 10.4 | 10.3 | 10.4 | pKd | 3 |
Homo sapiens | CaM-kinase kinase beta | 7.5 | 7.5 | 7.5 | pIC50 | 1 |
Homo sapiens | CaM-kinase kinase beta | 9.8 | 9.8 | 10.3 | pKd | 3 |
Bos taurus | cAMP-dependent protein kinase alpha-catalytic subunit | 7.4 | 7.4 | 7.4 | pIC50 | 1 |
Homo sapiens | cAMP-dependent protein kinase alpha-catalytic subunit | 8.8 | 8.6 | 9 | pIC50 | 3 |
Homo sapiens | cAMP-dependent protein kinase alpha-catalytic subunit | 7.7 | 7.7 | 7.7 | pKd | 2 |
Rattus norvegicus | cAMP-dependent protein kinase alpha-catalytic subunit | 7.6 | 6.9 | 7.8 | pIC50 | 3 |
Homo sapiens | cAMP-dependent protein kinase beta-1 catalytic subunit | 7.5 | 7.5 | 8.9 | pIC50 | 2 |
Homo sapiens | cAMP-dependent protein kinase beta-1 catalytic subunit | 7.5 | 7.5 | 7.5 | pKd | 2 |
Homo sapiens | cAMP-dependent protein kinase, gamma catalytic subunit | 8.2 | 8.2 | 8.2 | pIC50 | 1 |
Homo sapiens | Casein kinase I alpha | 5.4 | 5.4 | 5.4 | pIC50 | 2 |
Homo sapiens | Casein kinase I alpha | 6 | 6 | 6 | pKd | 1 |
Homo sapiens | Casein kinase I delta | 5.6 | 5.6 | 5.6 | pKd | 2 |
Homo sapiens | Casein kinase I epsilon | 7.1 | 6.2 | 7.1 | pKd | 3 |
Homo sapiens | Casein kinase I gamma 1 | 5.1 | 5.1 | 5.1 | pIC50 | 1 |
Homo sapiens | Casein kinase I gamma 1 | 5.5 | 5.5 | 5.5 | pKd | 1 |
Homo sapiens | Casein kinase I gamma 2 | 5.5 | 5.5 | 5.5 | pIC50 | 1 |
Homo sapiens | Casein kinase I gamma 2 | 6.1 | 5.9 | 6.1 | pKd | 3 |
Homo sapiens | Casein kinase II alpha | 5.4 | 5.4 | 5.4 | pIC50 | 1 |
Homo sapiens | Casein kinase II alpha | 6 | 6 | 7.4 | pKd | 2 |
Homo sapiens | Casein kinase II alpha (prime) | 6.1 | 6.1 | 6.1 | pIC50 | 1 |
Homo sapiens | Casein kinase II alpha (prime) | 6.6 | 6.6 | 8.2 | pKd | 2 |
Homo sapiens | Casein kinase I isoform alpha-like | 5.6 | 5.6 | 5.6 | pIC50 | 1 |
Homo sapiens | Casein kinase I isoform alpha-like | 6.6 | 6.6 | 6.6 | pKd | 2 |
Homo sapiens | Casein kinase I isoform gamma-3 | 5.5 | 5.5 | 5.5 | pIC50 | 1 |
Plasmodium falciparum (isolate 3D7) | Cell division control protein 2 homolog | 6.1 | 6.1 | 6.1 | pKd | 1 |
Homo sapiens | Cell division cycle 2-like protein kinase 6 | 6.7 | 6.7 | 6.7 | pKd | 2 |
Homo sapiens | Cell division protein kinase 8 | 6.3 | 6.3 | 6.3 | pKd | 2 |
Bos taurus | cGMP-dependent protein kinase 1 alpha | 7.8 | 7.8 | 7.8 | pIC50 | 2 |
Homo sapiens | cGMP-dependent protein kinase 1 beta | 8.6 | 8.3 | 8.9 | pIC50 | 3 |
Homo sapiens | cGMP-dependent protein kinase 1 beta | 7.5 | 7.5 | 7.5 | pKd | 2 |
Homo sapiens | cGMP-dependent protein kinase 2 | 8.2 | 8.2 | 8.2 | pIC50 | 1 |
Homo sapiens | cGMP-dependent protein kinase 2 | 7.8 | 7.8 | 7.8 | pKd | 2 |
Homo sapiens | Citron Rho-interacting kinase | 6 | 6 | 6 | pIC50 | 1 |
Homo sapiens | Citron Rho-interacting kinase | 6.5 | 6.5 | 6.5 | pKd | 2 |
Homo sapiens | c-Jun N-terminal kinase 1 | 6.2 | 5.5 | 6.4 | pIC50 | 5 |
Homo sapiens | c-Jun N-terminal kinase 1 | 6.7 | 6.3 | 6.7 | pKd | 3 |
Homo sapiens | c-Jun N-terminal kinase 2 | 5.6 | 5.5 | 5.7 | pIC50 | 3 |
Homo sapiens | c-Jun N-terminal kinase 2 | 6 | 6 | 6 | pKd | 2 |
Homo sapiens | c-Jun N-terminal kinase 3 | 7 | 6.5 | 7 | pKd | 3 |
Homo sapiens | Cyclin-dependent kinase 1 | 8.1 | 7.8 | 9.4 | pIC50 | 4 |
Mus musculus | Cyclin-dependent kinase 1 | 8.1 | 8.1 | 8.1 | pIC50 | 1 |
Homo sapiens | Cyclin-dependent kinase 13 | 7.2 | 7.2 | 7.2 | pKd | 1 |
Homo sapiens | Cyclin-dependent kinase 2 | 8.9 | 8.4 | 10 | pIC50 | 5 |
Homo sapiens | Cyclin-dependent kinase 2 | 8.2 | 8.1 | 8.2 | pKd | 3 |
Homo sapiens | Cyclin-dependent kinase 3 | 8.2 | 8.2 | 8.2 | pIC50 | 1 |
Homo sapiens | Cyclin-dependent kinase 3 | 7.5 | 7.5 | 7.5 | pKd | 2 |
Homo sapiens | Cyclin-dependent kinase 4 | 7.3 | 7.3 | 7.7 | pKd | 2 |
Homo sapiens | Cyclin-dependent kinase 5 | 7.1 | 7.1 | 7.1 | pKd | 3 |
Homo sapiens | Cyclin-dependent kinase 7 | 7.4 | 7.4 | 7.4 | pKd | 2 |
Homo sapiens | Cyclin-dependent kinase 9 | 7 | 7 | 7 | pKd | 2 |
Homo sapiens | Cyclin-dependent kinase-like 1 | 6.5 | 6.5 | 6.5 | pKd | 1 |
Homo sapiens | Cyclin-dependent kinase-like 2 | 6.3 | 6.3 | 6.3 | pKd | 1 |
Homo sapiens | Cyclin-dependent kinase-like 3 | 5.3 | 5.3 | 5.3 | pKd | 1 |
Homo sapiens | Cyclin-dependent kinase-like 5 | 6.5 | 6.5 | 6.5 | pKd | 1 |
Homo sapiens | Death-associated protein kinase 1 | 7.9 | 7.8 | 9.3 | pIC50 | 5 |
Homo sapiens | Death-associated protein kinase 1 | 8.9 | 8.9 | 8.9 | pKd | 2 |
Homo sapiens | Death-associated protein kinase 2 | 8.1 | 8.1 | 8.1 | pIC50 | 1 |
Homo sapiens | Death-associated protein kinase 2 | 8.8 | 8.5 | 8.8 | pKd | 3 |
Homo sapiens | Death-associated protein kinase 3 | 8.5 | 8.5 | 8.5 | pIC50 | 1 |
Homo sapiens | Death-associated protein kinase 3 | 9 | 5.8 | 9 | pKd | 4 |
Homo sapiens | Discoidin domain-containing receptor 2 | 8.9 | 8.9 | 8.9 | pIC50 | 1 |
Homo sapiens | Discoidin domain-containing receptor 2 | 7.4 | 7.4 | 7.4 | pKd | 2 |
Homo sapiens | Dual serine/threonine and tyrosine protein kinase | 7.2 | 7.2 | 7.2 | pIC50 | 2 |
Homo sapiens | Dual serine/threonine and tyrosine protein kinase | 8 | 8 | 8 | pKd | 1 |
Homo sapiens | Dual specificity mitogen-activated protein kinase kinase 1 | 7.6 | 6.2 | 8.6 | pIC50 | 9 |
Homo sapiens | Dual specificity mitogen-activated protein kinase kinase 1 | 7.7 | 7.7 | 7.7 | pKd | 2 |
Homo sapiens | Dual specificity mitogen-activated protein kinase kinase 2 | 7.4 | 7.4 | 7.4 | pIC50 | 1 |
Homo sapiens | Dual specificity mitogen-activated protein kinase kinase 2 | 7.6 | 7.6 | 7.6 | pKd | 2 |
Homo sapiens | Dual specificity mitogen-activated protein kinase kinase 3 | 7.8 | 7.8 | 7.8 | pIC50 | 1 |
Homo sapiens | Dual specificity mitogen-activated protein kinase kinase 3 | 8.3 | 8.3 | 8.3 | pKd | 2 |
Homo sapiens | Dual specificity mitogen-activated protein kinase kinase 4 | 5.8 | 5.8 | 5.8 | pIC50 | 1 |
Homo sapiens | Dual specificity mitogen-activated protein kinase kinase 4 | 7.2 | 7.2 | 7.2 | pKd | 2 |
Homo sapiens | Dual specificity mitogen-activated protein kinase kinase 5 | 7.4 | 7.4 | 7.4 | pIC50 | 1 |
Homo sapiens | Dual specificity mitogen-activated protein kinase kinase 5 | 8.5 | 8.5 | 8.5 | pKd | 1 |
Homo sapiens | Dual specificity mitogen-activated protein kinase kinase 6 | 8.1 | 8.1 | 8.1 | pIC50 | 1 |
Homo sapiens | Dual specificity mitogen-activated protein kinase kinase 6 | 8.5 | 8.5 | 8.5 | pKd | 2 |
Homo sapiens | Dual specificity mitogen-activated protein kinase kinase 7 | 5.9 | 5.9 | 5.9 | pIC50 | 1 |
Homo sapiens | Dual specificity mitogen-activated protein kinase kinase 7 | 7.5 | 7.5 | 7.5 | pKd | 1 |
Homo sapiens | Dual specificity protein kinase CLK2 | 8.3 | 8.3 | 8.3 | pIC50 | 1 |
