Search results (94 entries covering 48 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetails File
PRKACA (PKACa)PKAAGC5uzkAA2-{3-[3-(piperidin-4-yl)propoxy]phenyl}-n-[4-(1h-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamideHuman9726
PRKACA (PKACa)PKAAGC4ae9AA-Human5265
PRKACA (PKACa)PKAAGC4wb8AAadenosine-5'-triphosphateHuman5304
PRKACA (PKACa)PKAAGC3vqhAAn-[2-(4-bromocinnamylamino)ethyl]-5-isoquinoline sulfonamideHuman5271
PRKACA (PKACa)PKAAGC7y1gAB1-chloranyl-~{n}-[(~{s})-(3-chloranyl-4-cyano-phenyl)-[(2~{r},4~{s})-4-oxidanylpyrrolidin-2-yl]methyl]-7-methoxy-isoquinoline-6-carboxamideHuman14423
PRKACA (PKACa)PKAAGC4ujaAA7-{(3s,4r)-4-[(5-bromothiophen-2-yl)carbonyl]pyrrolidin-3-yl}quinazolin-4(3h)-oneHuman6549
PRKACA (PKACa)PKAAGC4ae9BA-Human5299
PRKACA (PKACa)PKAAGC5izjAB-Human6855
PRKACA (PKACa)PKAAGC5bx7AA1-benzothiophen-3-ylmethanolHuman7076
PRKACA (PKACa)PKAAGC3pooABn'-[(e)-(2,4-dihydroxy-6-methylphenyl)methylidene]-2-(3-methoxyphenyl)acetohydrazideHuman5285
PRKACA (PKACa)PKAAGC3aglB(10r,20r,23r)-1-[(2s,3s,4r,5r)-5-(6-amino-9h-purin-9-yl)-3,4-dihydroxytetrahydrofuran-2-yl]-20,23-bis(3-carbamimidamidopropyl)-10-methyl-1,8,11,18,21-pentaoxo-2,9,12,19,22-pentaazatetracosan-24-amideHuman5283
PRKACA (PKACa)PKAAGC3l9mB(2s)-n~1~-[5-(3-methyl-1h-indazol-5-yl)-1,3,4-thiadiazol-2-yl]-3-(4-methylphenyl)propane-1,2-diamineHuman5278
PRKACA (PKACa)PKAAGC6qj7AA~{n}'-[(2~{s})-2-[3,5-bis(fluoranyl)phenyl]-2-oxidanyl-ethanoyl]-2-ethyl-3-methyl-4-oxidanyl-benzohydrazideHuman11990
PRKACA (PKACa)PKAAGC4ae9AB-Human5307
PRKACA (PKACa)PKAAGC6bysE-Human11262
PRKACA (PKACa)PKAAGC3oogAA1-(4-hydroxy-3-methylphenyl)ethanoneHuman5281
PRKACA (PKACa)PKAAGC2gu8An-[(1s)-2-amino-1-(2,4-dichlorobenzyl)ethyl]-5-[2-(methylamino)pyrimidin-4-yl]thiophene-2-carboxamideHuman5295
PRKACA (PKACa)PKAAGC3owpAB(2s)-2-amino-n'-[(1e)-(3-bromo-4-hydroxyphenyl)methylidene]-2-phenylethanehydrazideHuman5296
PRKACA (PKACa)PKAAGC5bx7AB1-benzothiophen-3-ylmethanolHuman7077
PRKACA (PKACa)PKAAGC5izjAA-Human6857
PRKACA (PKACa)PKAAGC6no7A-Human11465
PRKACA (PKACa)PKAAGC4uj9A7-[(3s,4r)-4-[4-(trifluoromethyl)phenyl]carbonylpyrrolidin-3-yl]-3h-quinazolin-4-oneHuman6544
PRKACA (PKACa)PKAAGC4uj2AA7-[(3s,4r)-4-(3-iodanylphenyl)carbonylpyrrolidin-3-yl]-3h-quinazolin-4-oneHuman6550
PRKACA (PKACa)PKAAGC5j5xAA-Human6853
PRKACA (PKACa)PKAAGC5bx6AA4-chlorophthalazin-1(2h)-oneHuman7075
PRKACA (PKACa)PKAAGC3pooAAn'-[(e)-(2,4-dihydroxy-6-methylphenyl)methylidene]-2-(3-methoxyphenyl)acetohydrazideHuman5300
PRKACA (PKACa)PKAAGC4uj1A7-[(3s,4r)-4-(3-chlorophenyl)carbonylpyrrolidin-3-yl]-3h-quinazolin-4-oneHuman6548
PRKACA (PKACa)PKAAGC6wjgB-Human13007
