| HASPIN (Haspin) | Haspin | Other | 7avq | A | A | (2~{r})-2-[[3-(2~{h}-indazol-5-yl)imidazo[1,2-b]pyridazin-6-yl]amino]butan-1-ol | Human | 13176 | 0.42 | |
| ERN1 (IRE1) | IRE | Other | 4z7h | A | | 2-methoxy-4-[6-(propan-2-ylamino)imidazo[1,2-b]pyridazin-3-yl]benzamide | Human | 1794 | 0.41 | |
| PIM1 | PIM | CAMK | 2c3i | B | A | 1-(3-{6-[(cyclopropylmethyl)amino]imidazo[1,2-b]pyridazin-3-yl}phenyl)ethanone | Human | 2348 | 1.00 | |
| DAPK3 | DAPK | CAMK | 3bqr | A | A | 4-(6-{[(1r)-1-(hydroxymethyl)propyl]amino}imidazo[1,2-b]pyridazin-3-yl)benzoic acid | Human | 380 | 0.42 | |
| DAPK3 | DAPK | CAMK | 3bqr | A | B | 4-(6-{[(1r)-1-(hydroxymethyl)propyl]amino}imidazo[1,2-b]pyridazin-3-yl)benzoic acid | Human | 386 | 0.42 | |
| CLK1 | CLK | CMGC | 6yta | A | B | 1-(3-{6-[(cyclopropylmethyl)amino]imidazo[1,2-b]pyridazin-3-yl}phenyl)ethanone | Human | 12417 | 1.00 | |
| HASPIN (Haspin) | Haspin | Other | 3f2n | A | B | (2s)-2-{[3-(3-aminophenyl)imidazo[1,2-b]pyridazin-6-yl]amino}-3-methylbutan-1-ol | Human | 3813 | 0.46 | |
| ACVR1 (ALK2) | STKR | TKL | 4dym | A | | 1-(3-{6-[(cyclopropylmethyl)amino]imidazo[1,2-b]pyridazin-3-yl}phenyl)ethanone | Human | 1509 | 1.00 | |
| ACVR1 (ALK2) | STKR | TKL | 3oom | A | A | 1-{3-[6-(tetrahydro-2h-pyran-4-ylamino)imidazo[1,2-b]pyridazin-3-yl]phenyl}ethanone | Human | 1517 | 0.68 | |
| ACVR1 (ALK2) | STKR | TKL | 3oom | A | B | 1-{3-[6-(tetrahydro-2h-pyran-4-ylamino)imidazo[1,2-b]pyridazin-3-yl]phenyl}ethanone | Human | 1518 | 0.68 | |
| NTRK3 (TRKC) | Trk | TK | 4ymj | B | A | 4-[6-(benzylamino)imidazo[1,2-b]pyridazin-3-yl]benzonitrile | Human | 100 | 0.44 | |
| NTRK3 (TRKC) | Trk | TK | 4ymj | B | B | 4-[6-(benzylamino)imidazo[1,2-b]pyridazin-3-yl]benzonitrile | Human | 99 | 0.44 | |
| NTRK3 (TRKC) | Trk | TK | 4ymj | A | B | 4-[6-(benzylamino)imidazo[1,2-b]pyridazin-3-yl]benzonitrile | Human | 98 | 0.44 | |
| NTRK3 (TRKC) | Trk | TK | 4ymj | A | A | 4-[6-(benzylamino)imidazo[1,2-b]pyridazin-3-yl]benzonitrile | Human | 101 | 0.44 | |
| PIM1 | PIM | CAMK | 2c3i | B | B | 1-(3-{6-[(cyclopropylmethyl)amino]imidazo[1,2-b]pyridazin-3-yl}phenyl)ethanone | Human | 2374 | 1.00 | |
| ERN1 (IRE1) | IRE | Other | 4z7h | B | | 2-methoxy-4-[6-(propan-2-ylamino)imidazo[1,2-b]pyridazin-3-yl]benzamide | Human | 1801 | 0.41 | |
| CAMK2D (CaMK2d) | CAMK2 | CAMK | 6ayw | B | | n-[2-(dimethylamino)ethyl]-3-[6-(thiophen-2-yl)imidazo[1,2-b]pyridazin-3-yl]benzamide | Human | 8665 | 0.42 | |
| CAMK2D (CaMK2d) | CAMK2 | CAMK | 6ayw | A | | n-[2-(dimethylamino)ethyl]-3-[6-(thiophen-2-yl)imidazo[1,2-b]pyridazin-3-yl]benzamide | Human | 8666 | 0.42 | |
| CLK1 | CLK | CMGC | 6yta | A | A | 1-(3-{6-[(cyclopropylmethyl)amino]imidazo[1,2-b]pyridazin-3-yl}phenyl)ethanone | Human | 12423 | 1.00 | |
| HASPIN (Haspin) | Haspin | Other | 3f2n | A | A | (2s)-2-{[3-(3-aminophenyl)imidazo[1,2-b]pyridazin-6-yl]amino}-3-methylbutan-1-ol | Human | 3803 | 0.46 | |
| HASPIN (Haspin) | Haspin | Other | 7avq | A | B | (2~{r})-2-[[3-(2~{h}-indazol-5-yl)imidazo[1,2-b]pyridazin-6-yl]amino]butan-1-ol | Human | 13175 | 0.42 | |