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Search results (75 entries covering 34 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetails File
TGFBR1 (TGFbR1)STKRTKL1iasA-Human2113
TGFBR1 (TGFbR1)STKRTKL5qimABn-{4-[3-(5-methoxypyridin-2-yl)-1h-pyrrolo[3,2-b]pyridin-2-yl]pyridin-2-yl}acetamideHuman10661
TGFBR1 (TGFbR1)STKRTKL5usqABn-[2-(5-chloro-2-fluorophenyl)pyridin-4-yl]-2-[(piperidin-4-yl)methyl]-2h-pyrazolo[4,3-b]pyridin-7-amineHuman7557
TGFBR1 (TGFbR1)STKRTKL2wotAB4-[(5,6-dimethyl-2,2'-bipyridin-3-yl)oxy]-n-(3,4,5-trimethoxyphenyl)pyridin-2-amineHuman2092
TGFBR1 (TGFbR1)STKRTKL4x2jAB4-[(3-aminophenyl)amino]pyrido[2,3-d]pyrimidin-5(8h)-oneHuman2115
TGFBR1 (TGFbR1)STKRTKL5qikABn-{4-[3-(6-fluoropyridin-3-yl)-4-oxo-4,5,6,7-tetrahydro-1h-pyrrolo[3,2-c]pyridin-2-yl]pyridin-2-yl}acetamideHuman10662
TGFBR1 (TGFbR1)STKRTKL2x7oC(3z)-n-ethyl-n-methyl-2-oxo-3-(phenyl{[4-(piperidin-1-ylmethyl)phenyl]amino}methylidene)-2,3-dihydro-1h-indole-6-carboxamideHuman2104
TGFBR1 (TGFbR1)STKRTKL4x2jAA4-[(3-aminophenyl)amino]pyrido[2,3-d]pyrimidin-5(8h)-oneHuman2124
TGFBR1 (TGFbR1)STKRTKL2x7oE(3z)-n-ethyl-n-methyl-2-oxo-3-(phenyl{[4-(piperidin-1-ylmethyl)phenyl]amino}methylidene)-2,3-dihydro-1h-indole-6-carboxamideHuman2097
TGFBR1 (TGFbR1)STKRTKL3tzmAA4-[5-(1,3-benzodioxol-5-yl)-4-(pyridin-2-yl)-1h-imidazol-2-yl]benzamideHuman2095
TGFBR1 (TGFbR1)STKRTKL3tzmAB4-[5-(1,3-benzodioxol-5-yl)-4-(pyridin-2-yl)-1h-imidazol-2-yl]benzamideHuman2110
TGFBR1 (TGFbR1)STKRTKL4x2gAB4-[(4-aminophenyl)amino]pyrido[2,3-d]pyrimidin-5(6h)-oneHuman2114
TGFBR1 (TGFbR1)STKRTKL5e8uA-Human6616
TGFBR1 (TGFbR1)STKRTKL5usqAAn-[2-(5-chloro-2-fluorophenyl)pyridin-4-yl]-2-[(piperidin-4-yl)methyl]-2h-pyrazolo[4,3-b]pyridin-7-amineHuman7558
TGFBR1 (TGFbR1)STKRTKL4x2fAB4-amino-8-(4-aminophenyl)pyrido[2,3-d]pyrimidin-5(8h)-oneHuman6208
TGFBR1 (TGFbR1)STKRTKL1vjyA2-[5-(6-methylpyridin-2-yl)-2,3-dihydro-1h-pyrazol-4-yl]-1,5-naphthyridineHuman2096
TGFBR1 (TGFbR1)STKRTKL5qilABn-{4-[3-(6-methoxypyridin-3-yl)-1h-pyrrolo[3,2-b]pyridin-2-yl]pyridin-2-yl}acetamideHuman10660
TGFBR1 (TGFbR1)STKRTKL5e8sAA-Human6619
TGFBR1 (TGFbR1)STKRTKL5e8wAAstaurosporineHuman6611
TGFBR1 (TGFbR1)STKRTKL5e8sAB-Human6609
TGFBR1 (TGFbR1)STKRTKL5e90AB3-amino-6-[4-(2-hydroxyethyl)phenyl]-n-[4-(morpholin-4-yl)pyridin-3-yl]pyrazine-2-carboxamideHuman6607
TGFBR1 (TGFbR1)STKRTKL5qu0AA6-[4-(3-chloro-4-fluorophenyl)-1-(2-hydroxyethyl)-1h-imidazol-5-yl]imidazo[1,2-b]pyridazine-3-carbonitrileHuman11967
TGFBR1 (TGFbR1)STKRTKL3kcfB4-[3-(methoxymethyl)phenyl]-1,2-dimethyl-5-quinoxalin-6-yl-1,2-dihydro-3h-pyrazol-3-oneHuman2106
