Search results (8 entries covering 4 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetailsSimilarity (MFP)File
TGFBR1 (TGFbR1)STKRTKL5qimABn-{4-[3-(5-methoxypyridin-2-yl)-1h-pyrrolo[3,2-b]pyridin-2-yl]pyridin-2-yl}acetamideHuman106610.74
TGFBR1 (TGFbR1)STKRTKL5qikABn-{4-[3-(6-fluoropyridin-3-yl)-4-oxo-4,5,6,7-tetrahydro-1h-pyrrolo[3,2-c]pyridin-2-yl]pyridin-2-yl}acetamideHuman106620.46
TGFBR1 (TGFbR1)STKRTKL5qilABn-{4-[3-(6-methoxypyridin-3-yl)-1h-pyrrolo[3,2-b]pyridin-2-yl]pyridin-2-yl}acetamideHuman106601.00
TGFBR1 (TGFbR1)STKRTKL5qikAAn-{4-[3-(6-fluoropyridin-3-yl)-4-oxo-4,5,6,7-tetrahydro-1h-pyrrolo[3,2-c]pyridin-2-yl]pyridin-2-yl}acetamideHuman106570.46
TGFBR1 (TGFbR1)STKRTKL5qimAAn-{4-[3-(5-methoxypyridin-2-yl)-1h-pyrrolo[3,2-b]pyridin-2-yl]pyridin-2-yl}acetamideHuman106580.74
TGFBR2 (TGFbR2)STKRTKL5qinABn-{4-[3-(6-methoxypyridin-3-yl)-1h-pyrrolo[3,2-b]pyridin-2-yl]pyridin-2-yl}acetamideHuman106631.00
TGFBR2 (TGFbR2)STKRTKL5qinAAn-{4-[3-(6-methoxypyridin-3-yl)-1h-pyrrolo[3,2-b]pyridin-2-yl]pyridin-2-yl}acetamideHuman106641.00
TGFBR1 (TGFbR1)STKRTKL5qilAAn-{4-[3-(6-methoxypyridin-3-yl)-1h-pyrrolo[3,2-b]pyridin-2-yl]pyridin-2-yl}acetamideHuman106591.00