| AKT1 | Akt | AGC | 6hhh | A | | ~{n}-[4-[4-[[4-(5-oxidanylidene-3-phenyl-6~{h}-1,6-naphthyridin-2-yl)phenyl]methyl]piperazin-1-yl]phenyl]propanamide | Human | 10915 | |
| AKT1 | Akt | AGC | 4ekk | A | | phosphoaminophosphonic acid-adenylate ester | Human | 2541 | |
| AKT1 | Akt | AGC | 4ekk | B | | phosphoaminophosphonic acid-adenylate ester | Human | 2539 | |
| AKT1 | Akt | AGC | 6hhj | A | | ~{n}-[1-methyl-2-oxidanylidene-3-[1-[[4-(5-oxidanylidene-3-phenyl-6~{h}-1,6-naphthyridin-2-yl)phenyl]methyl]piperidin-4-yl]benzimidazol-5-yl]propanamide | Human | 10914 | |
| AKT1 | Akt | AGC | 6buu | B | C | - | Human | 10428 | |
| AKT1 | Akt | AGC | 3ocb | A | | (2s)-2-(4-chlorobenzyl)-3-oxo-3-[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperazin-1-yl]propan-1-amine | Human | 2548 | |
| AKT1 | Akt | AGC | 6buu | B | A | - | Human | 10430 | |
| AKT1 | Akt | AGC | 3mvh | A | B | n-{[(3s)-3-amino-1-(5-ethyl-7h-pyrrolo[2,3-d]pyrimidin-4-yl)pyrrolidin-3-yl]methyl}-2,4-difluorobenzamide | Human | 2531 | |
| AKT1 | Akt | AGC | 3cqu | A | B | n-[2-(5-methyl-4h-1,2,4-triazol-3-yl)phenyl]-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 6762 | |
| AKT1 | Akt | AGC | 6hhi | A | | ~{n}-[1-[[4-(5-oxidanylidene-3-phenyl-6~{h}-1,6-naphthyridin-2-yl)phenyl]methyl]piperidin-4-yl]-3-(propanoylamino)benzamide | Human | 10913 | |
| AKT1 | Akt | AGC | 3mv5 | A | A | (3r)-1-(5-methyl-7h-pyrrolo[2,3-d]pyrimidin-4-yl)pyrrolidin-3-amine | Human | 2537 | |
| AKT1 | Akt | AGC | 4ejn | A | | - | Human | 2542 | |
| AKT1 | Akt | AGC | 6ccy | A | B | (5r)-4-(4-{4-[4-fluoro-3-(trifluoromethyl)phenyl]-1-[2-(pyrrolidin-1-yl)ethyl]-1h-imidazol-2-yl}piperidin-1-yl)-5-methyl-5,8-dihydropyrido[2,3-d]pyrimidin-7(6h)-one | Human | 9869 | |
| AKT1 | Akt | AGC | 3qkm | A | | n-(2-ethoxyethyl)-n-{(2s)-2-hydroxy-3-[(5r)-2-(quinazolin-4-yl)-2,7-diazaspiro[4.5]dec-7-yl]propyl}-2,6-dimethylbenzenesulfonamide | Human | 2546 | |
| AKT1 | Akt | AGC | 3cqw | A | A | 5-(5-chloro-7h-pyrrolo[2,3-d]pyrimidin-4-yl)-4,5,6,7-tetrahydro-1h-imidazo[4,5-c]pyridine | Human | 6763 | |
| AKT1 | Akt | AGC | 6npz | B | A | - | Human | 10881 | |
| AKT1 | Akt | AGC | 6buu | A | B | - | Human | 10433 | |
| AKT1 | Akt | AGC | 6hhf | A | | borussertib | Human | 10970 | |
| AKT1 | Akt | AGC | 7nh5 | A | A | ~{n}-methyl-6-[4-[[4-[2-oxidanylidene-6-(propanoylamino)-3~{h}-benzimidazol-1-yl]piperidin-1-yl]methyl]phenyl]-5-phenyl-pyridine-3-carboxamide | Human | 13867 | |
| AKT1 | Akt | AGC | 6s9w | A | B | ~{n}-[3-[1-[[4-(5-methyl-6-oxidanylidene-3-phenyl-1~{h}-pyrazin-2-yl)phenyl]methyl]piperidin-4-yl]-2-oxidanylidene-1~{h}-benzimidazol-5-yl]propanamide | Human | 11747 | |
| AKT1 | Akt | AGC | 3mv5 | A | B | (3r)-1-(5-methyl-7h-pyrrolo[2,3-d]pyrimidin-4-yl)pyrrolidin-3-amine | Human | 2532 | |
| AKT1 | Akt | AGC | 3ow4 | A | | (2r)-3-(1h-indol-3-yl)-1-{4-[(5s)-5-methyl-5,7-dihydrothieno[3,4-d]pyrimidin-4-yl]piperazin-1-yl}-1-oxopropan-2-amine | Human | 2547 | |
| AKT1 | Akt | AGC | 7nh4 | A | A | ~{n}-[3-[1-[[4-[5-(hydroxymethyl)-3-phenyl-pyridin-2-yl]phenyl]methyl]piperidin-4-yl]-2-oxidanylidene-1~{h}-benzimidazol-5-yl]propanamide | Human | 13865 | |
| AKT1 | Akt | AGC | 3qkk | A | | n-(2-ethoxyethyl)-n-{(2s)-2-hydroxy-3-[(2r)-6-hydroxy-4-oxo-3,4-dihydro-1'h-spiro[chromene-2,3'-piperidin]-1'-yl]propyl}-2,6-dimethylbenzenesulfonamide | Human | 2535 | |
| AKT1 | Akt | AGC | 7apj | A | | - | Human | 13854 | |
