Search results (31 entries covering 5 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetails File
TNNI3K (HH498)MLKTKL4yffBB3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamideHuman6063
TNNI3K (HH498)MLKTKL6b5jABn-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamideHuman9800
TNNI3K (HH498)MLKTKL6b5jDCn-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamideHuman9795
TNNI3K (HH498)MLKTKL7mgjAn-methyl-4-[4-({[3-(trifluoromethyl)phenyl]carbamoyl}amino)phenoxy]pyridine-2-carboxamideHuman13969
TNNI3K (HH498)MLKTKL4yfiDAn-methyl-3-(9h-purin-6-ylamino)benzenesulfonamideHuman6072
TNNI3K (HH498)MLKTKL6b5jBAn-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamideHuman9802
TNNI3K (HH498)MLKTKL6b5jDAn-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamideHuman9792
TNNI3K (HH498)MLKTKL4yfiCAn-methyl-3-(9h-purin-6-ylamino)benzenesulfonamideHuman6070
TNNI3K (HH498)MLKTKL6b5jACn-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamideHuman9798
TNNI3K (HH498)MLKTKL6b5jBBn-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamideHuman9794
TNNI3K (HH498)MLKTKL4yffCB3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamideHuman6067
TNNI3K (HH498)MLKTKL4yfiDBn-methyl-3-(9h-purin-6-ylamino)benzenesulfonamideHuman6064
TNNI3K (HH498)MLKTKL4yffCA3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamideHuman6069
TNNI3K (HH498)MLKTKL6b5jAAn-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamideHuman9791
TNNI3K (HH498)MLKTKL4yffAA3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamideHuman6068
TNNI3K (HH498)MLKTKL4yffDB3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamideHuman6074
TNNI3K (HH498)MLKTKL6b5jCAn-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamideHuman9799
TNNI3K (HH498)MLKTKL6b5jCBn-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamideHuman9793
TNNI3K (HH498)MLKTKL7mgkABn-(3,5-dichloro-4-{[6-(methylamino)pyrimidin-4-yl]oxy}phenyl)-n'-[3-(trifluoromethyl)phenyl]ureaHuman13970
TNNI3K (HH498)MLKTKL4yfiCBn-methyl-3-(9h-purin-6-ylamino)benzenesulfonamideHuman6073
TNNI3K (HH498)MLKTKL7mgkAAn-(3,5-dichloro-4-{[6-(methylamino)pyrimidin-4-yl]oxy}phenyl)-n'-[3-(trifluoromethyl)phenyl]ureaHuman13968
TNNI3K (HH498)MLKTKL4yfiABn-methyl-3-(9h-purin-6-ylamino)benzenesulfonamideHuman6071
TNNI3K (HH498)MLKTKL4yffDA3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamideHuman6066
TNNI3K (HH498)MLKTKL6b5jBCn-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamideHuman9797
TNNI3K (HH498)MLKTKL4yfiAAn-methyl-3-(9h-purin-6-ylamino)benzenesulfonamideHuman6059
TNNI3K (HH498)MLKTKL4yffBA3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamideHuman6065
TNNI3K (HH498)MLKTKL6b5jDBn-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamideHuman9801
TNNI3K (HH498)MLKTKL4yfiBAn-methyl-3-(9h-purin-6-ylamino)benzenesulfonamideHuman6061
TNNI3K (HH498)MLKTKL6b5jCCn-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamideHuman9796
TNNI3K (HH498)MLKTKL4yffAB3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamideHuman6062
TNNI3K (HH498)MLKTKL4yfiBBn-methyl-3-(9h-purin-6-ylamino)benzenesulfonamideHuman6060