| RET | Ret | TK | 7dua | A | B | 4-azanyl-7-(1-methylcyclopropyl)-~{n}-(5-methyl-1~{h}-pyrazol-3-yl)pyrrolo[2,3-d]pyrimidine-5-carboxamide | Human | 14049 | |
| RET | Ret | TK | 6i82 | A | B | ~{n}-[3-(1,3-benzodioxol-5-yl)pyrazolo[1,5-a]pyrimidin-5-yl]-~{n}',~{n}'-dimethyl-propane-1,3-diamine | Human | 12054 | |
| RET | Ret | TK | 7run | A | | 1-(4-{(1s,3s)-3-[4-amino-5-(3-amino-4-chlorophenyl)-7h-pyrrolo[2,3-d]pyrimidin-7-yl]cyclobutyl}piperazin-1-yl)ethan-1-one | Human | 14072 | |
| RET | Ret | TK | 7du8 | A | B | selpercatinib | Human | 14095 | |
| RET | Ret | TK | 7dua | A | C | 4-azanyl-7-(1-methylcyclopropyl)-~{n}-(5-methyl-1~{h}-pyrazol-3-yl)pyrrolo[2,3-d]pyrimidine-5-carboxamide | Human | 14046 | |
| RET | Ret | TK | 6i82 | B | B | ~{n}-[3-(1,3-benzodioxol-5-yl)pyrazolo[1,5-a]pyrimidin-5-yl]-~{n}',~{n}'-dimethyl-propane-1,3-diamine | Human | 12053 | |
| RET | Ret | TK | 2x2m | A | | (3z)-3-[(3,5-dimethyl-1h-pyrrol-2-yl)methylidene]-1,3-dihydro-2h-indol-2-one | Human | 3366 | |
| RET | Ret | TK | 7ju6 | A | A | selpercatinib | Human | 13103 | |
| RET | Ret | TK | 6nec | A | B | methyl (3z)-3-{[(4-{methyl[(4-methylpiperazin-1-yl)acetyl]amino}phenyl)amino](phenyl)methylidene}-2-oxo-2,3-dihydro-1h-indole-6-carboxylate | Human | 11150 | |
| RET | Ret | TK | 6i82 | B | A | ~{n}-[3-(1,3-benzodioxol-5-yl)pyrazolo[1,5-a]pyrimidin-5-yl]-~{n}',~{n}'-dimethyl-propane-1,3-diamine | Human | 12052 | |
| RET | Ret | TK | 2x2k | A | B | (3z)-5-amino-3-[(3,5-dimethyl-1h-pyrrol-2-yl)methylidene]-1,3-dihydro-2h-indol-2-one | Human | 3358 | |
| RET | Ret | TK | 7ju5 | B | B | pralsetinib | Human | 13108 | |
| RET | Ret | TK | 4cki | A | C | adenosine | Human | 3368 | |
| RET | Ret | TK | 7ju5 | A | B | pralsetinib | Human | 13109 | |
| RET | Ret | TK | 6vhg | A | B | 3-(3,4-dimethoxyphenyl)-n~5~-(1-methylpiperidin-4-yl)-6-phenylpyrazolo[1,5-a]pyrimidine-5,7-diamine | Human | 11998 | |
| RET | Ret | TK | 2x2l | A | C | (3z)-5-amino-3-[(4-methoxyphenyl)methylidene]-1,3-dihydro-2h-indol-2-one | Human | 3367 | |
| RET | Ret | TK | 5fm2 | A | | 1-ter-butyl-3-p-tolyl-1h-pyrazolo[3,4-d]pyrimidin-4-ylamine | Human | 7328 | |
| RET | Ret | TK | 7ju6 | B | A | selpercatinib | Human | 13110 | |
| RET | Ret | TK | 2ivt | A | B | adenosine monophosphate | Human | 3365 | |
| RET | Ret | TK | 2x2m | B | | (3z)-3-[(3,5-dimethyl-1h-pyrrol-2-yl)methylidene]-1,3-dihydro-2h-indol-2-one | Human | 3375 | |
| RET | Ret | TK | 6ne7 | A | C | adenosine monophosphate | Human | 11152 | |
| RET | Ret | TK | 7ju6 | B | B | selpercatinib | Human | 13104 | |
| RET | Ret | TK | 7ju5 | B | A | pralsetinib | Human | 13105 | |
| RET | Ret | TK | 6fek | A | A | adenosine | Human | 9604 | |
| RET | Ret | TK | 4ckj | A | A | adenosine | Human | 3359 | |
| RET | Ret | TK | 7nzn | A | | 2-[4-[[4-[1-[2-(dimethylamino)ethyl]pyrazol-4-yl]-6-[(3-methyl-1~{h}-pyrazol-5-yl)amino]pyrimidin-2-yl]amino]phenyl]-~{n}-(3-fluorophenyl)ethanamide | Human | 14105 | |
| RET | Ret | TK | 4ckj | A | B | adenosine | Human | 3376 | |
| RET | Ret | TK | 2ivs | A | A | (3ar,4r,6r,6ar)-4-(6-amino-9h-purin-9-yl)-6-(hydroxymethyl)tetrahydrofuro[3,4-d][1,3,2]dioxaphosphol-2-ol 2-oxide | Human | 3372 | |
| RET | Ret | TK | 6nja | A | A | adenine | Human | 11146 | |