Homo sapiens | Dual specificity protein kinase CLK2 | 8.1 | 7.9 | 8.1 | pKd | 3 |
Homo sapiens | Dual specificity protein kinase CLK3 | 5.9 | 5.9 | 5.9 | pIC50 | 1 |
Homo sapiens | Dual specificity protein kinase CLK3 | 6 | 5.5 | 6 | pKd | 3 |
Homo sapiens | Dual specificity protein kinase CLK4 | 7.5 | 7.5 | 7.5 | pIC50 | 1 |
Homo sapiens | Dual specificity protein kinase CLK4 | 8 | 7.8 | 8 | pKd | 3 |
Homo sapiens | Dual specificity protein kinase TTK | 7.2 | 7 | 7.2 | pKd | 3 |
Homo sapiens | Dual specificity testis-specific protein kinase 1 | 6.6 | 6.6 | 6.6 | pIC50 | 1 |
Homo sapiens | Dual specificity testis-specific protein kinase 1 | 6.5 | 6.5 | 6.5 | pKd | 2 |
Homo sapiens | Dual-specificity tyrosine-phosphorylation regulated kinase 1A | 7.7 | 7.7 | 8.3 | pIC50 | 2 |
Homo sapiens | Dual-specificity tyrosine-phosphorylation regulated kinase 1A | 8.4 | 8.4 | 8.4 | pKd | 1 |
Homo sapiens | Dual specificity tyrosine-phosphorylation-regulated kinase 1B | 9 | 9 | 9 | pIC50 | 1 |
Homo sapiens | Dual specificity tyrosine-phosphorylation-regulated kinase 1B | 7.6 | 7.6 | 7.6 | pKd | 2 |
Homo sapiens | Dual-specificity tyrosine-phosphorylation regulated kinase 2 | 6.6 | 6.6 | 6.6 | pIC50 | 1 |
Homo sapiens | Dual-specificity tyrosine-phosphorylation regulated kinase 2 | 6.6 | 6.6 | 6.6 | pKd | 1 |
Homo sapiens | Dual-specificity tyrosine-phosphorylation regulated kinase 3 | 7.5 | 7.5 | 7.5 | pIC50 | 1 |
Homo sapiens | Dual specificty protein kinase CLK1 | 7.9 | 7.9 | 7.9 | pIC50 | 1 |
Homo sapiens | Dual specificty protein kinase CLK1 | 7.5 | 7.5 | 7.6 | pKd | 3 |
Homo sapiens | Ephrin type-A receptor 1 | 6.9 | 6.9 | 7.3 | pIC50 | 2 |
Homo sapiens | Ephrin type-A receptor 1 | 6.5 | 6.5 | 6.5 | pKd | 2 |
Homo sapiens | Ephrin type-A receptor 2 | 6.6 | 6.6 | 7.1 | pIC50 | 2 |
Homo sapiens | Ephrin type-A receptor 2 | 5.9 | 5.9 | 6.1 | pKd | 3 |
Homo sapiens | Ephrin type-A receptor 3 | 7.5 | 7.3 | 7.7 | pIC50 | 3 |
Homo sapiens | Ephrin type-A receptor 3 | 7.6 | 7.3 | 7.6 | pKd | 3 |
Homo sapiens | Ephrin type-A receptor 4 | 7.9 | 7.9 | 7.9 | pIC50 | 1 |
Homo sapiens | Ephrin type-A receptor 4 | 6.5 | 6.2 | 6.5 | pKd | 3 |
Homo sapiens | Ephrin type-A receptor 5 | 7.7 | 7.7 | 7.7 | pIC50 | 1 |
Homo sapiens | Ephrin type-A receptor 5 | 7 | 6.8 | 7 | pKd | 3 |
Homo sapiens | Ephrin type-A receptor 6 | 7.9 | 7.9 | 7.9 | pIC50 | 1 |
Homo sapiens | Ephrin type-A receptor 6 | 6.5 | 6.5 | 6.6 | pKd | 3 |
Homo sapiens | Ephrin type-A receptor 7 | 7.3 | 7.3 | 7.3 | pIC50 | 1 |
Homo sapiens | Ephrin type-A receptor 7 | 6.2 | 6.2 | 6.2 | pKd | 3 |
Homo sapiens | Ephrin type-A receptor 8 | 6.9 | 6.9 | 6.9 | pIC50 | 1 |
Homo sapiens | Ephrin type-A receptor 8 | 6.7 | 6.5 | 6.7 | pKd | 3 |
Homo sapiens | Ephrin type-B receptor 1 | 6.9 | 6.9 | 7.2 | pIC50 | 2 |
Homo sapiens | Ephrin type-B receptor 1 | 6.6 | 6.2 | 6.6 | pKd | 3 |
Homo sapiens | Ephrin type-B receptor 2 | 6.7 | 6.7 | 6.9 | pIC50 | 2 |
Homo sapiens | Ephrin type-B receptor 2 | 5.7 | 5.7 | 5.7 | pKd | 2 |
Homo sapiens | Ephrin type-B receptor 3 | 5.7 | 5.7 | 5.7 | pIC50 | 1 |
Homo sapiens | Ephrin type-B receptor 4 | 6.6 | 6.6 | 6.9 | pIC50 | 3 |
Homo sapiens | Ephrin type-B receptor 4 | 5.7 | 5.7 | 5.7 | pKd | 1 |
Homo sapiens | Ephrin type-B receptor 6 | 6.7 | 6.7 | 6.7 | pKd | 1 |
Homo sapiens | Epidermal growth factor receptor erbB1 | 7.3 | 6.6 | 9.5 | pIC50 | 27 |
Homo sapiens | Epidermal growth factor receptor erbB1 | 6.5 | 6 | 9.5 | pKd | 23 |
Homo sapiens | Epithelial discoidin domain-containing receptor 1 | 8.4 | 8.4 | 8.4 | pIC50 | 1 |
Homo sapiens | Epithelial discoidin domain-containing receptor 1 | 7.7 | 7.7 | 7.7 | pKd | 2 |
Homo sapiens | Eukaryotic translation initiation factor 2-alpha kinase 4 | 7.8 | 7.8 | 7.8 | pKd | 2 |
Homo sapiens | Fibroblast growth factor receptor 1 | 8.2 | 8.1 | 8.4 | pIC50 | 3 |
Homo sapiens | Fibroblast growth factor receptor 1 | 7.1 | 7.1 | 7.2 | pKd | 3 |
Homo sapiens | Fibroblast growth factor receptor 2 | 8.5 | 7.5 | 8.8 | pIC50 | 5 |
Homo sapiens | Fibroblast growth factor receptor 2 | 7 | 6.8 | 7 | pKd | 3 |
Homo sapiens | Fibroblast growth factor receptor 3 | 7.8 | 7.8 | 8 | pIC50 | 6 |
Homo sapiens | Fibroblast growth factor receptor 3 | 7 | 6.5 | 7.1 | pKd | 5 |
Homo sapiens | Fibroblast growth factor receptor 4 | 6.8 | 6.8 | 7 | pIC50 | 2 |
Homo sapiens | Fibroblast growth factor receptor 4 | 6.6 | 6.6 | 6.6 | pKd | 2 |
Homo sapiens | Focal adhesion kinase 1 | 7.3 | 5.5 | 8 | pIC50 | 10 |
Homo sapiens | Focal adhesion kinase 1 | 7.2 | 7.2 | 7.2 | pKd | 3 |
Homo sapiens | Glycogen synthase kinase-3 alpha | 7.6 | 7.6 | 8.6 | pIC50 | 2 |
Homo sapiens | Glycogen synthase kinase-3 alpha | 6.9 | 6.9 | 6.9 | pKd | 2 |
Homo sapiens | Glycogen synthase kinase-3 beta | 7.5 | 6.7 | 8.6 | pIC50 | 31 |
Homo sapiens | Glycogen synthase kinase-3 beta | 7.2 | 7.2 | 7.2 | pKd | 2 |
Homo sapiens | Glycogen synthase kinase-3 beta | 7.7 | 7.7 | 7.7 | pKi | 1 |
Homo sapiens | G-protein coupled receptor kinase 2 | 5.8 | 5.8 | 5.8 | pIC50 | 1 |
Homo sapiens | G protein-coupled receptor kinase 4 | 7 | 7 | 7 | pIC50 | 1 |
Homo sapiens | G protein-coupled receptor kinase 4 | 7.4 | 7.4 | 7.4 | pKd | 1 |
Homo sapiens | G protein-coupled receptor kinase 5 | 7.1 | 7.1 | 7.1 | pIC50 | 1 |
Homo sapiens | G protein-coupled receptor kinase 6 | 4.5 | 4.5 | 7.2 | pIC50 | 2 |
Homo sapiens | G protein-coupled receptor kinase 7 | 8.2 | 8.2 | 8.2 | pIC50 | 1 |
Homo sapiens | G protein-coupled receptor kinase 7 | 9.1 | 9.1 | 9.1 | pKd | 1 |
Homo sapiens | Hepatocyte growth factor receptor | 6.9 | 6 | 7.2 | pIC50 | 15 |
Homo sapiens | Hepatocyte growth factor receptor | 6.7 | 6.7 | 6.9 | pKd | 4 |
Homo sapiens | Hexokinase type IV | 9.1 | 9.1 | 9.1 | pIC50 | 1 |
Homo sapiens | Homeodomain-interacting protein kinase 1 | 5.6 | 5.6 | 5.6 | pIC50 | 1 |
Homo sapiens | Homeodomain-interacting protein kinase 1 | 5.6 | 5.6 | 5.6 | pKd | 1 |
Homo sapiens | Homeodomain-interacting protein kinase 2 | 6.2 | 6.2 | 6.2 | pIC50 | 1 |
Homo sapiens | Homeodomain-interacting protein kinase 2 | 6.7 | 6.7 | 6.7 | pKd | 1 |
Homo sapiens | Homeodomain-interacting protein kinase 3 | 6.2 | 6.2 | 6.2 | pIC50 | 1 |
Homo sapiens | Homeodomain-interacting protein kinase 3 | 7.1 | 7.1 | 7.1 | pKd | 1 |
Homo sapiens | Homeodomain-interacting protein kinase 4 | 6.5 | 6.5 | 6.5 | pIC50 | 1 |
Homo sapiens | Homeodomain-interacting protein kinase 4 | 6.4 | 6.4 | 6.4 | pKd | 1 |
Homo sapiens | Hormonally up-regulated neu tumor-associated kinase | 6.2 | 6.2 | 6.2 | pKd | 1 |
Homo sapiens | Inhibitor of nuclear factor kappa B kinase alpha subunit | 6.6 | 6.6 | 7.4 | pIC50 | 3 |
