Search results (101 entries covering 45 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetails File
ACVR1 (ALK2)STKRTKL5s7mAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13666
ACVR1 (ALK2)STKRTKL5s7dAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13668
ACVR1 (ALK2)STKRTKL5s80AB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13669
ACVR1 (ALK2)STKRTKL5s7qAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13670
ACVR1 (ALK2)STKRTKL5s7fAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13671
ACVR1 (ALK2)STKRTKL5s75AA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13714
ACVR1 (ALK2)STKRTKL5s7tAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13723
ACVR1 (ALK2)STKRTKL5s86AB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13729
ACVR1 (ALK2)STKRTKL5s7dAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13730
ACVR1 (ALK2)STKRTKL5s7gAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13713
ACVR1 (ALK2)STKRTKL5s87AA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13738
ACVR1 (ALK2)STKRTKL5s78AA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13716
ACVR1 (ALK2)STKRTKL5s7gAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13717
ACVR1 (ALK2)STKRTKL5s7fAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13737
ACVR1 (ALK2)STKRTKL5s7eAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13715
ACVR1 (ALK2)STKRTKL5s7bAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13719
ACVR1 (ALK2)STKRTKL5s75AB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13718
ACVR1 (ALK2)STKRTKL5s80AA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13728
ACVR1 (ALK2)STKRTKL5s86AA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13724
ACVR1 (ALK2)STKRTKL5s7mAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13739
ACVR1 (ALK2)STKRTKL5s7oAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13733
ACVR1 (ALK2)STKRTKL5s7rAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13731
ACVR1 (ALK2)STKRTKL5s7kAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13732
ACVR1 (ALK2)STKRTKL5s84AA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13734
ACVR1 (ALK2)STKRTKL5s87AB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13735
ACVR1 (ALK2)STKRTKL6srhBB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman11633
ACVR1 (ALK2)STKRTKL5s7eAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13643
ACVR1 (ALK2)STKRTKL5s7xAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13646
ACVR1 (ALK2)STKRTKL5s7kAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13649
ACVR1 (ALK2)STKRTKL5s7zAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13652
ACVR1 (ALK2)STKRTKL5s7rAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13654
ACVR1 (ALK2)STKRTKL5s7wAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13662
ACVR1 (ALK2)STKRTKL5s7iAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13663
ACVR1 (ALK2)STKRTKL5s7oAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13664
ACVR1 (ALK2)STKRTKL5s76AB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13672
ACVR1 (ALK2)STKRTKL5s7lAC-Human13665
ACVR1 (ALK2)STKRTKL5s89AA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13673
ACVR1 (ALK2)STKRTKL5s7lAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13676
ACVR1 (ALK2)STKRTKL5s7sAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13677
ACVR1 (ALK2)STKRTKL5s83AB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13685
ACVR1 (ALK2)STKRTKL5s78AB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13686
ACVR1 (ALK2)STKRTKL5s7xAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13692
ACVR1 (ALK2)STKRTKL5s8aAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13693
ACVR1 (ALK2)STKRTKL5s7lAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13736
ACVR1 (ALK2)STKRTKL5s7sAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13667
ACVR1 (ALK2)STKRTKL5s7cAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13689
ACVR1 (ALK2)STKRTKL5s7pAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13687
ACVR1 (ALK2)STKRTKL5s7pAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13695
ACVR1 (ALK2)STKRTKL5s7uAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13696
ACVR1 (ALK2)STKRTKL5s81AB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13697
ACVR1 (ALK2)STKRTKL5s77AB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13698
ACVR1 (ALK2)STKRTKL5s7iAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13699
ACVR1 (ALK2)STKRTKL5s7cAC-Human13702
ACVR1 (ALK2)STKRTKL5s79AB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13708
ACVR1 (ALK2)STKRTKL5s7tAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13709
ACVR1 (ALK2)STKRTKL5s7vAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13711
ACVR1 (ALK2)STKRTKL5s8bAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13721
ACVR1 (ALK2)STKRTKL5s8bAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13726
ACVR1 (ALK2)STKRTKL5s85AB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13720
ACVR1 (ALK2)STKRTKL5s8aAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13725
ACVR1 (ALK2)STKRTKL5s89AB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13688
ACVR1 (ALK2)STKRTKL5s77AA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13694
ACVR1 (ALK2)STKRTKL5s7cAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13690
ACVR1 (ALK2)STKRTKL5s7aAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13644
ACVR1 (ALK2)STKRTKL5s7oAC-Human13647
ACVR1 (ALK2)STKRTKL5s7nAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13655
ACVR1 (ALK2)STKRTKL5s7uAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13675
ACVR1 (ALK2)STKRTKL5s7zAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13674
ACVR1 (ALK2)STKRTKL5s7cAD-Human13680
ACVR1 (ALK2)STKRTKL5s7jAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13648
ACVR1 (ALK2)STKRTKL5s7qAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13678
ACVR1 (ALK2)STKRTKL5s85AC4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13679
ACVR1 (ALK2)STKRTKL5s82AA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13681
ACVR1 (ALK2)STKRTKL5s7hAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13682
ACVR1 (ALK2)STKRTKL5s7aAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13683
ACVR1 (ALK2)STKRTKL5s7yAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13684
ACVR1 (ALK2)STKRTKL5s81AA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13661
ACVR1 (ALK2)STKRTKL5s76AA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13691
ACVR1 (ALK2)STKRTKL5s7wAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13700
ACVR1 (ALK2)STKRTKL5s82AB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13701
ACVR1 (ALK2)STKRTKL5s7mAC-Human13705
ACVR1 (ALK2)STKRTKL5s84AC4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13722
ACVR1 (ALK2)STKRTKL5s7yAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13727
ACVR1 (ALK2)STKRTKL6srhAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman11632
ACVR1 (ALK2)STKRTKL6srhAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman11630
ACVR1 (ALK2)STKRTKL6srhBA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman11631
ACVR1 (ALK2)STKRTKL5s88AB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13703
ACVR1 (ALK2)STKRTKL5s79AA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13704
ACVR1 (ALK2)STKRTKL5s7vAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13707
ACVR1 (ALK2)STKRTKL5s83AA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13706
ACVR1 (ALK2)STKRTKL5s7jAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13712
ACVR1 (ALK2)STKRTKL5s7bAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13650
ACVR1 (ALK2)STKRTKL5s7iAC4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13653
ACVR1 (ALK2)STKRTKL5s9kAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13645
ACVR1 (ALK2)STKRTKL5s84AB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13656
ACVR1 (ALK2)STKRTKL5s9kAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13658
ACVR1 (ALK2)STKRTKL5s7hAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13660
ACVR1 (ALK2)STKRTKL5s7sAC4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13651
ACVR1 (ALK2)STKRTKL5s88AA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13657
ACVR1 (ALK2)STKRTKL5s7nAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13659
ACVR1 (ALK2)STKRTKL5s85AA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13710