| RET | Ret | TK | 2x2l | A | A | (3z)-5-amino-3-[(4-methoxyphenyl)methylidene]-1,3-dihydro-2h-indol-2-one | Human | 3363 | |
| RET | Ret | TK | 6i82 | A | A | ~{n}-[3-(1,3-benzodioxol-5-yl)pyrazolo[1,5-a]pyrimidin-5-yl]-~{n}',~{n}'-dimethyl-propane-1,3-diamine | Human | 12050 | |
| RET | Ret | TK | 7du9 | A | B | pralsetinib | Human | 14047 | |
| RET | Ret | TK | 5amn | A | | 4-[3-hydroxyanilino]-6,7-dimethoxyquinazoline | Human | 6412 | |
| RET | Ret | TK | 2ivv | A | | 1-ter-butyl-3-p-tolyl-1h-pyrazolo[3,4-d]pyrimidin-4-ylamine | Human | 3373 | |
| RET | Ret | TK | 6nec | C | A | methyl (3z)-3-{[(4-{methyl[(4-methylpiperazin-1-yl)acetyl]amino}phenyl)amino](phenyl)methylidene}-2-oxo-2,3-dihydro-1h-indole-6-carboxylate | Human | 11147 | |
| RET | Ret | TK | 6fek | A | B | adenosine | Human | 9603 | |
| RET | Ret | TK | 6nec | A | A | methyl (3z)-3-{[(4-{methyl[(4-methylpiperazin-1-yl)acetyl]amino}phenyl)amino](phenyl)methylidene}-2-oxo-2,3-dihydro-1h-indole-6-carboxylate | Human | 11151 | |
| RET | Ret | TK | 6ne7 | A | A | adenosine monophosphate | Human | 11149 | |
| RET | Ret | TK | 2x2l | A | B | (3z)-5-amino-3-[(4-methoxyphenyl)methylidene]-1,3-dihydro-2h-indol-2-one | Human | 3371 | |
| RET | Ret | TK | 6ne7 | A | B | adenosine monophosphate | Human | 11148 | |
| RET | Ret | TK | 6i83 | A | | 4-[5-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-3-yl]benzamide | Human | 12051 | |
| RET | Ret | TK | 6nja | A | B | adenine | Human | 11145 | |
| RET | Ret | TK | 7ju5 | A | A | pralsetinib | Human | 13106 | |
| RET | Ret | TK | 2ivs | B | B | (3ar,4r,6r,6ar)-4-(6-amino-9h-purin-9-yl)-6-(hydroxymethyl)tetrahydrofuro[3,4-d][1,3,2]dioxaphosphol-2-ol 2-oxide | Human | 3374 | |
| RET | Ret | TK | 7dua | A | A | 4-azanyl-7-(1-methylcyclopropyl)-~{n}-(5-methyl-1~{h}-pyrazol-3-yl)pyrrolo[2,3-d]pyrimidine-5-carboxamide | Human | 14048 | |
| RET | Ret | TK | 4cki | A | B | adenosine | Human | 3370 | |
| RET | Ret | TK | 2x2k | A | A | (3z)-5-amino-3-[(3,5-dimethyl-1h-pyrrol-2-yl)methylidene]-1,3-dihydro-2h-indol-2-one | Human | 3360 | |
| RET | Ret | TK | 7ju6 | A | B | selpercatinib | Human | 13107 | |
| RET | Ret | TK | 6nec | C | B | methyl (3z)-3-{[(4-{methyl[(4-methylpiperazin-1-yl)acetyl]amino}phenyl)amino](phenyl)methylidene}-2-oxo-2,3-dihydro-1h-indole-6-carboxylate | Human | 11153 | |
| RET | Ret | TK | 7du8 | A | A | selpercatinib | Human | 14096 | |
| RET | Ret | TK | 2ivs | B | A | (3ar,4r,6r,6ar)-4-(6-amino-9h-purin-9-yl)-6-(hydroxymethyl)tetrahydrofuro[3,4-d][1,3,2]dioxaphosphol-2-ol 2-oxide | Human | 3357 | |
| RET | Ret | TK | 4cki | A | A | adenosine | Human | 3362 | |
| RET | Ret | TK | 5fm3 | A | | 1-ter-butyl-3-p-tolyl-1h-pyrazolo[3,4-d]pyrimidin-4-ylamine | Human | 7327 | |
| RET | Ret | TK | 7du9 | A | A | pralsetinib | Human | 14050 | |
| RET | Ret | TK | 6vhg | A | A | 3-(3,4-dimethoxyphenyl)-n~5~-(1-methylpiperidin-4-yl)-6-phenylpyrazolo[1,5-a]pyrimidine-5,7-diamine | Human | 11997 | |
| RET | Ret | TK | 2ivs | A | B | (3ar,4r,6r,6ar)-4-(6-amino-9h-purin-9-yl)-6-(hydroxymethyl)tetrahydrofuro[3,4-d][1,3,2]dioxaphosphol-2-ol 2-oxide | Human | 3369 | |
| RET | Ret | TK | 2ivu | A | | 4-bromo-2-fluoro-n-[(4e)-6-methoxy-7-[(1-methylpiperidin-4-yl)methoxy]quinazolin-4(1h)-ylidene]aniline | Human | 3364 | |
| RET | Ret | TK | 2ivt | A | A | adenosine monophosphate | Human | 3361 | |