Homo sapiens | Inhibitor of nuclear factor kappa B kinase alpha subunit | 8.2 | 8.2 | 8.2 | pKd | 1 |
Homo sapiens | Inhibitor of nuclear factor kappa B kinase beta subunit | 6.3 | 5.9 | 9.1 | pIC50 | 8 |
Homo sapiens | Inhibitor of nuclear factor kappa B kinase beta subunit | 7.5 | 7.5 | 7.5 | pKd | 1 |
Homo sapiens | Inhibitor of nuclear factor kappa B kinase epsilon subunit | 9.4 | 9.4 | 9.4 | pIC50 | 1 |
Homo sapiens | Inhibitor of nuclear factor kappa B kinase epsilon subunit | 8.3 | 8.3 | 8.3 | pKd | 2 |
Homo sapiens | Insulin-like growth factor I receptor | 6.7 | 5.8 | 7.5 | pIC50 | 12 |
Homo sapiens | Insulin-like growth factor I receptor | 6.7 | 6.7 | 6.7 | pKd | 2 |
Homo sapiens | Insulin receptor | 7.8 | 7.1 | 8.1 | pIC50 | 4 |
Homo sapiens | Insulin receptor | 7 | 7 | 7.1 | pKd | 3 |
Mus musculus | Insulin receptor | 6.7 | 6.7 | 6.7 | pIC50 | 1 |
Homo sapiens | Insulin receptor-related protein | 7.8 | 7.8 | 7.8 | pIC50 | 1 |
Homo sapiens | Insulin receptor-related protein | 7.1 | 7.1 | 7.1 | pKd | 2 |
Homo sapiens | Interferon-induced, double-stranded RNA-activated protein kinase | 6.4 | 6.4 | 6.4 | pKd | 2 |
Homo sapiens | Interleukin-1 receptor-associated kinase 1 | 7.2 | 7.2 | 7.2 | pIC50 | 1 |
Homo sapiens | Interleukin-1 receptor-associated kinase 1 | 7.4 | 7.4 | 7.4 | pKd | 1 |
Homo sapiens | Interleukin-1 receptor-associated kinase 3 | 7.9 | 7.9 | 7.9 | pKd | 2 |
Homo sapiens | Interleukin-1 receptor-associated kinase 4 | 8.2 | 7.5 | 8.4 | pIC50 | 3 |
Homo sapiens | Interleukin-1 receptor-associated kinase 4 | 8.8 | 8.8 | 8.8 | pKd | 1 |
Homo sapiens | Kinase suppressor of Ras 1 | 5.1 | 5.1 | 5.1 | pIC50 | 1 |
Homo sapiens | Kinase suppressor of Ras 2 | 5.2 | 5.2 | 5.2 | pIC50 | 1 |
Homo sapiens | Leucine-rich repeat serine/threonine-protein kinase 2 | 7.8 | 7.8 | 9 | pIC50 | 2 |
Homo sapiens | Leucine-rich repeat serine/threonine-protein kinase 2 | 8.5 | 8.5 | 9.4 | pKd | 2 |
Homo sapiens | Leukocyte tyrosine kinase receptor | 7.5 | 7.5 | 8.4 | pIC50 | 2 |
Homo sapiens | Leukocyte tyrosine kinase receptor | 7.4 | 7.4 | 7.4 | pKd | 2 |
Homo sapiens | LIM domain kinase 1 | 8.6 | 8.6 | 8.6 | pIC50 | 1 |
Homo sapiens | LIM domain kinase 1 | 6.3 | 6.2 | 6.3 | pKd | 3 |
Homo sapiens | LIM domain kinase 2 | 7 | 7 | 7 | pIC50 | 1 |
Homo sapiens | LIM domain kinase 2 | 5 | 5 | 5 | pKd | 2 |
Homo sapiens | Macrophage colony stimulating factor receptor | 8.5 | 6 | 8.9 | pIC50 | 4 |
Homo sapiens | Macrophage colony stimulating factor receptor | 7.9 | 7.9 | 7.9 | pKd | 2 |
Homo sapiens | Macrophage-stimulating protein receptor | 6.5 | 6.4 | 7 | pIC50 | 4 |
Homo sapiens | Macrophage-stimulating protein receptor | 6.4 | 6.4 | 6.4 | pKd | 1 |
Homo sapiens | MAP kinase-activated protein kinase 2 | 6.4 | 5.5 | 7.4 | pIC50 | 9 |
Homo sapiens | MAP kinase-activated protein kinase 2 | 6.1 | 6.1 | 6.1 | pKd | 2 |
Homo sapiens | MAP kinase-activated protein kinase 3 | 5.5 | 5.5 | 5.5 | pIC50 | 1 |
Homo sapiens | MAP kinase-activated protein kinase 5 | 6.5 | 6.5 | 6.5 | pIC50 | 1 |
Homo sapiens | MAP kinase-activated protein kinase 5 | 6.6 | 6.6 | 6.6 | pKd | 1 |
Homo sapiens | MAP kinase ERK1 | 5.2 | 4.5 | 5.9 | pIC50 | 10 |
Homo sapiens | MAP kinase ERK1 | 5.1 | 5.1 | 5.1 | pKd | 2 |
Homo sapiens | MAP kinase ERK2 | 5.9 | 4.5 | 8.6 | pIC50 | 9 |
Homo sapiens | MAP kinase ERK2 | 5.1 | 5.1 | 5.1 | pKd | 2 |
Homo sapiens | MAP kinase-interacting serine/threonine-protein kinase MNK1 | 7.3 | 7.3 | 7.3 | pIC50 | 1 |
Homo sapiens | MAP kinase-interacting serine/threonine-protein kinase MNK1 | 6.8 | 6.8 | 6.8 | pKd | 2 |
Homo sapiens | MAP kinase p38 alpha | 5.2 | 5.2 | 8 | pIC50 | 2 |
Homo sapiens | MAP kinase p38 delta | 6.8 | 6.8 | 6.8 | pIC50 | 1 |
Homo sapiens | MAP kinase p38 delta | 6.6 | 6.6 | 6.6 | pKd | 1 |
Homo sapiens | MAP kinase p38 gamma | 6.6 | 6.6 | 6.6 | pIC50 | 1 |
Homo sapiens | MAP kinase p38 gamma | 7.4 | 7 | 7.4 | pKd | 3 |
Homo sapiens | MAP kinase signal-integrating kinase 2 | 7.6 | 7.6 | 7.7 | pIC50 | 2 |
Homo sapiens | MAP kinase signal-integrating kinase 2 | 7.8 | 7.7 | 7.8 | pKd | 3 |
Homo sapiens | MAP/microtubule affinity-regulating kinase 2 | 9.9 | 9.9 | 9.9 | pIC50 | 1 |
Homo sapiens | MAP/microtubule affinity-regulating kinase 2 | 9.2 | 9.2 | 10 | pKd | 3 |
Homo sapiens | MAP/microtubule affinity-regulating kinase 4 | 9.9 | 9.9 | 9.9 | pIC50 | 1 |
Homo sapiens | MAP/microtubule affinity-regulating kinase 4 | 8.3 | 8.3 | 8.3 | pKd | 2 |
Homo sapiens | Maternal embryonic leucine zipper kinase | 9.3 | 9.3 | 9.3 | pIC50 | 1 |
Homo sapiens | Maternal embryonic leucine zipper kinase | 7.5 | 7.5 | 7.5 | pKd | 2 |
Homo sapiens | Microtubule-associated serine/threonine-protein kinase 1 | 6.8 | 6.8 | 6.8 | pKd | 1 |
Homo sapiens | Misshapen-like kinase 1 | 9.3 | 9.3 | 9.4 | pIC50 | 3 |
Homo sapiens | Misshapen-like kinase 1 | 9 | 9 | 9 | pKd | 1 |
Homo sapiens | Mitogen-activated protein kinase 15 | 8.1 | 8.1 | 8.1 | pIC50 | 2 |
Homo sapiens | Mitogen-activated protein kinase 15 | 7.5 | 7.5 | 7.5 | pKd | 2 |
Homo sapiens | Mitogen-activated protein kinase 6 | 5.5 | 5.5 | 5.5 | pKd | 1 |
Homo sapiens | Mitogen-activated protein kinase 7 | 5.2 | 4.9 | 6.9 | pIC50 | 3 |
Homo sapiens | Mitogen-activated protein kinase 7 | 5.8 | 5.8 | 5.8 | pKd | 2 |
Homo sapiens | Mitogen-activated protein kinase kinase kinase 1 | 6.3 | 6.3 | 6.3 | pIC50 | 1 |
Homo sapiens | Mitogen-activated protein kinase kinase kinase 1 | 6.5 | 6.5 | 6.5 | pKd | 1 |
Homo sapiens | Mitogen-activated protein kinase kinase kinase 10 | 8.6 | 8.6 | 8.6 | pIC50 | 1 |
Homo sapiens | Mitogen-activated protein kinase kinase kinase 10 | 7.3 | 7.3 | 7.3 | pKd | 2 |
Homo sapiens | Mitogen-activated protein kinase kinase kinase 11 | 8.4 | 8.4 | 8.4 | pIC50 | 1 |
Homo sapiens | Mitogen-activated protein kinase kinase kinase 11 | 7.7 | 7.7 | 7.7 | pKd | 3 |
Homo sapiens | Mitogen-activated protein kinase kinase kinase 12 | 6.8 | 6.8 | 6.8 | pIC50 | 1 |
Homo sapiens | Mitogen-activated protein kinase kinase kinase 12 | 5.8 | 5.8 | 5.8 | pKd | 1 |
Homo sapiens | Mitogen-activated protein kinase kinase kinase 13 | 6.7 | 6.7 | 6.7 | pKd | 1 |
Homo sapiens | Mitogen-activated protein kinase kinase kinase 14 | 5.6 | 5.6 | 5.6 | pIC50 | 1 |
Homo sapiens | Mitogen-activated protein kinase kinase kinase 15 | 8.6 | 8.6 | 8.6 | pKd | 1 |
Homo sapiens | Mitogen-activated protein kinase kinase kinase 2 | 7.4 | 7.4 | 7.4 | pIC50 | 1 |
Homo sapiens | Mitogen-activated protein kinase kinase kinase 2 | 8.6 | 8.6 | 8.6 | pKd | 1 |
Homo sapiens | Mitogen-activated protein kinase kinase kinase 3 | 8 | 8 | 8 | pIC50 | 1 |
Homo sapiens | Mitogen-activated protein kinase kinase kinase 3 | 5.6 | 5.6 | 5.6 | pKd | 1 |
