Search results (15 entries covering 7 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetailsSimilarity (MFP)File
MAPK1 (Erk2)MAPKCMGC8ao6AB~{n}-(1~{h}-indazol-5-ylmethyl)ethanamideHuman143960.50
MAPK1 (Erk2)MAPKCMGC8ao2AB~{n}-(1~{h}-indazol-5-ylmethyl)propanamideHuman143940.46
MAPK1 (Erk2)MAPKCMGC8ao4AA~{n}-(1~{h}-indazol-5-yl)ethanesulfonamideHuman144160.44
MAPK1 (Erk2)MAPKCMGC8ao2AA~{n}-(1~{h}-indazol-5-ylmethyl)propanamideHuman144150.46
MAPK1 (Erk2)MAPKCMGC8ao4AB~{n}-(1~{h}-indazol-5-yl)ethanesulfonamideHuman143990.44
ROCK1DMPKAGC3v8sA1-(1h-indazol-5-yl)-3-(2-phenylethyl)ureaHuman27161.00
MAPK1 (Erk2)MAPKCMGC8ao5AB~{n}-(1~{h}-indazol-5-ylmethyl)ethanesulfonamideHuman144000.40
RPS6KA3-b (RSK2-b)RSKbCAMK4jg6A(2s)-2-cyano-3-(1h-indazol-5-yl)propanamideHuman14950.40
MAPK1 (Erk2)MAPKCMGC8ao6AA~{n}-(1~{h}-indazol-5-ylmethyl)ethanamideHuman143970.50
MAPK1 (Erk2)MAPKCMGC8ao3AB2-chloranyl-~{n}-(1~{h}-indazol-5-ylmethyl)ethanamideHuman144140.48
MAPK1 (Erk2)MAPKCMGC8ao3AA2-chloranyl-~{n}-(1~{h}-indazol-5-ylmethyl)ethanamideHuman143860.48
MAPK1 (Erk2)MAPKCMGC8ao5AA~{n}-(1~{h}-indazol-5-ylmethyl)ethanesulfonamideHuman143920.40
ROCK1DMPKAGC3v8sD1-(1h-indazol-5-yl)-3-(2-phenylethyl)ureaHuman26921.00
ROCK1DMPKAGC3v8sB1-(1h-indazol-5-yl)-3-(2-phenylethyl)ureaHuman27091.00
ROCK1DMPKAGC3v8sC1-(1h-indazol-5-yl)-3-(2-phenylethyl)ureaHuman27021.00