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Search results (191 entries covering 21 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetails File
VRK1VRKCK16bp0AB-Human8738
VRK1VRKCK12rsvA10-Human4873
VRK1VRKCK12lavA16-Human4888
VRK1VRKCK16ac9DAphosphoaminophosphonic acid-adenylate esterHuman10821
VRK1VRKCK15uvfA(7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(3-methylbutyl)-7,8-dihydropteridin-6(5h)-oneHuman7521
VRK1VRKCK13op5AA[4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrileHuman4870
VRK1VRKCK16dd4AB-Human9939
VRK1VRKCK16cnxAB(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-8-(3-methylbutyl)-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman9810
VRK1VRKCK16dd4DA(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-dipropyl-7,8-dihydropteridin-6(5h)-oneHuman9938
VRK1VRKCK16bp0AA-Human8744
VRK1VRKCK12kulA9-Human4869
VRK1VRKCK16cqhCA-Human9772
VRK1VRKCK12lavA5-Human4891
VRK1VRKCK16cmmDA(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman9764
VRK1VRKCK16cswBB(7r)-5-butyl-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7,8-dimethyl-7,8-dihydropteridin-6(5h)-oneHuman9808
VRK1VRKCK12ktyA17-Human4920
VRK1VRKCK12kulA10-Human4901
VRK1VRKCK16bruCB-Human9086
VRK1VRKCK12ktyA14-Human4926
VRK1VRKCK12lavA12-Human4946
VRK1VRKCK16bp0DB(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7,8-trimethyl-7,8-dihydropteridin-6(5h)-oneHuman8739
VRK1VRKCK12ktyA13-Human4922
VRK1VRKCK16bu6DA4,4'-(2-aminopyridine-3,5-diyl)bis(2,6-difluorophenol)Human9413
VRK1VRKCK16npnB(7r)-7-methyl-2-[(3-oxo-2,3-dihydro-1h-indazol-6-yl)amino]-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman11244
VRK1VRKCK13op5CA[4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrileHuman4886
VRK1VRKCK15ukfC4-{[(z)-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}benzene-1-sulfonamideHuman8027
VRK1VRKCK16cnxDA(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-8-(3-methylbutyl)-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman9814
VRK1VRKCK16cqhDA(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-ethyl-7-methyl-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman9771
VRK1VRKCK12kulA2-Human4921
VRK1VRKCK16vzhD(7~{r})-2-[[3,5-bis(fluoranyl)-4-oxidanyl-phenyl]amino]-5,7-dimethyl-8-prop-2-ynyl-7~{h}-pteridin-6-oneHuman12055
VRK1VRKCK16dd4DB(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-dipropyl-7,8-dihydropteridin-6(5h)-oneHuman9934
VRK1VRKCK15ukfD4-{[(z)-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}benzene-1-sulfonamideHuman8028
VRK1VRKCK12kulA17-Human4893
VRK1VRKCK16cswCA-Human9816
VRK1VRKCK12lavA18-Human4927
VRK1VRKCK12ktyA5-Human4900
VRK1VRKCK12rsvA12-Human4952
VRK1VRKCK16bu6CB-Human9414
VRK1VRKCK12lavA1-Human4930
VRK1VRKCK16bruAA-Human9085
VRK1VRKCK16bu6DB4,4'-(2-aminopyridine-3,5-diyl)bis(2,6-difluorophenol)Human9410
VRK1VRKCK13op5DB[4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrileHuman4892
VRK1VRKCK16cswCB-Human9811
VRK1VRKCK12ktyA18-Human4904
VRK1VRKCK12rsvA5-Human4899
VRK1VRKCK16dd4CA-Human9940
VRK1VRKCK12ktyA1-Human4877
VRK1VRKCK16cfmBB(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman9725
VRK1VRKCK16bp0BA(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7,8-trimethyl-7,8-dihydropteridin-6(5h)-oneHuman8740
VRK1VRKCK13op5DA[4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrileHuman4878
VRK1VRKCK12ktyA4-Human4938
VRK1VRKCK12rsvA4-Human4907
VRK1VRKCK16cfmBA(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman9724
VRK1VRKCK12kulA20-Human4915
VRK1VRKCK16cnxAA(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-8-(3-methylbutyl)-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman9815
VRK1VRKCK16btwDA2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-phenyl-7,8-dihydropteridin-6(5h)-oneHuman9415
VRK1VRKCK12rsvA15-Human4911
VRK1VRKCK12lavA19-Human4940
VRK1VRKCK16cfmDA(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman9721
VRK1VRKCK16bruBB(7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7,8-trimethyl-7,8-dihydropteridin-6(5h)-oneHuman9087
VRK1VRKCK12ktyA2-Human4947
