| JAK2 | JakA | TK | 6drw | A | A | 4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamide | Human | 10512 | 1.00 | |
| JAK2 | JakA | TK | 5usy | B | B | 4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamide | Human | 8104 | 1.00 | |
| CLK3 | CLK | CMGC | 2wu6 | A | B | 5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamide | Human | 1821 | 0.71 | |
| CLK3 | CLK | CMGC | 2wu6 | A | A | 5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamide | Human | 1823 | 0.71 | |
| JAK2 | JakA | TK | 5usy | A | A | 4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamide | Human | 8101 | 1.00 | |
| JAK2 | JakA | TK | 5usy | A | B | 4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamide | Human | 8102 | 1.00 | |
| CDK2 | CDK | CMGC | 3r9h | A | B | 4-amino-n-(2,6-difluorophenyl)-2-[(4-sulfamoylphenyl)amino]-1,3-thiazole-5-carboxamide | Human | 4336 | 0.47 | |
| CSNK1G3 (CK1g3) | CK1 | CK1 | 2chl | A | B | 5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamide | Human | 2217 | 0.71 | |
| CDK2 | CDK | CMGC | 3qtz | A | A | 4-{[4-amino-5-(3-fluorobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamide | Human | 4109 | 0.44 | |
| CDK2 | CDK | CMGC | 3r9d | A | A | 4-amino-n-(3-fluorophenyl)-2-[(4-sulfamoylphenyl)amino]-1,3-thiazole-5-carboxamide | Human | 4562 | 0.41 | |
| CDK2 | CDK | CMGC | 3qtz | A | B | 4-{[4-amino-5-(3-fluorobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamide | Human | 4337 | 0.44 | |
| CDK2 | CDK | CMGC | 3rpy | A | A | 4-amino-2-[(4-sulfamoylphenyl)amino]-1,3-thiazole-5-carboxamide | Human | 4261 | 0.40 | |
| CDK2 | CDK | CMGC | 3rpy | A | B | 4-amino-2-[(4-sulfamoylphenyl)amino]-1,3-thiazole-5-carboxamide | Human | 4519 | 0.40 | |
| AURKA (AurA) | Aur | Other | 5dpv | A | B | 4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamide | Human | 6826 | 1.00 | |
| CDK2 | CDK | CMGC | 5iey | A | A | 4-[(4-{[(2r,3r)-3-hydroxybutan-2-yl]amino}pyrimidin-2-yl)amino]benzene-1-sulfonamide | Human | 6566 | 0.40 | |
| SLK | STE20 | STE | 2jfl | A | | 5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamide | Human | 1838 | 0.71 | |
| CDK2 | CDK | CMGC | 7mkx | A | | 2-[(5-bromo-2-{4-[(cyanomethyl)sulfamoyl]anilino}pyrimidin-4-yl)amino]-6-fluorobenzamide | Human | 14490 | 0.46 | |
| AURKA (AurA) | Aur | Other | 5dt0 | A | B | 4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamide | Human | 6803 | 1.00 | |
| PRKACA (PKACa) | PKA | AGC | 3ama | A | | 4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamide | Human | 5284 | 1.00 | |
| CDK2 | CDK | CMGC | 5iey | A | B | 4-[(4-{[(2r,3r)-3-hydroxybutan-2-yl]amino}pyrimidin-2-yl)amino]benzene-1-sulfonamide | Human | 6573 | 0.40 | |
| JAK2-b | JakB | TK | 6occ | A | | 2-[4-({5-amino-3-[(4-sulfamoylphenyl)amino]-1h-1,2,4-triazole-1-carbonyl}amino)phenyl]-1,3-oxazole-4-carboxylic acid | Human | 12100 | 0.51 | |
| JAK2-b | JakB | TK | 6obb | A | | 5-amino-n-phenyl-3-[(4-sulfamoylphenyl)amino]-1h-1,2,4-triazole-1-carboxamide | Human | 12097 | 0.64 | |
| STK24 (MST3) | STE20 | STE | 4qmu | A | A | 4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamide | Human | 5606 | 1.00 | |
| AURKA (AurA) | Aur | Other | 5dr6 | A | B | 4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamide | Human | 6805 | 1.00 | |
| SLK | STE20 | STE | 2j51 | A | | 5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamide | Human | 1833 | 0.71 | |
