Search results (59 entries covering 40 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetails File
STK24 (MST3)STE20STE4o27Badenosine-5'-diphosphateHuman5602
STK24 (MST3)STE20STE7b33A8-[(5-azanyl-1,3-dioxan-2-yl)methyl]-6-[4-[6-[bis(fluoranyl)methyl]pyridin-2-yl]-2-chloranyl-phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7-oneHuman13048
STK24 (MST3)STE20STE4qmnAB4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrileHuman5604
STK24 (MST3)STE20STE8bzjAB8-(4-azanylbutyl)-6-[2-chloranyl-4-(6-methylpyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7-oneHuman14583
STK24 (MST3)STE20STE8bzjAA8-(4-azanylbutyl)-6-[2-chloranyl-4-(6-methylpyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7-oneHuman14586
STK24 (MST3)STE20STE8bziAB8-(4-azanylbutyl)-6-[2,5-bis(fluoranyl)-4-(6-methylpyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7-oneHuman14584
STK24 (MST3)STE20STE3a7fA-Human5596
STK24 (MST3)STE20STE4qmvAn-{2-[(1s,4r)-6-{[4-(cyclobutylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino}-1,2,3,4-tetrahydro-1,4-epiminonaphthalen-9-yl]-2-oxoethyl}acetamideHuman5581
STK24 (MST3)STE20STE4qmqAA1-{2-[5-(2-methoxyethoxy)-1h-benzimidazol-1-yl]quinolin-8-yl}piperidin-4-amineHuman5607
STK24 (MST3)STE20STE3a7jAadenosine-5'-diphosphateHuman5594
STK24 (MST3)STE20STE7b31AA1-[(5-azanyl-1,3-dioxan-2-yl)methyl]-3-[2-chloranyl-4-(3-fluoranylpyridin-2-yl)phenyl]-7-(methylamino)-1,6-naphthyridin-2-oneHuman13045
STK24 (MST3)STE20STE7b34A8-[(5-azanyl-1,3-dioxan-2-yl)methyl]-6-[2-chloranyl-4-(3-fluoranyl-6-methyl-pyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7-oneHuman13051
STK24 (MST3)STE20STE7b35B8-[(5-azanyl-1,3-dioxan-2-yl)methyl]-6-[2-chloranyl-4-(3-methoxy-6-methyl-pyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7-oneHuman13046
STK24 (MST3)STE20STE4qmzAn-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman5578
STK24 (MST3)STE20STE4qmsABn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman5608
STK24 (MST3)STE20STE4qmsAAn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman5590
STK24 (MST3)STE20STE3ckwAA-Human5580
STK24 (MST3)STE20STE3zhpC-Human5593
STK24 (MST3)STE20STE3zhpD-Human5588
STK24 (MST3)STE20STE4qmxAn-(5-chloro-1,3-benzodioxol-4-yl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]-5-(tetrahydro-2h-pyran-4-yloxy)quinazolin-4-amineHuman5609
STK24 (MST3)STE20STE4qmtAn-[2-oxo-3-((e)-phenyl{[4-(piperidin-1-ylmethyl)phenyl]imino}methyl)-2,6-dihydro-1h-indol-5-yl]ethanesulfonamideHuman5613
STK24 (MST3)STE20STE4u8zA3-[4-(morpholin-4-yl)-7h-pyrrolo[2,3-d]pyrimidin-5-yl]benzonitrileHuman5610
STK24 (MST3)STE20STE4qmlAphosphoaminophosphonic acid-adenylate esterHuman5605
STK24 (MST3)STE20STE7b30A8-[(trans-5-amino-1,3-dioxan-2-yl)methyl]-6-[2-chloro-4-(6-methylpyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7(8h)-oneHuman13047
STK24 (MST3)STE20STE3a7gA-Human5612
STK24 (MST3)STE20STE4qmwAA1-cyclopentyl-3-(1h-pyrrolo[2,3-b]pyridin-5-yl)-1h-pyrazolo[3,4-d]pyrimidin-4-amineHuman5577
STK24 (MST3)STE20STE7b32A8-[(5-azanyl-1,3-dioxan-2-yl)methyl]-6-[2-chloranyl-4-(6-methylpyridin-2-yl)phenyl]-2-[(2-methoxyphenyl)amino]pyrido[2,3-d]pyrimidin-7-oneHuman13049
STK24 (MST3)STE20STE3a7iAadenineHuman5611
STK24 (MST3)STE20STE3ckxAstaurosporineHuman5599