Homo sapiens | Mitogen-activated protein kinase kinase kinase 4 | 5.9 | 5.7 | 5.9 | pKd | 3 |
Homo sapiens | Mitogen-activated protein kinase kinase kinase 5 | 7.4 | 6 | 9.2 | pIC50 | 4 |
Homo sapiens | Mitogen-activated protein kinase kinase kinase 5 | 7 | 6.9 | 7 | pKd | 4 |
Homo sapiens | Mitogen-activated protein kinase kinase kinase 6 | 6.3 | 6.3 | 6.3 | pIC50 | 1 |
Homo sapiens | Mitogen-activated protein kinase kinase kinase 6 | 6.6 | 6.6 | 6.6 | pKd | 1 |
Homo sapiens | Mitogen-activated protein kinase kinase kinase 7 | 7.4 | 7.2 | 7.5 | pIC50 | 3 |
Homo sapiens | Mitogen-activated protein kinase kinase kinase 7 | 7.2 | 7.2 | 7.2 | pKd | 1 |
Homo sapiens | Mitogen-activated protein kinase kinase kinase 9 | 8.8 | 8.8 | 8.8 | pIC50 | 1 |
Homo sapiens | Mitogen-activated protein kinase kinase kinase 9 | 8 | 8 | 8 | pKd | 2 |
Homo sapiens | Mitogen-activated protein kinase kinase kinase kinase 1 | 8.4 | 8.4 | 8.4 | pKd | 2 |
Homo sapiens | Mitogen-activated protein kinase kinase kinase kinase 2 | 8.1 | 8.1 | 8.1 | pKd | 1 |
Homo sapiens | Mitogen-activated protein kinase kinase kinase kinase 3 | 10.1 | 10.1 | 10.1 | pIC50 | 1 |
Homo sapiens | Mitogen-activated protein kinase kinase kinase kinase 3 | 8.1 | 8.1 | 8.1 | pKd | 2 |
Homo sapiens | Mitogen-activated protein kinase kinase kinase kinase 4 | 9.2 | 9.2 | 9.2 | pIC50 | 1 |
Homo sapiens | Mitogen-activated protein kinase kinase kinase kinase 4 | 7.6 | 7.6 | 7.6 | pKd | 2 |
Homo sapiens | Mitogen-activated protein kinase kinase kinase kinase 5 | 9.5 | 9.5 | 9.5 | pIC50 | 1 |
Homo sapiens | Mitogen-activated protein kinase kinase kinase kinase 5 | 7.8 | 7.6 | 7.8 | pKd | 3 |
Homo sapiens | Mitogen-activated protein kinase kinase kinase MLK4 | 5.8 | 5.8 | 5.8 | pIC50 | 1 |
Homo sapiens | Muscle, skeletal receptor tyrosine protein kinase | 6.5 | 6.5 | 8.4 | pIC50 | 2 |
Homo sapiens | Muscle, skeletal receptor tyrosine protein kinase | 7.1 | 7.1 | 7.1 | pKd | 2 |
Homo sapiens | Myosin IIIA | 7.4 | 7.4 | 7.4 | pIC50 | 1 |
Homo sapiens | Myosin IIIA | 6.3 | 6.3 | 6.3 | pKd | 2 |
Homo sapiens | Myosin-IIIB | 8.2 | 8.2 | 8.2 | pIC50 | 1 |
Homo sapiens | Myosin-IIIB | 6.5 | 6.5 | 6.5 | pKd | 2 |
Homo sapiens | Myosin light chain kinase | 6.9 | 6.9 | 6.9 | pIC50 | 1 |
Homo sapiens | Myosin light chain kinase | 6.9 | 6.9 | 6.9 | pKd | 1 |
Homo sapiens | myosin light chain kinase 2 | 7.9 | 7.9 | 7.9 | pIC50 | 1 |
Homo sapiens | myosin light chain kinase 2 | 7.2 | 7 | 7.2 | pKd | 3 |
Homo sapiens | Myosin light chain kinase family member 4 | 7.3 | 7.3 | 7.3 | pIC50 | 1 |
Homo sapiens | Myosin light chain kinase family member 4 | 6.3 | 6.3 | 6.3 | pKd | 2 |
Gallus gallus | Myosin light chain kinase, smooth muscle | 8 | 8 | 8 | pIC50 | 1 |
Gallus gallus | Myosin light chain kinase, smooth muscle | 6.9 | 6.9 | 6.9 | pKd | 1 |
Homo sapiens | Myosin light chain kinase, smooth muscle | 7.4 | 7.3 | 8 | pIC50 | 3 |
Homo sapiens | Myosin light chain kinase, smooth muscle | 7.8 | 7.8 | 7.8 | pKd | 2 |
Homo sapiens | Myotonin-protein kinase | 7 | 7 | 7 | pIC50 | 1 |
Homo sapiens | Myotonin-protein kinase | 8.5 | 8.5 | 8.5 | pKd | 2 |
Homo sapiens | Nerve growth factor receptor Trk-A | 8.8 | 8.1 | 9.3 | pIC50 | 6 |
Homo sapiens | Nerve growth factor receptor Trk-A | 8.4 | 8.4 | 8.7 | pKd | 3 |
Homo sapiens | Neurotrophic tyrosine kinase receptor type 2 | 9 | 8.4 | 10.2 | pIC50 | 3 |
Homo sapiens | Neurotrophic tyrosine kinase receptor type 2 | 8.4 | 8.4 | 8.4 | pKd | 2 |
Homo sapiens | Non-receptor tyrosine-protein kinase TNK1 | 9.2 | 9.2 | 9.2 | pIC50 | 1 |
Homo sapiens | Non-receptor tyrosine-protein kinase TNK1 | 8.6 | 8.6 | 8.6 | pKd | 2 |
Homo sapiens | NT-3 growth factor receptor | 9.7 | 9.7 | 9.7 | pIC50 | 1 |
Homo sapiens | NT-3 growth factor receptor | 7.8 | 7.8 | 7.8 | pKd | 2 |
Homo sapiens | NUAK family SNF1-like kinase 1 | 8.9 | 8.1 | 8.9 | pIC50 | 3 |
Homo sapiens | NUAK family SNF1-like kinase 1 | 8.4 | 8.4 | 8.4 | pKd | 2 |
Homo sapiens | NUAK family SNF1-like kinase 2 | 8.8 | 8.8 | 8.8 | pIC50 | 1 |
Homo sapiens | NUAK family SNF1-like kinase 2 | 10.1 | 10.1 | 10.1 | pKd | 2 |
Homo sapiens | PAS domain-containing serine/threonine-protein kinase | 7.8 | 7.8 | 7.8 | pIC50 | 1 |
Homo sapiens | PDZ-binding kinase | 7.1 | 7.1 | 7.1 | pIC50 | 1 |
Homo sapiens | Peripheral plasma membrane protein CASK | 7.7 | 7.7 | 7.7 | pKd | 1 |
Homo sapiens | Phosphatidylinositol-4-phosphate 3-kinase C2 domain-containing subunit gamma | 6.4 | 6.4 | 6.4 | pKd | 1 |
Homo sapiens | Phosphatidylinositol-4-phosphate 5-kinase type-1 alpha | 7.4 | 7.4 | 7.4 | pKd | 2 |
Homo sapiens | Phosphatidylinositol-4-phosphate 5-kinase type-1 gamma | 5.6 | 5.6 | 5.6 | pKd | 1 |
Homo sapiens | Phosphatidylinositol-5-phosphate 4-kinase type-2 beta | 7.1 | 7.1 | 7.1 | pKd | 2 |
Homo sapiens | Phosphorylase kinase gamma subunit 1 | 8.6 | 8.6 | 8.6 | pIC50 | 1 |
Homo sapiens | Phosphorylase kinase gamma subunit 1 | 9.2 | 9.2 | 9.3 | pKd | 3 |
Homo sapiens | Phosphorylase kinase gamma subunit 2 | 9.2 | 9.2 | 9.3 | pIC50 | 2 |
Homo sapiens | Phosphorylase kinase gamma subunit 2 | 9.9 | 9 | 9.9 | pKd | 3 |
Homo sapiens | PI3-kinase p110-alpha subunit | 6.4 | 6.4 | 6.4 | pKd | 1 |
Homo sapiens | PI3-kinase p110-gamma subunit | 5.8 | 5.8 | 5.8 | pKd | 1 |
Homo sapiens | PI4-kinase beta subunit | 6.3 | 6.3 | 6.3 | pKd | 1 |
Homo sapiens | Platelet-derived growth factor receptor alpha | 9.2 | 9.1 | 9.4 | pIC50 | 4 |
Homo sapiens | Platelet-derived growth factor receptor alpha | 8 | 8 | 8 | pKd | 2 |
Homo sapiens | Platelet-derived growth factor receptor beta | 8.4 | 6.7 | 9.2 | pIC50 | 6 |
Homo sapiens | Platelet-derived growth factor receptor beta | 8.7 | 8.6 | 8.7 | pKd | 3 |
Homo sapiens | Protein kinase C alpha | 8.6 | 7.4 | 9.4 | pIC50 | 14 |
Homo sapiens | Protein kinase C alpha | 7.3 | 7.3 | 7.3 | pKd | 1 |
Homo sapiens | Protein kinase C beta | 7.7 | 7.1 | 8.8 | pIC50 | 14 |
Homo sapiens | Protein kinase C delta | 7.4 | 6.2 | 9.9 | pIC50 | 8 |
Homo sapiens | Protein kinase C delta | 8.8 | 8.8 | 8.8 | pKd | 2 |
Homo sapiens | Protein kinase C epsilon | 8.8 | 7.7 | 9.7 | pIC50 | 9 |
Homo sapiens | Protein kinase C epsilon | 9.6 | 9.6 | 9.6 | pKd | 2 |
Homo sapiens | Protein kinase C eta | 8.3 | 8.3 | 9.6 | pIC50 | 3 |
Homo sapiens | Protein kinase C eta | 8.3 | 8.3 | 8.3 | pKd | 2 |
Homo sapiens | Protein kinase C gamma | 7.2 | 7 | 8.9 | pIC50 | 8 |
Rattus norvegicus | Protein kinase C gamma | 8.1 | 8.1 | 8.1 | pIC50 | 1 |
Homo sapiens | Protein kinase C iota | 6.4 | 6.4 | 7.5 | pIC50 | 2 |
Homo sapiens | Protein kinase C iota | 7.6 | 7.6 | 7.6 | pKd | 1 |
