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Search results (10 entries covering 6 PDB structures)
#
Kinase
Family
Group
PDB
Chain
(Alternate) Model
Orthosteric ligand
Organism
Details
File
AURKA (AurA)
Aur
Other
6cpg
A
1-cyclopropyl-3-{3-[5-(morpholin-4-ylmethyl)-1h-benzimidazol-2-yl]-1h-pyrazol-4-yl}urea
Human
10032
PRKACA (PKACa)
PKA
AGC
5n23
A
A
1-cyclopropyl-3-{3-[5-(morpholin-4-ylmethyl)-1h-benzimidazol-2-yl]-1h-pyrazol-4-yl}urea
Human
9747
JAK2-b
JakB
TK
6d2i
B
1-cyclopropyl-3-{3-[5-(morpholin-4-ylmethyl)-1h-benzimidazol-2-yl]-1h-pyrazol-4-yl}urea
Human
10966
STK24 (MST3)
STE20
STE
4qmm
A
1-cyclopropyl-3-{3-[5-(morpholin-4-ylmethyl)-1h-benzimidazol-2-yl]-1h-pyrazol-4-yl}urea
Human
5583
AURKA (AurA)
Aur
Other
6cpg
D
1-cyclopropyl-3-{3-[5-(morpholin-4-ylmethyl)-1h-benzimidazol-2-yl]-1h-pyrazol-4-yl}urea
Human
10034
JAK2-b
JakB
TK
5ut0
A
B
1-cyclopropyl-3-{3-[5-(morpholin-4-ylmethyl)-1h-benzimidazol-2-yl]-1h-pyrazol-4-yl}urea
Human
8047
PRKACA (PKACa)
PKA
AGC
5n23
A
B
1-cyclopropyl-3-{3-[5-(morpholin-4-ylmethyl)-1h-benzimidazol-2-yl]-1h-pyrazol-4-yl}urea
Human
9746
JAK2-b
JakB
TK
6d2i
A
1-cyclopropyl-3-{3-[5-(morpholin-4-ylmethyl)-1h-benzimidazol-2-yl]-1h-pyrazol-4-yl}urea
Human
10967
JAK2-b
JakB
TK
5wim
A
1-cyclopropyl-3-{3-[5-(morpholin-4-ylmethyl)-1h-benzimidazol-2-yl]-1h-pyrazol-4-yl}urea
Human
10385
JAK2-b
JakB
TK
5ut0
A
A
1-cyclopropyl-3-{3-[5-(morpholin-4-ylmethyl)-1h-benzimidazol-2-yl]-1h-pyrazol-4-yl}urea
Human
8041
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