Search results (15 entries covering 10 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetails File
MAPK1 (Erk2)MAPKCMGC1pmeA4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridineHuman2583
MAPK14 (p38a)MAPKCMGC3zs5AA4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridineHuman4987
MAPK14 (p38a)MAPKCMGC3gcpAB4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridineHuman5157
RIPK2RIPKTKL5ar4B4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridineHuman6187
MAPK14 (p38a)MAPKCMGC3gcpAA4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridineHuman5194
MAPK14 (p38a)MAPKCMGC1a9uA4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridineHuman5229
MAPK14 (p38a)MAPKCMGC3obgA4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridineHuman5211
Mapk14 (p38a)MAPKCMGC2ewaAB4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridineMouse5870
RIPK2RIPKTKL5ar4A4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridineHuman6180
Mapk14 (p38a)MAPKCMGC8acoAA4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridineMouse15095
Mapk14 (p38a)MAPKCMGC8acoAB4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridineMouse15094
Mapk14 (p38a)MAPKCMGC8acmA4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridineMouse15096
MAPK14 (p38a)MAPKCMGC3zs5AB4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridineHuman4977
MAPK14 (p38a)MAPKCMGC3mpaA4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridineHuman5026
Mapk14 (p38a)MAPKCMGC2ewaAA4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridineMouse5859