| VRK1 | VRK | CK1 | 6bp0 | A | B | - | Human | 8738 | |
| VRK1 | VRK | CK1 | 2rsv | A | 10 | - | Human | 4873 | |
| VRK1 | VRK | CK1 | 2lav | A | 16 | - | Human | 4888 | |
| VRK1 | VRK | CK1 | 6ac9 | D | A | phosphoaminophosphonic acid-adenylate ester | Human | 10821 | |
| VRK1 | VRK | CK1 | 5uvf | A | | (7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(3-methylbutyl)-7,8-dihydropteridin-6(5h)-one | Human | 7521 | |
| VRK1 | VRK | CK1 | 3op5 | A | A | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrile | Human | 4870 | |
| VRK1 | VRK | CK1 | 6dd4 | A | B | - | Human | 9939 | |
| VRK1 | VRK | CK1 | 6cnx | A | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-8-(3-methylbutyl)-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9810 | |
| VRK1 | VRK | CK1 | 6dd4 | D | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-dipropyl-7,8-dihydropteridin-6(5h)-one | Human | 9938 | |
| VRK1 | VRK | CK1 | 6bp0 | A | A | - | Human | 8744 | |
| VRK1 | VRK | CK1 | 2kul | A | 9 | - | Human | 4869 | |
| VRK1 | VRK | CK1 | 6cqh | C | A | - | Human | 9772 | |
| VRK1 | VRK | CK1 | 2lav | A | 5 | - | Human | 4891 | |
| VRK1 | VRK | CK1 | 6cmm | D | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9764 | |
| VRK1 | VRK | CK1 | 6csw | B | B | (7r)-5-butyl-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7,8-dimethyl-7,8-dihydropteridin-6(5h)-one | Human | 9808 | |
| VRK1 | VRK | CK1 | 2kty | A | 17 | - | Human | 4920 | |
| VRK1 | VRK | CK1 | 2kul | A | 10 | - | Human | 4901 | |
| VRK1 | VRK | CK1 | 6bru | C | B | - | Human | 9086 | |
| VRK1 | VRK | CK1 | 2kty | A | 14 | - | Human | 4926 | |
| VRK1 | VRK | CK1 | 2lav | A | 12 | - | Human | 4946 | |
| VRK1 | VRK | CK1 | 6bp0 | D | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7,8-trimethyl-7,8-dihydropteridin-6(5h)-one | Human | 8739 | |
| VRK1 | VRK | CK1 | 2kty | A | 13 | - | Human | 4922 | |
| VRK1 | VRK | CK1 | 6bu6 | D | A | 4,4'-(2-aminopyridine-3,5-diyl)bis(2,6-difluorophenol) | Human | 9413 | |
| VRK1 | VRK | CK1 | 6npn | B | | (7r)-7-methyl-2-[(3-oxo-2,3-dihydro-1h-indazol-6-yl)amino]-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 11244 | |
| VRK1 | VRK | CK1 | 3op5 | C | A | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrile | Human | 4886 | |
| VRK1 | VRK | CK1 | 5ukf | C | | 4-{[(z)-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}benzene-1-sulfonamide | Human | 8027 | |
| VRK1 | VRK | CK1 | 6cnx | D | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-8-(3-methylbutyl)-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9814 | |
| VRK1 | VRK | CK1 | 6cqh | D | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-ethyl-7-methyl-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9771 | |
| VRK1 | VRK | CK1 | 2kul | A | 2 | - | Human | 4921 | |
| VRK1 | VRK | CK1 | 6vzh | D | | (7~{r})-2-[[3,5-bis(fluoranyl)-4-oxidanyl-phenyl]amino]-5,7-dimethyl-8-prop-2-ynyl-7~{h}-pteridin-6-one | Human | 12055 | |
| VRK1 | VRK | CK1 | 6dd4 | D | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-dipropyl-7,8-dihydropteridin-6(5h)-one | Human | 9934 | |
| VRK1 | VRK | CK1 | 5ukf | D | | 4-{[(z)-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}benzene-1-sulfonamide | Human | 8028 | |
| VRK1 | VRK | CK1 | 2kul | A | 17 | - | Human | 4893 | |
| VRK1 | VRK | CK1 | 6csw | C | A | - | Human | 9816 | |
| VRK1 | VRK | CK1 | 2lav | A | 18 | - | Human | 4927 | |
| VRK1 | VRK | CK1 | 2kty | A | 5 | - | Human | 4900 | |
