Search results (9 entries covering 7 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetailsSimilarity (MFP)File
TGFBR1 (TGFbR1)STKRTKL5friABn-[4-[(6-chloro-[1,3]dioxolo[4,5-b]pyridin-7-yl)amino]-2-pyridyl]cyclopropanecarboxamideHuman68930.40
JAK2JakATK4gmyA2,6-dichloro-n-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}benzamideHuman36840.57
TYK2JakATK4gihAA2,6-dichloro-n-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}benzamideHuman33390.57
TYK2-bJakBTK4oliA2-chloro-n-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}benzamideHuman21980.49
TYK2JakATK4gj3A2,6-dichloro-4-cyano-n-[2-({[(1r,2r)-2-fluorocyclopropyl]carbonyl}amino)pyridin-4-yl]benzamideHuman33451.00
TYK2JakATK4gj2A2,6-dichloro-n-[2-({[(1r,2r)-2-fluorocyclopropyl]carbonyl}amino)pyridin-4-yl]benzamideHuman33440.75
TYK2JakATK4gihAB2,6-dichloro-n-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}benzamideHuman33320.57
TYK2JakATK4giiA2,6-dichloro-4-cyano-n-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}benzamideHuman33310.77
TGFBR1 (TGFbR1)STKRTKL5friAAn-[4-[(6-chloro-[1,3]dioxolo[4,5-b]pyridin-7-yl)amino]-2-pyridyl]cyclopropanecarboxamideHuman68940.40