| AKT1 | Akt | AGC | 3o96 | A | | - | Human | 2545 | |
| AKT1 | Akt | AGC | 3ocb | B | | (2s)-2-(4-chlorobenzyl)-3-oxo-3-[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperazin-1-yl]propan-1-amine | Human | 2534 | |
| AKT1 | Akt | AGC | 6ccy | A | A | (5r)-4-(4-{4-[4-fluoro-3-(trifluoromethyl)phenyl]-1-[2-(pyrrolidin-1-yl)ethyl]-1h-imidazol-2-yl}piperidin-1-yl)-5-methyl-5,8-dihydropyrido[2,3-d]pyrimidin-7(6h)-one | Human | 9868 | |
| AKT1 | Akt | AGC | 6npz | B | B | - | Human | 10879 | |
| AKT1 | Akt | AGC | 4gv1 | A | A | 4-amino-n-[(1s)-1-(4-chlorophenyl)-3-hydroxypropyl]-1-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperidine-4-carboxamide | Human | 2543 | |
| AKT1 | Akt | AGC | 3cqw | A | B | 5-(5-chloro-7h-pyrrolo[2,3-d]pyrimidin-4-yl)-4,5,6,7-tetrahydro-1h-imidazo[4,5-c]pyridine | Human | 6765 | |
| AKT1 | Akt | AGC | 6buu | B | B | - | Human | 10439 | |
| AKT1 | Akt | AGC | 6hhg | A | | ~{n}-[2-chloranyl-5-[[1-[[4-(5-oxidanylidene-3-phenyl-6~{h}-1,6-naphthyridin-2-yl)phenyl]methyl]piperidin-4-yl]carbamoylamino]phenyl]propanamide | Human | 10916 | |
| AKT1 | Akt | AGC | 3ow4 | B | | (2r)-3-(1h-indol-3-yl)-1-{4-[(5s)-5-methyl-5,7-dihydrothieno[3,4-d]pyrimidin-4-yl]piperazin-1-yl}-1-oxopropan-2-amine | Human | 2533 | |
| AKT1 | Akt | AGC | 4ekl | A | | (2s)-2-(4-chlorophenyl)-1-{4-[(5r,7r)-7-hydroxy-5-methyl-6,7-dihydro-5h-cyclopenta[d]pyrimidin-4-yl]piperazin-1-yl}-3-(propan-2-ylamino)propan-1-one | Human | 2540 | |
| AKT1 | Akt | AGC | 7nh5 | A | B | ~{n}-methyl-6-[4-[[4-[2-oxidanylidene-6-(propanoylamino)-3~{h}-benzimidazol-1-yl]piperidin-1-yl]methyl]phenyl]-5-phenyl-pyridine-3-carboxamide | Human | 13868 | |
| AKT1 | Akt | AGC | 3qkl | A | | n-{(2s)-3-[(3s)-8',9'-dihydro-1h,3'h-spiro[piperidine-3,7'-pyrano[3,2-e]indazol]-1-yl]-2-hydroxypropyl}-n-(2-ethoxyethyl)-2,6-dimethylbenzenesulfonamide | Human | 2544 | |
| AKT1 | Akt | AGC | 3mvh | A | A | n-{[(3s)-3-amino-1-(5-ethyl-7h-pyrrolo[2,3-d]pyrimidin-4-yl)pyrrolidin-3-yl]methyl}-2,4-difluorobenzamide | Human | 2538 | |
| AKT1 | Akt | AGC | 6npz | A | A | - | Human | 10880 | |
| AKT1 | Akt | AGC | 6buu | A | C | - | Human | 10438 | |
| AKT1 | Akt | AGC | 5kcv | A | | 3-[3-[4-(1-azanylcyclobutyl)phenyl]-5-phenyl-imidazo[4,5-b]pyridin-2-yl]pyridin-2-amine | Human | 6708 | |
| AKT1 | Akt | AGC | 3cqu | A | A | n-[2-(5-methyl-4h-1,2,4-triazol-3-yl)phenyl]-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 6764 | |
| AKT1 | Akt | AGC | 6npz | A | B | - | Human | 10882 | |
| AKT1 | Akt | AGC | 7nh4 | A | B | ~{n}-[3-[1-[[4-[5-(hydroxymethyl)-3-phenyl-pyridin-2-yl]phenyl]methyl]piperidin-4-yl]-2-oxidanylidene-1~{h}-benzimidazol-5-yl]propanamide | Human | 13866 | |
| AKT1 | Akt | AGC | 4gv1 | A | B | 4-amino-n-[(1s)-1-(4-chlorophenyl)-3-hydroxypropyl]-1-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperidine-4-carboxamide | Human | 2536 | |
| AKT1 | Akt | AGC | 6s9x | A | | ~{n}-[3-[1-[[4-[5-[(4-hydroxyphenyl)methyl]-6-oxidanylidene-2-phenyl-1~{h}-pyrazin-3-yl]phenyl]methyl]piperidin-4-yl]-2-oxidanylidene-1~{h}-benzimidazol-5-yl]propanamide | Human | 11746 | |
| AKT1 | Akt | AGC | 6s9w | A | A | ~{n}-[3-[1-[[4-(5-methyl-6-oxidanylidene-3-phenyl-1~{h}-pyrazin-2-yl)phenyl]methyl]piperidin-4-yl]-2-oxidanylidene-1~{h}-benzimidazol-5-yl]propanamide | Human | 11748 | |
| AKT1 | Akt | AGC | 6buu | A | A | - | Human | 10432 | |