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Search results (7 entries covering 4 PDB structures)
#
Kinase
Family
Group
PDB
Chain
(Alternate) Model
Orthosteric ligand
Organism
Details
Similarity (MFP)
File
GRK2 (BARK1)
GRK
AGC
5wg4
A
B
2-fluoro-5-[(3s,4r)-3-{[(1h-indazol-5-yl)oxy]methyl}piperidin-4-yl]-n-[(pyridin-2-yl)methyl]benzamide
Human
9438
0.48
GRK2 (BARK1)
GRK
AGC
5he1
A
B
(4~{s})-4-[4-fluoranyl-3-(isoquinolin-1-ylmethylcarbamoyl)phenyl]-~{n}-(1~{h}-indazol-5-yl)-6-methyl-2-oxidanylidene-3,4-dihydro-1~{h}-pyrimidine-5-carboxamide
Human
6606
1.00
GRK2 (BARK1)
GRK
AGC
5wg3
A
2-fluoro-5-[(3s,4r)-3-{[(1h-indazol-5-yl)oxy]methyl}piperidin-4-yl]-n-[(1h-pyrazol-3-yl)methyl]benzamide
Human
9439
0.43
GRK2 (BARK1)
GRK
AGC
4pnk
A
B
(4s)-4-(4-fluorophenyl)-n-(2h-indazol-5-yl)-6-methyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
Human
1708
0.46
GRK2 (BARK1)
GRK
AGC
4pnk
A
A
(4s)-4-(4-fluorophenyl)-n-(2h-indazol-5-yl)-6-methyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
Human
1703
0.46
GRK2 (BARK1)
GRK
AGC
5wg4
A
A
2-fluoro-5-[(3s,4r)-3-{[(1h-indazol-5-yl)oxy]methyl}piperidin-4-yl]-n-[(pyridin-2-yl)methyl]benzamide
Human
9441
0.48
GRK2 (BARK1)
GRK
AGC
5he1
A
A
(4~{s})-4-[4-fluoranyl-3-(isoquinolin-1-ylmethylcarbamoyl)phenyl]-~{n}-(1~{h}-indazol-5-yl)-6-methyl-2-oxidanylidene-3,4-dihydro-1~{h}-pyrimidine-5-carboxamide
Human
6605
1.00
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