| STK24 (MST3) | STE20 | STE | 4o27 | B | | adenosine-5'-diphosphate | Human | 5602 | |
| STK24 (MST3) | STE20 | STE | 7b33 | A | | 8-[(5-azanyl-1,3-dioxan-2-yl)methyl]-6-[4-[6-[bis(fluoranyl)methyl]pyridin-2-yl]-2-chloranyl-phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7-one | Human | 13048 | |
| STK24 (MST3) | STE20 | STE | 4qmn | A | B | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | 5604 | |
| STK24 (MST3) | STE20 | STE | 8bzj | A | B | 8-(4-azanylbutyl)-6-[2-chloranyl-4-(6-methylpyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7-one | Human | 14583 | |
| STK24 (MST3) | STE20 | STE | 8bzj | A | A | 8-(4-azanylbutyl)-6-[2-chloranyl-4-(6-methylpyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7-one | Human | 14586 | |
| STK24 (MST3) | STE20 | STE | 8bzi | A | B | 8-(4-azanylbutyl)-6-[2,5-bis(fluoranyl)-4-(6-methylpyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7-one | Human | 14584 | |
| STK24 (MST3) | STE20 | STE | 3a7f | A | | - | Human | 5596 | |
| STK24 (MST3) | STE20 | STE | 4qmv | A | | n-{2-[(1s,4r)-6-{[4-(cyclobutylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino}-1,2,3,4-tetrahydro-1,4-epiminonaphthalen-9-yl]-2-oxoethyl}acetamide | Human | 5581 | |
| STK24 (MST3) | STE20 | STE | 4qmq | A | A | 1-{2-[5-(2-methoxyethoxy)-1h-benzimidazol-1-yl]quinolin-8-yl}piperidin-4-amine | Human | 5607 | |
| STK24 (MST3) | STE20 | STE | 3a7j | A | | adenosine-5'-diphosphate | Human | 5594 | |
| STK24 (MST3) | STE20 | STE | 7b31 | A | A | 1-[(5-azanyl-1,3-dioxan-2-yl)methyl]-3-[2-chloranyl-4-(3-fluoranylpyridin-2-yl)phenyl]-7-(methylamino)-1,6-naphthyridin-2-one | Human | 13045 | |
| STK24 (MST3) | STE20 | STE | 7b34 | A | | 8-[(5-azanyl-1,3-dioxan-2-yl)methyl]-6-[2-chloranyl-4-(3-fluoranyl-6-methyl-pyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7-one | Human | 13051 | |
| STK24 (MST3) | STE20 | STE | 7b35 | B | | 8-[(5-azanyl-1,3-dioxan-2-yl)methyl]-6-[2-chloranyl-4-(3-methoxy-6-methyl-pyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7-one | Human | 13046 | |
| STK24 (MST3) | STE20 | STE | 4qmz | A | | n-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 5578 | |
| STK24 (MST3) | STE20 | STE | 4qms | A | B | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 5608 | |
| STK24 (MST3) | STE20 | STE | 4qms | A | A | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 5590 | |
| STK24 (MST3) | STE20 | STE | 3ckw | A | A | - | Human | 5580 | |
| STK24 (MST3) | STE20 | STE | 3zhp | C | | - | Human | 5593 | |
| STK24 (MST3) | STE20 | STE | 3zhp | D | | - | Human | 5588 | |
| STK24 (MST3) | STE20 | STE | 4qmx | A | | n-(5-chloro-1,3-benzodioxol-4-yl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]-5-(tetrahydro-2h-pyran-4-yloxy)quinazolin-4-amine | Human | 5609 | |