VRK1VRKCK16cqhDB(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-ethyl-7-methyl-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman9767
VRK1VRKCK12kulA12-Human4883
VRK1VRKCK12ktyA19-Human4875
VRK1VRKCK16ac9DBphosphoaminophosphonic acid-adenylate esterHuman10820
VRK1VRKCK12lavA14-Human4898
VRK1VRKCK16ac9CAphosphoaminophosphonic acid-adenylate esterHuman10822
VRK1VRKCK16vxuB(7r)-8-(cyclopropylmethyl)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman13362
VRK1VRKCK16cfmAA(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman9723
VRK1VRKCK12lavA6-Human4871
VRK1VRKCK16cnxBA(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-8-(3-methylbutyl)-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman9803
VRK1VRKCK15uvfD(7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(3-methylbutyl)-7,8-dihydropteridin-6(5h)-oneHuman7522
VRK1VRKCK16cnxCB(7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-8-(3-methylbutyl)-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman9804
VRK1VRKCK12rsvA3-Human4913
VRK1VRKCK16cmmBB(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman9761
VRK1VRKCK16ac9CBphosphoaminophosphonic acid-adenylate esterHuman10819
VRK1VRKCK16dd4BB(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-dipropyl-7,8-dihydropteridin-6(5h)-oneHuman9933
VRK1VRKCK16cmmAB-Human9760
VRK1VRKCK16dd4AA-Human9935
VRK1VRKCK16cmmBA(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman9766
VRK1VRKCK12kulA14-Human4909
VRK1VRKCK16cswDA(7r)-5-butyl-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7,8-dimethyl-7,8-dihydropteridin-6(5h)-oneHuman9817
VRK1VRKCK12rsvA13-Human4935
VRK1VRKCK12ktyA6-Human4929
VRK1VRKCK12kulA6-Human4949
VRK1VRKCK16btwCA-Human9419
VRK1VRKCK16cmmCA-Human9765
VRK1VRKCK13op5CB[4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrileHuman4879
VRK1VRKCK16ac9ABphosphoaminophosphonic acid-adenylate esterHuman10817
VRK1VRKCK16bp0DA(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7,8-trimethyl-7,8-dihydropteridin-6(5h)-oneHuman8745
VRK1VRKCK16btwCB-Human9416
VRK1VRKCK12ktyA3-Human4874
VRK1VRKCK12lavA15-Human4931
VRK1VRKCK16vzhB(7~{r})-2-[[3,5-bis(fluoranyl)-4-oxidanyl-phenyl]amino]-5,7-dimethyl-8-prop-2-ynyl-7~{h}-pteridin-6-oneHuman12056
VRK1VRKCK15ukfB4-{[(z)-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}benzene-1-sulfonamideHuman8029
VRK1VRKCK12ktyA16-Human4937
VRK1VRKCK12lavA7-Human4936
VRK1VRKCK16bp0BB(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7,8-trimethyl-7,8-dihydropteridin-6(5h)-oneHuman8741
VRK1VRKCK12ktyA8-Human4939
VRK1VRKCK16npnA(7r)-7-methyl-2-[(3-oxo-2,3-dihydro-1h-indazol-6-yl)amino]-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman11243
VRK1VRKCK12lavA17-Human4950
VRK1VRKCK12lavA10-Human4882
VRK1VRKCK16bu6BB4,4'-(2-aminopyridine-3,5-diyl)bis(2,6-difluorophenol)Human9422
VRK1VRKCK12rsvA7-Human4889
VRK1VRKCK16bu6CA-Human9412
VRK1VRKCK12rsvA17-Human4951
VRK1VRKCK16bu6AB4,4'-(2-aminopyridine-3,5-diyl)bis(2,6-difluorophenol)Human9417
VRK1VRKCK16cmmAA-Human9763
VRK1VRKCK16bruCA-Human9089
VRK1VRKCK16cqhAB(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-ethyl-7-methyl-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman9768
VRK1VRKCK12ktyA15-Human4953
VRK1VRKCK15uvfB(7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(3-methylbutyl)-7,8-dihydropteridin-6(5h)-oneHuman7523
VRK1VRKCK16ac9BAphosphoaminophosphonic acid-adenylate esterHuman10818
VRK1VRKCK12kulA5-Human4954
VRK1VRKCK12rsvA2-Human4914
VRK1VRKCK12ktyA12-Human4897
VRK1VRKCK16bu6AA4,4'-(2-aminopyridine-3,5-diyl)bis(2,6-difluorophenol)Human9423
VRK1VRKCK16cnxBB(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-8-(3-methylbutyl)-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman9806
VRK1VRKCK12rsvA14-Human4925
VRK1VRKCK12rsvA18-Human4934
VRK1VRKCK16cswBA(7r)-5-butyl-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7,8-dimethyl-7,8-dihydropteridin-6(5h)-oneHuman9812
VRK1VRKCK13op5BA[4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrileHuman4894
VRK1VRKCK12rsvA6-Human4943
VRK1VRKCK16npnC(7r)-7-methyl-2-[(3-oxo-2,3-dihydro-1h-indazol-6-yl)amino]-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman11241
