| PRKACA (PKACa) | PKA | AGC | 5uzk | A | A | 2-{3-[3-(piperidin-4-yl)propoxy]phenyl}-n-[4-(1h-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamide | Human | 9726 | 0.44 | |
| ROCK1 | DMPK | AGC | 5uzj | A | | n-[4-(2-aminopyridin-4-yl)-1,3-thiazol-2-yl]-2-(3-methoxyphenyl)acetamide | Human | 9706 | 0.77 | |
| PRKACA (PKACa) | PKA | AGC | 3poo | A | B | n'-[(e)-(2,4-dihydroxy-6-methylphenyl)methylidene]-2-(3-methoxyphenyl)acetohydrazide | Human | 5285 | 0.40 | |
| PRKACA (PKACa) | PKA | AGC | 3poo | A | A | n'-[(e)-(2,4-dihydroxy-6-methylphenyl)methylidene]-2-(3-methoxyphenyl)acetohydrazide | Human | 5300 | 0.40 | |
| PRKACA (PKACa) | PKA | AGC | 3ovv | A | A | n'-[(1e)-(4-hydroxyphenyl)methylidene]-2-(3-methoxyphenyl)acetohydrazide | Human | 5266 | 0.43 | |
| ROCK1 | DMPK | AGC | 4yvc | A | | 2-fluoro-n-[4-(pyridin-4-yl)-1,3-thiazol-2-yl]benzamide | Human | 2715 | 0.46 | |
| ROCK1 | DMPK | AGC | 5hvu | B | | 2-{3-[3-(piperidin-4-yl)propoxy]phenyl}-n-[4-(pyridin-4-yl)-1,3-thiazol-2-yl]acetamide | Human | 7415 | 0.63 | |
| ROCK1 | DMPK | AGC | 5kkt | A | | 2-[3-[3-(4-methylpiperazin-1-yl)propoxy]phenyl]-~{n}-[4-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]ethanamide | Human | 8182 | 0.46 | |
| ROCK1 | DMPK | AGC | 5kks | B | | 2-[3-(methylsulfonylamino)phenyl]-~{n}-[4-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]ethanamide | Human | 8181 | 0.46 | |
| ROCK1 | DMPK | AGC | 3tv7 | B | | 1-[(1r)-1-(3-methoxyphenyl)ethyl]-3-(4-pyridin-4-yl-1,3-thiazol-2-yl)urea | Human | 2703 | 0.63 | |
| ROCK1 | DMPK | AGC | 4yve | A | | 2-(3-methoxyphenyl)-n-[4-(pyridin-4-yl)-1,3-thiazol-2-yl]acetamide | Human | 2693 | 1.00 | |
| PRKACA (PKACa) | PKA | AGC | 3ovv | A | B | n'-[(1e)-(4-hydroxyphenyl)methylidene]-2-(3-methoxyphenyl)acetohydrazide | Human | 5269 | 0.43 | |
| ROCK1 | DMPK | AGC | 3twj | C | | 1-[(3-hydroxyphenyl)methyl]-3-(4-pyridin-4-yl-1,3-thiazol-2-yl)urea | Human | 2689 | 0.54 | |
| ROCK1 | DMPK | AGC | 5hvu | A | | 2-{3-[3-(piperidin-4-yl)propoxy]phenyl}-n-[4-(pyridin-4-yl)-1,3-thiazol-2-yl]acetamide | Human | 7414 | 0.63 | |
| ROCK1 | DMPK | AGC | 5kks | A | | 2-[3-(methylsulfonylamino)phenyl]-~{n}-[4-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]ethanamide | Human | 8183 | 0.46 | |
| ROCK1 | DMPK | AGC | 3twj | A | | 1-[(3-hydroxyphenyl)methyl]-3-(4-pyridin-4-yl-1,3-thiazol-2-yl)urea | Human | 2710 | 0.54 | |
| ROCK1 | DMPK | AGC | 4yve | B | | 2-(3-methoxyphenyl)-n-[4-(pyridin-4-yl)-1,3-thiazol-2-yl]acetamide | Human | 2706 | 1.00 | |
| ROCK1 | DMPK | AGC | 4yvc | B | | 2-fluoro-n-[4-(pyridin-4-yl)-1,3-thiazol-2-yl]benzamide | Human | 2727 | 0.46 | |
| ROCK1 | DMPK | AGC | 5kkt | B | | 2-[3-[3-(4-methylpiperazin-1-yl)propoxy]phenyl]-~{n}-[4-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]ethanamide | Human | 8184 | 0.46 | |
| ROCK1 | DMPK | AGC | 3tv7 | D | | 1-[(1r)-1-(3-methoxyphenyl)ethyl]-3-(4-pyridin-4-yl-1,3-thiazol-2-yl)urea | Human | 2725 | 0.63 | |
| ROCK1 | DMPK | AGC | 3tv7 | C | | 1-[(1r)-1-(3-methoxyphenyl)ethyl]-3-(4-pyridin-4-yl-1,3-thiazol-2-yl)urea | Human | 2717 | 0.63 | |
| ROCK1 | DMPK | AGC | 5uzj | B | | n-[4-(2-aminopyridin-4-yl)-1,3-thiazol-2-yl]-2-(3-methoxyphenyl)acetamide | Human | 9707 | 0.77 | |
| ROCK1 | DMPK | AGC | 3tv7 | A | | 1-[(1r)-1-(3-methoxyphenyl)ethyl]-3-(4-pyridin-4-yl-1,3-thiazol-2-yl)urea | Human | 2697 | 0.63 | |