| VRK1 | VRK | CK1 | 2rsv | A | 12 | - | Human | 4952 | |
| VRK1 | VRK | CK1 | 6bu6 | C | B | - | Human | 9414 | |
| VRK1 | VRK | CK1 | 2lav | A | 1 | - | Human | 4930 | |
| VRK1 | VRK | CK1 | 6bru | A | A | - | Human | 9085 | |
| VRK1 | VRK | CK1 | 6bu6 | D | B | 4,4'-(2-aminopyridine-3,5-diyl)bis(2,6-difluorophenol) | Human | 9410 | |
| VRK1 | VRK | CK1 | 3op5 | D | B | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrile | Human | 4892 | |
| VRK1 | VRK | CK1 | 6csw | C | B | - | Human | 9811 | |
| VRK1 | VRK | CK1 | 2kty | A | 18 | - | Human | 4904 | |
| VRK1 | VRK | CK1 | 2rsv | A | 5 | - | Human | 4899 | |
| VRK1 | VRK | CK1 | 6dd4 | C | A | - | Human | 9940 | |
| VRK1 | VRK | CK1 | 2kty | A | 1 | - | Human | 4877 | |
| VRK1 | VRK | CK1 | 6cfm | B | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9725 | |
| VRK1 | VRK | CK1 | 6bp0 | B | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7,8-trimethyl-7,8-dihydropteridin-6(5h)-one | Human | 8740 | |
| VRK1 | VRK | CK1 | 3op5 | D | A | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrile | Human | 4878 | |
| VRK1 | VRK | CK1 | 2kty | A | 4 | - | Human | 4938 | |
| VRK1 | VRK | CK1 | 2rsv | A | 4 | - | Human | 4907 | |
| VRK1 | VRK | CK1 | 6cfm | B | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9724 | |
| VRK1 | VRK | CK1 | 2kul | A | 20 | - | Human | 4915 | |
| VRK1 | VRK | CK1 | 6cnx | A | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-8-(3-methylbutyl)-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9815 | |
| VRK1 | VRK | CK1 | 6btw | D | A | 2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-phenyl-7,8-dihydropteridin-6(5h)-one | Human | 9415 | |
| VRK1 | VRK | CK1 | 2rsv | A | 15 | - | Human | 4911 | |
| VRK1 | VRK | CK1 | 2lav | A | 19 | - | Human | 4940 | |
| VRK1 | VRK | CK1 | 6cfm | D | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9721 | |
| VRK1 | VRK | CK1 | 6bru | B | B | (7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7,8-trimethyl-7,8-dihydropteridin-6(5h)-one | Human | 9087 | |
| VRK1 | VRK | CK1 | 2kty | A | 2 | - | Human | 4947 | |
| VRK1 | VRK | CK1 | 6cqh | D | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-ethyl-7-methyl-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9767 | |
| VRK1 | VRK | CK1 | 2kul | A | 12 | - | Human | 4883 | |
| VRK1 | VRK | CK1 | 2kty | A | 19 | - | Human | 4875 | |
| VRK1 | VRK | CK1 | 6ac9 | D | B | phosphoaminophosphonic acid-adenylate ester | Human | 10820 | |
| VRK1 | VRK | CK1 | 2lav | A | 14 | - | Human | 4898 | |
| VRK1 | VRK | CK1 | 6ac9 | C | A | phosphoaminophosphonic acid-adenylate ester | Human | 10822 | |
| VRK1 | VRK | CK1 | 6vxu | B | | (7r)-8-(cyclopropylmethyl)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 13362 | |
| VRK1 | VRK | CK1 | 6cfm | A | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9723 | |
| VRK1 | VRK | CK1 | 2lav | A | 6 | - | Human | 4871 | |
| VRK1 | VRK | CK1 | 6cnx | B | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-8-(3-methylbutyl)-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9803 | |
| VRK1 | VRK | CK1 | 5uvf | D | | (7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(3-methylbutyl)-7,8-dihydropteridin-6(5h)-one | Human | 7522 | |
| VRK1 | VRK | CK1 | 6cnx | C | B | (7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-8-(3-methylbutyl)-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9804 | |
| VRK1 | VRK | CK1 | 2rsv | A | 3 | - | Human | 4913 | |
