| SYK | Syk | TK | 4yjr | A | A | 3-(1h-indazol-4-yl{2-[(1-methyl-1h-indazol-5-yl)amino]pyrimidin-4-yl}amino)propan-1-ol | Human | 6113 | 1.00 | |
| SYK | Syk | TK | 4xg7 | A | B | 1-[(3-methyl-1-{2-[(1-methyl-1h-indazol-5-yl)amino]pyrimidin-4-yl}-1h-pyrazol-4-yl)methyl]azetidin-3-ol | Human | 6318 | 0.41 | |
| SYK | Syk | TK | 4yjr | A | C | 3-(1h-indazol-4-yl{2-[(1-methyl-1h-indazol-5-yl)amino]pyrimidin-4-yl}amino)propan-1-ol | Human | 6122 | 1.00 | |
| SYK | Syk | TK | 4yjq | A | B | 3-[1h-indazol-4-yl(2-{[3-(4-methyl-1,3-oxazol-5-yl)phenyl]amino}pyrimidin-4-yl)amino]propan-1-ol | Human | 6123 | 0.68 | |
| SYK | Syk | TK | 4yjo | A | B | 5-chloro-n~2~-(1,1-dioxido-2,3-dihydro-1,2-benzothiazol-6-yl)-n~4~-ethyl-n~4~-(1h-indazol-4-yl)pyrimidine-2,4-diamine | Human | 6119 | 0.40 | |
| SYK | Syk | TK | 4yjp | A | | 2-[{2-[(1,1-dioxido-2,3-dihydro-1,2-benzothiazol-6-yl)amino]pyrimidin-4-yl}(1h-indazol-4-yl)amino]ethanol | Human | 6115 | 0.59 | |
| SYK | Syk | TK | 4yjt | A | A | n~2~-(1,1-dioxido-2,3-dihydro-1,2-benzothiazol-6-yl)-n~4~-ethyl-5-fluoro-n~4~-(1h-indazol-4-yl)pyrimidine-2,4-diamine | Human | 6125 | 0.40 | |
| SYK | Syk | TK | 4yjq | A | A | 3-[1h-indazol-4-yl(2-{[3-(4-methyl-1,3-oxazol-5-yl)phenyl]amino}pyrimidin-4-yl)amino]propan-1-ol | Human | 6114 | 0.68 | |
| SYK | Syk | TK | 4yjo | A | A | 5-chloro-n~2~-(1,1-dioxido-2,3-dihydro-1,2-benzothiazol-6-yl)-n~4~-ethyl-n~4~-(1h-indazol-4-yl)pyrimidine-2,4-diamine | Human | 6120 | 0.40 | |
| SYK | Syk | TK | 4yjv | A | B | 3-[6-({4-[ethyl(1h-indazol-4-yl)amino]-5-fluoropyrimidin-2-yl}amino)-2,4-dihydro-1h-indazol-1-yl]propan-1-ol | Human | 6148 | 0.41 | |
| SYK | Syk | TK | 4yjs | A | | 3-[{2-[(1,1-dioxido-2,3-dihydro-1,2-benzothiazol-6-yl)amino]pyrimidin-4-yl}(1h-indazol-4-yl)amino]propan-1-ol | Human | 6117 | 0.65 | |
| SYK | Syk | TK | 4yjt | A | B | n~2~-(1,1-dioxido-2,3-dihydro-1,2-benzothiazol-6-yl)-n~4~-ethyl-5-fluoro-n~4~-(1h-indazol-4-yl)pyrimidine-2,4-diamine | Human | 6118 | 0.40 | |
| SYK | Syk | TK | 4xg7 | A | A | 1-[(3-methyl-1-{2-[(1-methyl-1h-indazol-5-yl)amino]pyrimidin-4-yl}-1h-pyrazol-4-yl)methyl]azetidin-3-ol | Human | 6316 | 0.41 | |
| SYK | Syk | TK | 4yjt | A | C | n~2~-(1,1-dioxido-2,3-dihydro-1,2-benzothiazol-6-yl)-n~4~-ethyl-5-fluoro-n~4~-(1h-indazol-4-yl)pyrimidine-2,4-diamine | Human | 6124 | 0.40 | |
| SYK | Syk | TK | 4yjv | A | C | 3-[6-({4-[ethyl(1h-indazol-4-yl)amino]-5-fluoropyrimidin-2-yl}amino)-2,4-dihydro-1h-indazol-1-yl]propan-1-ol | Human | 6149 | 0.41 | |
| SYK | Syk | TK | 4yjr | A | B | 3-(1h-indazol-4-yl{2-[(1-methyl-1h-indazol-5-yl)amino]pyrimidin-4-yl}amino)propan-1-ol | Human | 6116 | 1.00 | |
| SYK | Syk | TK | 4yjv | A | A | 3-[6-({4-[ethyl(1h-indazol-4-yl)amino]-5-fluoropyrimidin-2-yl}amino)-2,4-dihydro-1h-indazol-1-yl]propan-1-ol | Human | 6150 | 0.41 | |