Homo sapiens | Protein kinase C mu | 8.4 | 8.4 | 8.4 | pIC50 | 1 |
Homo sapiens | Protein kinase C mu | 7.6 | 7.6 | 7.6 | pKd | 2 |
Homo sapiens | Protein kinase C nu | 8.8 | 8.8 | 8.8 | pIC50 | 1 |
Homo sapiens | Protein kinase C nu | 7.8 | 7.8 | 7.8 | pKd | 2 |
Homo sapiens | Protein kinase C theta | 8.8 | 8.8 | 8.8 | pIC50 | 1 |
Homo sapiens | Protein kinase C theta | 8.1 | 8.1 | 8.1 | pKd | 2 |
Homo sapiens | Protein kinase C zeta | 6.7 | 6.7 | 7.1 | pIC50 | 2 |
Homo sapiens | Protein kinase N1 | 8.9 | 8.4 | 9 | pIC50 | 3 |
Homo sapiens | Protein kinase N1 | 8.9 | 8.9 | 8.9 | pKd | 2 |
Homo sapiens | Protein kinase N2 | 8.7 | 7.9 | 8.7 | pIC50 | 3 |
Homo sapiens | Protein kinase N2 | 8.6 | 8.6 | 8.6 | pKd | 2 |
Plasmodium falciparum | Protein kinase Pfmrk | 5.4 | 5.4 | 5.4 | pIC50 | 2 |
Homo sapiens | Protein tyrosine kinase 2 beta | 8 | 8 | 8 | pIC50 | 1 |
Homo sapiens | Protein tyrosine kinase 2 beta | 8.5 | 8.5 | 8.5 | pKd | 2 |
Homo sapiens | Proto-oncogene tyrosine-protein kinase MER | 7.1 | 7.1 | 7.9 | pIC50 | 2 |
Homo sapiens | Proto-oncogene tyrosine-protein kinase MER | 8.2 | 8.2 | 8.2 | pKd | 2 |
Homo sapiens | Proto-oncogene tyrosine-protein kinase ROS | 9.8 | 9.7 | 10.2 | pIC50 | 3 |
Homo sapiens | Proto-oncogene tyrosine-protein kinase ROS | 7.5 | 7.5 | 7.5 | pKd | 2 |
Homo sapiens | Pseudopodium-enriched atypical kinase 1 | 8.5 | 8.5 | 8.5 | pIC50 | 1 |
Homo sapiens | Putative uncharacterized serine/threonine-protein kinase SgK110 | 7.6 | 7.6 | 7.6 | pKd | 1 |
Homo sapiens | Pyruvate dehydrogenase kinase isoform 1 | 9.3 | 9.3 | 9.3 | pIC50 | 1 |
Homo sapiens | Receptor-interacting serine/threonine-protein kinase 4 | 7 | 7 | 7 | pKd | 1 |
Homo sapiens | Receptor protein-tyrosine kinase erbB-2 | 7 | 6.9 | 7.5 | pIC50 | 6 |
Homo sapiens | Receptor protein-tyrosine kinase erbB-2 | 6.7 | 6.7 | 6.7 | pKd | 1 |
Homo sapiens | Receptor protein-tyrosine kinase erbB-4 | 6.6 | 6.3 | 7.6 | pIC50 | 5 |
Homo sapiens | Receptor protein-tyrosine kinase erbB-4 | 6.1 | 6.1 | 6.1 | pKd | 1 |
Homo sapiens | Rho-associated protein kinase 1 | 9.1 | 7.7 | 9.2 | pIC50 | 5 |
Homo sapiens | Rho-associated protein kinase 1 | 9.6 | 9.6 | 9.6 | pKd | 1 |
Homo sapiens | Rho-associated protein kinase 2 | 8.1 | 8.1 | 9 | pIC50 | 3 |
Homo sapiens | Rho-associated protein kinase 2 | 9.6 | 9.6 | 9.6 | pKd | 1 |
Homo sapiens | Rhodopsin kinase | 7.2 | 7.2 | 7.2 | pIC50 | 1 |
Homo sapiens | Rhodopsin kinase | 9 | 9 | 9 | pKd | 1 |
Homo sapiens | Ribosomal protein S6 kinase 1 | 9 | 9 | 9.3 | pIC50 | 2 |
Homo sapiens | Ribosomal protein S6 kinase 1 | 8.9 | 8.9 | 8.9 | pKd | 1 |
Homo sapiens | Ribosomal protein S6 kinase 2 | 8.6 | 8.6 | 8.6 | pIC50 | 1 |
Homo sapiens | Ribosomal protein S6 kinase alpha 1 | 9.9 | 8.9 | 10.1 | pIC50 | 6 |
Homo sapiens | Ribosomal protein S6 kinase alpha 1 | 5.9 | 5.9 | 7.4 | pKd | 8 |
Homo sapiens | Ribosomal protein S6 kinase alpha 2 | 9.6 | 9.6 | 9.6 | pIC50 | 2 |
Homo sapiens | Ribosomal protein S6 kinase alpha 2 | 8 | 6.7 | 8.1 | pKd | 10 |
Homo sapiens | Ribosomal protein S6 kinase alpha 3 | 9.9 | 9.9 | 9.9 | pIC50 | 2 |
Homo sapiens | Ribosomal protein S6 kinase alpha 3 | 7.2 | 7.2 | 7.2 | pKd | 6 |
Homo sapiens | Ribosomal protein S6 kinase alpha 4 | 8 | 8 | 8 | pIC50 | 2 |
Homo sapiens | Ribosomal protein S6 kinase alpha 4 | 5.7 | 5.7 | 6.9 | pKd | 8 |
Homo sapiens | Ribosomal protein S6 kinase alpha 5 | 8.9 | 8.9 | 8.9 | pIC50 | 4 |
Homo sapiens | Ribosomal protein S6 kinase alpha 5 | 7.4 | 6.1 | 7.7 | pKd | 10 |
Homo sapiens | Ribosomal protein S6 kinase alpha 6 | 9.8 | 9.8 | 9.8 | pIC50 | 2 |
Homo sapiens | Ribosomal protein S6 kinase alpha 6 | 5.5 | 5.5 | 7.8 | pKd | 8 |
Homo sapiens | Serine/threonine-protein kinase 10 | 8 | 8 | 8 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase 10 | 10.4 | 10.4 | 10.5 | pKd | 3 |
Homo sapiens | Serine/threonine-protein kinase 11 | 7.2 | 7.2 | 7.2 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase 11 | 7.2 | 7.2 | 7.2 | pKd | 2 |
Homo sapiens | Serine/threonine-protein kinase 16 | 6.6 | 6.6 | 6.6 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase 16 | 6.6 | 6.6 | 6.7 | pKd | 3 |
Homo sapiens | Serine/threonine-protein kinase 17A | 7.5 | 7.5 | 7.5 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase 17A | 7.9 | 7.6 | 7.9 | pKd | 3 |
Homo sapiens | Serine/threonine-protein kinase 17B | 7.6 | 7.6 | 7.6 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase 17B | 7.7 | 7.6 | 7.7 | pKd | 3 |
Homo sapiens | Serine/threonine-protein kinase 2 | 7.8 | 7.8 | 7.8 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase 2 | 10.6 | 10.6 | 10.7 | pKd | 3 |
Homo sapiens | Serine/threonine-protein kinase 24 | 8.4 | 8.4 | 8.5 | pIC50 | 2 |
Homo sapiens | Serine/threonine-protein kinase 24 | 6.9 | 6.9 | 6.9 | pKd | 2 |
Homo sapiens | Serine/threonine-protein kinase 25 | 8.6 | 8.6 | 8.7 | pIC50 | 2 |
Homo sapiens | Serine/threonine-protein kinase 25 | 7 | 7 | 7 | pKd | 2 |
Homo sapiens | Serine/threonine-protein kinase 32A | 7.9 | 7.9 | 7.9 | pKd | 1 |
Homo sapiens | Serine/threonine-protein kinase 32B | 7.3 | 7.3 | 7.3 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase 32B | 7 | 7 | 7 | pKd | 2 |
Homo sapiens | Serine/threonine-protein kinase 32C | 6.5 | 6.5 | 6.5 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase 32C | 6.5 | 6.5 | 6.5 | pKd | 2 |
Homo sapiens | Serine/threonine-protein kinase 33 | 7.4 | 7.4 | 7.4 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase 33 | 8.7 | 8.7 | 8.7 | pKd | 2 |
Homo sapiens | Serine/threonine-protein kinase 35 | 6.9 | 6.9 | 6.9 | pKd | 1 |
Homo sapiens | Serine/threonine-protein kinase 36 | 5.2 | 5.2 | 5.5 | pKd | 3 |
Homo sapiens | Serine/threonine-protein kinase 38 | 9.2 | 9.2 | 9.2 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase 38 | 7.3 | 7.3 | 7.3 | pKd | 1 |
Homo sapiens | Serine/threonine-protein kinase 38-like | 8.8 | 8.8 | 8.8 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase 38-like | 7.6 | 7.1 | 7.6 | pKd | 3 |
Homo sapiens | Serine/threonine-protein kinase AKT | 6.3 | 6.3 | 6.3 | pEC50 | 2 |
Homo sapiens | Serine/threonine-protein kinase AKT | 8 | 6.5 | 8.8 | pIC50 | 21 |
Homo sapiens | Serine/threonine-protein kinase AKT | 7.7 | 7.7 | 7.7 | pKd | 2 |
Homo sapiens | Serine/threonine-protein kinase AKT2 | 8.1 | 7.4 | 8.2 | pIC50 | 5 |
Homo sapiens | Serine/threonine-protein kinase AKT2 | 7.4 | 7.4 | 7.4 | pKd | 2 |
Homo sapiens | Serine/threonine-protein kinase AKT3 | 8 | 7.9 | 9.2 | pIC50 | 6 |
Homo sapiens | Serine/threonine-protein kinase AKT3 | 6.8 | 6.8 | 6.8 | pKd | 2 |
Homo sapiens | Serine/threonine-protein kinase Aurora-A | 8.1 | 7.4 | 9.2 | pIC50 | 16 |