| STK24 (MST3) | STE20 | STE | 4qmt | A | | n-[2-oxo-3-((e)-phenyl{[4-(piperidin-1-ylmethyl)phenyl]imino}methyl)-2,6-dihydro-1h-indol-5-yl]ethanesulfonamide | Human | 5613 | |
| STK24 (MST3) | STE20 | STE | 4u8z | A | | 3-[4-(morpholin-4-yl)-7h-pyrrolo[2,3-d]pyrimidin-5-yl]benzonitrile | Human | 5610 | |
| STK24 (MST3) | STE20 | STE | 4qml | A | | phosphoaminophosphonic acid-adenylate ester | Human | 5605 | |
| STK24 (MST3) | STE20 | STE | 7b30 | A | | 8-[(trans-5-amino-1,3-dioxan-2-yl)methyl]-6-[2-chloro-4-(6-methylpyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7(8h)-one | Human | 13047 | |
| STK24 (MST3) | STE20 | STE | 3a7g | A | | - | Human | 5612 | |
| STK24 (MST3) | STE20 | STE | 4qmw | A | A | 1-cyclopentyl-3-(1h-pyrrolo[2,3-b]pyridin-5-yl)-1h-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 5577 | |
| STK24 (MST3) | STE20 | STE | 7b32 | A | | 8-[(5-azanyl-1,3-dioxan-2-yl)methyl]-6-[2-chloranyl-4-(6-methylpyridin-2-yl)phenyl]-2-[(2-methoxyphenyl)amino]pyrido[2,3-d]pyrimidin-7-one | Human | 13049 | |
| STK24 (MST3) | STE20 | STE | 3a7i | A | | adenine | Human | 5611 | |
| STK24 (MST3) | STE20 | STE | 3ckx | A | | staurosporine | Human | 5599 | |
| STK24 (MST3) | STE20 | STE | 7b31 | A | B | 1-[(5-azanyl-1,3-dioxan-2-yl)methyl]-3-[2-chloranyl-4-(3-fluoranylpyridin-2-yl)phenyl]-7-(methylamino)-1,6-naphthyridin-2-one | Human | 13050 | |
| STK24 (MST3) | STE20 | STE | 4qmy | A | | staurosporine | Human | 5592 | |
| STK24 (MST3) | STE20 | STE | 4w8d | A | | 5-(1-methyl-1h-pyrazol-4-yl)-4-(morpholin-4-yl)-7h-pyrrolo[2,3-d]pyrimidine | Human | 5614 | |
| STK24 (MST3) | STE20 | STE | 4qmu | A | A | 4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamide | Human | 5606 | |
| STK24 (MST3) | STE20 | STE | 4qmm | A | | 1-cyclopropyl-3-{3-[5-(morpholin-4-ylmethyl)-1h-benzimidazol-2-yl]-1h-pyrazol-4-yl}urea | Human | 5583 | |
| STK24 (MST3) | STE20 | STE | 8qlt | A | B | 8-(4-azanylbutyl)-6-[2-chloranyl-4-(6-methylpyridin-2-yl)phenyl]-2-[3-(2-oxidanylidenepyrrolidin-1-yl)propylamino]pyrido[2,3-d]pyrimidin-7-one | Human | 14869 | |
| STK24 (MST3) | STE20 | STE | 8qlq | A | A | macrocyclic inhibitor | Human | 14873 | |
| STK24 (MST3) | STE20 | STE | 8qlt | A | A | 8-(4-azanylbutyl)-6-[2-chloranyl-4-(6-methylpyridin-2-yl)phenyl]-2-[3-(2-oxidanylidenepyrrolidin-1-yl)propylamino]pyrido[2,3-d]pyrimidin-7-one | Human | 14874 | |
| STK24 (MST3) | STE20 | STE | 8qls | A | B | 8-(4-azanylbutyl)-6-[2-chloranyl-4-(6-methylpyridin-2-yl)phenyl]-2-(3-morpholin-4-ylpropylamino)pyrido[2,3-d]pyrimidin-7-one | Human | 14876 | |
| STK24 (MST3) | STE20 | STE | 8qlr | A | | 8-(4-azanylbutyl)-2-[1,3-bis(oxidanyl)propan-2-ylamino]-6-[2-chloranyl-4-(6-methylpyridin-2-yl)phenyl]pyrido[2,3-d]pyrimidin-7-one | Human | 14875 | |
