| DYRK1A | DYRK | CMGC | 6eif | A | | 4-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)benzenesulfonamide | Human | 10534 | 0.45 | |
| CHUK (IKKa) | IKK | Other | 5ebz | B | | 2-azanyl-5-phenyl-3-(4-sulfamoylphenyl)benzamide | Human | 7145 | 0.40 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2wtc | A | | 4-[2-amino-5-(4-hydroxy-3-methoxyphenyl)pyridin-3-yl]benzamide | Human | 4767 | 0.40 | |
| VRK2 | VRK | CK1 | 6ncg | B | | 4-[6-amino-5-(3,5-difluoro-4-hydroxyphenyl)pyridin-3-yl]benzene-1-sulfonamide | Human | 10851 | 1.00 | |
| VRK1 | VRK | CK1 | 6bu6 | D | A | 4,4'-(2-aminopyridine-3,5-diyl)bis(2,6-difluorophenol) | Human | 9413 | 0.71 | |
| DYRK1A | DYRK | CMGC | 6eif | B | | 4-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)benzenesulfonamide | Human | 10544 | 0.45 | |
| CHUK (IKKa) | IKK | Other | 5ebz | K | | 2-azanyl-5-phenyl-3-(4-sulfamoylphenyl)benzamide | Human | 7150 | 0.40 | |
| CHUK (IKKa) | IKK | Other | 5ebz | L | | 2-azanyl-5-phenyl-3-(4-sulfamoylphenyl)benzamide | Human | 7147 | 0.40 | |
| CHUK (IKKa) | IKK | Other | 5ebz | D | | 2-azanyl-5-phenyl-3-(4-sulfamoylphenyl)benzamide | Human | 7144 | 0.40 | |
| CHUK (IKKa) | IKK | Other | 5ebz | J | | 2-azanyl-5-phenyl-3-(4-sulfamoylphenyl)benzamide | Human | 7148 | 0.40 | |
| VRK1 | VRK | CK1 | 6bu6 | D | B | 4,4'-(2-aminopyridine-3,5-diyl)bis(2,6-difluorophenol) | Human | 9410 | 0.71 | |
| CHUK (IKKa) | IKK | Other | 5ebz | A | | 2-azanyl-5-phenyl-3-(4-sulfamoylphenyl)benzamide | Human | 7153 | 0.40 | |
| CHUK (IKKa) | IKK | Other | 5ebz | G | | 2-azanyl-5-phenyl-3-(4-sulfamoylphenyl)benzamide | Human | 7154 | 0.40 | |
| CHUK (IKKa) | IKK | Other | 5ebz | I | | 2-azanyl-5-phenyl-3-(4-sulfamoylphenyl)benzamide | Human | 7152 | 0.40 | |
| CHUK (IKKa) | IKK | Other | 5ebz | C | | 2-azanyl-5-phenyl-3-(4-sulfamoylphenyl)benzamide | Human | 7146 | 0.40 | |
| CHUK (IKKa) | IKK | Other | 5ebz | F | | 2-azanyl-5-phenyl-3-(4-sulfamoylphenyl)benzamide | Human | 7149 | 0.40 | |
| CHUK (IKKa) | IKK | Other | 5ebz | H | | 2-azanyl-5-phenyl-3-(4-sulfamoylphenyl)benzamide | Human | 7155 | 0.40 | |
| CHUK (IKKa) | IKK | Other | 5ebz | E | | 2-azanyl-5-phenyl-3-(4-sulfamoylphenyl)benzamide | Human | 7151 | 0.40 | |
| DYRK1A | DYRK | CMGC | 6eif | C | | 4-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)benzenesulfonamide | Human | 10525 | 0.45 | |
| DYRK1A | DYRK | CMGC | 6eif | D | | 4-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)benzenesulfonamide | Human | 10532 | 0.45 | |
| VRK2 | VRK | CK1 | 6ncg | A | | 4-[6-amino-5-(3,5-difluoro-4-hydroxyphenyl)pyridin-3-yl]benzene-1-sulfonamide | Human | 10852 | 1.00 | |
| MAP4K4 (HGK) | STE20 | STE | 5di1 | A | | 4-{6-amino-5-[4-(methylsulfonyl)phenyl]pyridin-3-yl}phenol | Human | 6354 | 0.55 | |
| VRK1 | VRK | CK1 | 6bu6 | B | B | 4,4'-(2-aminopyridine-3,5-diyl)bis(2,6-difluorophenol) | Human | 9422 | 0.71 | |
| VRK1 | VRK | CK1 | 6bu6 | A | B | 4,4'-(2-aminopyridine-3,5-diyl)bis(2,6-difluorophenol) | Human | 9417 | 0.71 | |
| VRK1 | VRK | CK1 | 6bu6 | A | A | 4,4'-(2-aminopyridine-3,5-diyl)bis(2,6-difluorophenol) | Human | 9423 | 0.71 | |
| VRK1 | VRK | CK1 | 6bu6 | B | A | 4,4'-(2-aminopyridine-3,5-diyl)bis(2,6-difluorophenol) | Human | 9421 | 0.71 | |