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Search results (8 entries covering 4 PDB structures)
#
Kinase
Family
Group
PDB
Chain
(Alternate) Model
Orthosteric ligand
Organism
Details
Similarity (MFP)
File
PAK4
STE20
STE
5vef
A
A
5-(1,4-diazepan-1-sulfonyl)isoquinoline
Human
8569
0.43
ROCK1
DMPK
AGC
3d9v
A
(s)-2-methyl-1-[(4-methyl-5-isoquinoline)sulfonyl]-homopiperazine
Human
2696
1.00
ROCK1
DMPK
AGC
3d9v
B
(s)-2-methyl-1-[(4-methyl-5-isoquinoline)sulfonyl]-homopiperazine
Human
2701
1.00
CDC42BPB (MRCKb)
DMPK
AGC
3tku
A
5-(1,4-diazepan-1-sulfonyl)isoquinoline
Human
4862
0.43
CDC42BPB (MRCKb)
DMPK
AGC
3tku
B
5-(1,4-diazepan-1-sulfonyl)isoquinoline
Human
4859
0.43
PAK4
STE20
STE
5vef
A
B
5-(1,4-diazepan-1-sulfonyl)isoquinoline
Human
8571
0.43
ROCK1
DMPK
AGC
2esm
A
5-(1,4-diazepan-1-sulfonyl)isoquinoline
Human
2726
0.43
ROCK1
DMPK
AGC
2esm
B
5-(1,4-diazepan-1-sulfonyl)isoquinoline
Human
2714
0.43
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