| VRK1 | VRK | CK1 | 6cmm | B | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9761 | |
| VRK1 | VRK | CK1 | 6ac9 | C | B | phosphoaminophosphonic acid-adenylate ester | Human | 10819 | |
| VRK1 | VRK | CK1 | 6dd4 | B | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-dipropyl-7,8-dihydropteridin-6(5h)-one | Human | 9933 | |
| VRK1 | VRK | CK1 | 6cmm | A | B | - | Human | 9760 | |
| VRK1 | VRK | CK1 | 6dd4 | A | A | - | Human | 9935 | |
| VRK1 | VRK | CK1 | 6cmm | B | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9766 | |
| VRK1 | VRK | CK1 | 2kul | A | 14 | - | Human | 4909 | |
| VRK1 | VRK | CK1 | 6csw | D | A | (7r)-5-butyl-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7,8-dimethyl-7,8-dihydropteridin-6(5h)-one | Human | 9817 | |
| VRK1 | VRK | CK1 | 2rsv | A | 13 | - | Human | 4935 | |
| VRK1 | VRK | CK1 | 2kty | A | 6 | - | Human | 4929 | |
| VRK1 | VRK | CK1 | 2kul | A | 6 | - | Human | 4949 | |
| VRK1 | VRK | CK1 | 6btw | C | A | - | Human | 9419 | |
| VRK1 | VRK | CK1 | 6cmm | C | A | - | Human | 9765 | |
| VRK1 | VRK | CK1 | 3op5 | C | B | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrile | Human | 4879 | |
| VRK1 | VRK | CK1 | 6ac9 | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 10817 | |
| VRK1 | VRK | CK1 | 6bp0 | D | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7,8-trimethyl-7,8-dihydropteridin-6(5h)-one | Human | 8745 | |
| VRK1 | VRK | CK1 | 6btw | C | B | - | Human | 9416 | |
| VRK1 | VRK | CK1 | 2kty | A | 3 | - | Human | 4874 | |
| VRK1 | VRK | CK1 | 2lav | A | 15 | - | Human | 4931 | |
| VRK1 | VRK | CK1 | 6vzh | B | | (7~{r})-2-[[3,5-bis(fluoranyl)-4-oxidanyl-phenyl]amino]-5,7-dimethyl-8-prop-2-ynyl-7~{h}-pteridin-6-one | Human | 12056 | |
| VRK1 | VRK | CK1 | 5ukf | B | | 4-{[(z)-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}benzene-1-sulfonamide | Human | 8029 | |
| VRK1 | VRK | CK1 | 2kty | A | 16 | - | Human | 4937 | |
| VRK1 | VRK | CK1 | 2lav | A | 7 | - | Human | 4936 | |
| VRK1 | VRK | CK1 | 6bp0 | B | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7,8-trimethyl-7,8-dihydropteridin-6(5h)-one | Human | 8741 | |
| VRK1 | VRK | CK1 | 2kty | A | 8 | - | Human | 4939 | |
| VRK1 | VRK | CK1 | 6npn | A | | (7r)-7-methyl-2-[(3-oxo-2,3-dihydro-1h-indazol-6-yl)amino]-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 11243 | |
| VRK1 | VRK | CK1 | 2lav | A | 17 | - | Human | 4950 | |
| VRK1 | VRK | CK1 | 2lav | A | 10 | - | Human | 4882 | |
| VRK1 | VRK | CK1 | 6bu6 | B | B | 4,4'-(2-aminopyridine-3,5-diyl)bis(2,6-difluorophenol) | Human | 9422 | |
| VRK1 | VRK | CK1 | 2rsv | A | 7 | - | Human | 4889 | |
| VRK1 | VRK | CK1 | 6bu6 | C | A | - | Human | 9412 | |
| VRK1 | VRK | CK1 | 2rsv | A | 17 | - | Human | 4951 | |
| VRK1 | VRK | CK1 | 6bu6 | A | B | 4,4'-(2-aminopyridine-3,5-diyl)bis(2,6-difluorophenol) | Human | 9417 | |
| VRK1 | VRK | CK1 | 6cmm | A | A | - | Human | 9763 | |
| VRK1 | VRK | CK1 | 6bru | C | A | - | Human | 9089 | |
| VRK1 | VRK | CK1 | 6cqh | A | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-ethyl-7-methyl-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9768 | |
| VRK1 | VRK | CK1 | 2kty | A | 15 | - | Human | 4953 | |
| VRK1 | VRK | CK1 | 5uvf | B | | (7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(3-methylbutyl)-7,8-dihydropteridin-6(5h)-one | Human | 7523 | |
| VRK1 | VRK | CK1 | 6ac9 | B | A | phosphoaminophosphonic acid-adenylate ester | Human | 10818 | |
| VRK1 | VRK | CK1 | 2kul | A | 5 | - | Human | 4954 | |
