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Search results (14 entries covering 7 PDB structures)
#
Kinase
Family
Group
PDB
Chain
(Alternate) Model
Orthosteric ligand
Organism
Details
File
RPS6KA5-b (MSK1-b)
RSKb
CAMK
7up4
A
A
(5m)-5-(2,5-dichloropyrimidin-4-yl)-5h-pyrrolo[3,2-d]pyrimidine
Human
14277
RPS6KA5-b (MSK1-b)
RSKb
CAMK
7up7
A
A
(2s)-2-cyano-n-(1-hydroxy-2-methylpropan-2-yl)-3-[3-(3,4,5-trimethoxyphenyl)-1h-indazol-5-yl]propanamide
Human
14318
RPS6KA5-b (MSK1-b)
RSKb
CAMK
7up5
A
A
(2m)-6-chloro-2-(5h-pyrrolo[3,2-d]pyrimidin-5-yl)pyridine-3-carbonitrile
Human
14280
RPS6KA5-b (MSK1-b)
RSKb
CAMK
3kn5
A
phosphoaminophosphonic acid-adenylate ester
Human
4603
RPS6KA5-b (MSK1-b)
RSKb
CAMK
7up4
A
B
(5m)-5-(2,5-dichloropyrimidin-4-yl)-5h-pyrrolo[3,2-d]pyrimidine
Human
14279
RPS6KA5-b (MSK1-b)
RSKb
CAMK
7up6
A
A
(e)-3-(3-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)phenyl)-2-cyanoacrylamide bound form
Human
14353
RPS6KA5-b (MSK1-b)
RSKb
CAMK
7up8
A
B
(5m)-5-(5-bromo-2-chloropyrimidin-4-yl)-5h-pyrrolo[3,2-d]pyrimidine
Human
14281
RPS6KA5-b (MSK1-b)
RSKb
CAMK
7up8
A
A
(5m)-5-(5-bromo-2-chloropyrimidin-4-yl)-5h-pyrrolo[3,2-d]pyrimidine
Human
14282
RPS6KA5-b (MSK1-b)
RSKb
CAMK
7up6
A
B
(e)-3-(3-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)phenyl)-2-cyanoacrylamide bound form
Human
14354
RPS6KA5-b (MSK1-b)
RSKb
CAMK
3kn6
A
-
Human
4602
RPS6KA5-b (MSK1-b)
RSKb
CAMK
3kn6
B
-
Human
4601
RPS6KA5-b (MSK1-b)
RSKb
CAMK
7up7
A
B
(2s)-2-cyano-n-(1-hydroxy-2-methylpropan-2-yl)-3-[3-(3,4,5-trimethoxyphenyl)-1h-indazol-5-yl]propanamide
Human
14317
RPS6KA5-b (MSK1-b)
RSKb
CAMK
7up5
A
B
(2m)-6-chloro-2-(5h-pyrrolo[3,2-d]pyrimidin-5-yl)pyridine-3-carbonitrile
Human
14278
RPS6KA5-b (MSK1-b)
RSKb
CAMK
3kn5
B
phosphoaminophosphonic acid-adenylate ester
Human
4600
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