| CDK2 | CDK | CMGC | 1fvv | A | | 4-[(7-oxo-7h-thiazolo[5,4-e]indol-8-ylmethyl)-amino]-n-pyridin-2-yl-benzenesulfonamide | Human | 4065 | 0.45 | |
| CDK2 | CDK | CMGC | 4fks | A | A | n-[(4-{[(z)-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}phenyl)sulfonyl]acetamide | Human | 4412 | 0.48 | |
| CDK2 | CDK | CMGC | 6guc | C | | (3z)-3-(1h-imidazol-5-ylmethylene)-5-methoxy-1h-indol-2(3h)-one | Human | 10766 | 0.45 | |
| PAK1 | STE20 | STE | 7vto | A | B | 4-[(7-oxo-7h-thiazolo[5,4-e]indol-8-ylmethyl)-amino]-n-pyridin-2-yl-benzenesulfonamide | Human | 14484 | 0.45 | |
| PAK1 | STE20 | STE | 7vto | A | A | 4-[(7-oxo-7h-thiazolo[5,4-e]indol-8-ylmethyl)-amino]-n-pyridin-2-yl-benzenesulfonamide | Human | 14483 | 0.45 | |
| CDK2 | CDK | CMGC | 1pf8 | A | | (3z)-3-(1h-imidazol-5-ylmethylene)-5-methoxy-1h-indol-2(3h)-one | Human | 3861 | 0.45 | |
| CDK2 | CDK | CMGC | 1fvv | C | | 4-[(7-oxo-7h-thiazolo[5,4-e]indol-8-ylmethyl)-amino]-n-pyridin-2-yl-benzenesulfonamide | Human | 4461 | 0.45 | |
| CDK2 | CDK | CMGC | 3py0 | A | B | (3z)-3-(1h-imidazol-5-ylmethylene)-5-methoxy-1h-indol-2(3h)-one | Human | 3869 | 0.45 | |
| CDK2 | CDK | CMGC | 4fkr | A | A | (8z)-8-{[(2,2-dioxido-1,3-dihydro-2-benzothiophen-5-yl)amino]methylidene}-6,8-dihydro-7h-[1,3]thiazolo[5,4-e]indol-7-one | Human | 4149 | 0.50 | |
| CDK2 | CDK | CMGC | 3py1 | A | B | (3z)-3-(1h-imidazol-5-ylmethylene)-5-methoxy-1h-indol-2(3h)-one | Human | 4444 | 0.45 | |
| CDK2 | CDK | CMGC | 1ke6 | A | | n-methyl-{4-[2-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)hydrazino]phenyl}methanesulfonamide | Human | 4219 | 0.40 | |
| CDK2 | CDK | CMGC | 3py1 | A | A | (3z)-3-(1h-imidazol-5-ylmethylene)-5-methoxy-1h-indol-2(3h)-one | Human | 4361 | 0.45 | |
| VRK1 | VRK | CK1 | 5ukf | C | | 4-{[(z)-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}benzene-1-sulfonamide | Human | 8027 | 0.52 | |
| VRK1 | VRK | CK1 | 5ukf | D | | 4-{[(z)-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}benzene-1-sulfonamide | Human | 8028 | 0.52 | |
| CDK2 | CDK | CMGC | 4fkr | A | B | (8z)-8-{[(2,2-dioxido-1,3-dihydro-2-benzothiophen-5-yl)amino]methylidene}-6,8-dihydro-7h-[1,3]thiazolo[5,4-e]indol-7-one | Human | 4535 | 0.50 | |
| STK24 (MST3) | STE20 | STE | 4qmo | A | A | (8z)-8-(1h-imidazol-5-ylmethylidene)-6,8-dihydro-7h-[1,3]thiazolo[5,4-e]indol-7-one | Human | 5585 | 1.00 | |
| STK24 (MST3) | STE20 | STE | 4qmo | A | B | (8z)-8-(1h-imidazol-5-ylmethylidene)-6,8-dihydro-7h-[1,3]thiazolo[5,4-e]indol-7-one | Human | 5597 | 1.00 | |
| VRK1 | VRK | CK1 | 5ukf | B | | 4-{[(z)-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}benzene-1-sulfonamide | Human | 8029 | 0.52 | |
| CDK2 | CDK | CMGC | 4fks | A | C | n-[(4-{[(z)-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}phenyl)sulfonyl]acetamide | Human | 4315 | 0.48 | |
| CDK2 | CDK | CMGC | 6guc | A | | (3z)-3-(1h-imidazol-5-ylmethylene)-5-methoxy-1h-indol-2(3h)-one | Human | 10767 | 0.45 | |
| CDK2 | CDK | CMGC | 4fks | A | B | n-[(4-{[(z)-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}phenyl)sulfonyl]acetamide | Human | 4489 | 0.48 | |
| MAP2K7 | STE7 | STE | 6yg4 | A | | (3z)-3-(1h-imidazol-5-ylmethylene)-5-methoxy-1h-indol-2(3h)-one | Human | 12693 | 0.45 | |
| CDK2 | CDK | CMGC | 3py0 | A | A | (3z)-3-(1h-imidazol-5-ylmethylene)-5-methoxy-1h-indol-2(3h)-one | Human | 3995 | 0.45 | |
| VRK1 | VRK | CK1 | 5ukf | A | | 4-{[(z)-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}benzene-1-sulfonamide | Human | 8030 | 0.52 | |