Homo sapiens | Serine/threonine-protein kinase Aurora-A | 7.8 | 7 | 7.8 | pKd | 3 |
Homo sapiens | Serine/threonine-protein kinase Aurora-B | 8.2 | 8 | 9 | pIC50 | 9 |
Homo sapiens | Serine/threonine-protein kinase Aurora-B | 7.7 | 7.7 | 7.7 | pKd | 2 |
Homo sapiens | Serine/threonine-protein kinase Aurora-C | 8.6 | 8.6 | 8.6 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase Aurora-C | 7.6 | 7.6 | 8 | pKd | 3 |
Homo sapiens | Serine/threonine-protein kinase B-raf | 8.3 | 7.9 | 8.4 | pIC50 | 5 |
Homo sapiens | Serine/threonine-protein kinase Chk1 | 8.7 | 8 | 9.8 | pIC50 | 7 |
Homo sapiens | Serine/threonine-protein kinase Chk1 | 8.5 | 8.5 | 8.5 | pKd | 2 |
Homo sapiens | Serine/threonine-protein kinase Chk2 | 7.6 | 4.6 | 8.5 | pIC50 | 8 |
Homo sapiens | Serine/threonine-protein kinase Chk2 | 7.1 | 7.1 | 7.1 | pKd | 1 |
Homo sapiens | Serine/threonine-protein kinase c-TAK1 | 9.4 | 9.4 | 9.4 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase c-TAK1 | 8.5 | 8.5 | 8.5 | pKd | 2 |
Homo sapiens | Serine/threonine-protein kinase D2 | 8.9 | 8.9 | 8.9 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase D2 | 7.1 | 7.1 | 7.1 | pKd | 2 |
Homo sapiens | Serine/threonine-protein kinase DCLK1 | 6.8 | 6.8 | 6.8 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase DCLK1 | 7 | 7 | 7 | pKd | 2 |
Homo sapiens | Serine/threonine-protein kinase DCLK2 | 7.1 | 7.1 | 7.1 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase DCLK2 | 7.1 | 7.1 | 7.1 | pKd | 2 |
Homo sapiens | Serine/threonine-protein kinase DCLK3 | 7.8 | 7.8 | 7.8 | pKd | 2 |
Homo sapiens | Serine/threonine-protein kinase/endoribonuclease IRE1 | 6.7 | 6.7 | 6.7 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase/endoribonuclease IRE1 | 7.7 | 7.7 | 7.7 | pKd | 1 |
Homo sapiens | Serine/threonine-protein kinase/endoribonuclease IRE2 | 7.2 | 7.2 | 7.2 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase GAK | 7.8 | 7.2 | 7.8 | pKd | 3 |
Homo sapiens | Serine/threonine-protein kinase haspin | 7.1 | 7.1 | 7.7 | pIC50 | 2 |
Homo sapiens | Serine/threonine-protein kinase ICK | 7.3 | 7.3 | 7.4 | pIC50 | 2 |
Homo sapiens | Serine/threonine-protein kinase ICK | 7.8 | 7.8 | 7.8 | pKd | 1 |
Homo sapiens | Serine/threonine-protein kinase LATS1 | 7.9 | 7.9 | 7.9 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase LATS1 | 7.4 | 7.4 | 7.4 | pKd | 2 |
Homo sapiens | Serine/threonine-protein kinase LATS2 | 8.4 | 8.4 | 8.4 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase LATS2 | 7.8 | 7.8 | 7.8 | pKd | 2 |
Homo sapiens | Serine/threonine-protein kinase MAK | 7.5 | 7.5 | 7.5 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase MAK | 5.6 | 5.6 | 5.6 | pKd | 1 |
Homo sapiens | Serine/threonine-protein kinase MARK1 | 9.4 | 9.4 | 9.4 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase MARK1 | 8.4 | 8.4 | 8.4 | pKd | 2 |
Homo sapiens | Serine/threonine-protein kinase MRCK-A | 8.3 | 8.3 | 8.3 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase MRCK-A | 7.2 | 7.2 | 7.2 | pKd | 2 |
Homo sapiens | Serine/threonine-protein kinase MRCK beta | 8.3 | 8.3 | 8.3 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase MRCK beta | 7.4 | 7.4 | 7.4 | pKd | 2 |
Homo sapiens | Serine/threonine-protein kinase MRCK gamma | 9.1 | 9.1 | 9.1 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase MRCK gamma | 7.4 | 7.4 | 7.4 | pKd | 2 |
Homo sapiens | Serine/threonine-protein kinase MST1 | 8.8 | 8.8 | 8.8 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase MST1 | 9.7 | 9.7 | 9.7 | pKd | 3 |
Homo sapiens | Serine/threonine-protein kinase MST2 | 8.3 | 8.3 | 9.4 | pIC50 | 3 |
Homo sapiens | Serine/threonine-protein kinase MST2 | 9.7 | 9.7 | 9.7 | pKd | 2 |
Mus musculus | Serine/threonine-protein kinase MST2 | 9.8 | 9.8 | 9.8 | pKd | 1 |
Homo sapiens | Serine/threonine-protein kinase MST4 | 8.5 | 8.5 | 8.5 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase MST4 | 6.9 | 6.9 | 6.9 | pKd | 2 |
Homo sapiens | Serine/threonine-protein kinase N3 | 7.9 | 7.9 | 7.9 | pIC50 | 2 |
Homo sapiens | Serine/threonine-protein kinase Nek1 | 7.7 | 7.7 | 7.7 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase Nek1 | 6.1 | 6.1 | 6.1 | pKd | 2 |
Homo sapiens | Serine/threonine-protein kinase Nek11 | 6.1 | 6.1 | 6.1 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase Nek11 | 5.5 | 5.5 | 5.5 | pKd | 1 |
Homo sapiens | Serine/threonine-protein kinase NEK2 | 5.3 | 5.3 | 6.5 | pIC50 | 2 |
Homo sapiens | Serine/threonine-protein kinase NEK2 | 6.1 | 6.1 | 6.1 | pKd | 3 |
Homo sapiens | Serine/threonine-protein kinase Nek3 | 4.6 | 4.6 | 4.6 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase Nek4 | 7 | 7 | 7 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase Nek5 | 7 | 7 | 7 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase Nek5 | 6.1 | 6.1 | 6.1 | pKd | 2 |
Homo sapiens | Serine/threonine-protein kinase NEK7 | 5.4 | 5.4 | 5.4 | pKd | 2 |
Homo sapiens | Serine/threonine-protein kinase Nek8 | 7.8 | 7.8 | 7.8 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase NEK9 | 6.9 | 6.9 | 6.9 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase NEK9 | 5.5 | 5.2 | 5.5 | pKd | 3 |
Homo sapiens | Serine/threonine-protein kinase NIM1 | 6.9 | 6.9 | 6.9 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase NIM1 | 6.9 | 6.9 | 6.9 | pKd | 1 |
Homo sapiens | Serine/threonine protein kinase NLK | 7.1 | 7.1 | 7.1 | pIC50 | 1 |
Homo sapiens | Serine/threonine protein kinase NLK | 6.7 | 6.7 | 6.7 | pKd | 2 |
Homo sapiens | Serine/threonine-protein kinase OSR1 | 6.4 | 6.4 | 6.4 | pKd | 1 |
Homo sapiens | Serine/threonine-protein kinase PAK 1 | 9.3 | 9.3 | 9.5 | pIC50 | 2 |
Homo sapiens | Serine/threonine-protein kinase PAK 1 | 9.2 | 8.7 | 9.2 | pKd | 3 |
Homo sapiens | Serine/threonine-protein kinase PAK 2 | 8.6 | 8.5 | 9 | pIC50 | 3 |
Homo sapiens | Serine/threonine-protein kinase PAK 2 | 8.5 | 8.5 | 8.5 | pKd | 2 |
Homo sapiens | Serine/threonine-protein kinase PAK 3 | 9.5 | 9.5 | 9.5 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase PAK 3 | 8.2 | 8.2 | 9.3 | pKd | 3 |
Homo sapiens | Serine/threonine-protein kinase PAK 4 | 8.7 | 7.6 | 9 | pIC50 | 3 |
Homo sapiens | Serine/threonine-protein kinase PAK 4 | 8.2 | 8.1 | 8.2 | pKd | 3 |
Homo sapiens | Serine/threonine-protein kinase PAK6 | 7.5 | 7.5 | 7.5 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase PAK6 | 9.2 | 9.2 | 9.4 | pKd | 3 |
Homo sapiens | Serine/threonine-protein kinase PAK7 | 8.3 | 8.3 | 8.3 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase PAK7 | 8.9 | 8.5 | 8.9 | pKd | 3 |
Homo sapiens | Serine/threonine-protein kinase PCTAIRE-1 | 7.6 | 7.6 | 7.6 | pKd | 3 |
