| RPS6KA3 (RSK2) | RSK | AGC | 5d9k | B | | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(3-methylbutyl)-7,8-dihydropteridin-6(5h)-one | Human | 5987 | |
| VRK1 | VRK | CK1 | 5uge | B | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(3-methylbutyl)-7,8-dihydropteridin-6(5h)-one | Human | 7424 | |
| RPS6KA3 (RSK2) | RSK | AGC | 5d9k | A | | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(3-methylbutyl)-7,8-dihydropteridin-6(5h)-one | Human | 5988 | |
| VRK1 | VRK | CK1 | 5uge | D | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(3-methylbutyl)-7,8-dihydropteridin-6(5h)-one | Human | 7423 | |
| VRK1 | VRK | CK1 | 5uge | B | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(3-methylbutyl)-7,8-dihydropteridin-6(5h)-one | Human | 7420 | |
| VRK1 | VRK | CK1 | 5uge | A | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(3-methylbutyl)-7,8-dihydropteridin-6(5h)-one | Human | 7418 | |
| VRK1 | VRK | CK1 | 5uge | C | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(3-methylbutyl)-7,8-dihydropteridin-6(5h)-one | Human | 7419 | |
| VRK1 | VRK | CK1 | 5uge | A | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(3-methylbutyl)-7,8-dihydropteridin-6(5h)-one | Human | 7421 | |
| JAK2-b | JakB | TK | 5wik | B | | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(3-methylbutyl)-7,8-dihydropteridin-6(5h)-one | Human | 10387 | |
| VRK1 | VRK | CK1 | 5uge | D | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(3-methylbutyl)-7,8-dihydropteridin-6(5h)-one | Human | 7425 | |
| VRK1 | VRK | CK1 | 5uge | C | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(3-methylbutyl)-7,8-dihydropteridin-6(5h)-one | Human | 7422 | |