Search results (20 entries covering 11 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetailsSimilarity (MFP)File
CHEK1 (CHK1)CAMKLCAMK7bjeAAadenineHuman137670.41
CHEK1 (CHK1)CAMKLCAMK7bknAadenineHuman137690.41
PDPK1 (PDK1)PDK1AGC5lvmAAadenineHuman71120.41
TGFBR1 (TGFbR1)STKRTKL4x2jAB4-[(3-aminophenyl)amino]pyrido[2,3-d]pyrimidin-5(8h)-oneHuman21150.58
TGFBR1 (TGFbR1)STKRTKL4x2jAA4-[(3-aminophenyl)amino]pyrido[2,3-d]pyrimidin-5(8h)-oneHuman21240.58
TGFBR1 (TGFbR1)STKRTKL4x2fAB4-amino-8-(4-aminophenyl)pyrido[2,3-d]pyrimidin-5(8h)-oneHuman62080.40
CHEK1 (CHK1)CAMKLCAMK7bjeABadenineHuman137730.41
STK24 (MST3)STE20STE3a7iAadenineHuman56110.41
CAMK1D (CaMK1d)CAMK1CAMK8bfsAA3~{h}-pyrrolo[2,3-c]isoquinolin-5-amineHuman145060.40
CAMK1D (CaMK1d)CAMK1CAMK8bfsAB3~{h}-pyrrolo[2,3-c]isoquinolin-5-amineHuman145050.40
ACVR2B (ACTR2B)STKRTKL2qluAadenineHuman29400.41
TGFBR1 (TGFbR1)STKRTKL4x2fAA4-amino-8-(4-aminophenyl)pyrido[2,3-d]pyrimidin-5(8h)-oneHuman62070.40
PDPK1 (PDK1)PDK1AGC5lvmACadenineHuman71380.41
PDPK1 (PDK1)PDK1AGC5lvmABadenineHuman71030.41
RETRetTK6njaAAadenineHuman111460.41
RETRetTK6njaABadenineHuman111450.41
TGFBR1 (TGFbR1)STKRTKL4x0mAB4-aminopyrido[2,3-d]pyrimidin-5(8h)-oneHuman21211.00
TGFBR1 (TGFbR1)STKRTKL4x0mAA4-aminopyrido[2,3-d]pyrimidin-5(8h)-oneHuman21221.00
Prkci (PKCi)PKCAGC4dc2ABadenineMouse58290.41
Prkci (PKCi)PKCAGC4dc2AAadenineMouse58300.41