VRK1VRKCK16cswDB(7r)-5-butyl-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7,8-dimethyl-7,8-dihydropteridin-6(5h)-oneHuman9809
VRK1VRKCK16bruBA(7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7,8-trimethyl-7,8-dihydropteridin-6(5h)-oneHuman9088
VRK1VRKCK12lavA13-Human4872
VRK1VRKCK16cmmDB(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman9759
VRK1VRKCK16bp0CB-Human8742
VRK1VRKCK16cfmDB(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman9722
VRK1VRKCK16btwAB2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-phenyl-7,8-dihydropteridin-6(5h)-oneHuman9425
VRK1VRKCK12lavA2-Human4903
VRK1VRKCK12ktyA10-Human4932
VRK1VRKCK16cswAA-Human9818
VRK1VRKCK16bruAB-Human9082
VRK1VRKCK12kulA7-Human4908
VRK1VRKCK12kulA3-Human4895
VRK1VRKCK12kulA11-Human4923
VRK1VRKCK16cfmAB(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman9718
VRK1VRKCK16bruDA(7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7,8-trimethyl-7,8-dihydropteridin-6(5h)-oneHuman9084
VRK1VRKCK16bp0CA-Human8743
VRK1VRKCK12ktyA11-Human4917
VRK1VRKCK16cfmCA-Human9719
VRK1VRKCK16cqhBB(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-ethyl-7-methyl-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman9770
VRK1VRKCK16cqhBA(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-ethyl-7-methyl-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman9769
VRK1VRKCK12kulA18-Human4896
VRK1VRKCK12rsvA9-Human4928
VRK1VRKCK12kulA15-Human4876
VRK1VRKCK12kulA16-Human4924
VRK1VRKCK16dd4CB-Human9936
VRK1VRKCK16cfmCB-Human9720
VRK1VRKCK12ktyA20-Human4890
VRK1VRKCK16cqhAA(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-ethyl-7-methyl-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman9774
VRK1VRKCK16vzhA-Human12057
VRK1VRKCK16btwBA2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-phenyl-7,8-dihydropteridin-6(5h)-oneHuman9424
VRK1VRKCK16cmmCB-Human9762
VRK1VRKCK12lavA9-Human4945
VRK1VRKCK16btwAA2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-phenyl-7,8-dihydropteridin-6(5h)-oneHuman9418
VRK1VRKCK12kulA19-Human4906
VRK1VRKCK16btwBB2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-phenyl-7,8-dihydropteridin-6(5h)-oneHuman9411
VRK1VRKCK12lavA4-Human4884
VRK1VRKCK16cnxDB(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-8-(3-methylbutyl)-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman9807
VRK1VRKCK13op5BB[4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrileHuman4944
VRK1VRKCK16npnD(7r)-7-methyl-2-[(3-oxo-2,3-dihydro-1h-indazol-6-yl)amino]-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman11242
VRK1VRKCK16cqhCB-Human9773
VRK1VRKCK12kulA13-Human4941
VRK1VRKCK12ktyA9-Human4885
VRK1VRKCK12ktyA7-Human4880
VRK1VRKCK12lavA20-Human4933
VRK1VRKCK12rsvA16-Human4905
VRK1VRKCK12kulA8-Human4887
VRK1VRKCK16ac9BBphosphoaminophosphonic acid-adenylate esterHuman10823
VRK1VRKCK12rsvA11-Human4902
VRK1VRKCK12kulA1-Human4919
VRK1VRKCK16btwDB2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-phenyl-7,8-dihydropteridin-6(5h)-oneHuman9420
VRK1VRKCK16ac9AAphosphoaminophosphonic acid-adenylate esterHuman10816
VRK1VRKCK16vzhC-Human12058
VRK1VRKCK16bu6BA4,4'-(2-aminopyridine-3,5-diyl)bis(2,6-difluorophenol)Human9421
VRK1VRKCK12rsvA1-Human4910
VRK1VRKCK16bruDB(7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7,8-trimethyl-7,8-dihydropteridin-6(5h)-oneHuman9083
VRK1VRKCK16cnxCA(7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-8-(3-methylbutyl)-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman9805
VRK1VRKCK13op5AB[4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrileHuman4942
VRK1VRKCK12kulA4-Human4948
VRK1VRKCK16cswAB-Human9813
VRK1VRKCK15ukfA4-{[(z)-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}benzene-1-sulfonamideHuman8030
VRK1VRKCK16dd4BA(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-dipropyl-7,8-dihydropteridin-6(5h)-oneHuman9937
VRK1VRKCK12lavA11-Human4916
VRK1VRKCK15uvfC(7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(3-methylbutyl)-7,8-dihydropteridin-6(5h)-oneHuman7520
VRK1VRKCK12rsvA8-Human4918
VRK1VRKCK12lavA3-Human4912
VRK1VRKCK12lavA8-Human4881
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