Search results (24 entries covering 6 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetails File
PTK6 (BRK)SrcTK5h2uBBn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman7337
PTK6 (BRK)SrcTK5h2uDAn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman7344
PTK6 (BRK)SrcTK6cz3AB(3-fluoro-4-{[6-methyl-3-(1h-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-yl]amino}phenyl)(morpholin-4-yl)methanoneHuman9999
PTK6 (BRK)SrcTK5d7vDB-Human6952
PTK6 (BRK)SrcTK5d7vDA-Human6948
PTK6 (BRK)SrcTK5h2uDBn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman7340
PTK6 (BRK)SrcTK5d7vAA-Human6953
PTK6 (BRK)SrcTK5h2uCBn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman7342
PTK6 (BRK)SrcTK5da3AB(2-chloro-4-{[6-cyclopropyl-3-(1h-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-yl]amino}phenyl)(morpholin-4-yl)methanoneHuman6988
PTK6 (BRK)SrcTK6cz2AB-Human10031
PTK6 (BRK)SrcTK5d7vCA-Human6949
PTK6 (BRK)SrcTK6cz4AB2-{[(3r,4s)-3-fluoro-1-{[4-(trifluoromethoxy)phenyl]acetyl}piperidin-4-yl]oxy}-5-(1-methyl-1h-imidazol-4-yl)pyridine-3-carboxamideHuman10000
PTK6 (BRK)SrcTK5d7vBB-Human6951
PTK6 (BRK)SrcTK6cz3AA(3-fluoro-4-{[6-methyl-3-(1h-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-yl]amino}phenyl)(morpholin-4-yl)methanoneHuman10001
PTK6 (BRK)SrcTK5da3AA(2-chloro-4-{[6-cyclopropyl-3-(1h-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-yl]amino}phenyl)(morpholin-4-yl)methanoneHuman6989
PTK6 (BRK)SrcTK6cz2AA-Human10030
PTK6 (BRK)SrcTK6cz4AA2-{[(3r,4s)-3-fluoro-1-{[4-(trifluoromethoxy)phenyl]acetyl}piperidin-4-yl]oxy}-5-(1-methyl-1h-imidazol-4-yl)pyridine-3-carboxamideHuman9998
PTK6 (BRK)SrcTK5d7vCB-Human6954
PTK6 (BRK)SrcTK5h2uCAn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman7341
PTK6 (BRK)SrcTK5d7vAB-Human6950
PTK6 (BRK)SrcTK5h2uBAn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman7339
PTK6 (BRK)SrcTK5h2uAAn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman7338
PTK6 (BRK)SrcTK5d7vBA-Human6955
PTK6 (BRK)SrcTK5h2uABn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman7343