Homo sapiens | Serine/threonine-protein kinase PCTAIRE-2 | 7 | 7 | 7 | pKd | 2 |
Homo sapiens | Serine/threonine-protein kinase PCTAIRE-3 | 6.6 | 6.6 | 6.6 | pKd | 2 |
Homo sapiens | Serine/threonine-protein kinase PFTAIRE-1 | 6.8 | 6.8 | 6.8 | pKd | 2 |
Homo sapiens | Serine/threonine-protein kinase PFTAIRE-2 | 6.6 | 6.6 | 6.6 | pKd | 1 |
Homo sapiens | Serine/threonine-protein kinase PIM1 | 8 | 7 | 8.6 | pIC50 | 12 |
Homo sapiens | Serine/threonine-protein kinase PIM1 | 8.5 | 7.8 | 8.9 | pKd | 4 |
Homo sapiens | Serine/threonine-protein kinase PIM2 | 7.6 | 6.5 | 8.2 | pIC50 | 4 |
Homo sapiens | Serine/threonine-protein kinase PIM2 | 8.7 | 8.4 | 8.7 | pKd | 3 |
Homo sapiens | Serine/threonine-protein kinase PIM3 | 9.9 | 9.9 | 10.1 | pIC50 | 2 |
Homo sapiens | Serine/threonine-protein kinase PIM3 | 9.3 | 9.3 | 9.3 | pKd | 2 |
Mycobacterium tuberculosis | Serine/threonine-protein kinase pknB | 7.1 | 7.1 | 7.1 | pKd | 1 |
Homo sapiens | Serine/threonine-protein kinase PLK1 | 6.3 | 4.7 | 6.7 | pIC50 | 7 |
Homo sapiens | Serine/threonine-protein kinase PLK1 | 6.7 | 6.7 | 6.7 | pKd | 2 |
Homo sapiens | Serine/threonine-protein kinase PLK2 | 6.3 | 6 | 6.7 | pIC50 | 5 |
Homo sapiens | Serine/threonine-protein kinase PLK2 | 6.7 | 6.7 | 6.7 | pKd | 1 |
Homo sapiens | Serine/threonine-protein kinase PLK3 | 6.7 | 6.7 | 6.7 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase PLK3 | 6 | 6 | 6 | pKd | 2 |
Homo sapiens | Serine/threonine-protein kinase PLK4 | 8 | 8 | 8 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase PLK4 | 9.1 | 9.1 | 9.1 | pKd | 3 |
Homo sapiens | Serine/threonine-protein kinase PRKX | 8.9 | 8.9 | 8.9 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase PRKX | 7.9 | 7.9 | 7.9 | pKd | 2 |
Homo sapiens | Serine/threonine-protein kinase PRP4 homolog | 6.7 | 6.7 | 6.7 | pKd | 1 |
Homo sapiens | Serine/threonine-protein kinase RAF | 6.9 | 6.6 | 6.9 | pIC50 | 3 |
Homo sapiens | Serine/threonine-protein kinase receptor R3 | 6.1 | 6.1 | 6.1 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase RIO1 | 6.9 | 6.9 | 6.9 | pKd | 2 |
Homo sapiens | Serine/threonine-protein kinase RIO2 | 6.4 | 6.4 | 6.4 | pKd | 1 |
Homo sapiens | Serine/threonine-protein kinase RIO3 | 7.1 | 7.1 | 7.1 | pKd | 2 |
Homo sapiens | Serine/threonine-protein kinase RIPK2 | 6.5 | 6.5 | 6.5 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase RIPK2 | 5.3 | 5.3 | 5.3 | pKd | 3 |
Homo sapiens | Serine/threonine-protein kinase SBK1 | 7 | 7 | 7 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase SBK1 | 8.5 | 8.5 | 8.5 | pKd | 1 |
Homo sapiens | Serine/threonine-protein kinase Sgk1 | 7.9 | 7.9 | 8.2 | pIC50 | 2 |
Homo sapiens | Serine/threonine-protein kinase Sgk2 | 7.8 | 7.8 | 7.8 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase Sgk3 | 7.1 | 7.1 | 7.1 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase Sgk3 | 8.5 | 8.5 | 8.5 | pKd | 1 |
Homo sapiens | Serine/threonine-protein kinase SIK1 | 8.9 | 8.9 | 8.9 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase SIK1 | 8.7 | 8.7 | 8.7 | pKd | 2 |
Homo sapiens | Serine/threonine-protein kinase SIK2 | 9.4 | 9.4 | 9.4 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase SIK2 | 9 | 9 | 9 | pKd | 2 |
Homo sapiens | Serine/threonine-protein kinase SIK3 | 8.9 | 8.9 | 8.9 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase SIK3 | 9.3 | 9.3 | 9.3 | pKd | 1 |
Homo sapiens | Serine/threonine-protein kinase SRPK1 | 7.6 | 7.6 | 7.6 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase SRPK1 | 8.3 | 8.3 | 8.3 | pKd | 2 |
Homo sapiens | Serine/threonine-protein kinase SRPK2 | 6.6 | 6.6 | 6.6 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase SRPK2 | 7.2 | 7.2 | 7.2 | pKd | 2 |
Homo sapiens | Serine/threonine-protein kinase SRPK3 | 5.7 | 5.7 | 5.7 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase SRPK3 | 7.1 | 7.1 | 7.1 | pKd | 1 |
Homo sapiens | Serine/threonine-protein kinase TAO1 | 8.9 | 8.9 | 8.9 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase TAO1 | 9.4 | 9.4 | 9.4 | pKd | 1 |
Homo sapiens | Serine/threonine-protein kinase TAO2 | 7.9 | 7.9 | 7.9 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase TAO2 | 7.9 | 7.9 | 7.9 | pKd | 1 |
Homo sapiens | Serine/threonine-protein kinase TAO3 | 8.7 | 8.7 | 8.7 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase TAO3 | 9.7 | 9.7 | 9.7 | pKd | 1 |
Homo sapiens | Serine/threonine-protein kinase TBK1 | 8.7 | 8.7 | 8.7 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase TBK1 | 9.1 | 9.1 | 9.1 | pKd | 1 |
Homo sapiens | Serine/threonine-protein kinase TNNI3K | 6 | 6 | 6 | pKd | 2 |
Homo sapiens | Serine/threonine-protein kinase tousled-like 1 | 7.5 | 7.5 | 7.7 | pIC50 | 2 |
Homo sapiens | Serine/threonine-protein kinase tousled-like 1 | 7.6 | 7.6 | 7.6 | pKd | 2 |
Homo sapiens | Serine/threonine-protein kinase tousled-like 2 | 8.4 | 8.4 | 8.4 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase tousled-like 2 | 7.8 | 7.8 | 7.8 | pKd | 2 |
Homo sapiens | Serine/threonine-protein kinase ULK1 | 8.1 | 8.1 | 8.1 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase ULK1 | 8 | 8 | 8 | pKd | 1 |
Homo sapiens | Serine/threonine-protein kinase ULK2 | 8.6 | 8.6 | 8.6 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase ULK2 | 9.1 | 9.1 | 9.1 | pKd | 1 |
Homo sapiens | Serine/threonine-protein kinase ULK3 | 8.4 | 8.4 | 8.4 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase ULK3 | 8.9 | 8.9 | 8.9 | pKd | 1 |
Homo sapiens | Serine/threonine-protein kinase WEE1 | 5.8 | 5.8 | 5.8 | pKd | 2 |
Homo sapiens | Serine/threonine-protein kinase WNK1 | 4.9 | 4.9 | 4.9 | pIC50 | 1 |
Homo sapiens | Serine/threonine-protein kinase WNK2 | 5.8 | 5.8 | 5.8 | pIC50 | 1 |
Homo sapiens | SNF-related serine/threonine-protein kinase | 8.1 | 8.1 | 8.1 | pIC50 | 1 |
Homo sapiens | SNF-related serine/threonine-protein kinase | 7.1 | 7.1 | 7.1 | pKd | 1 |
Homo sapiens | SPS1/STE20-related protein kinase YSK4 | 7.8 | 7.8 | 7.8 | pIC50 | 1 |
Homo sapiens | SPS1/STE20-related protein kinase YSK4 | 9.1 | 9.1 | 9.1 | pKd | 1 |
Homo sapiens | STE20/SPS1-related proline-alanine-rich protein kinase | 7.8 | 7.8 | 7.8 | pIC50 | 1 |
Homo sapiens | STE20/SPS1-related proline-alanine-rich protein kinase | 6.9 | 6.9 | 6.9 | pKd | 1 |
Homo sapiens | Stem cell growth factor receptor | 7.6 | 7.1 | 8.4 | pIC50 | 8 |
Homo sapiens | Stem cell growth factor receptor | 7.8 | 7 | 9.4 | pKd | 16 |
Homo sapiens | Testis-specific serine/threonine-protein kinase 1 | 10.3 | 10.3 | 10.3 | pIC50 | 1 |
Homo sapiens | Testis-specific serine/threonine-protein kinase 1 | 7.6 | 7.6 | 7.6 | pKd | 2 |
Mus musculus | Testis-specific serine/threonine-protein kinase 1 | 9.5 | 9.5 | 9.5 | pIC50 | 1 |
