Search results (14 entries covering 7 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetails File
PRKAA1 (AMPKa1)CAMKLCAMK7jhgA6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHuman13816
PRKAA1 (AMPKa1)CAMKLCAMK7m74A6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHuman14017
ACVR2A (ACTR2)STKRTKL3q4tBA6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHuman2680
ACVR2A (ACTR2)STKRTKL3q4tAA6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHuman2682
ACVR1 (ALK2)STKRTKL4c02AA6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHuman1525
ACVR2A (ACTR2)STKRTKL3q4tAB6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHuman2686
ACVR1 (ALK2)STKRTKL3h9rA6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHuman1531
MELKCAMKLCAMK6gvxAA6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHuman11137
MELKCAMKLCAMK6gvxAB6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHuman11139
MELKCAMKLCAMK6gvxBA6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHuman11136
MELKCAMKLCAMK6gvxBB6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHuman11138
ACVR2A (ACTR2)STKRTKL3q4tBB6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHuman2684
ACVR1 (ALK2)STKRTKL4c02AB6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHuman1532
PRKAA2 (AMPKa2)CAMKLCAMK3aqvA6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHuman193