4HZR - chain B (model A) | Tyrosine kinase, non-receptor, 2
Structure information
PDB:4HZR
PubMed:23342057
Release date:2013-02-06
Resolution:1.31 Å
 
Kinase:TNK2 (ACK)
Family:Ack
Group:TK
Species:HUMAN
 
Quality Score:5.6
Missing Residues:6
Missing Atoms:0
DFG conformation:in
αC-helix conformation:in
Salt bridge KIII.17 and EαC.24:Yes (2.8Å)
 
 
ASP rotation (xDFG.81) :15°
PHE rotation (xDFG.82) :14°
Activation loop position:-5Å
αC-helix position:18.5Å
 
G-rich loop angle:-
G-rich loop distance:-
G-rich loop rotation:-
Other models from this PDB:
2D & 3D views

The orthosteric binding pocket
Binding pocket waters
The following waters were found in the defined clusters:
I1
H-bond protein
I3
No H-bonds
I5
No H-bonds
I6
No H-bonds
I8
H-bond protein
I10
No H-bonds
I11
No H-bonds
Binding pocket sequence
UniprotEKLGDGSFGVVRRVAVKCLDFIREVNAMHSLDRNLIRLYGVKMVTELAPLGSLLDRLRKYLESKRFIHRDLAARNLLLIGDFGLM
Structure:EKLG_____VVRRVAVKC_DFIREVNAMHSLDRNLIRLYGVKMVTELAPLGSLLDRLRKYLESKRFIHRDLAARNLLLIGDFGLM


Modified residues
No modified residues identified.