| VRK1 | VRK | CK1 | 2rsv | A | 2 | - | Human | 4914 | |
| VRK1 | VRK | CK1 | 2kty | A | 12 | - | Human | 4897 | |
| VRK1 | VRK | CK1 | 6bu6 | A | A | 4,4'-(2-aminopyridine-3,5-diyl)bis(2,6-difluorophenol) | Human | 9423 | |
| VRK1 | VRK | CK1 | 6cnx | B | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-8-(3-methylbutyl)-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9806 | |
| VRK1 | VRK | CK1 | 2rsv | A | 14 | - | Human | 4925 | |
| VRK1 | VRK | CK1 | 2rsv | A | 18 | - | Human | 4934 | |
| VRK1 | VRK | CK1 | 6csw | B | A | (7r)-5-butyl-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7,8-dimethyl-7,8-dihydropteridin-6(5h)-one | Human | 9812 | |
| VRK1 | VRK | CK1 | 3op5 | B | A | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrile | Human | 4894 | |
| VRK1 | VRK | CK1 | 2rsv | A | 6 | - | Human | 4943 | |
| VRK1 | VRK | CK1 | 6npn | C | | (7r)-7-methyl-2-[(3-oxo-2,3-dihydro-1h-indazol-6-yl)amino]-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 11241 | |
| VRK1 | VRK | CK1 | 6csw | D | B | (7r)-5-butyl-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7,8-dimethyl-7,8-dihydropteridin-6(5h)-one | Human | 9809 | |
| VRK1 | VRK | CK1 | 6bru | B | A | (7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7,8-trimethyl-7,8-dihydropteridin-6(5h)-one | Human | 9088 | |
| VRK1 | VRK | CK1 | 2lav | A | 13 | - | Human | 4872 | |
| VRK1 | VRK | CK1 | 6cmm | D | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9759 | |
| VRK1 | VRK | CK1 | 6bp0 | C | B | - | Human | 8742 | |
| VRK1 | VRK | CK1 | 6cfm | D | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9722 | |
| VRK1 | VRK | CK1 | 6btw | A | B | 2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-phenyl-7,8-dihydropteridin-6(5h)-one | Human | 9425 | |
| VRK1 | VRK | CK1 | 2lav | A | 2 | - | Human | 4903 | |
| VRK1 | VRK | CK1 | 2kty | A | 10 | - | Human | 4932 | |
| VRK1 | VRK | CK1 | 6csw | A | A | - | Human | 9818 | |
| VRK1 | VRK | CK1 | 6bru | A | B | - | Human | 9082 | |
| VRK1 | VRK | CK1 | 2kul | A | 7 | - | Human | 4908 | |
| VRK1 | VRK | CK1 | 2kul | A | 3 | - | Human | 4895 | |
| VRK1 | VRK | CK1 | 2kul | A | 11 | - | Human | 4923 | |
| VRK1 | VRK | CK1 | 6cfm | A | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9718 | |
| VRK1 | VRK | CK1 | 6bru | D | A | (7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7,8-trimethyl-7,8-dihydropteridin-6(5h)-one | Human | 9084 | |
| VRK1 | VRK | CK1 | 6bp0 | C | A | - | Human | 8743 | |
| VRK1 | VRK | CK1 | 2kty | A | 11 | - | Human | 4917 | |
| VRK1 | VRK | CK1 | 6cfm | C | A | - | Human | 9719 | |
| VRK1 | VRK | CK1 | 6cqh | B | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-ethyl-7-methyl-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9770 | |
| VRK1 | VRK | CK1 | 6cqh | B | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-ethyl-7-methyl-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9769 | |
| VRK1 | VRK | CK1 | 2kul | A | 18 | - | Human | 4896 | |
| VRK1 | VRK | CK1 | 2rsv | A | 9 | - | Human | 4928 | |
| VRK1 | VRK | CK1 | 2kul | A | 15 | - | Human | 4876 | |
| VRK1 | VRK | CK1 | 2kul | A | 16 | - | Human | 4924 | |
| VRK1 | VRK | CK1 | 6dd4 | C | B | - | Human | 9936 | |
| VRK1 | VRK | CK1 | 6cfm | C | B | - | Human | 9720 | |
| VRK1 | VRK | CK1 | 2kty | A | 20 | - | Human | 4890 | |
| VRK1 | VRK | CK1 | 6cqh | A | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-ethyl-7-methyl-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9774 | |
