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Search results (11 entries covering 6 PDB structures)
#
Kinase
Family
Group
PDB
Chain
(Alternate) Model
Orthosteric ligand
Organism
Details
Similarity (MFP)
File
PRKACA (PKACa)
PKA
AGC
5uzk
A
A
2-{3-[3-(piperidin-4-yl)propoxy]phenyl}-n-[4-(1h-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamide
Human
9726
1.00
ROCK1
DMPK
AGC
5uzj
A
n-[4-(2-aminopyridin-4-yl)-1,3-thiazol-2-yl]-2-(3-methoxyphenyl)acetamide
Human
9706
0.46
ROCK1
DMPK
AGC
5hvu
B
2-{3-[3-(piperidin-4-yl)propoxy]phenyl}-n-[4-(pyridin-4-yl)-1,3-thiazol-2-yl]acetamide
Human
7415
0.74
ROCK1
DMPK
AGC
5kkt
A
2-[3-[3-(4-methylpiperazin-1-yl)propoxy]phenyl]-~{n}-[4-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]ethanamide
Human
8182
0.69
ROCK1
DMPK
AGC
5kks
B
2-[3-(methylsulfonylamino)phenyl]-~{n}-[4-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]ethanamide
Human
8181
0.60
ROCK1
DMPK
AGC
4yve
A
2-(3-methoxyphenyl)-n-[4-(pyridin-4-yl)-1,3-thiazol-2-yl]acetamide
Human
2693
0.44
ROCK1
DMPK
AGC
5hvu
A
2-{3-[3-(piperidin-4-yl)propoxy]phenyl}-n-[4-(pyridin-4-yl)-1,3-thiazol-2-yl]acetamide
Human
7414
0.74
ROCK1
DMPK
AGC
5kks
A
2-[3-(methylsulfonylamino)phenyl]-~{n}-[4-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]ethanamide
Human
8183
0.60
ROCK1
DMPK
AGC
4yve
B
2-(3-methoxyphenyl)-n-[4-(pyridin-4-yl)-1,3-thiazol-2-yl]acetamide
Human
2706
0.44
ROCK1
DMPK
AGC
5kkt
B
2-[3-[3-(4-methylpiperazin-1-yl)propoxy]phenyl]-~{n}-[4-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]ethanamide
Human
8184
0.69
ROCK1
DMPK
AGC
5uzj
B
n-[4-(2-aminopyridin-4-yl)-1,3-thiazol-2-yl]-2-(3-methoxyphenyl)acetamide
Human
9707
0.46
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