| STK24 (MST3) | STE20 | STE | 4qmo | A | A | (8z)-8-(1h-imidazol-5-ylmethylidene)-6,8-dihydro-7h-[1,3]thiazolo[5,4-e]indol-7-one | Human | 5585 | |
| STK24 (MST3) | STE20 | STE | 3a7g | B | | - | Human | 5598 | |
| STK24 (MST3) | STE20 | STE | 4qna | A | | 2-(4,6-diamino-1,3,5-triazin-2-yl)phenol | Human | 5579 | |
| STK24 (MST3) | STE20 | STE | 4qo9 | A | | n-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamide | Human | 5586 | |
| STK24 (MST3) | STE20 | STE | 4qmq | A | B | 1-{2-[5-(2-methoxyethoxy)-1h-benzimidazol-1-yl]quinolin-8-yl}piperidin-4-amine | Human | 5595 | |
| STK24 (MST3) | STE20 | STE | 4qmo | A | B | (8z)-8-(1h-imidazol-5-ylmethylidene)-6,8-dihydro-7h-[1,3]thiazolo[5,4-e]indol-7-one | Human | 5597 | |
| STK24 (MST3) | STE20 | STE | 4qo9 | B | | n-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamide | Human | 5591 | |
| STK24 (MST3) | STE20 | STE | 3a7h | A | | adenosine-5'-triphosphate | Human | 5600 | |
| STK24 (MST3) | STE20 | STE | 8qlq | A | B | macrocyclic inhibitor | Human | 14870 | |
| STK24 (MST3) | STE20 | STE | 4qmu | A | B | 4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamide | Human | 5603 | |
| STK24 (MST3) | STE20 | STE | 3ckw | A | B | - | Human | 5601 | |
| STK24 (MST3) | STE20 | STE | 8qls | A | C | 8-(4-azanylbutyl)-6-[2-chloranyl-4-(6-methylpyridin-2-yl)phenyl]-2-(3-morpholin-4-ylpropylamino)pyrido[2,3-d]pyrimidin-7-one | Human | 14871 | |
| STK24 (MST3) | STE20 | STE | 4w8e | A | | 3-{4-[(2r)-2-(5-methyl-1,2,4-oxadiazol-3-yl)morpholin-4-yl]-7h-pyrrolo[2,3-d]pyrimidin-5-yl}benzonitrile | Human | 5589 | |
| STK24 (MST3) | STE20 | STE | 8bzi | A | A | 8-(4-azanylbutyl)-6-[2,5-bis(fluoranyl)-4-(6-methylpyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7-one | Human | 14585 | |
| STK24 (MST3) | STE20 | STE | 8qls | A | A | 8-(4-azanylbutyl)-6-[2-chloranyl-4-(6-methylpyridin-2-yl)phenyl]-2-(3-morpholin-4-ylpropylamino)pyrido[2,3-d]pyrimidin-7-one | Human | 14872 | |
| STK24 (MST3) | STE20 | STE | 3a7h | B | | adenosine-5'-triphosphate | Human | 5576 | |
| STK24 (MST3) | STE20 | STE | 4qmn | A | A | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | 5587 | |
| STK24 (MST3) | STE20 | STE | 4qmw | A | B | 1-cyclopentyl-3-(1h-pyrrolo[2,3-b]pyridin-5-yl)-1h-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 5582 | |
| STK24 (MST3) | STE20 | STE | 4qmp | A | | 5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamide | Human | 5584 | |
| STK24 (MST3) | STE20 | STE | 7b35 | A | | 8-[(5-azanyl-1,3-dioxan-2-yl)methyl]-6-[2-chloranyl-4-(3-methoxy-6-methyl-pyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7-one | Human | 13052 | |