| VRK1 | VRK | CK1 | 6vzh | A | | - | Human | 12057 | |
| VRK1 | VRK | CK1 | 6btw | B | A | 2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-phenyl-7,8-dihydropteridin-6(5h)-one | Human | 9424 | |
| VRK1 | VRK | CK1 | 6cmm | C | B | - | Human | 9762 | |
| VRK1 | VRK | CK1 | 2lav | A | 9 | - | Human | 4945 | |
| VRK1 | VRK | CK1 | 6btw | A | A | 2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-phenyl-7,8-dihydropteridin-6(5h)-one | Human | 9418 | |
| VRK1 | VRK | CK1 | 2kul | A | 19 | - | Human | 4906 | |
| VRK1 | VRK | CK1 | 6btw | B | B | 2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-phenyl-7,8-dihydropteridin-6(5h)-one | Human | 9411 | |
| VRK1 | VRK | CK1 | 2lav | A | 4 | - | Human | 4884 | |
| VRK1 | VRK | CK1 | 6cnx | D | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-8-(3-methylbutyl)-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9807 | |
| VRK1 | VRK | CK1 | 3op5 | B | B | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrile | Human | 4944 | |
| VRK1 | VRK | CK1 | 6npn | D | | (7r)-7-methyl-2-[(3-oxo-2,3-dihydro-1h-indazol-6-yl)amino]-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 11242 | |
| VRK1 | VRK | CK1 | 6cqh | C | B | - | Human | 9773 | |
| VRK1 | VRK | CK1 | 2kul | A | 13 | - | Human | 4941 | |
| VRK1 | VRK | CK1 | 2kty | A | 9 | - | Human | 4885 | |
| VRK1 | VRK | CK1 | 2kty | A | 7 | - | Human | 4880 | |
| VRK1 | VRK | CK1 | 2lav | A | 20 | - | Human | 4933 | |
| VRK1 | VRK | CK1 | 2rsv | A | 16 | - | Human | 4905 | |
| VRK1 | VRK | CK1 | 2kul | A | 8 | - | Human | 4887 | |
| VRK1 | VRK | CK1 | 6ac9 | B | B | phosphoaminophosphonic acid-adenylate ester | Human | 10823 | |
| VRK1 | VRK | CK1 | 2rsv | A | 11 | - | Human | 4902 | |
| VRK1 | VRK | CK1 | 2kul | A | 1 | - | Human | 4919 | |
| VRK1 | VRK | CK1 | 6btw | D | B | 2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-phenyl-7,8-dihydropteridin-6(5h)-one | Human | 9420 | |
| VRK1 | VRK | CK1 | 6ac9 | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 10816 | |
| VRK1 | VRK | CK1 | 6vzh | C | | - | Human | 12058 | |
| VRK1 | VRK | CK1 | 6bu6 | B | A | 4,4'-(2-aminopyridine-3,5-diyl)bis(2,6-difluorophenol) | Human | 9421 | |
| VRK1 | VRK | CK1 | 2rsv | A | 1 | - | Human | 4910 | |
| VRK1 | VRK | CK1 | 6bru | D | B | (7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7,8-trimethyl-7,8-dihydropteridin-6(5h)-one | Human | 9083 | |
| VRK1 | VRK | CK1 | 6cnx | C | A | (7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-8-(3-methylbutyl)-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9805 | |
| VRK1 | VRK | CK1 | 3op5 | A | B | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrile | Human | 4942 | |
| VRK1 | VRK | CK1 | 2kul | A | 4 | - | Human | 4948 | |
| VRK1 | VRK | CK1 | 6csw | A | B | - | Human | 9813 | |
| VRK1 | VRK | CK1 | 5ukf | A | | 4-{[(z)-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}benzene-1-sulfonamide | Human | 8030 | |
| VRK1 | VRK | CK1 | 6dd4 | B | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-dipropyl-7,8-dihydropteridin-6(5h)-one | Human | 9937 | |
| VRK1 | VRK | CK1 | 2lav | A | 11 | - | Human | 4916 | |
| VRK1 | VRK | CK1 | 5uvf | C | | (7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(3-methylbutyl)-7,8-dihydropteridin-6(5h)-one | Human | 7520 | |
| VRK1 | VRK | CK1 | 2rsv | A | 8 | - | Human | 4918 | |
| VRK1 | VRK | CK1 | 2lav | A | 3 | - | Human | 4912 | |
| VRK1 | VRK | CK1 | 2lav | A | 8 | - | Human | 4881 | |