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Search results (12 entries covering 7 PDB structures)
#
Kinase
Family
Group
PDB
Chain
(Alternate) Model
Orthosteric ligand
Organism
Details
Similarity (MFP)
File
GRK2 (BARK1)
GRK
AGC
6u7c
A
5-[(3s,4r)-3-{[(2h-1,3-benzodioxol-5-yl)oxy]methyl}piperidin-4-yl]-2-fluoro-n-[(2h-indazol-3-yl)methyl]benzamide
Human
12162
0.57
GRK2 (BARK1)
GRK
AGC
3v5w
A
A
paroxetine
Human
1705
1.00
GRK2 (BARK1)
GRK
AGC
5ukk
A
B
5-[(3s,4r)-3-{[(2h-1,3-benzodioxol-5-yl)oxy]methyl}piperidin-4-yl]-2-fluoro-n-[(pyridin-2-yl)methyl]benzamide
Human
7530
0.60
GRK2 (BARK1)
GRK
AGC
5ukk
A
A
5-[(3s,4r)-3-{[(2h-1,3-benzodioxol-5-yl)oxy]methyl}piperidin-4-yl]-2-fluoro-n-[(pyridin-2-yl)methyl]benzamide
Human
7529
0.60
GRK2 (BARK1)
GRK
AGC
5ukl
A
A
2-{5-[(3s,4r)-3-{[(2h-1,3-benzodioxol-5-yl)oxy]methyl}piperidin-4-yl]-2-fluorophenyl}-n-[2-(1h-pyrazol-4-yl)ethyl]acetamide
Human
7528
0.57
GRK2 (BARK1)
GRK
AGC
3v5w
A
B
paroxetine
Human
1711
1.00
GRK2 (BARK1)
GRK
AGC
4mk0
A
A
5-{[(3s,4r)-4-(4-fluorophenyl)piperidin-3-yl]methoxy}-1h-isoindol-1-one
Human
1710
0.59
GRK2 (BARK1)
GRK
AGC
5wg5
A
B
5-{[(3s,4r)-4-(4-fluorophenyl)piperidin-3-yl]methoxy}-2h-indazole
Human
9440
0.61
GRK2 (BARK1)
GRK
AGC
5wg5
A
A
5-{[(3s,4r)-4-(4-fluorophenyl)piperidin-3-yl]methoxy}-2h-indazole
Human
9437
0.61
GRK2 (BARK1)
GRK
AGC
4mk0
A
B
5-{[(3s,4r)-4-(4-fluorophenyl)piperidin-3-yl]methoxy}-1h-isoindol-1-one
Human
1704
0.59
GRK2 (BARK1)
GRK
AGC
5wg3
A
2-fluoro-5-[(3s,4r)-3-{[(1h-indazol-5-yl)oxy]methyl}piperidin-4-yl]-n-[(1h-pyrazol-3-yl)methyl]benzamide
Human
9439
0.42
GRK2 (BARK1)
GRK
AGC
5ukl
A
B
2-{5-[(3s,4r)-3-{[(2h-1,3-benzodioxol-5-yl)oxy]methyl}piperidin-4-yl]-2-fluorophenyl}-n-[2-(1h-pyrazol-4-yl)ethyl]acetamide
Human
7531
0.57
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