PRKACA (PKACa)PKAAGC3oxtA(2s)-2-amino-n'-[(1e)-(2,4-dihydroxy-6-methylphenyl)methylidene]-2-phenylethanehydrazideHuman5268
PRKACA (PKACa)PKAAGC5izjBA-Human6851
PRKACA (PKACa)PKAAGC6bysA-Human11259
PRKACA (PKACa)PKAAGC3mvjA(3r)-1-(5-methyl-7h-pyrrolo[2,3-d]pyrimidin-4-yl)pyrrolidin-3-amineHuman5289
PRKACA (PKACa)PKAAGC4ae6BB-Human5298
PRKACA (PKACa)PKAAGC3ovvAAn'-[(1e)-(4-hydroxyphenyl)methylidene]-2-(3-methoxyphenyl)acetohydrazideHuman5266
PRKACA (PKACa)PKAAGC3p0mAA(2r)-4-amino-n'-[(1e)-(3-bromo-4-hydroxyphenyl)methylidene]-2-phenylbutanehydrazideHuman5297
PRKACA (PKACa)PKAAGC4wb7BAadenosine-5'-triphosphateHuman6875
PRKACA (PKACa)PKAAGC6byrAadenosine-5'-triphosphateHuman11256
PRKACA (PKACa)PKAAGC4ujbAB7-[(3s,4r)-4-(3-fluorophenyl)carbonylpyrrolidin-3-yl]-3h-quinazolin-4-oneHuman6545
PRKACA (PKACa)PKAAGC3vqhABn-[2-(4-bromocinnamylamino)ethyl]-5-isoquinoline sulfonamideHuman5275
PRKACA (PKACa)PKAAGC3aglA(10r,20r,23r)-1-[(2s,3s,4r,5r)-5-(6-amino-9h-purin-9-yl)-3,4-dihydroxytetrahydrofuran-2-yl]-20,23-bis(3-carbamimidamidopropyl)-10-methyl-1,8,11,18,21-pentaoxo-2,9,12,19,22-pentaazatetracosan-24-amideHuman5267
PRKACA (PKACa)PKAAGC4ae9BB-Human5286
PRKACA (PKACa)PKAAGC3amaA4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHuman5284
PRKACA (PKACa)PKAAGC4uj2AB7-[(3s,4r)-4-(3-iodanylphenyl)carbonylpyrrolidin-3-yl]-3h-quinazolin-4-oneHuman6551
PRKACA (PKACa)PKAAGC6wjfA-Human13008
PRKACA (PKACa)PKAAGC6wjfB-Human13009
PRKACA (PKACa)PKAAGC5n23AA1-cyclopropyl-3-{3-[5-(morpholin-4-ylmethyl)-1h-benzimidazol-2-yl]-1h-pyrazol-4-yl}ureaHuman9747
PRKACA (PKACa)PKAAGC4wb6Aadenosine-5'-triphosphateHuman5303
PRKACA (PKACa)PKAAGC4ujbAA7-[(3s,4r)-4-(3-fluorophenyl)carbonylpyrrolidin-3-yl]-3h-quinazolin-4-oneHuman6546
PRKACA (PKACa)PKAAGC3l9lA5-[2-({(2s)-2-amino-3-[4-(trifluoromethyl)phenyl]propyl}amino)-1,3-thiazol-5-yl]-1,3-dihydro-2h-indol-2-oneHuman5305
PRKACA (PKACa)PKAAGC3p0mAB(2r)-4-amino-n'-[(1e)-(3-bromo-4-hydroxyphenyl)methylidene]-2-phenylbutanehydrazideHuman5279
PRKACA (PKACa)PKAAGC4ae6BA-Human5290
PRKACA (PKACa)PKAAGC7y1gAA1-chloranyl-~{n}-[(~{s})-(3-chloranyl-4-cyano-phenyl)-[(2~{r},4~{s})-4-oxidanylpyrrolidin-2-yl]methyl]-7-methoxy-isoquinoline-6-carboxamideHuman14422
PRKACA (PKACa)PKAAGC5izjBB-Human6858
PRKACA (PKACa)PKAAGC3mvjE(3r)-1-(5-methyl-7h-pyrrolo[2,3-d]pyrimidin-4-yl)pyrrolidin-3-amineHuman5291
PRKACA (PKACa)PKAAGC3owpAA(2s)-2-amino-n'-[(1e)-(3-bromo-4-hydroxyphenyl)methylidene]-2-phenylethanehydrazideHuman5273
PRKACA (PKACa)PKAAGC8fecA6-[(6p)-6-(4-bromo-1-methyl-1h-imidazol-5-yl)-2,3-dihydro-4h-1,4-thiazin-4-yl]-7h-purineHuman14890
PRKACA (PKACa)PKAAGC8fe5A6-[(6p)-6-(1-methyl-1h-imidazol-5-yl)-2,3-dihydro-4h-1,4-thiazin-4-yl]-7,9-dihydro-8h-purin-8-oneHuman14888
