| STK24 (MST3) | STE20 | STE | 4qmv | A | | n-{2-[(1s,4r)-6-{[4-(cyclobutylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino}-1,2,3,4-tetrahydro-1,4-epiminonaphthalen-9-yl]-2-oxoethyl}acetamide | Human | 5581 | 1.00 | |
| ULK1 | ULK | Other | 6qas | B | A | n-{2-[(1s,4r)-6-{[4-(cyclobutylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino}-1,2,3,4-tetrahydro-1,4-epiminonaphthalen-9-yl]-2-oxoethyl}acetamide | Human | 10932 | 1.00 | |
| ULK1 | ULK | Other | 6qas | A | B | n-{2-[(1s,4r)-6-{[4-(cyclobutylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino}-1,2,3,4-tetrahydro-1,4-epiminonaphthalen-9-yl]-2-oxoethyl}acetamide | Human | 10931 | 1.00 | |
| ULK1 | ULK | Other | 6qas | A | A | n-{2-[(1s,4r)-6-{[4-(cyclobutylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino}-1,2,3,4-tetrahydro-1,4-epiminonaphthalen-9-yl]-2-oxoethyl}acetamide | Human | 10930 | 1.00 | |
| ULK2 | ULK | Other | 6qav | A | A | ~{n}-[3-[[5-cyclopropyl-2-[(2-methyl-3,4-dihydro-1~{h}-isoquinolin-6-yl)amino]pyrimidin-4-yl]amino]propyl]cyclobutanecarboxamide | Human | 11231 | 0.40 | |
| ULK2 | ULK | Other | 6qav | B | A | ~{n}-[3-[[5-cyclopropyl-2-[(2-methyl-3,4-dihydro-1~{h}-isoquinolin-6-yl)amino]pyrimidin-4-yl]amino]propyl]cyclobutanecarboxamide | Human | 11224 | 0.40 | |
| ULK1 | ULK | Other | 6qas | B | B | n-{2-[(1s,4r)-6-{[4-(cyclobutylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino}-1,2,3,4-tetrahydro-1,4-epiminonaphthalen-9-yl]-2-oxoethyl}acetamide | Human | 10933 | 1.00 | |
| WEE1 (Wee1) | WEE | Other | 5vd2 | A | | n-{2-[(1s,4r)-6-{[4-(cyclobutylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino}-1,2,3,4-tetrahydro-1,4-epiminonaphthalen-9-yl]-2-oxoethyl}acetamide | Human | 8330 | 1.00 | |
| PTK2B (PYK2) | FAK | TK | 3h3c | A | | 4-{[4-{[(1r,2r)-2-(dimethylamino)cyclopentyl]amino}-5-(trifluoromethyl)pyrimidin-2-yl]amino}-n-methylbenzenesulfonamide | Human | 96 | 0.43 | |
| ULK2 | ULK | Other | 6qav | D | B | ~{n}-[3-[[5-cyclopropyl-2-[(2-methyl-3,4-dihydro-1~{h}-isoquinolin-6-yl)amino]pyrimidin-4-yl]amino]propyl]cyclobutanecarboxamide | Human | 11238 | 0.40 | |
| ULK2 | ULK | Other | 6qav | C | B | ~{n}-[3-[[5-cyclopropyl-2-[(2-methyl-3,4-dihydro-1~{h}-isoquinolin-6-yl)amino]pyrimidin-4-yl]amino]propyl]cyclobutanecarboxamide | Human | 11228 | 0.40 | |
| ULK2 | ULK | Other | 6qav | B | B | ~{n}-[3-[[5-cyclopropyl-2-[(2-methyl-3,4-dihydro-1~{h}-isoquinolin-6-yl)amino]pyrimidin-4-yl]amino]propyl]cyclobutanecarboxamide | Human | 11237 | 0.40 | |
| PTK2 (FAK) | FAK | TK | 6yvy | C | A | 4-{[4-{[(1r,2r)-2-(dimethylamino)cyclopentyl]amino}-5-(trifluoromethyl)pyrimidin-2-yl]amino}-n-methylbenzenesulfonamide | Human | 13269 | 0.43 | |
| PTK2 (FAK) | FAK | TK | 6yvy | C | B | 4-{[4-{[(1r,2r)-2-(dimethylamino)cyclopentyl]amino}-5-(trifluoromethyl)pyrimidin-2-yl]amino}-n-methylbenzenesulfonamide | Human | 13268 | 0.43 | |
| PTK2 (FAK) | FAK | TK | 6yvy | A | B | 4-{[4-{[(1r,2r)-2-(dimethylamino)cyclopentyl]amino}-5-(trifluoromethyl)pyrimidin-2-yl]amino}-n-methylbenzenesulfonamide | Human | 13270 | 0.43 | |
| PTK2 (FAK) | FAK | TK | 6yvy | D | A | 4-{[4-{[(1r,2r)-2-(dimethylamino)cyclopentyl]amino}-5-(trifluoromethyl)pyrimidin-2-yl]amino}-n-methylbenzenesulfonamide | Human | 13273 | 0.43 | |
| PTK2 (FAK) | FAK | TK | 6yvy | A | A | 4-{[4-{[(1r,2r)-2-(dimethylamino)cyclopentyl]amino}-5-(trifluoromethyl)pyrimidin-2-yl]amino}-n-methylbenzenesulfonamide | Human | 13275 | 0.43 | |
| PTK2 (FAK) | FAK | TK | 6yvy | D | B | 4-{[4-{[(1r,2r)-2-(dimethylamino)cyclopentyl]amino}-5-(trifluoromethyl)pyrimidin-2-yl]amino}-n-methylbenzenesulfonamide | Human | 13274 | 0.43 | |
| PTK2 (FAK) | FAK | TK | 6yvy | B | A | 4-{[4-{[(1r,2r)-2-(dimethylamino)cyclopentyl]amino}-5-(trifluoromethyl)pyrimidin-2-yl]amino}-n-methylbenzenesulfonamide | Human | 13276 | 0.43 | |
| PTK2 (FAK) | FAK | TK | 6yvy | B | B | 4-{[4-{[(1r,2r)-2-(dimethylamino)cyclopentyl]amino}-5-(trifluoromethyl)pyrimidin-2-yl]amino}-n-methylbenzenesulfonamide | Human | 13267 | 0.43 | |
| ULK2 | ULK | Other | 6qav | A | B | ~{n}-[3-[[5-cyclopropyl-2-[(2-methyl-3,4-dihydro-1~{h}-isoquinolin-6-yl)amino]pyrimidin-4-yl]amino]propyl]cyclobutanecarboxamide | Human | 11239 | 0.40 | |
| ULK2 | ULK | Other | 6qav | D | A | ~{n}-[3-[[5-cyclopropyl-2-[(2-methyl-3,4-dihydro-1~{h}-isoquinolin-6-yl)amino]pyrimidin-4-yl]amino]propyl]cyclobutanecarboxamide | Human | 11234 | 0.40 | |
| ULK2 | ULK | Other | 6qav | C | A | ~{n}-[3-[[5-cyclopropyl-2-[(2-methyl-3,4-dihydro-1~{h}-isoquinolin-6-yl)amino]pyrimidin-4-yl]amino]propyl]cyclobutanecarboxamide | Human | 11223 | 0.40 | |