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Search results (8 entries covering 2 PDB structures)
#
Kinase
Family
Group
PDB
Chain
(Alternate) Model
Orthosteric ligand
Organism
Details
Similarity (MFP)
File
TYK2-b
JakB
TK
6nsl
B
B
6-{[1-(4-cyanophenyl)-2-oxo-1,2-dihydropyridin-3-yl]amino}-n-cyclopropyl-8-(methylamino)imidazo[1,2-b]pyridazine-3-carboxamide
Human
11953
0.45
TYK2-b
JakB
TK
6nsl
B
A
6-{[1-(4-cyanophenyl)-2-oxo-1,2-dihydropyridin-3-yl]amino}-n-cyclopropyl-8-(methylamino)imidazo[1,2-b]pyridazine-3-carboxamide
Human
11955
0.45
TYK2-b
JakB
TK
5tkd
A
B
6-[(3,5-dimethylphenyl)amino]-8-(methylamino)imidazo[1,2-b]pyridazine-3-carboxamide
Human
7326
1.00
TYK2-b
JakB
TK
6nsl
A
A
6-{[1-(4-cyanophenyl)-2-oxo-1,2-dihydropyridin-3-yl]amino}-n-cyclopropyl-8-(methylamino)imidazo[1,2-b]pyridazine-3-carboxamide
Human
11952
0.45
TYK2-b
JakB
TK
5tkd
B
B
6-[(3,5-dimethylphenyl)amino]-8-(methylamino)imidazo[1,2-b]pyridazine-3-carboxamide
Human
7324
1.00
TYK2-b
JakB
TK
6nsl
A
B
6-{[1-(4-cyanophenyl)-2-oxo-1,2-dihydropyridin-3-yl]amino}-n-cyclopropyl-8-(methylamino)imidazo[1,2-b]pyridazine-3-carboxamide
Human
11954
0.45
TYK2-b
JakB
TK
5tkd
A
A
6-[(3,5-dimethylphenyl)amino]-8-(methylamino)imidazo[1,2-b]pyridazine-3-carboxamide
Human
7323
1.00
TYK2-b
JakB
TK
5tkd
B
A
6-[(3,5-dimethylphenyl)amino]-8-(methylamino)imidazo[1,2-b]pyridazine-3-carboxamide
Human
7325
1.00
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