TGFBR1 (TGFbR1)STKRTKL3faaEn-[4-(5-fluoro-6-methylpyridin-2-yl)-5-quinoxalin-6-yl-1h-imidazol-2-yl]acetamideHuman2098
TGFBR1 (TGFbR1)STKRTKL5qtzAA6-[1-(2,2-difluoroethyl)-4-(6-methylpyridin-2-yl)-1h-imidazol-5-yl]imidazo[1,2-a]pyridineHuman11965
TGFBR1 (TGFbR1)STKRTKL5e8tAA-Human6608
TGFBR1 (TGFbR1)STKRTKL1b6cD-Human2126
TGFBR1 (TGFbR1)STKRTKL5e90AA3-amino-6-[4-(2-hydroxyethyl)phenyl]-n-[4-(morpholin-4-yl)pyridin-3-yl]pyrazine-2-carboxamideHuman6610
TGFBR1 (TGFbR1)STKRTKL1rw8A3-(4-fluorophenyl)-2-(6-methylpyridin-2-yl)-5,6-dihydro-4h-pyrrolo[1,2-b]pyrazoleHuman2100
TGFBR1 (TGFbR1)STKRTKL5friABn-[4-[(6-chloro-[1,3]dioxolo[4,5-b]pyridin-7-yl)amino]-2-pyridyl]cyclopropanecarboxamideHuman6893
TGFBR1 (TGFbR1)STKRTKL3kcfC4-[3-(methoxymethyl)phenyl]-1,2-dimethyl-5-quinoxalin-6-yl-1,2-dihydro-3h-pyrazol-3-oneHuman2093
TGFBR1 (TGFbR1)STKRTKL6b8yAAn-(3-fluoropyridin-4-yl)-2-[6-(trifluoromethyl)pyridin-2-yl]-7h-pyrrolo[2,3-d]pyrimidin-4-amineHuman9553
TGFBR1 (TGFbR1)STKRTKL5e8zAA3-amino-6-[4-(2-hydroxyethyl)phenyl]-n-[4-(morpholin-4-yl)pyridin-3-yl]pyrazine-2-carboxamideHuman6618
TGFBR1 (TGFbR1)STKRTKL5qu0AB6-[4-(3-chloro-4-fluorophenyl)-1-(2-hydroxyethyl)-1h-imidazol-5-yl]imidazo[1,2-b]pyridazine-3-carbonitrileHuman11964
TGFBR1 (TGFbR1)STKRTKL2x7oA(3z)-n-ethyl-n-methyl-2-oxo-3-(phenyl{[4-(piperidin-1-ylmethyl)phenyl]amino}methylidene)-2,3-dihydro-1h-indole-6-carboxamideHuman2127
TGFBR1 (TGFbR1)STKRTKL5qikAAn-{4-[3-(6-fluoropyridin-3-yl)-4-oxo-4,5,6,7-tetrahydro-1h-pyrrolo[3,2-c]pyridin-2-yl]pyridin-2-yl}acetamideHuman10657
TGFBR1 (TGFbR1)STKRTKL4x2kAA4-[(3-aminophenyl)amino]pyrido[2,3-d]pyrimidin-5(6h)-oneHuman2135
TGFBR1 (TGFbR1)STKRTKL3faaCn-[4-(5-fluoro-6-methylpyridin-2-yl)-5-quinoxalin-6-yl-1h-imidazol-2-yl]acetamideHuman2130
TGFBR1 (TGFbR1)STKRTKL5qimAAn-{4-[3-(5-methoxypyridin-2-yl)-1h-pyrrolo[3,2-b]pyridin-2-yl]pyridin-2-yl}acetamideHuman10658
TGFBR1 (TGFbR1)STKRTKL3kcfD4-[3-(methoxymethyl)phenyl]-1,2-dimethyl-5-quinoxalin-6-yl-1,2-dihydro-3h-pyrazol-3-oneHuman2119
TGFBR1 (TGFbR1)STKRTKL3faaDn-[4-(5-fluoro-6-methylpyridin-2-yl)-5-quinoxalin-6-yl-1h-imidazol-2-yl]acetamideHuman2132
TGFBR1 (TGFbR1)STKRTKL4x2gAA4-[(4-aminophenyl)amino]pyrido[2,3-d]pyrimidin-5(6h)-oneHuman2123
TGFBR1 (TGFbR1)STKRTKL1iasD-Human2131
TGFBR1 (TGFbR1)STKRTKL1iasB-Human2102
TGFBR1 (TGFbR1)STKRTKL5e8xABstaurosporineHuman6617
TGFBR1 (TGFbR1)STKRTKL5qilAAn-{4-[3-(6-methoxypyridin-3-yl)-1h-pyrrolo[3,2-b]pyridin-2-yl]pyridin-2-yl}acetamideHuman10659
TGFBR1 (TGFbR1)STKRTKL3gxlAn-1h-indazol-5-yl-2-(6-methylpyridin-2-yl)quinazolin-4-amineHuman2116