Homo sapiens | Testis-specific serine/threonine-protein kinase 2 | 8.4 | 8.4 | 8.4 | pIC50 | 1 |
Homo sapiens | Testis-specific serine/threonine-protein kinase 3 | 8.2 | 8.2 | 8.2 | pIC50 | 1 |
Homo sapiens | Testis-specific serine/threonine-protein kinase 6 | 6.7 | 6.7 | 6.7 | pIC50 | 1 |
Homo sapiens | TGF-beta receptor type I | 5.2 | 5.2 | 5.2 | pIC50 | 1 |
Homo sapiens | TGF-beta receptor type I | 5.7 | 5.7 | 5.7 | pKd | 2 |
Homo sapiens | TRAF2- and NCK-interacting kinase | 8.9 | 7.4 | 9.3 | pIC50 | 3 |
Homo sapiens | TRAF2- and NCK-interacting kinase | 8.3 | 8.2 | 8.3 | pKd | 3 |
Homo sapiens | Tyrosine kinase non-receptor protein 2 | 7.5 | 7.5 | 7.5 | pIC50 | 1 |
Homo sapiens | Tyrosine kinase non-receptor protein 2 | 7.8 | 7.8 | 7.8 | pKd | 3 |
Homo sapiens | Tyrosine-protein kinase ABL | 6.9 | 6.5 | 7.5 | pIC50 | 10 |
Homo sapiens | Tyrosine-protein kinase ABL | 7 | 5.6 | 8.5 | pKd | 29 |
Homo sapiens | Tyrosine-protein kinase ABL2 | 7.1 | 7.1 | 7.8 | pIC50 | 2 |
Homo sapiens | Tyrosine-protein kinase ABL2 | 7 | 6.8 | 7 | pKd | 3 |
Homo sapiens | Tyrosine-protein kinase BLK | 9 | 9 | 9 | pIC50 | 1 |
Homo sapiens | Tyrosine-protein kinase BLK | 7.8 | 7.8 | 7.8 | pKd | 2 |
Mus musculus | Tyrosine-protein kinase BLK | 6.4 | 6.4 | 6.4 | pIC50 | 1 |
Homo sapiens | Tyrosine-protein kinase BMX | 8.2 | 8.2 | 8.2 | pIC50 | 1 |
Homo sapiens | Tyrosine-protein kinase BMX | 6.8 | 6.4 | 6.8 | pKd | 3 |
Homo sapiens | Tyrosine-protein kinase BRK | 6.6 | 5.9 | 6.6 | pIC50 | 3 |
Homo sapiens | Tyrosine-protein kinase BRK | 5.6 | 5.6 | 5.6 | pKd | 2 |
Homo sapiens | Tyrosine-protein kinase BTK | 7.6 | 4.8 | 7.9 | pIC50 | 7 |
Homo sapiens | Tyrosine-protein kinase BTK | 6.7 | 6.2 | 6.7 | pKd | 3 |
Homo sapiens | Tyrosine-protein kinase CSK | 7.8 | 7.8 | 7.8 | pIC50 | 1 |
Homo sapiens | Tyrosine-protein kinase CSK | 6.5 | 6.4 | 6.5 | pKd | 3 |
Homo sapiens | Tyrosine-protein kinase CTK | 6.3 | 6.3 | 6.3 | pIC50 | 1 |
Homo sapiens | Tyrosine-protein kinase CTK | 6.6 | 6.6 | 6.6 | pKd | 1 |
Homo sapiens | Tyrosine-protein kinase FER | 8.7 | 8.7 | 9.4 | pIC50 | 2 |
Homo sapiens | Tyrosine-protein kinase FER | 7.6 | 7.5 | 7.6 | pKd | 3 |
Homo sapiens | Tyrosine-protein kinase FES | 8.1 | 8.1 | 8.8 | pIC50 | 2 |
Homo sapiens | Tyrosine-protein kinase FES | 7.6 | 7.6 | 7.6 | pKd | 2 |
Homo sapiens | Tyrosine-protein kinase FGR | 8.9 | 8.9 | 8.9 | pIC50 | 1 |
Homo sapiens | Tyrosine-protein kinase FGR | 7.8 | 7.5 | 7.8 | pKd | 3 |
Homo sapiens | Tyrosine-protein kinase FRK | 7.8 | 7.8 | 7.8 | pIC50 | 1 |
Homo sapiens | Tyrosine-protein kinase FRK | 7.4 | 6.6 | 7.4 | pKd | 3 |
Homo sapiens | Tyrosine-protein kinase FYN | 7.8 | 6.3 | 8.7 | pIC50 | 9 |
Homo sapiens | Tyrosine-protein kinase FYN | 7.5 | 7.3 | 7.5 | pKd | 3 |
Homo sapiens | Tyrosine-protein kinase HCK | 8.7 | 8.7 | 8.7 | pIC50 | 1 |
Homo sapiens | Tyrosine-protein kinase HCK | 7.7 | 7.7 | 7.9 | pKd | 3 |
Homo sapiens | Tyrosine-protein kinase ITK/TSK | 7.9 | 4.8 | 8.4 | pIC50 | 5 |
Homo sapiens | Tyrosine-protein kinase ITK/TSK | 7.7 | 7.7 | 7.7 | pKd | 2 |
Homo sapiens | Tyrosine-protein kinase JAK1 | 8.5 | 7.9 | 9.2 | pIC50 | 10 |
Homo sapiens | Tyrosine-protein kinase JAK1 | 8.2 | 8.2 | 8.2 | pKd | 2 |
Homo sapiens | Tyrosine-protein kinase JAK2 | 8.7 | 8.3 | 9.7 | pIC50 | 16 |
Homo sapiens | Tyrosine-protein kinase JAK2 | 8 | 8 | 8 | pKd | 6 |
Homo sapiens | Tyrosine-protein kinase JAK3 | 9.3 | 8.2 | 10 | pIC50 | 20 |
Homo sapiens | Tyrosine-protein kinase JAK3 | 7.9 | 7.9 | 8 | pKd | 4 |
Homo sapiens | Tyrosine-protein kinase LCK | 8.7 | 5.7 | 9 | pIC50 | 11 |
Homo sapiens | Tyrosine-protein kinase LCK | 7.5 | 7.5 | 7.7 | pKd | 3 |
Homo sapiens | Tyrosine-protein kinase Lyn | 8.9 | 8.6 | 9.3 | pIC50 | 8 |
Homo sapiens | Tyrosine-protein kinase Lyn | 7.4 | 6.7 | 7.4 | pKd | 3 |
Homo sapiens | Tyrosine-protein kinase receptor FLT3 | 8.9 | 8.3 | 9.7 | pIC50 | 16 |
Homo sapiens | Tyrosine-protein kinase receptor FLT3 | 8.6 | 8.5 | 9.7 | pKd | 14 |
Homo sapiens | Tyrosine-protein kinase receptor RET | 8.5 | 8.3 | 9.3 | pIC50 | 5 |
Homo sapiens | Tyrosine-protein kinase receptor RET | 7.8 | 7.6 | 7.9 | pKd | 6 |
Homo sapiens | Tyrosine-protein kinase receptor Tie-1 | 7.2 | 7.2 | 7.2 | pKd | 2 |
Homo sapiens | Tyrosine-protein kinase receptor TYRO3 | 7.3 | 7.3 | 8.6 | pIC50 | 2 |
Homo sapiens | Tyrosine-protein kinase receptor TYRO3 | 6.6 | 6.6 | 6.6 | pKd | 2 |
Homo sapiens | Tyrosine-protein kinase receptor UFO | 8.1 | 7.4 | 8.5 | pIC50 | 4 |
Homo sapiens | Tyrosine-protein kinase receptor UFO | 8.2 | 8.2 | 8.2 | pKd | 2 |
Homo sapiens | Tyrosine-protein kinase SRC | 8 | 5.5 | 9.1 | pIC50 | 24 |
Homo sapiens | Tyrosine-protein kinase SRC | 7.1 | 7 | 8.1 | pKd | 4 |
Homo sapiens | Tyrosine-protein kinase Srms | 5.1 | 5.1 | 5.1 | pIC50 | 1 |
Homo sapiens | Tyrosine-protein kinase Srms | 6.1 | 6.1 | 6.1 | pKd | 2 |
Homo sapiens | Tyrosine-protein kinase SYK | 8.9 | 7.2 | 9.7 | pIC50 | 7 |
Homo sapiens | Tyrosine-protein kinase SYK | 7.9 | 7.9 | 8.2 | pKd | 3 |
Homo sapiens | Tyrosine-protein kinase TEC | 7.4 | 7.4 | 7.4 | pIC50 | 1 |
Homo sapiens | Tyrosine-protein kinase TEC | 5.9 | 5.9 | 5.9 | pKd | 2 |
Homo sapiens | Tyrosine-protein kinase TIE-2 | 7.2 | 6.7 | 7.3 | pIC50 | 4 |
Homo sapiens | Tyrosine-protein kinase TIE-2 | 6.9 | 6.6 | 6.9 | pKd | 3 |
Homo sapiens | Tyrosine-protein kinase TXK | 7.7 | 7.7 | 7.7 | pIC50 | 1 |
Homo sapiens | Tyrosine-protein kinase TXK | 6.6 | 6.6 | 6.6 | pKd | 2 |
Homo sapiens | Tyrosine-protein kinase TYK2 | 9.5 | 9.2 | 9.7 | pIC50 | 6 |
Homo sapiens | Tyrosine-protein kinase TYK2 | 7.3 | 5.5 | 7.3 | pKd | 6 |
Homo sapiens | Tyrosine-protein kinase YES | 8.6 | 8.4 | 8.6 | pIC50 | 3 |
Homo sapiens | Tyrosine-protein kinase YES | 7.3 | 7.3 | 7.3 | pKd | 3 |
Homo sapiens | Tyrosine-protein kinase ZAP-70 | 7.9 | 7.3 | 8.9 | pIC50 | 6 |
Homo sapiens | Tyrosine-protein kinase ZAP-70 | 7.4 | 7.4 | 7.4 | pKd | 2 |
Mus musculus | ULK3 kinase | 8.5 | 8.5 | 8.5 | pKd | 1 |
Homo sapiens | Vascular endothelial growth factor receptor 1 | 7.8 | 7.5 | 8.3 | pIC50 | 6 |
Homo sapiens | Vascular endothelial growth factor receptor 1 | 6.8 | 6.8 | 6.8 | pKd | 2 |
Homo sapiens | Vascular endothelial growth factor receptor 2 | 8 | 4.7 | 8.9 | pIC50 | 28 |
Homo sapiens | Vascular endothelial growth factor receptor 2 | 6.7 | 6.6 | 6.7 | pKd | 3 |
Homo sapiens | Vascular endothelial growth factor receptor 2 | 8.8 | 8.8 | 8.8 | pKi | 1 |
Homo sapiens | Vascular endothelial growth factor receptor 3 | 8.5 | 7.2 | 9.1 | pIC50 | 8 |
Homo sapiens | Vascular endothelial growth factor receptor 3 | 7.6 | 7.5 | 7.6 | pKd | 3 |