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Search results (14 entries covering 7 PDB structures)
#
Kinase
Family
Group
PDB
Chain
(Alternate) Model
Orthosteric ligand
Organism
Details
File
PRKAA1 (AMPKa1)
CAMKL
CAMK
7jhg
A
6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine
Human
13816
PRKAA1 (AMPKa1)
CAMKL
CAMK
7m74
A
6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine
Human
14017
ACVR2A (ACTR2)
STKR
TKL
3q4t
B
A
6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine
Human
2680
ACVR2A (ACTR2)
STKR
TKL
3q4t
A
A
6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine
Human
2682
ACVR1 (ALK2)
STKR
TKL
4c02
A
A
6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine
Human
1525
ACVR2A (ACTR2)
STKR
TKL
3q4t
A
B
6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine
Human
2686
ACVR1 (ALK2)
STKR
TKL
3h9r
A
6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine
Human
1531
MELK
CAMKL
CAMK
6gvx
A
A
6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine
Human
11137
MELK
CAMKL
CAMK
6gvx
A
B
6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine
Human
11139
MELK
CAMKL
CAMK
6gvx
B
A
6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine
Human
11136
MELK
CAMKL
CAMK
6gvx
B
B
6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine
Human
11138
ACVR2A (ACTR2)
STKR
TKL
3q4t
B
B
6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine
Human
2684
ACVR1 (ALK2)
STKR
TKL
4c02
A
B
6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine
Human
1532
PRKAA2 (AMPKa2)
CAMKL
CAMK
3aqv
A
6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine
Human
193
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