Search results (8 entries covering 6 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetails File
RPS6KA3-b (RSK2-b)RSKbCAMK8xeyA-Human15207
RPS6KA3-b (RSK2-b)RSKbCAMK4jg7AA(2r)-2-cyano-3-[3-(1h-pyrrolo[2,3-b]pyridin-3-ylcarbonyl)phenyl]propanamideHuman1496
RPS6KA3-b (RSK2-b)RSKbCAMK4jg8AB(2s)-2-cyano-n-(1-hydroxy-2-methylpropan-2-yl)-3-[3-(3,4,5-trimethoxyphenyl)-1h-indazol-5-yl]propanamideHuman1498
RPS6KA3-b (RSK2-b)RSKbCAMK4jg7AB(2r)-2-cyano-3-[3-(1h-pyrrolo[2,3-b]pyridin-3-ylcarbonyl)phenyl]propanamideHuman1494
RPS6KA3-b (RSK2-b)RSKbCAMK4d9tAmethyl (2s)-3-{4-amino-7-[(1e)-3-hydroxyprop-1-en-1-yl]-5-(4-methylphenyl)-7h-pyrrolo[2,3-d]pyrimidin-6-yl}-2-cyanopropanoateHuman1493
RPS6KA3-b (RSK2-b)RSKbCAMK4d9uAtert-butyl (2s)-3-[4-amino-7-(3-hydroxypropyl)-5-(4-methylphenyl)-7h-pyrrolo[2,3-d]pyrimidin-6-yl]-2-cyanopropanoateHuman1499
RPS6KA3-b (RSK2-b)RSKbCAMK4jg6A(2s)-2-cyano-3-(1h-indazol-5-yl)propanamideHuman1495
RPS6KA3-b (RSK2-b)RSKbCAMK4jg8AA(2s)-2-cyano-n-(1-hydroxy-2-methylpropan-2-yl)-3-[3-(3,4,5-trimethoxyphenyl)-1h-indazol-5-yl]propanamideHuman1497