Search results (26 entries covering 7 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetails File
PRPF4B (PRP4)DYRKCMGC4ijpBB4-(5-{[(2-chloropyridin-4-yl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHuman5534
PRPF4B (PRP4)DYRKCMGC4iirAAphosphoaminophosphonic acid-adenylate esterHuman5545
PRPF4B (PRP4)DYRKCMGC4ianA-Human5543
PRPF4B (PRP4)DYRKCMGC4iirABphosphoaminophosphonic acid-adenylate esterHuman5539
PRPF4B (PRP4)DYRKCMGC4ijpBA4-(5-{[(2-chloropyridin-4-yl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHuman5541
PRPF4B (PRP4)DYRKCMGC4ifcAAadenosine-5'-diphosphateHuman5538
PRPF4B (PRP4)DYRKCMGC6pjjBA4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHuman11583
PRPF4B (PRP4)DYRKCMGC6pjjAB4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHuman11577
PRPF4B (PRP4)DYRKCMGC6pjjAA4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHuman11585
PRPF4B (PRP4)DYRKCMGC4iirBBphosphoaminophosphonic acid-adenylate esterHuman5537
PRPF4B (PRP4)DYRKCMGC4ifcBBadenosine-5'-diphosphateHuman5540
PRPF4B (PRP4)DYRKCMGC6pjjCB4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHuman11586
PRPF4B (PRP4)DYRKCMGC4ianB-Human5546
PRPF4B (PRP4)DYRKCMGC4ifcBAadenosine-5'-diphosphateHuman5542
PRPF4B (PRP4)DYRKCMGC4ifcABadenosine-5'-diphosphateHuman5544
PRPF4B (PRP4)DYRKCMGC4ijpAB4-(5-{[(2-chloropyridin-4-yl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHuman5535
PRPF4B (PRP4)DYRKCMGC6cnhAB4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamideHuman9775
PRPF4B (PRP4)DYRKCMGC6pjjDB4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHuman11579
PRPF4B (PRP4)DYRKCMGC6cnhAA4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamideHuman9776
PRPF4B (PRP4)DYRKCMGC6pjjBB4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHuman11581
PRPF4B (PRP4)DYRKCMGC6pk6AA4-(5-{[(2-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHuman11582
PRPF4B (PRP4)DYRKCMGC6pjjCA4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHuman11578
PRPF4B (PRP4)DYRKCMGC6pk6AB4-(5-{[(2-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHuman11584
PRPF4B (PRP4)DYRKCMGC4ijpAA4-(5-{[(2-chloropyridin-4-yl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHuman5547
PRPF4B (PRP4)DYRKCMGC6pjjDA4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHuman11580
PRPF4B (PRP4)DYRKCMGC4iirBAphosphoaminophosphonic acid-adenylate esterHuman5536