| CDK2 | CDK | CMGC | 1fvv | A | | 4-[(7-oxo-7h-thiazolo[5,4-e]indol-8-ylmethyl)-amino]-n-pyridin-2-yl-benzenesulfonamide | Human | 4065 | 0.70 | |
| CDK2 | CDK | CMGC | 4fks | A | A | n-[(4-{[(z)-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}phenyl)sulfonyl]acetamide | Human | 4412 | 0.74 | |
| CDK2 | CDK | CMGC | 1ke9 | A | | 3-{[4-([amino(imino)methyl]aminosulfonyl)anilino]methylene}-2-oxo-2,3-dihydro-1h-indole | Human | 4250 | 0.41 | |
| PAK1 | STE20 | STE | 7vto | A | B | 4-[(7-oxo-7h-thiazolo[5,4-e]indol-8-ylmethyl)-amino]-n-pyridin-2-yl-benzenesulfonamide | Human | 14484 | 0.70 | |
| PAK1 | STE20 | STE | 7vto | A | A | 4-[(7-oxo-7h-thiazolo[5,4-e]indol-8-ylmethyl)-amino]-n-pyridin-2-yl-benzenesulfonamide | Human | 14483 | 0.70 | |
| CDK2 | CDK | CMGC | 4fkq | A | A | 4-[(2z)-2-(7-oxidanylidene-3,6-dihydropyrrolo[3,2-e]benzotriazol-8-ylidene)hydrazinyl]benzenesulfonamide | Human | 3972 | 0.41 | |
| CDK2 | CDK | CMGC | 4fkp | A | C | 3-{[4-([amino(imino)methyl]aminosulfonyl)anilino]methylene}-2-oxo-2,3-dihydro-1h-indole | Human | 4468 | 0.41 | |
| CDK2 | CDK | CMGC | 1fvv | C | | 4-[(7-oxo-7h-thiazolo[5,4-e]indol-8-ylmethyl)-amino]-n-pyridin-2-yl-benzenesulfonamide | Human | 4461 | 0.70 | |
| CDK2 | CDK | CMGC | 4fkr | A | A | (8z)-8-{[(2,2-dioxido-1,3-dihydro-2-benzothiophen-5-yl)amino]methylidene}-6,8-dihydro-7h-[1,3]thiazolo[5,4-e]indol-7-one | Human | 4149 | 0.66 | |
| CDK2 | CDK | CMGC | 1ke6 | A | | n-methyl-{4-[2-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)hydrazino]phenyl}methanesulfonamide | Human | 4219 | 0.45 | |
| CDK2 | CDK | CMGC | 4fkp | A | A | 3-{[4-([amino(imino)methyl]aminosulfonyl)anilino]methylene}-2-oxo-2,3-dihydro-1h-indole | Human | 4035 | 0.41 | |
| CDK2 | CDK | CMGC | 1ke8 | A | | 4-{[(2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]amino}-n-(1,3-thiazol-2-yl)benzenesulfonamide | Human | 4048 | 0.43 | |
| VRK1 | VRK | CK1 | 5ukf | C | | 4-{[(z)-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}benzene-1-sulfonamide | Human | 8027 | 1.00 | |
| VRK1 | VRK | CK1 | 5ukf | D | | 4-{[(z)-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}benzene-1-sulfonamide | Human | 8028 | 1.00 | |
| CDK2 | CDK | CMGC | 4fkr | A | B | (8z)-8-{[(2,2-dioxido-1,3-dihydro-2-benzothiophen-5-yl)amino]methylidene}-6,8-dihydro-7h-[1,3]thiazolo[5,4-e]indol-7-one | Human | 4535 | 0.66 | |
| STK24 (MST3) | STE20 | STE | 4qmo | A | A | (8z)-8-(1h-imidazol-5-ylmethylidene)-6,8-dihydro-7h-[1,3]thiazolo[5,4-e]indol-7-one | Human | 5585 | 0.52 | |
| STK24 (MST3) | STE20 | STE | 4qmo | A | B | (8z)-8-(1h-imidazol-5-ylmethylidene)-6,8-dihydro-7h-[1,3]thiazolo[5,4-e]indol-7-one | Human | 5597 | 0.52 | |
| CDK2 | CDK | CMGC | 1ke5 | A | | n-methyl-4-{[(2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]amino}benzenesulfonamide | Human | 4376 | 0.41 | |
| VRK1 | VRK | CK1 | 5ukf | B | | 4-{[(z)-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}benzene-1-sulfonamide | Human | 8029 | 1.00 | |
| CDK2 | CDK | CMGC | 4fks | A | C | n-[(4-{[(z)-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}phenyl)sulfonyl]acetamide | Human | 4315 | 0.74 | |
| CDK2 | CDK | CMGC | 4fkp | A | B | 3-{[4-([amino(imino)methyl]aminosulfonyl)anilino]methylene}-2-oxo-2,3-dihydro-1h-indole | Human | 4313 | 0.41 | |
| CDK2 | CDK | CMGC | 4fkq | A | B | 4-[(2z)-2-(7-oxidanylidene-3,6-dihydropyrrolo[3,2-e]benzotriazol-8-ylidene)hydrazinyl]benzenesulfonamide | Human | 4026 | 0.41 | |
| CDK2 | CDK | CMGC | 4fks | A | B | n-[(4-{[(z)-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}phenyl)sulfonyl]acetamide | Human | 4489 | 0.74 | |
| VRK1 | VRK | CK1 | 5ukf | A | | 4-{[(z)-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}benzene-1-sulfonamide | Human | 8030 | 1.00 | |
