Search results (14 entries covering 7 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetails File
RPS6KA5-b (MSK1-b)RSKbCAMK7up4AA(5m)-5-(2,5-dichloropyrimidin-4-yl)-5h-pyrrolo[3,2-d]pyrimidineHuman14277
RPS6KA5-b (MSK1-b)RSKbCAMK7up7AA(2s)-2-cyano-n-(1-hydroxy-2-methylpropan-2-yl)-3-[3-(3,4,5-trimethoxyphenyl)-1h-indazol-5-yl]propanamideHuman14318
RPS6KA5-b (MSK1-b)RSKbCAMK7up5AA(2m)-6-chloro-2-(5h-pyrrolo[3,2-d]pyrimidin-5-yl)pyridine-3-carbonitrileHuman14280
RPS6KA5-b (MSK1-b)RSKbCAMK3kn5Aphosphoaminophosphonic acid-adenylate esterHuman4603
RPS6KA5-b (MSK1-b)RSKbCAMK7up4AB(5m)-5-(2,5-dichloropyrimidin-4-yl)-5h-pyrrolo[3,2-d]pyrimidineHuman14279
RPS6KA5-b (MSK1-b)RSKbCAMK7up6AA(e)-3-(3-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)phenyl)-2-cyanoacrylamide bound formHuman14353
RPS6KA5-b (MSK1-b)RSKbCAMK7up8AB(5m)-5-(5-bromo-2-chloropyrimidin-4-yl)-5h-pyrrolo[3,2-d]pyrimidineHuman14281
RPS6KA5-b (MSK1-b)RSKbCAMK7up8AA(5m)-5-(5-bromo-2-chloropyrimidin-4-yl)-5h-pyrrolo[3,2-d]pyrimidineHuman14282
RPS6KA5-b (MSK1-b)RSKbCAMK7up6AB(e)-3-(3-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)phenyl)-2-cyanoacrylamide bound formHuman14354
RPS6KA5-b (MSK1-b)RSKbCAMK3kn6A-Human4602
RPS6KA5-b (MSK1-b)RSKbCAMK3kn6B-Human4601
RPS6KA5-b (MSK1-b)RSKbCAMK7up7AB(2s)-2-cyano-n-(1-hydroxy-2-methylpropan-2-yl)-3-[3-(3,4,5-trimethoxyphenyl)-1h-indazol-5-yl]propanamideHuman14317
RPS6KA5-b (MSK1-b)RSKbCAMK7up5AB(2m)-6-chloro-2-(5h-pyrrolo[3,2-d]pyrimidin-5-yl)pyridine-3-carbonitrileHuman14278
RPS6KA5-b (MSK1-b)RSKbCAMK3kn5Bphosphoaminophosphonic acid-adenylate esterHuman4600