Search results (16 entries covering 6 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetailsSimilarity (MFP)File
ACVR1 (ALK2)STKRTKL3mtfBB3-[6-amino-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenolHuman15300.44
VRK2VRKCK16ncgB4-[6-amino-5-(3,5-difluoro-4-hydroxyphenyl)pyridin-3-yl]benzene-1-sulfonamideHuman108510.71
ACVR1 (ALK2)STKRTKL3mtfAA3-[6-amino-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenolHuman15130.44
VRK1VRKCK16bu6DA4,4'-(2-aminopyridine-3,5-diyl)bis(2,6-difluorophenol)Human94131.00
ACVR1 (ALK2)STKRTKL3mtfAB3-[6-amino-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenolHuman15210.44
ACVR1 (ALK2)STKRTKL3mtfBA3-[6-amino-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenolHuman15150.44
VRK1VRKCK16bu6DB4,4'-(2-aminopyridine-3,5-diyl)bis(2,6-difluorophenol)Human94101.00
ACVR1 (ALK2)STKRTKL6eixAB3-[6-amino-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenolHuman85330.44
MAP4K4 (HGK)STE20STE5j95A1-{4-[6-amino-5-(4-chlorophenyl)pyridin-3-yl]phenyl}cyclopentane-1-carboxylic acidHuman79990.40
VRK2VRKCK16ncgA4-[6-amino-5-(3,5-difluoro-4-hydroxyphenyl)pyridin-3-yl]benzene-1-sulfonamideHuman108520.71
MAP4K4 (HGK)STE20STE5di1A4-{6-amino-5-[4-(methylsulfonyl)phenyl]pyridin-3-yl}phenolHuman63540.44
VRK1VRKCK16bu6BB4,4'-(2-aminopyridine-3,5-diyl)bis(2,6-difluorophenol)Human94221.00
VRK1VRKCK16bu6AB4,4'-(2-aminopyridine-3,5-diyl)bis(2,6-difluorophenol)Human94171.00
VRK1VRKCK16bu6AA4,4'-(2-aminopyridine-3,5-diyl)bis(2,6-difluorophenol)Human94231.00
ACVR1 (ALK2)STKRTKL6eixAA3-[6-amino-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenolHuman85300.44
VRK1VRKCK16bu6BA4,4'-(2-aminopyridine-3,5-diyl)bis(2,6-difluorophenol)Human94211.00