| AURKA (AurA) | Aur | Other | 5dr6 | A | A | 4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamide | Human | 6811 | 1.00 | |
| STK24 (MST3) | STE20 | STE | 4qmu | A | B | 4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamide | Human | 5603 | 1.00 | |
| AURKA (AurA) | Aur | Other | 5dr9 | A | | 4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamide | Human | 6821 | 1.00 | |
| JAK2-b | JakB | TK | 5win | A | | 4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamide | Human | 10378 | 1.00 | |
| JAK2-b | JakB | TK | 5usz | A | B | 4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamide | Human | 8043 | 1.00 | |
| JAK2 | JakA | TK | 5usy | B | A | 4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamide | Human | 8103 | 1.00 | |
| CAMK4 (CaMK4) | CAMK1 | CAMK | 2w4o | A | | 5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamide | Human | 2687 | 0.71 | |
| CDK2 | CDK | CMGC | 3r9d | A | B | 4-amino-n-(3-fluorophenyl)-2-[(4-sulfamoylphenyl)amino]-1,3-thiazole-5-carboxamide | Human | 4565 | 0.41 | |
| STK24 (MST3) | STE20 | STE | 4qmp | A | | 5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamide | Human | 5584 | 0.71 | |
| CDK2 | CDK | CMGC | 1ykr | A | | 4-{[6-(2,6-dichlorobenzoyl)imidazo[1,2-a]pyridin-2-yl]amino}benzenesulfonamide | Human | 4578 | 0.42 | |
| JAK2 | JakA | TK | 6drw | A | B | 4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamide | Human | 10513 | 1.00 | |
| CDK2 | CDK | CMGC | 3r9h | A | A | 4-amino-n-(2,6-difluorophenyl)-2-[(4-sulfamoylphenyl)amino]-1,3-thiazole-5-carboxamide | Human | 3958 | 0.47 | |
| PIK3CG (p110g) | PIK | Atypical | 4ful | A | | 4-({4-[3-(piperidin-1-ylcarbonyl)phenyl]pyrimidin-2-yl}amino)benzenesulfonamide | Human | 9242 | 0.43 | |
| AURKA (AurA) | Aur | Other | 5obr | A | | 4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamide | Human | 8304 | 1.00 | |
| JAK2-b | JakB | TK | 5usz | A | A | 4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamide | Human | 8048 | 1.00 | |
| AURKA (AurA) | Aur | Other | 5dpv | A | A | 4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamide | Human | 6808 | 1.00 | |
| JAK2-b | JakB | TK | 6obf | A | | [4-({5-amino-3-[(4-sulfamoylphenyl)amino]-1h-1,2,4-triazole-1-carbonyl}amino)phenoxy]acetic acid | Human | 12098 | 0.52 | |
| JAK2-b | JakB | TK | 6oav | A | | 5-amino-3-[(4-cyanophenyl)amino]-n-phenyl-1h-1,2,4-triazole-1-carboxamide | Human | 12099 | 0.45 | |
| AURKA (AurA) | Aur | Other | 5dt0 | A | A | 4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamide | Human | 6806 | 1.00 | |
| CDK2 | CDK | CMGC | 1oit | A | | 4-[(4-imidazo[1,2-a]pyridin-3-ylpyrimidin-2-yl)amino]benzenesulfonamide | Human | 4025 | 0.40 | |
| CDKL2 | CDKL | CMGC | 4aaa | A | A | 5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamide | Human | 964 | 0.71 | |
| CDKL2 | CDKL | CMGC | 4aaa | A | B | 5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamide | Human | 962 | 0.71 | |
| ABL2 | Abl | TK | 3hmi | A | B | 5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamide | Human | 118 | 0.71 | |
| ABL2 | Abl | TK | 3hmi | A | A | 5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamide | Human | 115 | 0.71 | |
| STK26 (MST4) | STE20 | STE | 4fzf | B | | 5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamide | Human | 1803 | 0.71 | |
| CSNK1G3 (CK1g3) | CK1 | CK1 | 2chl | A | A | 5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamide | Human | 2220 | 0.71 | |