STK24 (MST3)STE20STE7b31AB1-[(5-azanyl-1,3-dioxan-2-yl)methyl]-3-[2-chloranyl-4-(3-fluoranylpyridin-2-yl)phenyl]-7-(methylamino)-1,6-naphthyridin-2-oneHuman13050
STK24 (MST3)STE20STE4qmyAstaurosporineHuman5592
STK24 (MST3)STE20STE4w8dA5-(1-methyl-1h-pyrazol-4-yl)-4-(morpholin-4-yl)-7h-pyrrolo[2,3-d]pyrimidineHuman5614
STK24 (MST3)STE20STE4qmuAA4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHuman5606
STK24 (MST3)STE20STE4qmmA1-cyclopropyl-3-{3-[5-(morpholin-4-ylmethyl)-1h-benzimidazol-2-yl]-1h-pyrazol-4-yl}ureaHuman5583
STK24 (MST3)STE20STE8qltAB8-(4-azanylbutyl)-6-[2-chloranyl-4-(6-methylpyridin-2-yl)phenyl]-2-[3-(2-oxidanylidenepyrrolidin-1-yl)propylamino]pyrido[2,3-d]pyrimidin-7-oneHuman14869
STK24 (MST3)STE20STE8qlqAAmacrocyclic inhibitorHuman14873
STK24 (MST3)STE20STE8qltAA8-(4-azanylbutyl)-6-[2-chloranyl-4-(6-methylpyridin-2-yl)phenyl]-2-[3-(2-oxidanylidenepyrrolidin-1-yl)propylamino]pyrido[2,3-d]pyrimidin-7-oneHuman14874
STK24 (MST3)STE20STE8qlsAB8-(4-azanylbutyl)-6-[2-chloranyl-4-(6-methylpyridin-2-yl)phenyl]-2-(3-morpholin-4-ylpropylamino)pyrido[2,3-d]pyrimidin-7-oneHuman14876
STK24 (MST3)STE20STE8qlrA8-(4-azanylbutyl)-2-[1,3-bis(oxidanyl)propan-2-ylamino]-6-[2-chloranyl-4-(6-methylpyridin-2-yl)phenyl]pyrido[2,3-d]pyrimidin-7-oneHuman14875
STK24 (MST3)STE20STE4qmoAA(8z)-8-(1h-imidazol-5-ylmethylidene)-6,8-dihydro-7h-[1,3]thiazolo[5,4-e]indol-7-oneHuman5585
STK24 (MST3)STE20STE3a7gB-Human5598
STK24 (MST3)STE20STE4qnaA2-(4,6-diamino-1,3,5-triazin-2-yl)phenolHuman5579
STK24 (MST3)STE20STE4qo9An-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamideHuman5586
STK24 (MST3)STE20STE4qmqAB1-{2-[5-(2-methoxyethoxy)-1h-benzimidazol-1-yl]quinolin-8-yl}piperidin-4-amineHuman5595
STK24 (MST3)STE20STE4qmoAB(8z)-8-(1h-imidazol-5-ylmethylidene)-6,8-dihydro-7h-[1,3]thiazolo[5,4-e]indol-7-oneHuman5597
STK24 (MST3)STE20STE4qo9Bn-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamideHuman5591
STK24 (MST3)STE20STE3a7hAadenosine-5'-triphosphateHuman5600
STK24 (MST3)STE20STE8qlqABmacrocyclic inhibitorHuman14870
STK24 (MST3)STE20STE4qmuAB4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHuman5603
STK24 (MST3)STE20STE3ckwAB-Human5601
STK24 (MST3)STE20STE8qlsAC8-(4-azanylbutyl)-6-[2-chloranyl-4-(6-methylpyridin-2-yl)phenyl]-2-(3-morpholin-4-ylpropylamino)pyrido[2,3-d]pyrimidin-7-oneHuman14871
STK24 (MST3)STE20STE4w8eA3-{4-[(2r)-2-(5-methyl-1,2,4-oxadiazol-3-yl)morpholin-4-yl]-7h-pyrrolo[2,3-d]pyrimidin-5-yl}benzonitrileHuman5589
STK24 (MST3)STE20STE8bziAA8-(4-azanylbutyl)-6-[2,5-bis(fluoranyl)-4-(6-methylpyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7-oneHuman14585
STK24 (MST3)STE20STE8qlsAA8-(4-azanylbutyl)-6-[2-chloranyl-4-(6-methylpyridin-2-yl)phenyl]-2-(3-morpholin-4-ylpropylamino)pyrido[2,3-d]pyrimidin-7-oneHuman14872
STK24 (MST3)STE20STE3a7hBadenosine-5'-triphosphateHuman5576
STK24 (MST3)STE20STE4qmnAA4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrileHuman5587
STK24 (MST3)STE20STE4qmwAB1-cyclopentyl-3-(1h-pyrrolo[2,3-b]pyridin-5-yl)-1h-pyrazolo[3,4-d]pyrimidin-4-amineHuman5582
STK24 (MST3)STE20STE4qmpA5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamideHuman5584
STK24 (MST3)STE20STE7b35A8-[(5-azanyl-1,3-dioxan-2-yl)methyl]-6-[2-chloranyl-4-(3-methoxy-6-methyl-pyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7-oneHuman13052