Search results (11 entries covering 8 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetailsSimilarity (MFP)File
TTKTTKOther5nadAbay 1217389Human79750.43
TTKTTKOther6tndABbay 1217389Human122720.43
TTKTTKOther6tncAn-cyclopropyl-4-{8-[(thiophen-2-ylmethyl)amino]imidazo[1,2-a]pyrazin-3-yl}benzamideHuman122700.44
ERN1 (IRE1)IREOther6hx1AB6-chloranyl-~{n}-(cyclopropylmethyl)-3-(2~{h}-indazol-5-yl)imidazo[1,2-b]pyridazin-8-amineHuman109290.44
ACVR1 (ALK2)STKRTKL3oomAA1-{3-[6-(tetrahydro-2h-pyran-4-ylamino)imidazo[1,2-b]pyridazin-3-yl]phenyl}ethanoneHuman15170.42
ACVR1 (ALK2)STKRTKL3oomAB1-{3-[6-(tetrahydro-2h-pyran-4-ylamino)imidazo[1,2-b]pyridazin-3-yl]phenyl}ethanoneHuman15180.42
TTKTTKOther3wzkAn-cyclopropyl-4-{8-[(thiophen-2-ylmethyl)amino]imidazo[1,2-a]pyrazin-3-yl}benzamideHuman47030.44
TTKTTKOther3wzjA4-{6-(cyclohexylamino)-8-[(tetrahydro-2h-pyran-4-ylmethyl)amino]imidazo[1,2-b]pyridazin-3-yl}-n-cyclopropylbenzamideHuman47041.00
ERN1 (IRE1)IREOther6hx1AA6-chloranyl-~{n}-(cyclopropylmethyl)-3-(2~{h}-indazol-5-yl)imidazo[1,2-b]pyridazin-8-amineHuman109270.44
TTKTTKOther5n84A~{n}-cyclopropyl-4-[8-(2-methylpropylamino)imidazo[1,2-a]pyrazin-3-yl]benzamideHuman79730.43
TTKTTKOther6tndAAbay 1217389Human122680.43