Search results (16 entries covering 8 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetailsSimilarity (MFP)File
FGFR1FGFRTK7ozbAA4-[3-(4-piperazin-4-ium-1-ylphenyl)-1h-indazol-6-yl]phenolHuman140100.40
FGFR2FGFRTK7ozyAA4-[3-(4-piperazin-4-ium-1-ylphenyl)-1h-indazol-6-yl]phenolHuman139990.40
FGFR2FGFRTK7ozyAB4-[3-(4-piperazin-4-ium-1-ylphenyl)-1h-indazol-6-yl]phenolHuman139980.40
PIM1PIMCAMK6aydAAn-[6-(4-hydroxyphenyl)-2h-indazol-3-yl]cyclopropanecarboxamideHuman94421.00
FGFR1FGFRTK7ozdAAn-[6-(4-hydroxyphenyl)-1h-indazol-3-yl]benzamideHuman140070.42
FGFR1FGFRTK4zsaAA4-(4-ethylpiperazin-1-yl)-n-[6-(3-methoxyphenyl)-2h-indazol-3-yl]benzamideHuman34910.44
AURKA (AurA)AurOther3lauAn-[6-(4-hydroxyphenyl)-1h-indazol-3-yl]butanamideHuman19710.42
PIM1PIMCAMK6aydABn-[6-(4-hydroxyphenyl)-2h-indazol-3-yl]cyclopropanecarboxamideHuman94431.00
BMP2K (BIKE)NAKOther5i3oBn-(6-{3-[(dimethylsulfamoyl)amino]phenyl}-1h-indazol-3-yl)cyclopropanecarboxamideHuman64340.40
BMP2K (BIKE)NAKOther5ikwAn-(6-{3-[(cyclopropylsulfonyl)amino]phenyl}-1h-indazol-3-yl)cyclopropanecarboxamideHuman67090.42
BMP2K (BIKE)NAKOther5i3oAn-(6-{3-[(dimethylsulfamoyl)amino]phenyl}-1h-indazol-3-yl)cyclopropanecarboxamideHuman64370.40
FGFR1FGFRTK7ozbAB4-[3-(4-piperazin-4-ium-1-ylphenyl)-1h-indazol-6-yl]phenolHuman140080.40
FGFR1FGFRTK7ozdABn-[6-(4-hydroxyphenyl)-1h-indazol-3-yl]benzamideHuman140090.42
FGFR1FGFRTK4zsaBA4-(4-ethylpiperazin-1-yl)-n-[6-(3-methoxyphenyl)-2h-indazol-3-yl]benzamideHuman35720.44
FGFR1FGFRTK4zsaBB4-(4-ethylpiperazin-1-yl)-n-[6-(3-methoxyphenyl)-2h-indazol-3-yl]benzamideHuman35120.44
FGFR1FGFRTK4zsaAB4-(4-ethylpiperazin-1-yl)-n-[6-(3-methoxyphenyl)-2h-indazol-3-yl]benzamideHuman34870.44