PRKACA (PKACa)PKAAGC8fe2A6-[(6m)-6-(1-methyl-1h-imidazol-5-yl)-2,3-dihydro-4h-1,4-thiazin-4-yl]-9h-purineHuman14889
PRKACA (PKACa)PKAAGC3ambAcyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amideHuman5276
PRKACA (PKACa)PKAAGC3nx8AA-Human5277
PRKACA (PKACa)PKAAGC4wb7ABadenosine-5'-triphosphateHuman6878
PRKACA (PKACa)PKAAGC6frxA~{n}-[3-[(5-chloranyl-2-phenylazanyl-pyrimidin-4-yl)amino]phenyl]prop-2-enamideHuman11261
PRKACA (PKACa)PKAAGC4ae6AB-Human5301
PRKACA (PKACa)PKAAGC3l9nA(2s)-n~1~-[5-(1h-indazol-5-yl)-1,3,4-thiadiazol-2-yl]-3-(4-methylphenyl)propane-1,2-diamineHuman5292
PRKACA (PKACa)PKAAGC4wb8ABadenosine-5'-triphosphateHuman5287
PRKACA (PKACa)PKAAGC6no7Eadenosine-5'-triphosphateHuman11463
PRKACA (PKACa)PKAAGC6c0uAn-[(3r,4r)-4-{[4-(2-fluoro-3-methoxy-6-propoxybenzene-1-carbonyl)benzene-1-carbonyl]amino}pyrrolidin-3-yl]-1h-indazole-5-carboxamideHuman9974
PRKACA (PKACa)PKAAGC4ae6AA-Human5274
PRKACA (PKACa)PKAAGC5izfA-Human6854
PRKACA (PKACa)PKAAGC3agmA-Human5282
PRKACA (PKACa)PKAAGC3l9lB5-[2-({(2s)-2-amino-3-[4-(trifluoromethyl)phenyl]propyl}amino)-1,3-thiazol-5-yl]-1,3-dihydro-2h-indol-2-oneHuman5302
PRKACA (PKACa)PKAAGC4wb7BBadenosine-5'-triphosphateHuman6877
PRKACA (PKACa)PKAAGC3nx8AB-Human5294
PRKACA (PKACa)PKAAGC5j5xAC-Human6852
PRKACA (PKACa)PKAAGC5n23AB1-cyclopropyl-3-{3-[5-(morpholin-4-ylmethyl)-1h-benzimidazol-2-yl]-1h-pyrazol-4-yl}ureaHuman9746
PRKACA (PKACa)PKAAGC6wjgA-Human13006
PRKACA (PKACa)PKAAGC6byrCadenosine-5'-triphosphateHuman11258
PRKACA (PKACa)PKAAGC3mvjB-Human5288
PRKACA (PKACa)PKAAGC6bysG-Human11260
PRKACA (PKACa)PKAAGC6no7C-Human11466
PRKACA (PKACa)PKAAGC6qj7AB~{n}'-[(2~{s})-2-[3,5-bis(fluoranyl)phenyl]-2-oxidanyl-ethanoyl]-2-ethyl-3-methyl-4-oxidanyl-benzohydrazideHuman11991
PRKACA (PKACa)PKAAGC4wb7AAadenosine-5'-triphosphateHuman6876
PRKACA (PKACa)PKAAGC3l9mA(2s)-n~1~-[5-(3-methyl-1h-indazol-5-yl)-1,3,4-thiadiazol-2-yl]-3-(4-methylphenyl)propane-1,2-diamineHuman5270
PRKACA (PKACa)PKAAGC4wb6Badenosine-5'-triphosphateHuman5293
PRKACA (PKACa)PKAAGC5bx6AB4-chlorophthalazin-1(2h)-oneHuman7078
PRKACA (PKACa)PKAAGC3ovvABn'-[(1e)-(4-hydroxyphenyl)methylidene]-2-(3-methoxyphenyl)acetohydrazideHuman5269
PRKACA (PKACa)PKAAGC6bysC-Human11257
PRKACA (PKACa)PKAAGC3oogAB1-(4-hydroxy-3-methylphenyl)ethanoneHuman5272
PRKACA (PKACa)PKAAGC4wb5ABadenosine-5'-triphosphateHuman5306
PRKACA (PKACa)PKAAGC4wb5AAadenosine-5'-triphosphateHuman5280
PRKACA (PKACa)PKAAGC6no7Gadenosine-5'-triphosphateHuman11464
PRKACA (PKACa)PKAAGC4ujaAB7-{(3s,4r)-4-[(5-bromothiophen-2-yl)carbonyl]pyrrolidin-3-yl}quinazolin-4(3h)-oneHuman6547
PRKACA (PKACa)PKAAGC8x5lA(2s)-2-(4-chlorophenyl)-2-hydroxy-2-[4-(1h-pyrazol-4-yl)phenyl]ethanaminiumHuman15111
PRKACA (PKACa)PKAAGC5j5xAB-Human6856