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Search results (16 entries covering 7 PDB structures)
#
Kinase
Family
Group
PDB
Chain
(Alternate) Model
Orthosteric ligand
Organism
Details
Similarity (MFP)
File
ROCK1
DMPK
AGC
5uzj
A
n-[4-(2-aminopyridin-4-yl)-1,3-thiazol-2-yl]-2-(3-methoxyphenyl)acetamide
Human
9706
0.42
ROCK1
DMPK
AGC
4yvc
A
2-fluoro-n-[4-(pyridin-4-yl)-1,3-thiazol-2-yl]benzamide
Human
2715
0.47
ROCK1
DMPK
AGC
5hvu
B
2-{3-[3-(piperidin-4-yl)propoxy]phenyl}-n-[4-(pyridin-4-yl)-1,3-thiazol-2-yl]acetamide
Human
7415
0.44
Map3k14 (NIK)
STE-Unique
STE
4g3g
A
A
4-fluoro-2-{[4-(pyridin-4-yl)-1,3-thiazol-2-yl]amino}phenol
Mouse
5793
0.43
ROCK1
DMPK
AGC
3tv7
B
1-[(1r)-1-(3-methoxyphenyl)ethyl]-3-(4-pyridin-4-yl-1,3-thiazol-2-yl)urea
Human
2703
0.49
ROCK1
DMPK
AGC
4yve
A
2-(3-methoxyphenyl)-n-[4-(pyridin-4-yl)-1,3-thiazol-2-yl]acetamide
Human
2693
0.54
Map3k14 (NIK)
STE-Unique
STE
4g3g
A
B
4-fluoro-2-{[4-(pyridin-4-yl)-1,3-thiazol-2-yl]amino}phenol
Mouse
5791
0.43
ROCK1
DMPK
AGC
3twj
C
1-[(3-hydroxyphenyl)methyl]-3-(4-pyridin-4-yl-1,3-thiazol-2-yl)urea
Human
2689
1.00
ROCK1
DMPK
AGC
5hvu
A
2-{3-[3-(piperidin-4-yl)propoxy]phenyl}-n-[4-(pyridin-4-yl)-1,3-thiazol-2-yl]acetamide
Human
7414
0.44
ROCK1
DMPK
AGC
3twj
A
1-[(3-hydroxyphenyl)methyl]-3-(4-pyridin-4-yl-1,3-thiazol-2-yl)urea
Human
2710
1.00
ROCK1
DMPK
AGC
4yve
B
2-(3-methoxyphenyl)-n-[4-(pyridin-4-yl)-1,3-thiazol-2-yl]acetamide
Human
2706
0.54
ROCK1
DMPK
AGC
4yvc
B
2-fluoro-n-[4-(pyridin-4-yl)-1,3-thiazol-2-yl]benzamide
Human
2727
0.47
ROCK1
DMPK
AGC
3tv7
D
1-[(1r)-1-(3-methoxyphenyl)ethyl]-3-(4-pyridin-4-yl-1,3-thiazol-2-yl)urea
Human
2725
0.49
ROCK1
DMPK
AGC
3tv7
C
1-[(1r)-1-(3-methoxyphenyl)ethyl]-3-(4-pyridin-4-yl-1,3-thiazol-2-yl)urea
Human
2717
0.49
ROCK1
DMPK
AGC
5uzj
B
n-[4-(2-aminopyridin-4-yl)-1,3-thiazol-2-yl]-2-(3-methoxyphenyl)acetamide
Human
9707
0.42
ROCK1
DMPK
AGC
3tv7
A
1-[(1r)-1-(3-methoxyphenyl)ethyl]-3-(4-pyridin-4-yl-1,3-thiazol-2-yl)urea
Human
2697
0.49
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