TGFBR1 (TGFbR1)STKRTKL4x2fAA4-amino-8-(4-aminophenyl)pyrido[2,3-d]pyrimidin-5(8h)-oneHuman6207
TGFBR1 (TGFbR1)STKRTKL5qtzAB6-[1-(2,2-difluoroethyl)-4-(6-methylpyridin-2-yl)-1h-imidazol-5-yl]imidazo[1,2-a]pyridineHuman11966
TGFBR1 (TGFbR1)STKRTKL5friAAn-[4-[(6-chloro-[1,3]dioxolo[4,5-b]pyridin-7-yl)amino]-2-pyridyl]cyclopropanecarboxamideHuman6894
TGFBR1 (TGFbR1)STKRTKL2x7oD(3z)-n-ethyl-n-methyl-2-oxo-3-(phenyl{[4-(piperidin-1-ylmethyl)phenyl]amino}methylidene)-2,3-dihydro-1h-indole-6-carboxamideHuman2107
TGFBR1 (TGFbR1)STKRTKL4x0mAB4-aminopyrido[2,3-d]pyrimidin-5(8h)-oneHuman2121
TGFBR1 (TGFbR1)STKRTKL4x2nAB-Human2109
TGFBR1 (TGFbR1)STKRTKL5e8zAB3-amino-6-[4-(2-hydroxyethyl)phenyl]-n-[4-(morpholin-4-yl)pyridin-3-yl]pyrazine-2-carboxamideHuman6612
TGFBR1 (TGFbR1)STKRTKL1py5A4-(3-pyridin-2-yl-1h-pyrazol-4-yl)quinolineHuman2094
TGFBR1 (TGFbR1)STKRTKL3hmmA2-(6-methylpyridin-2-yl)-n-pyridin-4-ylquinazolin-4-amineHuman2111
TGFBR1 (TGFbR1)STKRTKL1iasC-Human2117
TGFBR1 (TGFbR1)STKRTKL5e8tAB-Human6613
TGFBR1 (TGFbR1)STKRTKL1b6cB-Human2133
TGFBR1 (TGFbR1)STKRTKL4x0mAA4-aminopyrido[2,3-d]pyrimidin-5(8h)-oneHuman2122
TGFBR1 (TGFbR1)STKRTKL2wotAA4-[(5,6-dimethyl-2,2'-bipyridin-3-yl)oxy]-n-(3,4,5-trimethoxyphenyl)pyridin-2-amineHuman2120
TGFBR1 (TGFbR1)STKRTKL5e8xAAstaurosporineHuman6615
TGFBR1 (TGFbR1)STKRTKL1b6cF-Human2103
TGFBR1 (TGFbR1)STKRTKL3faaBn-[4-(5-fluoro-6-methylpyridin-2-yl)-5-quinoxalin-6-yl-1h-imidazol-2-yl]acetamideHuman2108
TGFBR1 (TGFbR1)STKRTKL2wouA4-({4-[(2,6-dimethylpyridin-3-yl)oxy]pyridin-2-yl}amino)benzenesulfonamideHuman2125
TGFBR1 (TGFbR1)STKRTKL1iasE-Human2134
TGFBR1 (TGFbR1)STKRTKL4x2nAA-Human2129
TGFBR1 (TGFbR1)STKRTKL3faaAn-[4-(5-fluoro-6-methylpyridin-2-yl)-5-quinoxalin-6-yl-1h-imidazol-2-yl]acetamideHuman2118
TGFBR1 (TGFbR1)STKRTKL1b6cH-Human2099
TGFBR1 (TGFbR1)STKRTKL6b8yABn-(3-fluoropyridin-4-yl)-2-[6-(trifluoromethyl)pyridin-2-yl]-7h-pyrrolo[2,3-d]pyrimidin-4-amineHuman9552
TGFBR1 (TGFbR1)STKRTKL3kcfE4-[3-(methoxymethyl)phenyl]-1,2-dimethyl-5-quinoxalin-6-yl-1,2-dihydro-3h-pyrazol-3-oneHuman2105
TGFBR1 (TGFbR1)STKRTKL5e8wABstaurosporineHuman6614
TGFBR1 (TGFbR1)STKRTKL3kcfA4-[3-(methoxymethyl)phenyl]-1,2-dimethyl-5-quinoxalin-6-yl-1,2-dihydro-3h-pyrazol-3-oneHuman2112
TGFBR1 (TGFbR1)STKRTKL2x7oB(3z)-n-ethyl-n-methyl-2-oxo-3-(phenyl{[4-(piperidin-1-ylmethyl)phenyl]amino}methylidene)-2,3-dihydro-1h-indole-6-carboxamideHuman2128
TGFBR1 (TGFbR1)STKRTKL4x2kAB4-[(3-aminophenyl)amino]pyrido[2,3-d]pyrimidin-5(6h)-oneHuman2101
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